Sfoglia per Autore CHIMENTI, Paola
Novel therapeutic opportunities for Toxoplasma gondii, Trichomonas vaginalis, and Giardia intestinalis infections
2023 Arrighi, Francesca; Granese, Arianna; Chimenti, Paola; Guglielmi, Paolo
Novel Insights on Human Carbonic Anhydrase Inhibitors Based on Coumalic Acid: Design, Synthesis, Molecular Modeling Investigation, and Biological Studies
2022 Pontecorvi, Virginia; Mori, Mattia; Picarazzi, Francesca; Zara, Susi; Carradori, Simone; Cataldi, Amelia; Angeli, Andrea; Berrino, Emanuela; Chimenti, Paola; Ciogli, Alessia; Secci, Daniela; Guglielmi, Paolo; Supuran, Claudiu T.
Novel insights on saccharin- and acesulfame-based carbonic anhydrase inhibitors: design, synthesis, modelling investigations and biological activity evaluation
2020 Guglielmi, P.; Rotondi, G.; Secci, D.; Angeli, A.; Chimenti, P.; Nocentini, A.; Bonardi, A.; Gratteri, P.; Carradori, S.; Supuran, C. T.
Phytochemical analyses and pharmacological screening of Neem oil
2019 Cesa, S.; Sisto, F.; Zengin, G.; Scaccabarozzi, D.; Kokolakis, A. K.; Scaltrito, M. M.; Grande, R.; Locatelli, M.; Cacciagrano, F.; Angiolella, L.; Campestre, C.; Granese, A.; Chimenti, P.; Basilico, N.
Benzo[b]tiophen-3-ol derivatives as effective inhibitors of human monoamine oxidase: design, synthesis, and biological activity
2019 Guglielmi, Paolo; Secci, Daniela; Petzer, Anél; Bagetta, Donatella; Chimenti, Paola; Rotondi, Giulia; Ferrante, Claudio; Recinella, Lucia; Leone, Sheila; Alcaro, Stefano; Zengin, Gokhan; Petzer, Jacobus P; Ortuso, Francesco; Carradori, Simone
Design, synthesis, docking studies and monoamine oxidase inhibition of a small library of 1-acetyl- and 1-thiocarbamoyl-3,5-diphenyl-4,5-dihydro-(1h)-pyrazoles
2019 Guglielmi, Paolo; Carradori, Simone; Poli, Giulio; Secci, Daniela; Cirilli, Roberto; Rotondi, Giulia; Chimenti, Paola; Petzer, Anél; Petzer, Jacobus P.
4-(3-Nitrophenyl)thiazol-2-ylhydrazone derivatives as antioxidants and selective hMAO-B inhibitors: synthesis, biological activity and computational analysis
2019 Secci, Daniela; Carradori, Simone; Petzer, Anél; Guglielmi, Paolo; D’Ascenzio, Melissa; Chimenti, Paola; Bagetta, Donatella; Alcaro, Stefano; Zengin, Gokhan; Petzer, Jacobus P.; Ortuso, Francesco
Synthesis and biological evaluation of anti-Toxoplasma gondii activity of a novel scaffold of thiazolidinone derivatives
2017 Carradori, Simone; Secci, Daniela; Bizzarri, Bruna; Chimenti, Paola; DE MONTE, Celeste; Guglielmi, Paolo; Campestre, Cristina; Rivanera, Daniela; Bordón, Claudia; Jones Brando, Lorraine
Novel 1,3-thiazolidin-4-one derivatives as promising anti-Candida agents endowed with anti-oxidant and chelating properties
2016 Secci, Daniela; Simone, Carradori; Bizzarri, Bruna; Chimenti, Paola; DE MONTE, Celeste; Adriano, Mollica; Rivanera, Daniela; Zicari, Alessandra; Emanuela, Mari; Gokhan, Zengin; Abdurrahman, Aktumsek
Inhibition of human monoamine oxidase: biological and molecular modeling studies on selected natural flavonoids
2016 Carradori, Simone; Gidaro, Maria Concetta; Petzer, Anél; Costa, Giosuè; Guglielmi, Paolo; Chimenti, Paola; Alcaro, Stefano; Petzer, Jacobus P.
Antimicrobial activity, synergism and inhibition of germ tube formation by Crocus sativus-derived compounds against Candida spp
2016 Carradori, Simone; Fazzari, Marina; Granese, Arianna; Chimenti, Paola; Angiolella, Letizia
(Thiazol-2-yl)hydrazone derivatives from acetylpyridines as dual inhibitors of MAO and AChE: synthesis, biological evaluation and molecular modeling studies
2015 D’Ascenzio, M; Chimenti, Paola; Gidaro, Mc; DE MONTE, Celeste; DE VITA, Daniela; Granese, Arianna; Scipione, Luigi; DI SANTO, Roberto; Costa, G; Alcaro, S; Yáñez, M; Carradori, S.
New amide derivatives of Probenecid as selective inhibitors of carbonic anhydrase IX and XII: Biological evaluation and molecular modelling studies
2015 Carradori, Simone; Mollica, Adriano; Ceruso, Mariangela; D'Ascenzio, Melissa; DE MONTE, Celeste; Chimenti, Paola; Sabia, Rocchina; Akdemir, Atilla; Supuran, Claudiu T.
