A simple, straightforward palladium-catalyzed approach to 2-(aminomethyl)-3-arylindoles from 3-(o-trifluoroacetamidoaryl)-1-propargylic alcohols, amines, and aryl iodides has been developed.

2-(Aminomethyl)-3-arylindoles from 3-(o-Trifluoroacetamidoaryl)-1-propargylic Alcohols, Aryl Halides, and Amines: A Domino Palladium-Catalyzed Three-Component Approach / Cacchi, Sandro; Fabrizi, Giancarlo; Goggiamani, Antonella; Iazzetti, Antonia; Verdiglione, Rosanna. - In: SYNTHESIS. - ISSN 0039-7881. - (2017). [10.1055/s-0036-1589016]

2-(Aminomethyl)-3-arylindoles from 3-(o-Trifluoroacetamidoaryl)-1-propargylic Alcohols, Aryl Halides, and Amines: A Domino Palladium-Catalyzed Three-Component Approach

CACCHI, Sandro;FABRIZI, Giancarlo;GOGGIAMANI, ANTONELLA;IAZZETTI, Antonia;VERDIGLIONE, ROSANNA
2017

Abstract

A simple, straightforward palladium-catalyzed approach to 2-(aminomethyl)-3-arylindoles from 3-(o-trifluoroacetamidoaryl)-1-propargylic alcohols, amines, and aryl iodides has been developed.
2-(aminomethyl)indoles; 3-(o-trifluoroacetamidoaryl)-1-propargylic alcohols; cyclization; domino reaction; multicomponent reaction; palladium; Catalysis; Organic Chemistry
01 Pubblicazione su rivista::01a Articolo in rivista
2-(Aminomethyl)-3-arylindoles from 3-(o-Trifluoroacetamidoaryl)-1-propargylic Alcohols, Aryl Halides, and Amines: A Domino Palladium-Catalyzed Three-Component Approach / Cacchi, Sandro; Fabrizi, Giancarlo; Goggiamani, Antonella; Iazzetti, Antonia; Verdiglione, Rosanna. - In: SYNTHESIS. - ISSN 0039-7881. - (2017). [10.1055/s-0036-1589016]
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Utilizza questo identificativo per citare o creare un link a questo documento: https://hdl.handle.net/11573/983694
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