RAGNO, Rino

RAGNO, Rino  

DIPARTIMENTO DI CHIMICA E TECNOLOGIE DEL FARMACO  

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Titolo Data di pubblicazione Autore(i) File
(((thienylcarbonyl)alkyl)oxy)phenyl)- and (((pyrrylcarbonyl)alkyl)oxy)phenyl)oxazoline derivatives with potent and selective antihuman rhinovirus activity 1995 Massa, S; Corelli, F; Mai, Antonello; Ragno, Rino; DE MONTIS, A; LOI A., G; Corrias, S; MARONGIU M., E; LA COLLA, P.; Artico, Marino
2,6-Bis(3,4,5-trihydroxybenzylydene) derivatives of cyclohexanone: novel potent HIV-1 integrase inhibitors that prevent HIV-1 multiplication in cell-based assays 2004 Costi, Roberta; DI SANTO, Roberto; Artico, Marino; S., Massa; Ragno, Rino; R., Loddo; M., La Colla; E., Tramomtano; P., La Colla; A., Pani
2-(Alkyl/aryl)amino-6-benzylpyrimidin-4(3H)-ones as inhibitors of wild-type and mutant HIV-1: enantioselectivity studies. 2012 Rotili, Dante; A., Samuele; Domenico, Tarantino; Ragno, Rino; Musmuca, Ira; Ballante, Flavio; G., Botta; Morera, Ludovica; Pierini, Marco; R., Cirilli; M. B., Nawrozkij; E., Gonzalez; B., Clotet; Marino, Artico; J. A., Este; G., Maga; Mai, Antonello
3-(4-Aroyl-1-methyl-1H-2-pyrrolyl)-N-hydroxy-2-alkylamides as a New Class of Synthetic Histone Deacetylase Inhibitors. 1. Design, Synthesis, Biological Evaluation, and Binding Mode Studies Performed through Three Different Docking Procedures 2003 Mai, Antonello; S., Massa; Ragno, Rino; I., Cerbara; F., Jesacher; P., Loidl; G., Brosch
3-(4-Aroyl-1-methyl-1H-2-pyrrolyl)-N-hydroxy-2-propenamides as a New Class of Synthetic Histone Deacetylase Inhibitors. 2. Effect of Pyrrole-C2 and/or -C4 Substitutions on Biological Activity 2004 Mai, Antonello; S., Massa; I., Cerbara; Valente, Sergio; Ragno, Rino; P., Bottoni; R., Scatena; P., Loidl; G., Brosch
3-(4-Aroyl-1-methyl-1H-pyrrol-2-yl)-N-hydroxy-2-propenamides as a new class of synthetic histone deacetylase inhibitors. 3. Discovery of novel lead compounds through structure-based drug design and docking studies. 2004 Ragno, Rino; Mai, Antonello; Massa, S; Cerbara, I; Valente, Sergio; Bottoni, P; Scatena, R; Jesacher, F; Loidl, P; Brosch, G.
3-(4-aroyl-1h-pyrrol-2-yl)-N-hydroxy-2-propenamides, a new class of synthetic histone deacetylase inhibitors 2001 Massa, S; Mai, Antonello; Sbardella, G; Esposito, M; Ragno, Rino; Loidl, P; Brosch, G.
3-D QSAR SERVER – A 3-D QSAR models database for virtual screening 2010 Patsilinakos, A; Ballante, Flavio; Musmuca, Ira; Ragno, Rino
3-D QSAR Studies on Histone Deacetylase Inhibitors. A GOLPE/GRID Approach on Different Series of Compounds. 2006 Ragno, Rino; Simeoni, S; Valente, Sergio; Massa, S; Mai, Antonello
3-D QSAutogrid/R: An alternative procedure to build 3-D QSAR models. methodologies and applications 2012 Ballante, Flavio; Ragno, Rino
3D QSAR and Molecular Modeling on a Set of New Anti Mycobacterial Compounds. 1998 Artico, M.; DI SANTO, Roberto; Costi, Roberta; Massa, S.; Marshall, G. R.; Ragno, Rino
5-Alkyl-2-alkylamino-6-(2,6-difluorophenylalkyl)-3,4-dihydropyrimidin-4(3H)-ones, a new series of potent, broad-spectrum non-nucleoside reverse transcriptase inhibitors belonging to the DABO family 2005 Mai, Antonello; Artico, Marino; Ragno, Rino; Gianluca, Sbardella; Silvio, Massa; Chiara, Musiu; Massimo, Mura; Flavia, Marturana; Alessandra, Cadeddu; Giovanni, Maga; Paolo La, Colla
5-Alkyl-6-benzyl-2-(2-oxo-2-phenylethylsulfanyl)pyrimidin-4(3H)-ones, a series of anti-HIV-1 agents of the dihydro-alkoxy-benzyl-oxopyrimidine family with peculiar structure-activity relationship profile. 2008 Nawrozkij, Mb; Rotili, Dante; Tarantino, Domenico; Botta, G; Eremiychuk, As; Musmuca, Ira; Ragno, Rino; Samuele, A; Zanoli, S; ARMAND UGÓN, M; CLOTET CODINA, I; Novakov, Ia; Orlinson, Bs; Maga, G; Esté, Ja; Artico, Marino; Mai, Antonello
6-Aryl-2,4-dioxo-5-hexenoic Acids, Novel Integrase Inhibitors Active Against HIV-1 Multiplication in Cell-Based Assays. 2004 Costi, Roberta; DI SANTO, Roberto; Artico, Marino; A., Roux; Ragno, Rino; S., Massa; E., Tramontano; M., LA COLLA; R., Loddo; M. E., Marongiu; A., Pani; P., LA COLLA
A Combination of Molecular Dynamics and Docking Calculations to Explore the Binding Mode of ADS-J1, a Polyanionic Compound Endowed with Anti-HIV-1 Activity 2006 F., Manetti; C., Tintori; M., ARMAND UGN; I., CLOTET CODINA; S., Massa; Ragno, Rino; J. A., Est; M., Botta
A combined structure and ligand-based application on BSAO as an encouraging approach in anti-cancer therapy. 2014 Ballante, Flavio; Tempera, Giampiero; Agostinelli, Enzo; Ragno, Rino
A comparative analysis of punicalagin interaction with PDIA1 and PDIA3 by biochemical and computational approaches 2021 Paglia, G.; Antonini, L.; Cervoni, L.; Ragno, R.; Sabatino, M.; Minacori, M.; Rubini, E.; Altieri, F.
A series of COX-2 inhibitors endowed with NO-releasing properties: synthesis, biological evaluation, and docking analysis 2016 Consalvi, Sara; Poce, Giovanna; Ragno, Rino; Sabatino, Manuela; Lamotta, Concettina; Sartini, Stefania; Calderone, Vincenzo; Martelli, Alma; Ghelardini, Carla; Dicesaremannelli, Lorenzo; Biava, Mariangela
Ab-initio and experimental study of pentose sugar dehydration mechanism in the gas phase 2018 Antonini, L.; Garzoli, S.; Ricci, A.; Troiani, A.; Salvitti, C.; Giacomello, P.; Ragno, R.; Patsilinakos, Alexandros; Di Rienzo, B.; Pepi, F.
Acidi 6-Aril-2,4-dioxo-5-esenoici, Nuovi Inibitori dell’Integrasi. Blocco la Replicazione dell’HIV-1 in Cellule Infettate. 2003 DI SANTO, Roberto; Costi, Roberta; M., Artico; A., Roux; Ragno, Rino; F., Esposito; L., Onidi; M., Marongiu; M., Atzori; P., LA COLLA