New insights into the biological properties of Crocus sativus L.: chemical modifications, human monoamine oxidases inhibition and molecular modeling studies
2014 DE MONTE, Celeste; Carradori, Simone; Chimenti, Paola; Secci, Daniela; Mannina, Luisa; Alcaro, F; Petzer, A; N'Da, Ci; Gidaro, Mc; Costa, G; Alcaro, S; Petzer, Jp
Selective MAO-B inhibitors: a lesson from natural products
2014 Carradori, Simone; D'Ascenzio, Melissa; Chimenti, Paola; Secci, Daniela; Bolasco, Adriana
Microwave and Ultrasound-Assisted Synthesis of Thiosemicarbazones and Their Corresponding (4,5-Substituted-thiazol-2-yl)hydrazines
2014 Carradori, S; Secci, Daniela; D'Ascenzio, M; Chimenti, Paola; Bolasco, Adriana
New thiadiazoline and thiadiazole analogues of K858: antiproliferative activity in a model of prostate carcinoma
2013 DE MONTE, Celeste; Carradori, S.; D’Ascenzio, M.; Chimenti, Paola; Secci, Daniela; Bolasco, Adriana; Nicolazzo, Chiara; Silvestri, Ida
Exploring (4-substituted-thiazol-2-yl)hydrazine derivatives of 2-, 3-, and 4-acetylpyridine as selective and reversible hMAO-B inhibitors.
2013 Chimenti, Paola; Petzer, A.; Carradori, S.; D’Ascenzio, M.; Silvestri, Romano; Alcaro, S.; Ortuso, F.; Petzer, J. J.; Secci, Daniela
Patent-related survey on new monoamine oxidase inhibitors and their therapeutic potential
2012 Carradori, Simone; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; D'Ascenzio, Melissa
Thiazolyl-hydrazine derivatives: synthesis, molecular modeling, SAR studies, and selective MAO-B inhibitory activity.
2011 Chimenti, Paola; Bolasco, A.; Bizzarri, Bruna; Rivanera, Daniela
The State of the Art of Pyrazole Derivatives as Monoamine Oxidase Inhibitors and Antidepressant/Anticonvulsant Agents
2011 Secci, Daniela; Bolasco, Adriana; Carradori, Simone; Chimenti, Paola
Synthesis and selective human monoamine oxidase inhibition of 3-carbonyl, 3-acyl, and 3-carboxyhydrazido coumarin derivatives
2011 Secci, Daniela; Carradori, Simone; Bolasco, Adriana; Chimenti, Paola; Yanez, Matilde; Ortuso, Francesco; Alcaro, Stefano
Synthesis and biological evaluation of novel 2,4-disubstituted-1,3-thiazoles as anti-Candida spp. agents
2011 Franco, Chimenti; Bizzarri, Bruna; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Granese, Arianna; Simone, Carradori; Melissa, D'Ascenzio; Lilli, Daniela; Rivanera, Daniela
A new series of flavones, thioflavones, and flavanones as selective monoamine oxidase-B inhibitors
2010 Chimenti, Franco; Fioravanti, Rossella; Bolasco, Adriana; Chimenti, Paola; Secci, Daniela; Rossi, Francesca; Matilde, Yanez; Francisco, Orallo; Francesco, Ortuso; Stefano, Alcaro; Roberto, Cirilli; Rosella, Ferretti; M., Luisa Sanna
Investigations on the 2-thiazolylhydrazyne scaffold: Synthesis and molecular modeling of selective human monoamine oxidase inhibitors
2010 Chimenti, Franco; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Arianna, Granese; Simone, Carradori; Matilde, Yanez; Francisco, Orallo; Francesco, Ortuso; Stefano, Alcaro
Synthesis and characterization of new 3-acyl-7-hydroxy-6,8-substituted-coumarin and 3-acyl-7-benzyloxy-6,8-substituted-coumarin derivatives
2010 Chimenti, Franco; Bolasco, Adriana; Secci, Daniela; Bizzarri, Bruna; Chimenti, Paola; Granese, A; Carradori, S.
Synthesis, selective anti-Helicobacter pylori activity, and cytotoxicity of novel N-substituted-2-oxo-2H-1-benzopyran-3-carboxamides
2010 Chimenti, Franco; Bizzarri, Bruna; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Granese, Arianna; Carradori, Simone; Rivanera, Daniela; Zicari, Alessandra; M., Maddalena Scaltrito; Francesca, Sisto
Synthesis, semipreparative HPLC separation, biological evaluation, and 3D-QSAR of hydrazothiazole derivatives as human monoamine oxidase B inhibitors
2010 Chimenti, Franco; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Arianna, Granese; Simone, Carradori; Elias, Maccioni; M., Cristina Cardia; Matilde, Yanez; Francisco, Orallo; Stefano, Alcaro; Francesco, Ortuso; Roberto, Cirilli; Rosella, Ferretti; Simona, Distinto; Johannes, Kirchmair; Thierry, Langer
Synthesis and selective inhibition of human monoamine oxidases of a large scaffold of (4,5-substituted-thiazol-2-yl)hydrazones
2010 Chimenti, Franco; Secci, Daniela; Chimenti, Paola; Granese, Arianna; Carradori, Simone; D'Ascenzio, Melissa; Matilde, Yanez; Francisco, Orallo; Bolasco, Adriana
Synthesis and anti-Helicobacter pylori activity of 4-(coumarin-3-yl)thiazol-2-ylhydrazone derivatives
2010 Chimenti, F; Bizzarri, Bruna; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Granese, A; Carradori, S; D'Ascenzio, M; SCALTRITO M., M; Sisto, F.
Synthesis and inhibitory activity against human monoamine oxidase of N1-thiocarbamoyl-3,5-di(hetero)aryl-4,5-dihydro-(1H)-pyrazole derivatives
2010 Chimenti, Franco; Carradori, Simone; Secci, Daniela; Bolasco, Adriana; Bizzarri, Bruna; Chimenti, Paola; Arianna, Granese; Matilde, Yanez; Francisco, Orallo
SYNTHESIS, STEREOCHEMICAL SEPARATION, AND BIOLOGICAL EVALUATION OF SELECTIVE INHIBITORS OF HUMAN MAO-B: 1-(4-ARYLTHIAZOL-2-YL)-2-(3-METHYLCYCLOHEXYLIDENE)HYDRAZINES
2010 Chimenti, Franco; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Granese, A; Carradori, S; Yanez, M; Orallo, F; Sanna, Ml; Gallinella, B; Cirilli, R.
