GUGLIELMI, PAOLO
GUGLIELMI, PAOLO
DIPARTIMENTO DI CHIMICA E TECNOLOGIE DEL FARMACO
1,3-Dipolar Cycloaddition, HPLC Enantioseparation, and Docking Studies of Saccharin/Isoxazole and Saccharin/Isoxazoline Derivatives as Selective Carbonic Anhydrase IX and XII Inhibitors
2020 D'Ascenzio, M.; Secci, D.; Carradori, S.; Zara, S.; Guglielmi, P.; Cirilli, R.; Pierini, M.; Poli, G.; Tuccinardi, T.; Angeli, A.; Supuran, C. T.
4-(3-Nitrophenyl)thiazol-2-ylhydrazone derivatives as antioxidants and selective hMAO-B inhibitors: synthesis, biological activity and computational analysis
2019 Secci, Daniela; Carradori, Simone; Petzer, Anél; Guglielmi, Paolo; D’Ascenzio, Melissa; Chimenti, Paola; Bagetta, Donatella; Alcaro, Stefano; Zengin, Gokhan; Petzer, Jacobus P.; Ortuso, Francesco
A Multitarget Approach against Neuroinflammation: Alkyl Substituted Coumarins as Inhibitors of Enzymes Involved in Neurodegeneration
2023 Berrino, E.; Carradori, S.; Carta, F.; Melfi, F.; Gallorini, M.; Poli, G.; Tuccinardi, T.; Fernandez-Bolanos, J. G.; Lopez, O.; Petzer, J. P.; Petzer, A.; Guglielmi, P.; Secci, D.; Supuran, C. T.
A novel library of saccharin and acesulfame derivatives as potent and selective inhibitors of carbonic anhydrase IX and XII isoforms
2016 Carradori, Simone; Secci, Daniela; DE MONTE, Celeste; Mollica, Adriano; Ceruso, Mariangela; Akdemir, Atilla; Sobolev, Anatoly P; Codispoti, Rossella; DE COSMI, Federica; Guglielmi, Paolo; Supuran, Claudiu T.
An innovative spectroscopic approach for qualitative and quantitative evaluation of Mb-CO from myoglobin carbonylation reaction through chemometrics methods
2021 Mansoldo, F. R. P.; Berrino, E.; Guglielmi, P.; Carradori, S.; Carta, F.; Secci, D.; Supuran, C. T.; Vermelho, A. B.
An updated patent review on monoamine oxidase (MAO) inhibitors
2022 Guglielmi, Paolo; Carradori, Simone; D'Agostino, Ilaria; Campestre, Cristina; Petzer, Jacobus P
Analysis of imidazoles and triazoles in biological samples after MicroExtraction by packed sorbent
2017 Campestre, Cristina; Locatelli, Marcello; Guglielmi, Paolo; De Luca, Elisa; Bellagamba, Giuseppe; Menta, Sergio; Zengin, Gokhan; Celia, Christian; Di Marzio, Luisa; Carradori, Simone
Antimalarial agents from medicinal plant and fungal sources
2020 Luisi, Grazia; Carradori, Simone; Grande, Rossella; Secci, Daniela; Guglielmi, Paolo
Aurone Scaffold and Structural Analogues for the Development of Monoamine Oxidase (MAO) Inhibitors
2022 Guglielmi, Paolo; Pontecorvi, Virginia; Akdemir, Atilla
Benzo[b]tiophen-3-ol derivatives as effective inhibitors of human monoamine oxidase: design, synthesis, and biological activity
2019 Guglielmi, Paolo; Secci, Daniela; Petzer, Anél; Bagetta, Donatella; Chimenti, Paola; Rotondi, Giulia; Ferrante, Claudio; Recinella, Lucia; Leone, Sheila; Alcaro, Stefano; Zengin, Gokhan; Petzer, Jacobus P; Ortuso, Francesco; Carradori, Simone
Chalcones: Unearthing their therapeutic possibility as monoamine oxidase B inhibitors
2020 Guglielmi, Paolo; Mathew, Bijo; Secci, Daniela; Carradori, Simone
Chiral hydroxy metabolite of Mebendazole. Analytical and semi-preparative high-performance liquid chromatography resolution and chiroptical properties
2024 Guglielmi, Paolo; Pulitelli, Gaia; Arrighi, Francesca; Secci, Daniela; Pierini, Marco; Cirilli, Roberto
Crystal structure of the Eg5 - K858 complex and implications for structure-based design of thiadiazole-containing inhibitors
2018 Talapatra, Sandeep K.; Tham, Chuin Lean; Guglielmi, Paolo; Cirilli, Roberto; Chandrasekaran, Balakumar; Karpoormath, Rajshekhar; Carradori, Simone; Kozielski, Frank
Design, synthesis and biochemical evaluation of novel multi-target inhibitors as potential anti-Parkinson agents
2018 Carradori, Simone; Ottuso, Francesco; Petzer, Anèl; Bagetta, Donatella; DE MONTE, Celeste; Secci, Daniela; DE VITA, Daniela; Guglielmi, Paolo; Zengin, Gokhan; Aktumsek, Abdurrahman; Alcaro, Stefano; Petzer, Jacobus P.
