ORTAR, Giorgio
ORTAR, Giorgio
DIPARTIMENTO DI CHIMICA E TECNOLOGIE DEL FARMACO
(-)Menthylamine derivatives as potent and selective antagonists of transient receptor potential melastatin type-8 (TRPM8) channels
2010 Ortar, Giorgio; LUCIANO DE, Petrocellis; Morera, Ludovica; ANIELLO SCHIANO, Moriello; Pierangelo, Orlando; Morera, Enrico; Nalli, Marianna; VINCENZO DI, Marzo
3-Aroyl-1,4-diarylpyrroles inhibit chronic myeloid leukemia cell growth through an interaction with tubulin
2017 LA REGINA, Giuseppe; Bai, R.; Coluccia, Antonio; Famiglini, Valeria; Passacantilli, Sara; Naccarato, Valentina; Ortar, Giorgio; Mazzoccoli, Carmela; Ruggieri, V.; Agriesti, F.; Piccoli, C.; Tataranni, T.; Nalli, Marianna; Brancale, A.; Vultaggio, S.; Mercurio, C.; Varasi, M.; Saponaro, C.; Sergio, S.; Maffia, M.; Coluccia, A. M. L.; Hamel, E.; Silvestri, Romano
3-Ylidenephthalides as a new class of transient receptor potential channel TRPA1 and TRPM8 modulators
2013 Ortar, Giorgio; Aniello Schiano, Moriello; Morera, Enrico; Nalli, Marianna; Vincenzo Di, Marzo; Luciano De, Petrocellis
A Concise Synthesis of Photoactivatable 4-Aroyl-L-phenylalanines
2000 Morera, Enrico; Ortar, Giorgio
A Convenient Preparation of Selectively Protected L-DOPA derivatives from 3-iodo-L-Tyrosine
2001 Morera, Enrico; Ortar, Giorgio
A Palladium-Catalyzed Carbonylative Route to Primary Amides
1998 Morera, Enrico; Ortar, Giorgio
An analytical approach to the forensic identification of different classes of new psychoactive substances (NPSs) in seized materials
2014 S., Strano Rossi; S., Odoardi; A., Gregori; G., Peluso; L., Ripani; Ortar, Giorgio; G., Serpelloni; F. S., Romolo
An Efficient Synthesis of 4-Aryl and 4-Vinylphenylalanines by Stille Cross-Coupling Reaction
1997 Morera, Enrico; Ortar, Giorgio
An Improved Preparation of 4-Hydroxymethyl-L-Phenylalanine
1998 Morera, Enrico; Ortar, Giorgio; Varani, A.
Antibacterial and antifungal agents. XV. Synthesis and antifungal activity of structural analogues of bifonazole and ketoconazole.
1992 Stefancich, Giorgio; Artico, Marco; Ortar, Giorgio; Silvestri, Romano; Simonetti, Giovanna; Germana, Apuzzo; Artico, Marino
Antinociceptive Effects of Tetrazole Inhibitors of Endocannabinoid Inactivation: Cannabinoid and Non-cannabinoid Receptor-mediated Mechanisms
2008 S., Maione; Morera, Enrico; I., Marabese; A., Ligresti; L., Luongo; Ortar, Giorgio; V., DI MARZO
Arylboronic acids as dual-action FAAH and TRPV1 ligands
2016 Morera, Enrico; Di Marzo, Vincenzo; Monti, Ludovica; Allarà, Marco; Schiano Moriello, Aniello; Nalli, Marianna; Ortar, Giorgio; De Petrocellis, Luciano
Biaryl tetrazolyl ureas inhibitors of endocannabinoid metabolism: modulation at the N-portion and distal phenyl ring
2013 Ortar, Giorgio; Morera, Enrico; Luciano De, Petrocellis; Alessia, Ligresti; Aniello Schiano, Moriello; Morera, Ludovica; Nalli, Marianna; Ragno, Rino; Pirolli, Adele; Vincenzo Di, Marzo
Bovine serum amine oxidase and spermine in association with anandamide cause cytotoxicity in melanoma and colon adenocarcinoma cells