Synthesis, Molecular Modeling, and Selective Inhibitory Activity against Human Monoamine Oxidases of 3-Carboxamido-7-Substituted Coumarins.
2009 Chimenti, Franco; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Bizzarri, Bruna; Granese, Arianna; Carradori, Simone; Yanez, Matilde; Orallo, Francisco; Ortuso, Francesco; Alcaro, Stefano
Chalcones: A Valid Scaffold for Monoamine Oxidases Inhibitors
2009 Franco, Chimenti; Fioravanti, Rossella; Rossella, ; Bolasco, Adriana; Adriana, ; Chimenti, Paola; Paola, ; Secci, Daniela; Daniela, ; Rossi, Francesca
Synthesis and Biological Evaluation of Novel Conjugated Coumarin-Thiazole Systems
2009 Chimenti, Franco; Carradori, Simone; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Granese, Arianna; Bizzarri, Bruna
A Novel Histone Acetyltransferase Inhibitor Modulating Gcn5 Network: Cyclopentylidene-[4-(4′-chlorophenyl)thiazol-2-yl)hydrazone
2009 Chimenti, Franco; Bizzarri, Bruna; Elias, Maccioni; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Fioravanti, Rossella; Granese, Arianna; Carradori, Simone; Federica, Tosi; Ballario, Paola; S., Vernarecci; Patrizia, Filetici
Synthesis and Evaluation of 4-Acyl-2- Thiazolylhydrazone Derivatives for anti-Toxoplasma Efficacy in Vitro
2009 Chimenti, Franco; Bizzarri, Bruna; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Carradori, Simone; A., Granese; Rivanera, Daniela; N., Frishberg; C., Bordón; L., JONES BRANDO
Synthesis, molecular modeling studies and selective inhibitory activity against MAO of N1-propanoyl-3,5-diphenyl-4,5-dihydro-(1H)-pyrazole derivatives
2008 Chimenti, Franco; Fioravanti, Rossella; Bolasco, Adriana; Manna, Fedele; Chimenti, Paola; Secci, Daniela; Rossi, Francesca; Turini, Paola; Francesco, Ortuso; Stefano, Alcaro; Maria Cristina, Cardia
Synthesis, Stereochemical Identification, and Selective Inhibitory Activity against Human Monoamine Oxidase-B of 2-Methylcyclohexylidene-(4-arylthiazol-2-yl)hydrazones
2008 Chimenti, F.; Maccioni, E.; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Granese, Arianna; Carradori, Simone; Alcaro, S.; Ortuso, F.; Yanez, M.; Orallo, F.; Cirilli, R.; Ferretti, R.; LA TORRE, F.
Monoamine oxidase isoform-dependent tautomeric influence in the recognition of 3,5-diaryl pyrazole inhibitors.
2007 Chimenti, Franco; Fioravanti, Rossella; Bolasco, Adriana; Manna, Fedele; Chimenti, Paola; Secci, Daniela; Befani, O; Turini, Paola; Ortuso, F; Alcaro, S.
A novel class of selective anti-Helicobacter pylori agents 2-Oxo-2H-chromene-3-carboxamide derivatives.
2007 Chimenti, Franco; Bizzarri, Bruna; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Carradori, Simone; Granese, Arianna; Rivanera, Daniela; Lilli, Daniela; Zicari, Alessandra; SCALTRITO M., M; Sisto, F.
Synthesis and in vitro activity of 2-thiazolylhydrazone derivatives compared with the activity of clotrimazole against clinical isolates of Candida spp.
2007 Chimenti, Franco; Bizzarri, Bruna; Elias, Maccioni; Secci, Daniela; Bolasco, Adriana; Fioravanti, Rossella; Chimenti, Paola; Granese, Arianna; Carradori, Simone; Rivanera, Daniela; Lilli, Daniela; Zicari, Alessandra; Simona, Distinto
Selective inhibitory activity against MAO and molecular modeling studies of 2-thiazolylhydrazone derivatives
2007 Chimenti, Franco; Elias, Maccioni; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Granese, Arianna; Olivia, Befani; Turini, Paola; Stefano, Alcaro; Francesco, Ortuso; Maria C., Cardia; Simona, Distinto
Synthesis, biological evaluation and 3D-QSAR of 1,3,5-trisubstituted-4,5-dihydro-(1H)-pyrazole derivatives as potent and highly selective monoamine oxidase-A inhibitors.
2006 Manna, Fedele; Chimenti, Paola; Granese, Arianna; Befani, O; Turini, Paola; Cirilli, R; LA TORRE, F; Alcaro, S; Ortuso, F; Langer, T.; Chimenti, Franco; Bolasco, Adriana; Secci, Daniela
Analytical and semipreparative high performance liquid chromatography enantioseparation of new substituted 1-thiocarbamoyl-3,5-diaryl-4,5-dihydro-(1H)-pyrazoles on polysaccharide-based chiral stationary phases in normal-phase, polar organic and reversed-phase conditions.
2006 Cirilli, R; Simonelli, A; Ferretti, R; Bolasco, Adriana; Chimenti, Paola; Secci, Daniela; Maccioni, E; LA TORRE, F.
Quercetin as the active principle of Hypericum hircinum exerts a selective inhibitory activity against MAO-A: Extraction, biological analysis, and computational study
2006 F., Chimenti; F., Cottiglia; L., Bonsignore; L., Casu; M., Casu; C., Floris; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Granese, Arianna; O., Befani; Turini, Paola; S., Alcaro; F., Ortuso; G., Trombetta; A., Loizzo; I., Guarino
Synthesis, molecular modeling studies, and selective inhibitory activity against monoamine oxidase of N,N'-bis[2-oxo-2H-benzopyran]-3-carboxamides
2006 Chimenti, Franco; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Granese, Arianna; Carradori, Simone; O., Befani; Turini, Paola; S., Alcaro; F., Ortuso
Synthesis and in vitro selective anti-Helicobacter pylori activity of N-substituted-2-oxo-2H-1-benzopyran-3-carboxamides
2006 Chimenti, Franco; Bizzarri, Bruna; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Carradori, Simone; Granese, Arianna; Rivanera, Daniela; Lilli, Daniela; Maddalena Scaltrito, M.; Immacolata Brenciaglia, M.
