Sfoglia per Autore
Development of the First Potential Covalent Inhibitors of Anandamide Cellular Uptake
2006 SCHIANO MORIELLO, A; Balas, L; Ligresti, A; CASCIO M., G; Durand, T; Morera, Enrico; Ortar, Giorgio; DI MARZO, V.
New N-Arachidonoylserotonin Analogues with Potential 'Dual' Mechanism Action against Pain
2007 Ortar, Giorgio; CASCIO MARIA, Grazia; DE PETROCELLIS, Luciano; Morera, Enrico; Rossi, Francesca; SCHIANO MORIELLO, Aniello; Nalli, Marianna; DE NOVELLIS, Vito; WOODWARD DAVID, F; Maione, Sabatino; DI MARZO, Vincenzo
New tetrazole-based selective anandamide uptake inhibitors
2008 Ortar, Giorgio; Aniello Schiano, Moriello; Maria Grazia, Cascio; Luciano De, Petrocellis; Alessia, Ligresti; Morera, Enrico; Nalli, Marianna; Vincenzo Di, Marzo
Antinociceptive Effects of Tetrazole Inhibitors of Endocannabinoid Inactivation: Cannabinoid and Non-cannabinoid Receptor-mediated Mechanisms
2008 S., Maione; Morera, Enrico; I., Marabese; A., Ligresti; L., Luongo; Ortar, Giorgio; V., DI MARZO
Carbamoyl tetrazoles as inhibitors of endocannabinoid inactivation: A critical revisitation
2008 Ortar, Giorgio; Maria Grazia, Cascio; A., Schiano Moriello; Mercedes, Camalli; Morera, Enrico; Nalli, Marianna; Vincenzo Di, Marzo
Development of a potent inhibitor of 2-arachidonoylglycerol hydrolysis with antinociceptive activity in vivo
2009 Tiziana, Bisogno; Ortar, Giorgio; Stefania, Petrosino; Morera, Enrico; Enza, Palazzo; Nalli, Marianna; Sabatino, Maione; Vincenzo Di, Marzo
Synthesis and biological evaluation of piperazinyl carbamates and ureas as fatty acid amide hydrolase (FAAH) and transient receptor potential (TRP) channel dual ligands
2009 Morera, Enrico; Luciano De, Petrocellis; Morera, Ludovica; Aniello Schiano, Moriello; Alessia, Ligresti; Nalli, Marianna; David F., Woodward; Vincenzo Di, Marzo; Ortar, Giorgio
Pharmacological Differentiation of Bimatoprost and Latanoprost Induced Ocular Hypotension by a Second Generation Prostamide Antagonist (AGN211336)
2010 WOODWARD D., F; Liang, Y; WANG J., W; Li, C; GUZMAN V., M; KHARLAMB A., B; WHEELER L., A; GARST M., E; CARLING R. W., C; CORNELL C., L; FLIRI H., G; MARTOS J., L; PETTIT S., N; HOPPER D., L; DI MARZO, V; Ortar, Giorgio
(-)Menthylamine derivatives as potent and selective antagonists of transient receptor potential melastatin type-8 (TRPM8) channels
2010 Ortar, Giorgio; LUCIANO DE, Petrocellis; Morera, Ludovica; ANIELLO SCHIANO, Moriello; Pierangelo, Orlando; Morera, Enrico; Nalli, Marianna; VINCENZO DI, Marzo
Cytotoxic effect induced by combination of polyamines metabolites and endocannabinoid, anandamide, on human cancer cells: a new anticancer strategy”
2010 Batista de Carvalho, A. L. M.; Tempera, Giampiero; Viceconte, N.; Saccoccio, Stefania; Bidollari, E.; Nalli, Marianna; Morera, Enrico; Ortar, Giorgio; Agostinelli, Enzo
Discussion Addendum for: Palladium-Catalyzed Reduction of Vinyl Trifluoromethanesulfonates to Alkenes: Cholesta-3,5-DieneOrganic Syntheses
2011 Cacchi, Sandro; Morera, Enrico; Ortar, Giorgio
Development and characterization of endocannabinoid hydrolases FAAH and MAGL inhibitors bearing a benzotriazol-1-yl carboxamide scaffold
2012 Morera, Ludovica; Geoffray, Labar; Ortar, Giorgio; Didier M., Lambert
Spermine enzymatic oxidation products alone and in association with anandamide induce cytotoxicity in human cancer cells
2012 Tempera, Giampiero; Bidollari, E.; Meringolo, M.; Coccia, M.; Calcabrini, A.; Ortar, Giorgio; Morera, Enrico; Nalli, Marianna; Arancia, G.; Molinari, A.; Agostinelli, Enzo