2012 Bidollari, E.; Tempera, Giampiero; Ueshima, T.; Calcabrini, A.; Ortar, Giorgio; Morera, Enrico; Nalli, Marianna; Condello, M.; Arancia, G.; Molinari, A.; Agostinelli, Enzo
Carbamoyl tetrazoles as inhibitors of endocannabinoid inactivation: A critical revisitation
2008 Ortar, Giorgio; Maria Grazia, Cascio; A., Schiano Moriello; Mercedes, Camalli; Morera, Enrico; Nalli, Marianna; Vincenzo Di, Marzo
Cytotoxic effect induced by combination of polyamines metabolites and endocannabinoid, anandamide, on human cancer cells: a new anticancer strategy”
2010 Batista de Carvalho, A. L. M.; Tempera, Giampiero; Viceconte, N.; Saccoccio, Stefania; Bidollari, E.; Nalli, Marianna; Morera, Enrico; Ortar, Giorgio; Agostinelli, Enzo
Development and characterization of endocannabinoid hydrolases FAAH and MAGL inhibitors bearing a benzotriazol-1-yl carboxamide scaffold
2012 Morera, Ludovica; Geoffray, Labar; Ortar, Giorgio; Didier M., Lambert
Development of a potent inhibitor of 2-arachidonoylglycerol hydrolysis with antinociceptive activity in vivo
2009 Tiziana, Bisogno; Ortar, Giorgio; Stefania, Petrosino; Morera, Enrico; Enza, Palazzo; Nalli, Marianna; Sabatino, Maione; Vincenzo Di, Marzo
Development of the First Potential Covalent Inhibitors of Anandamide Cellular Uptake
2006 SCHIANO MORIELLO, A; Balas, L; Ligresti, A; CASCIO M., G; Durand, T; Morera, Enrico; Ortar, Giorgio; DI MARZO, V.
Discussion Addendum for: Palladium-Catalyzed Reduction of Vinyl Trifluoromethanesulfonates to Alkenes: Cholesta-3,5-DieneOrganic Syntheses
2011 Cacchi, Sandro; Morera, Enrico; Ortar, Giorgio
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
(-)Menthylamine derivatives as potent and selective antagonists of transient receptor potential melastatin type-8 (TRPM8) channels | 2010 | Ortar, Giorgio; LUCIANO DE, Petrocellis; Morera, Ludovica; ANIELLO SCHIANO, Moriello; Pierangelo, Orlando; Morera, Enrico; Nalli, Marianna; VINCENZO DI, Marzo | |
3-Aroyl-1,4-diarylpyrroles inhibit chronic myeloid leukemia cell growth through an interaction with tubulin | 2017 | LA REGINA, Giuseppe; Bai, R.; Coluccia, Antonio; Famiglini, Valeria; Passacantilli, Sara; Naccarato, Valentina; Ortar, Giorgio; Mazzoccoli, Carmela; Ruggieri, V.; Agriesti, F.; Piccoli, C.; Tataranni, T.; Nalli, Marianna; Brancale, A.; Vultaggio, S.; Mercurio, C.; Varasi, M.; Saponaro, C.; Sergio, S.; Maffia, M.; Coluccia, A. M. L.; Hamel, E.; Silvestri, Romano | |
3-Ylidenephthalides as a new class of transient receptor potential channel TRPA1 and TRPM8 modulators | 2013 | Ortar, Giorgio; Aniello Schiano, Moriello; Morera, Enrico; Nalli, Marianna; Vincenzo Di, Marzo; Luciano De, Petrocellis | |
A Concise Synthesis of Photoactivatable 4-Aroyl-L-phenylalanines | 2000 | Morera, Enrico; Ortar, Giorgio | |
A Convenient Preparation of Selectively Protected L-DOPA derivatives from 3-iodo-L-Tyrosine | 2001 | Morera, Enrico; Ortar, Giorgio | |
A Palladium-Catalyzed Carbonylative Route to Primary Amides | 1998 | Morera, Enrico; Ortar, Giorgio | |
An analytical approach to the forensic identification of different classes of new psychoactive substances (NPSs) in seized materials | 2014 | S., Strano Rossi; S., Odoardi; A., Gregori; G., Peluso; L., Ripani; Ortar, Giorgio; G., Serpelloni; F. S., Romolo | |