Synthesis and molecular modelling of novel substituted-4,5-dihydro-(1H)-pyrazole derivatives as potent and highly selective monoamine oxidase-A inhibitors.
2006 Chimenti, Franco; Bolasco, Adriana; Manna, Fedele; Secci, Daniela; Chimenti, Paola; Granese, Arianna; Befani, O; Turini, Paola; Alcaro, S; Ortuso, F.
A environmentally friendly reversed-phase liquid chromatography method for phthalates determination in nail cosmetics
2006 DE ORSI, D; Gagliardi, L; Porra', R; Berri, S; Chimenti, Paola; Granese, Arianna; Carpani, I; Tonelli, D.
Synthesis and In Vitro Selective anti-Helicobacter pylori Activity of Pyrazoline Derivatives
2005 Chimenti, Franco; Bizzarri, Bruna; Manna, Fedele; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Granese, Arianna; Rivanera, Daniela; Lilli, Daniela; M. M., Scaltrito; M. I., Brenciaglia
LC Determination of Coumarin-3-acyl Derivatives for Evaluation of the Stability and Monoamine Oxidase Inhibition Mechanism.
2005 Chimenti, Paola; Granese, Arianna; Gagliardi, L; DE ORSI, D.; Chimenti, Franco; Secci, Daniela; Bolasco, Adriana
Pyrazole Derivatives as Potential Anticancer agents and their Affinity Binding to P-Glycoprotein
2005 F., Manna; Chimenti, Franco; Fioravanti, Rossella; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; C., Ferlini; G., Scambia
Synthesis, molecular modeling studies and selective inhibitory activity against MAO of 1-thiocarbamoyl-3,5-diaryl-4,5-dihydro-(1H)-pyrazole derivatives.
2005 Chimenti, Franco; Maccioni, E; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Granese, Arianna; Befani, Olivia; Turini, Paola; Alcaro, S; Ortuso, F; Cirilli, R; LA TORRE, F; Cardia, Mc; Distinto, S.
Cyclization of N ,N’-bis(salicylidene)diamines with Carbon Suboxide.
2005 Chimenti, Franco; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Granese, Arianna
Enantiomers of C5-chiral 1-acetyl-3,5-diphenyl-4,5-dihydro-(1H)-pyrazole derivatives: analytical and semipreparative HPLC separation, chiroptical properties, absolute configuration and inhibitory activity against monoamino oxidase
2004 Cirilli, R.; Ferretti, R.; Gallinella, B.; Turchetto, L.; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Pierini, Marco; Fares, V.; Befani, O.; LA TORRE, F.
Synthesis of New Diethynylbenzene Derivatives.
2004 Chimenti, Franco; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Granese, Arianna
Inhibition of Monoamine Oxidases by Coumarin-3-Acyl Derivatives: Biological Activity and Computational Study
2004 Chimenti, Franco; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Granese, Arianna; O., Befani; Turini, Paola; S., Alcaro; F., Ortuso
Development of an HPLC method for the identification and dosage of non-allowed substances in cosmetic products. Part I: local anaesthetics and antihistaminics
2004 R., Porra; Simona, Berri; Luigi, Gagliardi; Chimenti, Paola; Granese, Arianna; Daniela, Orsi; Irene, Carpani; Domenica, Tonelli
Analysis of corticosteroids by high performance liquid chromatography-electrospray mass spectrometry.
2004 Panusa, A; Ottaviani, M; Picardo, M; Camera, E; Gagliardi, L; Chimenti, Paola; Granese, Arianna; Tonelli, D.
Microwave-assisted synthesis of chiral pyrrolines with biological activity.
2004 Collina, S.; Loddo, G.; Barbieri, A.; Linati, L.; Alcaro, S.; Chimenti, Paola; Azzolina, O.
Synthesis and selective inhibitory activity against MAO of 1-acetyl-3,5-diphenyl-4,5-dihydro-(1H)-pyrazole derivatives.
2004 Chimenti, Franco; Bolasco, Adriana; Manna, Fedele; Secci, Daniela; Chimenti, Paola; Befani, O.; Turini, P.; Giovannini, V.; Mondovi', B.; Cirilli, R.; LA TORRE, F.
HPLC determination of imidazole antimycotis in antidandruff cosmetic products.
2003 Luigi, Gagliardi; Daniela De, Orsi; Chimenti, Paola; R., Porra'; Domenica, Tonelli
Development of a tandem thin-layer chromatography-high-performance liquid chromatography method for the identification and determination of corticosteroids in cosmetic products.
2002 Gagliardi, L.; De, Orsi; Del, Giudice; M. R., Gatta; F., Porra; Chimenti, Paola; Tonelli, D.
Efficacy of Hypericum and Calendula oils in the epithelial reconstruction of surgical wounds in childbirth with cesarean section.