Bovine serum amine oxidase and spermine in association with anandamide cause cytotoxicity in melanoma and colon adenocarcinoma cells
2012 Bidollari, E.; Tempera, Giampiero; Ueshima, T.; Calcabrini, A.; Ortar, Giorgio; Morera, Enrico; Nalli, Marianna; Condello, M.; Arancia, G.; Molinari, A.; Agostinelli, Enzo
Modulation of thermo-transient receptor potential (thermo-TRP) channels by thymol-based compounds
2012 Ortar, Giorgio; Morera, Ludovica; Aniello Schiano, Moriello; Morera, Enrico; Nalli, Marianna; Vincenzo Di, Marzo; Luciano De, Petrocellis
Synthesis and biological evaluation of [6]-gingerol analogues as transient receptor potential channel TRPV1 and TRPA1 modulators
2012 Morera, Enrico; Luciano De, Petrocellis; Morera, Ludovica; Aniello Schiano, Moriello; Nalli, Marianna; Vincenzo Di, Marzo; Ortar, Giorgio
Biaryl tetrazolyl ureas inhibitors of endocannabinoid metabolism: modulation at the N-portion and distal phenyl ring
2013 Ortar, Giorgio; Morera, Enrico; Luciano De, Petrocellis; Alessia, Ligresti; Aniello Schiano, Moriello; Morera, Ludovica; Nalli, Marianna; Ragno, Rino; Pirolli, Adele; Vincenzo Di, Marzo
Tetrahydro-beta-carboline derivatives targeting fatty acid amide hydrolase (FAAH) and transient receptor potential (TRP) channels
2013 Ortar, Giorgio; L., De Petrocellis; A., Schiano Moriello; M., Allara; Morera, Enrico; Nalli, Marianna; V., Di Marzo
Molecular Docking Of Biaryl Tetrazolyl Ureas As Inhibitors Of Endocannabinoid Metabolism
2013 Pirolli, Adele; Ballante, Flavio; Patsilinakos, A.; Ortar, Giorgio; Morera, Enrico; Ragno, Rino
The effects of an Inhibitor of Diglyceride Lipase on Collagen-induced Pltelet Activation
2013 E. C. G., Jackson; Ortar, Giorgio; A., Mcnicol
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Development of the First Potential Covalent Inhibitors of Anandamide Cellular Uptake | 2006 | SCHIANO MORIELLO, A; Balas, L; Ligresti, A; CASCIO M., G; Durand, T; Morera, Enrico; Ortar, Giorgio; DI MARZO, V. | |
New N-Arachidonoylserotonin Analogues with Potential 'Dual' Mechanism Action against Pain | 2007 | Ortar, Giorgio; CASCIO MARIA, Grazia; DE PETROCELLIS, Luciano; Morera, Enrico; Rossi, Francesca; SCHIANO MORIELLO, Aniello; Nalli, Marianna; DE NOVELLIS, Vito; WOODWARD DAVID, F; Maione, Sabatino; DI MARZO, Vincenzo | |
New tetrazole-based selective anandamide uptake inhibitors | 2008 | Ortar, Giorgio; Aniello Schiano, Moriello; Maria Grazia, Cascio; Luciano De, Petrocellis; Alessia, Ligresti; Morera, Enrico; Nalli, Marianna; Vincenzo Di, Marzo | |
Antinociceptive Effects of Tetrazole Inhibitors of Endocannabinoid Inactivation: Cannabinoid and Non-cannabinoid Receptor-mediated Mechanisms | 2008 | S., Maione; Morera, Enrico; I., Marabese; A., Ligresti; L., Luongo; Ortar, Giorgio; V., DI MARZO | |
Carbamoyl tetrazoles as inhibitors of endocannabinoid inactivation: A critical revisitation | 2008 | Ortar, Giorgio; Maria Grazia, Cascio; A., Schiano Moriello; Mercedes, Camalli; Morera, Enrico; Nalli, Marianna; Vincenzo Di, Marzo | |
Development of a potent inhibitor of 2-arachidonoylglycerol hydrolysis with antinociceptive activity in vivo | 2009 | Tiziana, Bisogno; Ortar, Giorgio; Stefania, Petrosino; Morera, Enrico; Enza, Palazzo; Nalli, Marianna; Sabatino, Maione; Vincenzo Di, Marzo | |
Synthesis and biological evaluation of piperazinyl carbamates and ureas as fatty acid amide hydrolase (FAAH) and transient receptor potential (TRP) channel dual ligands | 2009 | Morera, Enrico; Luciano De, Petrocellis; Morera, Ludovica; Aniello Schiano, Moriello; Alessia, Ligresti; Nalli, Marianna; David F., Woodward; Vincenzo Di, Marzo; Ortar, Giorgio | |