An Efficient Synthesis of 4-Aryl and 4-Vinylphenylalanines by Stille Cross-Coupling Reaction | 1997 | Morera, Enrico; Ortar, Giorgio | |
An Improved Preparation of 4-Hydroxymethyl-L-Phenylalanine | 1998 | Morera, Enrico; Ortar, Giorgio; Varani, A. | |
Antibacterial and antifungal agents. XV. Synthesis and antifungal activity of structural analogues of bifonazole and ketoconazole. | 1992 | Stefancich, Giorgio; Artico, Marco; Ortar, Giorgio; Silvestri, Romano; Simonetti, Giovanna; Germana, Apuzzo; Artico, Marino | |
Antinociceptive Effects of Tetrazole Inhibitors of Endocannabinoid Inactivation: Cannabinoid and Non-cannabinoid Receptor-mediated Mechanisms | 2008 | S., Maione; Morera, Enrico; I., Marabese; A., Ligresti; L., Luongo; Ortar, Giorgio; V., DI MARZO | |
Arylboronic acids as dual-action FAAH and TRPV1 ligands | 2016 | Morera, Enrico; Di Marzo, Vincenzo; Monti, Ludovica; Allarà, Marco; Schiano Moriello, Aniello; Nalli, Marianna; Ortar, Giorgio; De Petrocellis, Luciano | |
Biaryl tetrazolyl ureas inhibitors of endocannabinoid metabolism: modulation at the N-portion and distal phenyl ring | 2013 | Ortar, Giorgio; Morera, Enrico; Luciano De, Petrocellis; Alessia, Ligresti; Aniello Schiano, Moriello; Morera, Ludovica; Nalli, Marianna; Ragno, Rino; Pirolli, Adele; Vincenzo Di, Marzo | |
Bovine serum amine oxidase and spermine in association with anandamide cause cytotoxicity in melanoma and colon adenocarcinoma cells | 2012 | Bidollari, E.; Tempera, Giampiero; Ueshima, T.; Calcabrini, A.; Ortar, Giorgio; Morera, Enrico; Nalli, Marianna; Condello, M.; Arancia, G.; Molinari, A.; Agostinelli, Enzo | |
Carbamoyl tetrazoles as inhibitors of endocannabinoid inactivation: A critical revisitation | 2008 | Ortar, Giorgio; Maria Grazia, Cascio; A., Schiano Moriello; Mercedes, Camalli; Morera, Enrico; Nalli, Marianna; Vincenzo Di, Marzo | |
Cytotoxic effect induced by combination of polyamines metabolites and endocannabinoid, anandamide, on human cancer cells: a new anticancer strategy” | 2010 | Batista de Carvalho, A. L. M.; Tempera, Giampiero; Viceconte, N.; Saccoccio, Stefania; Bidollari, E.; Nalli, Marianna; Morera, Enrico; Ortar, Giorgio; Agostinelli, Enzo | |
Development and characterization of endocannabinoid hydrolases FAAH and MAGL inhibitors bearing a benzotriazol-1-yl carboxamide scaffold | 2012 | Morera, Ludovica; Geoffray, Labar; Ortar, Giorgio; Didier M., Lambert | |
Development of a potent inhibitor of 2-arachidonoylglycerol hydrolysis with antinociceptive activity in vivo | 2009 | Tiziana, Bisogno; Ortar, Giorgio; Stefania, Petrosino; Morera, Enrico; Enza, Palazzo; Nalli, Marianna; Sabatino, Maione; Vincenzo Di, Marzo | |
Development of the First Potential Covalent Inhibitors of Anandamide Cellular Uptake | 2006 | SCHIANO MORIELLO, A; Balas, L; Ligresti, A; CASCIO M., G; Durand, T; Morera, Enrico; Ortar, Giorgio; DI MARZO, V. | |
Discussion Addendum for: Palladium-Catalyzed Reduction of Vinyl Trifluoromethanesulfonates to Alkenes: Cholesta-3,5-DieneOrganic Syntheses | 2011 | Cacchi, Sandro; Morera, Enrico; Ortar, Giorgio |