2001 Lavagna, Silvio Massimo; Secci, Daniela; Chimenti, Paola; Bonsignore, L.; Ottaviani, A.; Bizzarri, Bruna
Structure-activity relationship studies on new DABOs: effect of substitutions at pyrimidine C-5 and C-6 positions on anti-HIV-1 activity
2001 Sbardella, G.; Mai, Antonello; Artico, M.; Chimenti, Paola; Massa, S.; Loddo, R.; Marongiu, M. E.; LA COLLA, P.; Pani, A.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Novel therapeutic opportunities for Toxoplasma gondii, Trichomonas vaginalis, and Giardia intestinalis infections | 2023 | Arrighi, Francesca; Granese, Arianna; Chimenti, Paola; Guglielmi, Paolo | |
Novel Insights on Human Carbonic Anhydrase Inhibitors Based on Coumalic Acid: Design, Synthesis, Molecular Modeling Investigation, and Biological Studies | 2022 | Pontecorvi, Virginia; Mori, Mattia; Picarazzi, Francesca; Zara, Susi; Carradori, Simone; Cataldi, Amelia; Angeli, Andrea; Berrino, Emanuela; Chimenti, Paola; Ciogli, Alessia; Secci, Daniela; Guglielmi, Paolo; Supuran, Claudiu T. | |
Novel insights on saccharin- and acesulfame-based carbonic anhydrase inhibitors: design, synthesis, modelling investigations and biological activity evaluation | 2020 | Guglielmi, P.; Rotondi, G.; Secci, D.; Angeli, A.; Chimenti, P.; Nocentini, A.; Bonardi, A.; Gratteri, P.; Carradori, S.; Supuran, C. T. | |
Phytochemical analyses and pharmacological screening of Neem oil | 2019 | Cesa, S.; Sisto, F.; Zengin, G.; Scaccabarozzi, D.; Kokolakis, A. K.; Scaltrito, M. M.; Grande, R.; Locatelli, M.; Cacciagrano, F.; Angiolella, L.; Campestre, C.; Granese, A.; Chimenti, P.; Basilico, N. | |
Benzo[b]tiophen-3-ol derivatives as effective inhibitors of human monoamine oxidase: design, synthesis, and biological activity | 2019 | Guglielmi, Paolo; Secci, Daniela; Petzer, Anél; Bagetta, Donatella; Chimenti, Paola; Rotondi, Giulia; Ferrante, Claudio; Recinella, Lucia; Leone, Sheila; Alcaro, Stefano; Zengin, Gokhan; Petzer, Jacobus P; Ortuso, Francesco; Carradori, Simone | |
Design, synthesis, docking studies and monoamine oxidase inhibition of a small library of 1-acetyl- and 1-thiocarbamoyl-3,5-diphenyl-4,5-dihydro-(1h)-pyrazoles | 2019 | Guglielmi, Paolo; Carradori, Simone; Poli, Giulio; Secci, Daniela; Cirilli, Roberto; Rotondi, Giulia; Chimenti, Paola; Petzer, Anél; Petzer, Jacobus P. | |
4-(3-Nitrophenyl)thiazol-2-ylhydrazone derivatives as antioxidants and selective hMAO-B inhibitors: synthesis, biological activity and computational analysis | 2019 | Secci, Daniela; Carradori, Simone; Petzer, Anél; Guglielmi, Paolo; D’Ascenzio, Melissa; Chimenti, Paola; Bagetta, Donatella; Alcaro, Stefano; Zengin, Gokhan; Petzer, Jacobus P.; Ortuso, Francesco | |
Synthesis and biological evaluation of anti-Toxoplasma gondii activity of a novel scaffold of thiazolidinone derivatives | 2017 | Carradori, Simone; Secci, Daniela; Bizzarri, Bruna; Chimenti, Paola; DE MONTE, Celeste; Guglielmi, Paolo; Campestre, Cristina; Rivanera, Daniela; Bordón, Claudia; Jones Brando, Lorraine | |
Novel 1,3-thiazolidin-4-one derivatives as promising anti-Candida agents endowed with anti-oxidant and chelating properties | 2016 | Secci, Daniela; Simone, Carradori; Bizzarri, Bruna; Chimenti, Paola; DE MONTE, Celeste; Adriano, Mollica; Rivanera, Daniela; Zicari, Alessandra; Emanuela, Mari; Gokhan, Zengin; Abdurrahman, Aktumsek | |
Inhibition of human monoamine oxidase: biological and molecular modeling studies on selected natural flavonoids | 2016 | Carradori, Simone; Gidaro, Maria Concetta; Petzer, Anél; Costa, Giosuè; Guglielmi, Paolo; Chimenti, Paola; Alcaro, Stefano; Petzer, Jacobus P. | |
Antimicrobial activity, synergism and inhibition of germ tube formation by Crocus sativus-derived compounds against Candida spp | 2016 | Carradori, Simone; Fazzari, Marina; Granese, Arianna; Chimenti, Paola; Angiolella, Letizia | |
(Thiazol-2-yl)hydrazone derivatives from acetylpyridines as dual inhibitors of MAO and AChE: synthesis, biological evaluation and molecular modeling studies | 2015 | D’Ascenzio, M; Chimenti, Paola; Gidaro, Mc; DE MONTE, Celeste; DE VITA, Daniela; Granese, Arianna; Scipione, Luigi; DI SANTO, Roberto; Costa, G; Alcaro, S; Yáñez, M; Carradori, S. | |
New amide derivatives of Probenecid as selective inhibitors of carbonic anhydrase IX and XII: Biological evaluation and molecular modelling studies | 2015 | Carradori, Simone; Mollica, Adriano; Ceruso, Mariangela; D'Ascenzio, Melissa; DE MONTE, Celeste; Chimenti, Paola; Sabia, Rocchina; Akdemir, Atilla; Supuran, Claudiu T. | |
New insights into the biological properties of Crocus sativus L.: chemical modifications, human monoamine oxidases inhibition and molecular modeling studies | 2014 | DE MONTE, Celeste; Carradori, Simone; Chimenti, Paola; Secci, Daniela; Mannina, Luisa; Alcaro, F; Petzer, A; N'Da, Ci; Gidaro, Mc; Costa, G; Alcaro, S; Petzer, Jp | |
Selective MAO-B inhibitors: a lesson from natural products | 2014 | Carradori, Simone; D'Ascenzio, Melissa; Chimenti, Paola; Secci, Daniela; Bolasco, Adriana | |
