SCIPIONE, Luigi
SCIPIONE, Luigi
DIPARTIMENTO DI CHIMICA E TECNOLOGIE DEL FARMACO
(Thiazol-2-yl)hydrazone derivatives from acetylpyridines as dual inhibitors of MAO and AChE: synthesis, biological evaluation and molecular modeling studies
2015 D’Ascenzio, M; Chimenti, Paola; Gidaro, Mc; DE MONTE, Celeste; DE VITA, Daniela; Granese, Arianna; Scipione, Luigi; DI SANTO, Roberto; Costa, G; Alcaro, S; Yáñez, M; Carradori, S.
4-aminopyridine derivatives with anticholinesterase and antiamnesic activity
2008 Scipione, Luigi; DE VITA, Daniela; Alessandra, Musella; Lisa, Flammini; Simona, Bertoni; Elisabetta, Barocelli
6-(1-Benzyl-1H-pyrrol-2-yl)-2,4-dioxo-5-hexenoic acids as dual inhibitors of recombinant HIV-1 integrase and ribonuclease H, synthesized by a parallel synthesis approach.
2013 Costi, Roberta; M., Metifiot; F., Esposito; CUZZUCOLI CRUCITTI, Giuliana; Pescatori, Luca; Messore, Antonella; Scipione, Luigi; Tortorella, Silvano; L., Zinzula; C., Marchand; Y., Pommier; E., Tramontano; DI SANTO, Roberto
Acetylcholinesterase inhibitors for the treatment of Alzheimer’s disease–a patent review (2016–present)
2021 Bortolami, M.; Rocco, D.; Messore, A.; Di Santo, R.; Costi, R.; Madia, V. N.; Scipione, L.; Pandolfi, F.
Activity of caffeic acid derivatives against Candida albicans biofilm
2014 DE VITA, Daniela; Friggeri, Laura; D'Auria, Felicia Diodata; Pandolfi, Fabiana; Francesco, Piccoli; Panella, Simona; Palamara, ANNA TERESA; Simonetti, Giovanna; Scipione, Luigi; R., Santo; DI SANTO, Roberto; Costi, Roberta; Tortorella, Silvano
Activity of Drugs Against Dormant Mycobacterium tuberculosis
2011 G., Piccaro; P., Filippini; F., Giannoni; Scipione, Luigi; Tortorella, Silvano; DE VITA, Daniela; Mellini, Paolo; L., Fattorini
Analytical characterization of an inulin-type fructooligosaccharide from root-tubers of Asphodelus ramosus L
2021 Madia, Valentina Noemi; De Vita, Daniela; Messore, Antonella; Toniolo, Chiara; Tudino, Valeria; De Leo, Alessandro; Pindinello, Ivano; Ialongo, Davide; Saccoliti, Francesco; D'Ursi, Anna Maria; Grimaldi, Manuela; Ceccobelli, Pietro; Scipione, Luigi; Di Santo, Roberto; Costi, Roberta
Anti-tumoral effects of a (1H-pyrrol-1-yl)methyl-1H-benzoimidazole carbamate ester derivative on head and neck squamous carcinoma cell lines
2021 Nicolai, Alice; Madia, Valentina Noemi; Messore, Antonella; De Vita, Daniela; De Leo, Alessandro; Ialongo, Davide; Tudino, Valeria; Tortorella, Elisabetta; Scipione, Luigi; Taurone, Samanta; Pergolizzi, Tiziano; Artico, Marco; Di Santo, Roberto; Costi, Roberta; Scarpa, Susanna
Article study on extra virgin olive oil: Quality evaluation by anti-radical activity, color analysis, and polyphenolic hplc-dad analysis
2021 Cairone, F.; Petralito, S.; Scipione, L.; Cesa, S.
Basic Quinolinonyl Diketo Acid Derivatives as Inhibitors of HIV Integrase and their Activity against RNase H Function of Reverse Transcriptase
2014 Costi, Roberta; Mathieu, Metifiot; Suhman, Chung; CUZZUCOLI CRUCITTI, Giuliana; Kasthuraiah, Maddali; Pescatori, Luca; Messore, Antonella; Madia, VALENTINA NOEMI; Giovanni, Pupo; Scipione, Luigi; Tortorella, Silvano; Francesco Saverio Di, Leva; Sandro, Cosconati; Luciana, Marinelli; Ettore, Novellino; Stuart F: J., Le Grice; Angela, Corona; Yves, Pommier; Christophe, Marchand; DI SANTO, Roberto
behavioral and electroencephalographic effects of choline esters able to delivery and release choline into the brain of animal model of Alzheimer disease.