Pharmacological Differentiation of Bimatoprost and Latanoprost Induced Ocular Hypotension by a Second Generation Prostamide Antagonist (AGN211336) | 2010 | WOODWARD D., F; Liang, Y; WANG J., W; Li, C; GUZMAN V., M; KHARLAMB A., B; WHEELER L., A; GARST M., E; CARLING R. W., C; CORNELL C., L; FLIRI H., G; MARTOS J., L; PETTIT S., N; HOPPER D., L; DI MARZO, V; Ortar, Giorgio | |
(-)Menthylamine derivatives as potent and selective antagonists of transient receptor potential melastatin type-8 (TRPM8) channels | 2010 | Ortar, Giorgio; LUCIANO DE, Petrocellis; Morera, Ludovica; ANIELLO SCHIANO, Moriello; Pierangelo, Orlando; Morera, Enrico; Nalli, Marianna; VINCENZO DI, Marzo | |
Cytotoxic effect induced by combination of polyamines metabolites and endocannabinoid, anandamide, on human cancer cells: a new anticancer strategy” | 2010 | Batista de Carvalho, A. L. M.; Tempera, Giampiero; Viceconte, N.; Saccoccio, Stefania; Bidollari, E.; Nalli, Marianna; Morera, Enrico; Ortar, Giorgio; Agostinelli, Enzo | |
Discussion Addendum for: Palladium-Catalyzed Reduction of Vinyl Trifluoromethanesulfonates to Alkenes: Cholesta-3,5-DieneOrganic Syntheses | 2011 | Cacchi, Sandro; Morera, Enrico; Ortar, Giorgio | |
Development and characterization of endocannabinoid hydrolases FAAH and MAGL inhibitors bearing a benzotriazol-1-yl carboxamide scaffold | 2012 | Morera, Ludovica; Geoffray, Labar; Ortar, Giorgio; Didier M., Lambert | |
Spermine enzymatic oxidation products alone and in association with anandamide induce cytotoxicity in human cancer cells | 2012 | Tempera, Giampiero; Bidollari, E.; Meringolo, M.; Coccia, M.; Calcabrini, A.; Ortar, Giorgio; Morera, Enrico; Nalli, Marianna; Arancia, G.; Molinari, A.; Agostinelli, Enzo | |
Bovine serum amine oxidase and spermine in association with anandamide cause cytotoxicity in melanoma and colon adenocarcinoma cells | 2012 | Bidollari, E.; Tempera, Giampiero; Ueshima, T.; Calcabrini, A.; Ortar, Giorgio; Morera, Enrico; Nalli, Marianna; Condello, M.; Arancia, G.; Molinari, A.; Agostinelli, Enzo | |
Modulation of thermo-transient receptor potential (thermo-TRP) channels by thymol-based compounds | 2012 | Ortar, Giorgio; Morera, Ludovica; Aniello Schiano, Moriello; Morera, Enrico; Nalli, Marianna; Vincenzo Di, Marzo; Luciano De, Petrocellis | |
Synthesis and biological evaluation of [6]-gingerol analogues as transient receptor potential channel TRPV1 and TRPA1 modulators | 2012 | Morera, Enrico; Luciano De, Petrocellis; Morera, Ludovica; Aniello Schiano, Moriello; Nalli, Marianna; Vincenzo Di, Marzo; Ortar, Giorgio | |
Biaryl tetrazolyl ureas inhibitors of endocannabinoid metabolism: modulation at the N-portion and distal phenyl ring | 2013 | Ortar, Giorgio; Morera, Enrico; Luciano De, Petrocellis; Alessia, Ligresti; Aniello Schiano, Moriello; Morera, Ludovica; Nalli, Marianna; Ragno, Rino; Pirolli, Adele; Vincenzo Di, Marzo | |
Tetrahydro-beta-carboline derivatives targeting fatty acid amide hydrolase (FAAH) and transient receptor potential (TRP) channels | 2013 | Ortar, Giorgio; L., De Petrocellis; A., Schiano Moriello; M., Allara; Morera, Enrico; Nalli, Marianna; V., Di Marzo | |
Molecular Docking Of Biaryl Tetrazolyl Ureas As Inhibitors Of Endocannabinoid Metabolism | 2013 | Pirolli, Adele; Ballante, Flavio; Patsilinakos, A.; Ortar, Giorgio; Morera, Enrico; Ragno, Rino | |
The effects of an Inhibitor of Diglyceride Lipase on Collagen-induced Pltelet Activation | 2013 | E. C. G., Jackson; Ortar, Giorgio; A., Mcnicol |
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