Microwave and Ultrasound-Assisted Synthesis of Thiosemicarbazones and Their Corresponding (4,5-Substituted-thiazol-2-yl)hydrazines | 2014 | Carradori, S; Secci, Daniela; D'Ascenzio, M; Chimenti, Paola; Bolasco, Adriana | |
New thiadiazoline and thiadiazole analogues of K858: antiproliferative activity in a model of prostate carcinoma | 2013 | DE MONTE, Celeste; Carradori, S.; D’Ascenzio, M.; Chimenti, Paola; Secci, Daniela; Bolasco, Adriana; Nicolazzo, Chiara; Silvestri, Ida | |
Exploring (4-substituted-thiazol-2-yl)hydrazine derivatives of 2-, 3-, and 4-acetylpyridine as selective and reversible hMAO-B inhibitors. | 2013 | Chimenti, Paola; Petzer, A.; Carradori, S.; D’Ascenzio, M.; Silvestri, Romano; Alcaro, S.; Ortuso, F.; Petzer, J. J.; Secci, Daniela | |
Patent-related survey on new monoamine oxidase inhibitors and their therapeutic potential | 2012 | Carradori, Simone; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; D'Ascenzio, Melissa | |
Thiazolyl-hydrazine derivatives: synthesis, molecular modeling, SAR studies, and selective MAO-B inhibitory activity. | 2011 | Chimenti, Paola; Bolasco, A.; Bizzarri, Bruna; Rivanera, Daniela | |
The State of the Art of Pyrazole Derivatives as Monoamine Oxidase Inhibitors and Antidepressant/Anticonvulsant Agents | 2011 | Secci, Daniela; Bolasco, Adriana; Carradori, Simone; Chimenti, Paola | |
Synthesis and selective human monoamine oxidase inhibition of 3-carbonyl, 3-acyl, and 3-carboxyhydrazido coumarin derivatives | 2011 | Secci, Daniela; Carradori, Simone; Bolasco, Adriana; Chimenti, Paola; Yanez, Matilde; Ortuso, Francesco; Alcaro, Stefano | |
Synthesis and biological evaluation of novel 2,4-disubstituted-1,3-thiazoles as anti-Candida spp. agents | 2011 | Franco, Chimenti; Bizzarri, Bruna; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Granese, Arianna; Simone, Carradori; Melissa, D'Ascenzio; Lilli, Daniela; Rivanera, Daniela | |
A new series of flavones, thioflavones, and flavanones as selective monoamine oxidase-B inhibitors | 2010 | Chimenti, Franco; Fioravanti, Rossella; Bolasco, Adriana; Chimenti, Paola; Secci, Daniela; Rossi, Francesca; Matilde, Yanez; Francisco, Orallo; Francesco, Ortuso; Stefano, Alcaro; Roberto, Cirilli; Rosella, Ferretti; M., Luisa Sanna | |
Investigations on the 2-thiazolylhydrazyne scaffold: Synthesis and molecular modeling of selective human monoamine oxidase inhibitors | 2010 | Chimenti, Franco; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Arianna, Granese; Simone, Carradori; Matilde, Yanez; Francisco, Orallo; Francesco, Ortuso; Stefano, Alcaro | |
Synthesis and characterization of new 3-acyl-7-hydroxy-6,8-substituted-coumarin and 3-acyl-7-benzyloxy-6,8-substituted-coumarin derivatives | 2010 | Chimenti, Franco; Bolasco, Adriana; Secci, Daniela; Bizzarri, Bruna; Chimenti, Paola; Granese, A; Carradori, S. | |
Synthesis, selective anti-Helicobacter pylori activity, and cytotoxicity of novel N-substituted-2-oxo-2H-1-benzopyran-3-carboxamides | 2010 | Chimenti, Franco; Bizzarri, Bruna; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Granese, Arianna; Carradori, Simone; Rivanera, Daniela; Zicari, Alessandra; M., Maddalena Scaltrito; Francesca, Sisto | |
Synthesis, semipreparative HPLC separation, biological evaluation, and 3D-QSAR of hydrazothiazole derivatives as human monoamine oxidase B inhibitors | 2010 | Chimenti, Franco; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Arianna, Granese; Simone, Carradori; Elias, Maccioni; M., Cristina Cardia; Matilde, Yanez; Francisco, Orallo; Stefano, Alcaro; Francesco, Ortuso; Roberto, Cirilli; Rosella, Ferretti; Simona, Distinto; Johannes, Kirchmair; Thierry, Langer | |
Synthesis and selective inhibition of human monoamine oxidases of a large scaffold of (4,5-substituted-thiazol-2-yl)hydrazones | 2010 | Chimenti, Franco; Secci, Daniela; Chimenti, Paola; Granese, Arianna; Carradori, Simone; D'Ascenzio, Melissa; Matilde, Yanez; Francisco, Orallo; Bolasco, Adriana | |
Synthesis and anti-Helicobacter pylori activity of 4-(coumarin-3-yl)thiazol-2-ylhydrazone derivatives | 2010 | Chimenti, F; Bizzarri, Bruna; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Granese, A; Carradori, S; D'Ascenzio, M; SCALTRITO M., M; Sisto, F. | |
Synthesis and inhibitory activity against human monoamine oxidase of N1-thiocarbamoyl-3,5-di(hetero)aryl-4,5-dihydro-(1H)-pyrazole derivatives | 2010 | Chimenti, Franco; Carradori, Simone; Secci, Daniela; Bolasco, Adriana; Bizzarri, Bruna; Chimenti, Paola; Arianna, Granese; Matilde, Yanez; Francisco, Orallo | |
SYNTHESIS, STEREOCHEMICAL SEPARATION, AND BIOLOGICAL EVALUATION OF SELECTIVE INHIBITORS OF HUMAN MAO-B: 1-(4-ARYLTHIAZOL-2-YL)-2-(3-METHYLCYCLOHEXYLIDENE)HYDRAZINES | 2010 | Chimenti, Franco; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Granese, A; Carradori, S; Yanez, M; Orallo, F; Sanna, Ml; Gallinella, B; Cirilli, R. | |