2001 Carelli, Vincenzo; Liberatore, Felice; Scipione, Luigi; Rispoli, V.; Rotiroti, D.
behavioral and electroencephalographic effects of choline esters able to delivery and release choline into the brain of animal models of alzheimer's disease
2001 Carelli, Vincenzo; Liberatore, Felice; Scipione, Luigi; V., Rispoli; D., Rotiroti
Biological evaluation and structure-activity relationships of imidazole-based compounds as antiprotozoal agents
2018 Saccoliti, Francesco; Madia, VALENTINA NOEMI; Tudino, Valeria; DE LEO, Alessandro; Pescatori, Luca; Messore, Antonella; DE VITA, Daniela; Scipione, Luigi; Brun, Reto; Kaiser, Marcel; Mäser, Pascal; Magalhaes Calvet, Claudia; K Jennings, Gareth; M Podust, Larissa; Costi, Roberta; DI SANTO, Roberto
Choline pivaloyl ester enhances brain expression of both nerve growth factor and high-affinity receptor TrkA, and reverses memory and cognitive deficits, in rats with excitotoxic lesion of nucleus basalis magnocellularis
2008 Rispoli, V.; Marra, R.; Costa, N.; Rotiroti, D.; Tirassa, P.; Scipione, Luigi; DE VITA, Daniela; Liberatore, F.; Carelli, V.
Choline pivaloyl ester strengthened the benefit effects of Tacrine and Galantamine on electroencephalographic and cognitive performances in nucleus basalis magnocellularis-lesioned and aged rats
2006 V., Rispoli; R., Marra; N., Costa; D., Rotiroti; Scipione, Luigi; DE VITA, Daniela; Felice, Liberatore; Vincenzo, Carelli
Choline pivaloyl esters improve in rats cognitive and memory performances impaired by scopolamine treatment or lesions of the nucleus basalis of Meynert
2004 Vincenzo, Rispoli; Domenicantonio, Rotiroti; Vincenzo, Carelli; Felice, Liberatore; Scipione, Luigi; Rosario, Marra; Gianfabio, Giorgioni; Antonio Di, Stefano
Comparison of different methods for the extraction of cannabinoids from cannabis
2019 De Vita, D.; Madia, V. N.; Tudino, V.; Saccoliti, F.; De Leo, A.; Messore, A.; Roscilli, P.; Botto, A.; Pindinello, I.; Santilli, G.; Scipione, L.; Costi, R.; Di Santo, R.
