PROIA, ELEONORA
PROIA, ELEONORA
DIPARTIMENTO DI CHIMICA E TECNOLOGIE DEL FARMACO
(Heteroarylmethyl)benzoic acids as a new class of bacterial cystathionine γ-lyase inhibitors. Synthesis, biological evaluation, and molecular modeling
2024 Golovina, Anastasia; Proia, Eleonora; Fiorentino, Francesco; Yunin, Maxim; Kasatkina, Maria; Zigangirova, Nailya; Soloveva, Anna; Sysolyatina, Elena; Ermolaeva, Svetlana; Novikov, Roman; Silonov, Sergei; Pushkin, Sergei; Mladenović, Milan; Isakova, Julia; Belik, Albina; Nawrozkij, Maxim; Rotili, Dante; Ragno, Rino; Ivanov, Roman
1,2,4-Oxadiazoles in medicinal chemistry: trends of the last years
2025 Cherkasova, Anastasia; Astolfi, Roberta; Nawrozkij, Maxim; Gladkikh, Boris; Proia, Eleonora; Giuliani, Lidia; Rotili, Dante; Ragno, Rino; Ivanov, Roman
Bovine serum amine oxidase and polyamine analogues: chemical synthesis and biological evaluation integrated with molecular docking and 3-D QSAR studies
2022 Ragno, Rino; Anna, Minarini; Proia, Eleonora; Antonini, Lorenzo; Andrea, Milelli; Vincenzo, Tumiatti; Marco, Fiore; Fino, Pasquale; Rutigliano, Lavinia; Fioravanti, Rossella; Tahara, Tomoaki; Pacella, Elena; Greco, Antonio; Canettieri, Gianluca; Maria Luisa Di Paolo, ; Agostinelli, Enzo
Essential oils as antimicrobials against Acinetobacter baumannii. Experimental and literature data to definite predictive quantitative composition–activity relationship models using machine learning algorithms
2025 Astolfi, Roberta; Oliva, Alessandra; Raffo, Antonio; Sapienza, Filippo; Ragno, Alessio; Proia, Eleonora; Mastroianni, Claudio M; Luceri, Cristina; Bozovic, Mijat; Mladenovic, Milan; Papa, Rosanna; Bottoni, Patrizia; Mazzinelli, Elena; Nocca, Giuseppina; Ragno, Rino
Ligand-based and structure-based studies to develop predictive models for {SARS}-{CoV}-2 main protease inhibitors through the 3d-qsar.com portal
2022 Proia, Eleonora; Ragno, Alessio; Antonini, Lorenzo; Sabatino, Manuela; Mladenović, Milan; Capobianco, Roberto; Ragno, Rino
Molecular docking assessment of cathinones as 5-HT2AR ligands. Developing of predictive structure-based bioactive conformations and three-dimensional structure-activity relationships models for future recognition of abuse drugs
2023 Tomašević, Nevena; Vujović, Maja; Kostić, Emilija; Ragavendran, Venkatesan; Arsić, Biljana; Matić, Sanja Lj.; Božović, Mijat; Fioravanti, Rossella; Proia, Eleonora; Ragno, Rino; Mladenović, Milan
Pyrimidine thioethers. A novel class of antidepressant agents, endowed with anxiolytic, performance enhancing and nootropic activity
2023 Fioravanti, Rossella; Proia, Eleonora; Tyurenkov, Ivan N; Kurkin, Denis V; Bakulin, Dmitry A; Kovalev, Nikolay S; Sheikin, Dmitry S; Kirillov, Ivan A; Nawrozkij, Maxim B; Vernigora, Andrey A; Brunilina, Leila L; Fiorentino, Francesco; Mladenović, Milan; Rotili, Dante; Ragno, Rino
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| (Heteroarylmethyl)benzoic acids as a new class of bacterial cystathionine γ-lyase inhibitors. Synthesis, biological evaluation, and molecular modeling | 2024 | Golovina, Anastasia; Proia, Eleonora; Fiorentino, Francesco; Yunin, Maxim; Kasatkina, Maria; Zigangirova, Nailya; Soloveva, Anna; Sysolyatina, Elena; Ermolaeva, Svetlana; Novikov, Roman; Silonov, Sergei; Pushkin, Sergei; Mladenović, Milan; Isakova, Julia; Belik, Albina; Nawrozkij, Maxim; Rotili, Dante; Ragno, Rino; Ivanov, Roman | |
| 1,2,4-Oxadiazoles in medicinal chemistry: trends of the last years | 2025 | Cherkasova, Anastasia; Astolfi, Roberta; Nawrozkij, Maxim; Gladkikh, Boris; Proia, Eleonora; Giuliani, Lidia; Rotili, Dante; Ragno, Rino; Ivanov, Roman | |
| Bovine serum amine oxidase and polyamine analogues: chemical synthesis and biological evaluation integrated with molecular docking and 3-D QSAR studies | 2022 | Ragno, Rino; Anna, Minarini; Proia, Eleonora; Antonini, Lorenzo; Andrea, Milelli; Vincenzo, Tumiatti; Marco, Fiore; Fino, Pasquale; Rutigliano, Lavinia; Fioravanti, Rossella; Tahara, Tomoaki; Pacella, Elena; Greco, Antonio; Canettieri, Gianluca; Maria Luisa Di Paolo, ; Agostinelli, Enzo | |
| Essential oils as antimicrobials against Acinetobacter baumannii. Experimental and literature data to definite predictive quantitative composition–activity relationship models using machine learning algorithms | 2025 | Astolfi, Roberta; Oliva, Alessandra; Raffo, Antonio; Sapienza, Filippo; Ragno, Alessio; Proia, Eleonora; Mastroianni, Claudio M; Luceri, Cristina; Bozovic, Mijat; Mladenovic, Milan; Papa, Rosanna; Bottoni, Patrizia; Mazzinelli, Elena; Nocca, Giuseppina; Ragno, Rino | |
| Ligand-based and structure-based studies to develop predictive models for {SARS}-{CoV}-2 main protease inhibitors through the 3d-qsar.com portal | 2022 | Proia, Eleonora; Ragno, Alessio; Antonini, Lorenzo; Sabatino, Manuela; Mladenović, Milan; Capobianco, Roberto; Ragno, Rino | |
| Molecular docking assessment of cathinones as 5-HT2AR ligands. Developing of predictive structure-based bioactive conformations and three-dimensional structure-activity relationships models for future recognition of abuse drugs | 2023 | Tomašević, Nevena; Vujović, Maja; Kostić, Emilija; Ragavendran, Venkatesan; Arsić, Biljana; Matić, Sanja Lj.; Božović, Mijat; Fioravanti, Rossella; Proia, Eleonora; Ragno, Rino; Mladenović, Milan | |
| Pyrimidine thioethers. A novel class of antidepressant agents, endowed with anxiolytic, performance enhancing and nootropic activity | 2023 | Fioravanti, Rossella; Proia, Eleonora; Tyurenkov, Ivan N; Kurkin, Denis V; Bakulin, Dmitry A; Kovalev, Nikolay S; Sheikin, Dmitry S; Kirillov, Ivan A; Nawrozkij, Maxim B; Vernigora, Andrey A; Brunilina, Leila L; Fiorentino, Francesco; Mladenović, Milan; Rotili, Dante; Ragno, Rino |