Synthesis, Molecular Modeling, and Selective Inhibitory Activity against Human Monoamine Oxidases of 3-Carboxamido-7-Substituted Coumarins. | 2009 | Chimenti, Franco; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Bizzarri, Bruna; Granese, Arianna; Carradori, Simone; Yanez, Matilde; Orallo, Francisco; Ortuso, Francesco; Alcaro, Stefano | |
Chalcones: A Valid Scaffold for Monoamine Oxidases Inhibitors | 2009 | Franco, Chimenti; Fioravanti, Rossella; Rossella, ; Bolasco, Adriana; Adriana, ; Chimenti, Paola; Paola, ; Secci, Daniela; Daniela, ; Rossi, Francesca | |
Synthesis and Biological Evaluation of Novel Conjugated Coumarin-Thiazole Systems | 2009 | Chimenti, Franco; Carradori, Simone; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Granese, Arianna; Bizzarri, Bruna | |
A Novel Histone Acetyltransferase Inhibitor Modulating Gcn5 Network: Cyclopentylidene-[4-(4′-chlorophenyl)thiazol-2-yl)hydrazone | 2009 | Chimenti, Franco; Bizzarri, Bruna; Elias, Maccioni; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Fioravanti, Rossella; Granese, Arianna; Carradori, Simone; Federica, Tosi; Ballario, Paola; S., Vernarecci; Patrizia, Filetici | |
Synthesis and Evaluation of 4-Acyl-2- Thiazolylhydrazone Derivatives for anti-Toxoplasma Efficacy in Vitro | 2009 | Chimenti, Franco; Bizzarri, Bruna; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Carradori, Simone; A., Granese; Rivanera, Daniela; N., Frishberg; C., Bordón; L., JONES BRANDO | |
Synthesis, molecular modeling studies and selective inhibitory activity against MAO of N1-propanoyl-3,5-diphenyl-4,5-dihydro-(1H)-pyrazole derivatives | 2008 | Chimenti, Franco; Fioravanti, Rossella; Bolasco, Adriana; Manna, Fedele; Chimenti, Paola; Secci, Daniela; Rossi, Francesca; Turini, Paola; Francesco, Ortuso; Stefano, Alcaro; Maria Cristina, Cardia | |
Synthesis, Stereochemical Identification, and Selective Inhibitory Activity against Human Monoamine Oxidase-B of 2-Methylcyclohexylidene-(4-arylthiazol-2-yl)hydrazones | 2008 | Chimenti, F.; Maccioni, E.; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Granese, Arianna; Carradori, Simone; Alcaro, S.; Ortuso, F.; Yanez, M.; Orallo, F.; Cirilli, R.; Ferretti, R.; LA TORRE, F. | |
Monoamine oxidase isoform-dependent tautomeric influence in the recognition of 3,5-diaryl pyrazole inhibitors. | 2007 | Chimenti, Franco; Fioravanti, Rossella; Bolasco, Adriana; Manna, Fedele; Chimenti, Paola; Secci, Daniela; Befani, O; Turini, Paola; Ortuso, F; Alcaro, S. | |
A novel class of selective anti-Helicobacter pylori agents 2-Oxo-2H-chromene-3-carboxamide derivatives. | 2007 | Chimenti, Franco; Bizzarri, Bruna; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Carradori, Simone; Granese, Arianna; Rivanera, Daniela; Lilli, Daniela; Zicari, Alessandra; SCALTRITO M., M; Sisto, F. | |
Synthesis and in vitro activity of 2-thiazolylhydrazone derivatives compared with the activity of clotrimazole against clinical isolates of Candida spp. | 2007 | Chimenti, Franco; Bizzarri, Bruna; Elias, Maccioni; Secci, Daniela; Bolasco, Adriana; Fioravanti, Rossella; Chimenti, Paola; Granese, Arianna; Carradori, Simone; Rivanera, Daniela; Lilli, Daniela; Zicari, Alessandra; Simona, Distinto | |
Selective inhibitory activity against MAO and molecular modeling studies of 2-thiazolylhydrazone derivatives | 2007 | Chimenti, Franco; Elias, Maccioni; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Granese, Arianna; Olivia, Befani; Turini, Paola; Stefano, Alcaro; Francesco, Ortuso; Maria C., Cardia; Simona, Distinto | |
Synthesis, biological evaluation and 3D-QSAR of 1,3,5-trisubstituted-4,5-dihydro-(1H)-pyrazole derivatives as potent and highly selective monoamine oxidase-A inhibitors. | 2006 | Manna, Fedele; Chimenti, Paola; Granese, Arianna; Befani, O; Turini, Paola; Cirilli, R; LA TORRE, F; Alcaro, S; Ortuso, F; Langer, T.; Chimenti, Franco; Bolasco, Adriana; Secci, Daniela | |
Analytical and semipreparative high performance liquid chromatography enantioseparation of new substituted 1-thiocarbamoyl-3,5-diaryl-4,5-dihydro-(1H)-pyrazoles on polysaccharide-based chiral stationary phases in normal-phase, polar organic and reversed-phase conditions. | 2006 | Cirilli, R; Simonelli, A; Ferretti, R; Bolasco, Adriana; Chimenti, Paola; Secci, Daniela; Maccioni, E; LA TORRE, F. | |
Quercetin as the active principle of Hypericum hircinum exerts a selective inhibitory activity against MAO-A: Extraction, biological analysis, and computational study | 2006 | F., Chimenti; F., Cottiglia; L., Bonsignore; L., Casu; M., Casu; C., Floris; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Granese, Arianna; O., Befani; Turini, Paola; S., Alcaro; F., Ortuso; G., Trombetta; A., Loizzo; I., Guarino | |
Synthesis, molecular modeling studies, and selective inhibitory activity against monoamine oxidase of N,N'-bis[2-oxo-2H-benzopyran]-3-carboxamides | 2006 | Chimenti, Franco; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Granese, Arianna; Carradori, Simone; O., Befani; Turini, Paola; S., Alcaro; F., Ortuso | |