derivati della colina per il trattamento della malattia di Alzheimer
2000 Carelli, V.; Liberatore, Felice; Scipione, Luigi; Rotiroti, D.; Rispoli, V.; Cardellini, M.
Design, synthesis and biological evaluation of a series of iron and copper chelating deferiprone derivatives as new agents active against Candida albicans
2021 Bortolami, Martina; Pandolfi, Fabiana; Messore, Antonella; Rocco, Daniele; Feroci, Marta; DI SANTO, Roberto; DE VITA, Daniela; Costi, Roberta; Cascarino, Paola; Simonetti, Giovanna; Scipione, Luigi
Design, synthesis and biological evaluation of new pyrimidine derivatives as anticancer agents
2021 Madia, Valentina Noemi; Nicolai, Alice; Messore, Antonella; De Leo, Alessandro; Ialongo, Davide; Tudino, Valeria; Saccoliti, Francesco; De Vita, Daniela; Scipione, Luigi; Artico, Marco; Taurone, Samanta; Taglieri, Ludovica; Di Santo, Roberto; Scarpa, Susanna; Costi, Roberta
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
(Thiazol-2-yl)hydrazone derivatives from acetylpyridines as dual inhibitors of MAO and AChE: synthesis, biological evaluation and molecular modeling studies | 2015 | D’Ascenzio, M; Chimenti, Paola; Gidaro, Mc; DE MONTE, Celeste; DE VITA, Daniela; Granese, Arianna; Scipione, Luigi; DI SANTO, Roberto; Costa, G; Alcaro, S; Yáñez, M; Carradori, S. | |
4-aminopyridine derivatives with anticholinesterase and antiamnesic activity | 2008 | Scipione, Luigi; DE VITA, Daniela; Alessandra, Musella; Lisa, Flammini; Simona, Bertoni; Elisabetta, Barocelli | |
6-(1-Benzyl-1H-pyrrol-2-yl)-2,4-dioxo-5-hexenoic acids as dual inhibitors of recombinant HIV-1 integrase and ribonuclease H, synthesized by a parallel synthesis approach. | 2013 | Costi, Roberta; M., Metifiot; F., Esposito; CUZZUCOLI CRUCITTI, Giuliana; Pescatori, Luca; Messore, Antonella; Scipione, Luigi; Tortorella, Silvano; L., Zinzula; C., Marchand; Y., Pommier; E., Tramontano; DI SANTO, Roberto | |
Acetylcholinesterase inhibitors for the treatment of Alzheimer’s disease–a patent review (2016–present) | 2021 | Bortolami, M.; Rocco, D.; Messore, A.; Di Santo, R.; Costi, R.; Madia, V. N.; Scipione, L.; Pandolfi, F. | |
Activity of caffeic acid derivatives against Candida albicans biofilm | 2014 | DE VITA, Daniela; Friggeri, Laura; D'Auria, Felicia Diodata; Pandolfi, Fabiana; Francesco, Piccoli; Panella, Simona; Palamara, ANNA TERESA; Simonetti, Giovanna; Scipione, Luigi; R., Santo; DI SANTO, Roberto; Costi, Roberta; Tortorella, Silvano | |
Activity of Drugs Against Dormant Mycobacterium tuberculosis | 2011 | G., Piccaro; P., Filippini; F., Giannoni; Scipione, Luigi; Tortorella, Silvano; DE VITA, Daniela; Mellini, Paolo; L., Fattorini | |
Analytical characterization of an inulin-type fructooligosaccharide from root-tubers of Asphodelus ramosus L | 2021 | Madia, Valentina Noemi; De Vita, Daniela; Messore, Antonella; Toniolo, Chiara; Tudino, Valeria; De Leo, Alessandro; Pindinello, Ivano; Ialongo, Davide; Saccoliti, Francesco; D'Ursi, Anna Maria; Grimaldi, Manuela; Ceccobelli, Pietro; Scipione, Luigi; Di Santo, Roberto; Costi, Roberta | |
Anti-tumoral effects of a (1H-pyrrol-1-yl)methyl-1H-benzoimidazole carbamate ester derivative on head and neck squamous carcinoma cell lines | 2021 | Nicolai, Alice; Madia, Valentina Noemi; Messore, Antonella; De Vita, Daniela; De Leo, Alessandro; Ialongo, Davide; Tudino, Valeria; Tortorella, Elisabetta; Scipione, Luigi; Taurone, Samanta; Pergolizzi, Tiziano; Artico, Marco; Di Santo, Roberto; Costi, Roberta; Scarpa, Susanna | |
Article study on extra virgin olive oil: Quality evaluation by anti-radical activity, color analysis, and polyphenolic hplc-dad analysis | 2021 | Cairone, F.; Petralito, S.; Scipione, L.; Cesa, S. | |
Basic Quinolinonyl Diketo Acid Derivatives as Inhibitors of HIV Integrase and their Activity against RNase H Function of Reverse Transcriptase | 2014 | Costi, Roberta; Mathieu, Metifiot; Suhman, Chung; CUZZUCOLI CRUCITTI, Giuliana; Kasthuraiah, Maddali; Pescatori, Luca; Messore, Antonella; Madia, VALENTINA NOEMI; Giovanni, Pupo; Scipione, Luigi; Tortorella, Silvano; Francesco Saverio Di, Leva; Sandro, Cosconati; Luciana, Marinelli; Ettore, Novellino; Stuart F: J., Le Grice; Angela, Corona; Yves, Pommier; Christophe, Marchand; DI SANTO, Roberto | |
behavioral and electroencephalographic effects of choline esters able to delivery and release choline into the brain of animal model of Alzheimer disease. | 2001 | Carelli, Vincenzo; Liberatore, Felice; Scipione, Luigi; Rispoli, V.; Rotiroti, D. | |
behavioral and electroencephalographic effects of choline esters able to delivery and release choline into the brain of animal models of alzheimer's disease | 2001 | Carelli, Vincenzo; Liberatore, Felice; Scipione, Luigi; V., Rispoli; D., Rotiroti | |
Biological evaluation and structure-activity relationships of imidazole-based compounds as antiprotozoal agents | 2018 | Saccoliti, Francesco; Madia, VALENTINA NOEMI; Tudino, Valeria; DE LEO, Alessandro; Pescatori, Luca; Messore, Antonella; DE VITA, Daniela; Scipione, Luigi; Brun, Reto; Kaiser, Marcel; Mäser, Pascal; Magalhaes Calvet, Claudia; K Jennings, Gareth; M Podust, Larissa; Costi, Roberta; DI SANTO, Roberto | |
Choline pivaloyl ester enhances brain expression of both nerve growth factor and high-affinity receptor TrkA, and reverses memory and cognitive deficits, in rats with excitotoxic lesion of nucleus basalis magnocellularis | 2008 | Rispoli, V.; Marra, R.; Costa, N.; Rotiroti, D.; Tirassa, P.; Scipione, Luigi; DE VITA, Daniela; Liberatore, F.; Carelli, V. | |
Choline pivaloyl ester strengthened the benefit effects of Tacrine and Galantamine on electroencephalographic and cognitive performances in nucleus basalis magnocellularis-lesioned and aged rats | 2006 | V., Rispoli; R., Marra; N., Costa; D., Rotiroti; Scipione, Luigi; DE VITA, Daniela; Felice, Liberatore; Vincenzo, Carelli | |
Choline pivaloyl esters improve in rats cognitive and memory performances impaired by scopolamine treatment or lesions of the nucleus basalis of Meynert | 2004 | Vincenzo, Rispoli; Domenicantonio, Rotiroti; Vincenzo, Carelli; Felice, Liberatore; Scipione, Luigi; Rosario, Marra; Gianfabio, Giorgioni; Antonio Di, Stefano | |
Comparison of different methods for the extraction of cannabinoids from cannabis | 2019 | De Vita, D.; Madia, V. N.; Tudino, V.; Saccoliti, F.; De Leo, A.; Messore, A.; Roscilli, P.; Botto, A.; Pindinello, I.; Santilli, G.; Scipione, L.; Costi, R.; Di Santo, R. | |
derivati della colina per il trattamento della malattia di Alzheimer | 2000 | Carelli, V.; Liberatore, Felice; Scipione, Luigi; Rotiroti, D.; Rispoli, V.; Cardellini, M. | |
Design, synthesis and biological evaluation of a series of iron and copper chelating deferiprone derivatives as new agents active against Candida albicans | 2021 | Bortolami, Martina; Pandolfi, Fabiana; Messore, Antonella; Rocco, Daniele; Feroci, Marta; DI SANTO, Roberto; DE VITA, Daniela; Costi, Roberta; Cascarino, Paola; Simonetti, Giovanna; Scipione, Luigi | |
Design, synthesis and biological evaluation of new pyrimidine derivatives as anticancer agents | 2021 | Madia, Valentina Noemi; Nicolai, Alice; Messore, Antonella; De Leo, Alessandro; Ialongo, Davide; Tudino, Valeria; Saccoliti, Francesco; De Vita, Daniela; Scipione, Luigi; Artico, Marco; Taurone, Samanta; Taglieri, Ludovica; Di Santo, Roberto; Scarpa, Susanna; Costi, Roberta |