Synthesis and in vitro selective anti-Helicobacter pylori activity of N-substituted-2-oxo-2H-1-benzopyran-3-carboxamides | 2006 | Chimenti, Franco; Bizzarri, Bruna; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Carradori, Simone; Granese, Arianna; Rivanera, Daniela; Lilli, Daniela; Maddalena Scaltrito, M.; Immacolata Brenciaglia, M. | |
Synthesis and molecular modelling of novel substituted-4,5-dihydro-(1H)-pyrazole derivatives as potent and highly selective monoamine oxidase-A inhibitors. | 2006 | Chimenti, Franco; Bolasco, Adriana; Manna, Fedele; Secci, Daniela; Chimenti, Paola; Granese, Arianna; Befani, O; Turini, Paola; Alcaro, S; Ortuso, F. | |
A environmentally friendly reversed-phase liquid chromatography method for phthalates determination in nail cosmetics | 2006 | DE ORSI, D; Gagliardi, L; Porra', R; Berri, S; Chimenti, Paola; Granese, Arianna; Carpani, I; Tonelli, D. | |
Synthesis and In Vitro Selective anti-Helicobacter pylori Activity of Pyrazoline Derivatives | 2005 | Chimenti, Franco; Bizzarri, Bruna; Manna, Fedele; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Granese, Arianna; Rivanera, Daniela; Lilli, Daniela; M. M., Scaltrito; M. I., Brenciaglia | |
LC Determination of Coumarin-3-acyl Derivatives for Evaluation of the Stability and Monoamine Oxidase Inhibition Mechanism. | 2005 | Chimenti, Paola; Granese, Arianna; Gagliardi, L; DE ORSI, D.; Chimenti, Franco; Secci, Daniela; Bolasco, Adriana | |
Pyrazole Derivatives as Potential Anticancer agents and their Affinity Binding to P-Glycoprotein | 2005 | F., Manna; Chimenti, Franco; Fioravanti, Rossella; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; C., Ferlini; G., Scambia | |
Synthesis, molecular modeling studies and selective inhibitory activity against MAO of 1-thiocarbamoyl-3,5-diaryl-4,5-dihydro-(1H)-pyrazole derivatives. | 2005 | Chimenti, Franco; Maccioni, E; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Granese, Arianna; Befani, Olivia; Turini, Paola; Alcaro, S; Ortuso, F; Cirilli, R; LA TORRE, F; Cardia, Mc; Distinto, S. | |
Cyclization of N ,N’-bis(salicylidene)diamines with Carbon Suboxide. | 2005 | Chimenti, Franco; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Granese, Arianna | |
Enantiomers of C5-chiral 1-acetyl-3,5-diphenyl-4,5-dihydro-(1H)-pyrazole derivatives: analytical and semipreparative HPLC separation, chiroptical properties, absolute configuration and inhibitory activity against monoamino oxidase | 2004 | Cirilli, R.; Ferretti, R.; Gallinella, B.; Turchetto, L.; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Pierini, Marco; Fares, V.; Befani, O.; LA TORRE, F. | |
Synthesis of New Diethynylbenzene Derivatives. | 2004 | Chimenti, Franco; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Granese, Arianna | |
Inhibition of Monoamine Oxidases by Coumarin-3-Acyl Derivatives: Biological Activity and Computational Study | 2004 | Chimenti, Franco; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Granese, Arianna; O., Befani; Turini, Paola; S., Alcaro; F., Ortuso | |
Development of an HPLC method for the identification and dosage of non-allowed substances in cosmetic products. Part I: local anaesthetics and antihistaminics | 2004 | R., Porra; Simona, Berri; Luigi, Gagliardi; Chimenti, Paola; Granese, Arianna; Daniela, Orsi; Irene, Carpani; Domenica, Tonelli | |
Analysis of corticosteroids by high performance liquid chromatography-electrospray mass spectrometry. | 2004 | Panusa, A; Ottaviani, M; Picardo, M; Camera, E; Gagliardi, L; Chimenti, Paola; Granese, Arianna; Tonelli, D. | |
Microwave-assisted synthesis of chiral pyrrolines with biological activity. | 2004 | Collina, S.; Loddo, G.; Barbieri, A.; Linati, L.; Alcaro, S.; Chimenti, Paola; Azzolina, O. | |
Synthesis and selective inhibitory activity against MAO of 1-acetyl-3,5-diphenyl-4,5-dihydro-(1H)-pyrazole derivatives. | 2004 | Chimenti, Franco; Bolasco, Adriana; Manna, Fedele; Secci, Daniela; Chimenti, Paola; Befani, O.; Turini, P.; Giovannini, V.; Mondovi', B.; Cirilli, R.; LA TORRE, F. | |
HPLC determination of imidazole antimycotis in antidandruff cosmetic products. | 2003 | Luigi, Gagliardi; Daniela De, Orsi; Chimenti, Paola; R., Porra'; Domenica, Tonelli | |
Development of a tandem thin-layer chromatography-high-performance liquid chromatography method for the identification and determination of corticosteroids in cosmetic products. | 2002 | Gagliardi, L.; De, Orsi; Del, Giudice; M. R., Gatta; F., Porra; Chimenti, Paola; Tonelli, D. | |
Efficacy of Hypericum and Calendula oils in the epithelial reconstruction of surgical wounds in childbirth with cesarean section. | 2001 | Lavagna, Silvio Massimo; Secci, Daniela; Chimenti, Paola; Bonsignore, L.; Ottaviani, A.; Bizzarri, Bruna | |
Structure-activity relationship studies on new DABOs: effect of substitutions at pyrimidine C-5 and C-6 positions on anti-HIV-1 activity | 2001 | Sbardella, G.; Mai, Antonello; Artico, M.; Chimenti, Paola; Massa, S.; Loddo, R.; Marongiu, M. E.; LA COLLA, P.; Pani, A. |
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