Design, synthesis and biological activity of selective hCAs inhibitors based on 2-(benzylsulfinyl)benzoic acid scaffold
2019 Rotondi, G.; Guglielmi, P.; Carradori, S.; Secci, D.; De Monte, C.; De Filippis, B.; Maccallini, C.; Amoroso, R.; Cirilli, R.; Akdemir, A.; Angeli, A.; Supuran, C. T.
Design, synthesis, docking studies and monoamine oxidase inhibition of a small library of 1-acetyl- and 1-thiocarbamoyl-3,5-diphenyl-4,5-dihydro-(1h)-pyrazoles
2019 Guglielmi, Paolo; Carradori, Simone; Poli, Giulio; Secci, Daniela; Cirilli, Roberto; Rotondi, Giulia; Chimenti, Paola; Petzer, Anél; Petzer, Jacobus P.
Dual carbonic anhydrase ix/xii inhibitors and carbon monoxide releasing molecules modulate LPS-mediated inflammation in mouse macrophages
2021 Berrino, E.; Carradori, S.; Angeli, A.; Carta, F.; Supuran, C. T.; Guglielmi, P.; Coletti, C.; Paciotti, R.; Schweikl, H.; Maestrelli, F.; Cerbai, E.; Gallorini, M.
Enantiomers of triclabendazole sulfoxide: analytical and semipreparative HPLC separation, absolute configuration assignment, and transformation into sodium salt
2017 Ferretti, Rosella; Carradori, Simone; Guglielmi, Paolo; Pierini, Marco; Casulli, Adriano; Cirilli, Roberto
High-performance liquid chromatography enantioseparation of chiral 2-(benzylsulfinyl)benzamide derivatives on cellulose tris(3,5-dichlorophenylcarbamate) chiral stationary phase
2020 Carradori, S.; Secci, D.; Guglielmi, P.; Pierini, M.; Cirilli, R.
Indoleamine 2,3-dioxygenase
2023 Coluccia, Michele; Secci, Daniela; Guglielmi, Paolo
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| 1,3-Dipolar Cycloaddition, HPLC Enantioseparation, and Docking Studies of Saccharin/Isoxazole and Saccharin/Isoxazoline Derivatives as Selective Carbonic Anhydrase IX and XII Inhibitors | 2020 | D'Ascenzio, M.; Secci, D.; Carradori, S.; Zara, S.; Guglielmi, P.; Cirilli, R.; Pierini, M.; Poli, G.; Tuccinardi, T.; Angeli, A.; Supuran, C. T. | |
| 4-(3-Nitrophenyl)thiazol-2-ylhydrazone derivatives as antioxidants and selective hMAO-B inhibitors: synthesis, biological activity and computational analysis | 2019 | Secci, Daniela; Carradori, Simone; Petzer, Anél; Guglielmi, Paolo; D’Ascenzio, Melissa; Chimenti, Paola; Bagetta, Donatella; Alcaro, Stefano; Zengin, Gokhan; Petzer, Jacobus P.; Ortuso, Francesco | |
| A Multitarget Approach against Neuroinflammation: Alkyl Substituted Coumarins as Inhibitors of Enzymes Involved in Neurodegeneration | 2023 | Berrino, E.; Carradori, S.; Carta, F.; Melfi, F.; Gallorini, M.; Poli, G.; Tuccinardi, T.; Fernandez-Bolanos, J. G.; Lopez, O.; Petzer, J. P.; Petzer, A.; Guglielmi, P.; Secci, D.; Supuran, C. T. | |
| A novel library of saccharin and acesulfame derivatives as potent and selective inhibitors of carbonic anhydrase IX and XII isoforms | 2016 | Carradori, Simone; Secci, Daniela; DE MONTE, Celeste; Mollica, Adriano; Ceruso, Mariangela; Akdemir, Atilla; Sobolev, Anatoly P; Codispoti, Rossella; DE COSMI, Federica; Guglielmi, Paolo; Supuran, Claudiu T. | |
| An innovative spectroscopic approach for qualitative and quantitative evaluation of Mb-CO from myoglobin carbonylation reaction through chemometrics methods | 2021 | Mansoldo, F. R. P.; Berrino, E.; Guglielmi, P.; Carradori, S.; Carta, F.; Secci, D.; Supuran, C. T.; Vermelho, A. B. | |
| An updated patent review on monoamine oxidase (MAO) inhibitors | 2022 | Guglielmi, Paolo; Carradori, Simone; D'Agostino, Ilaria; Campestre, Cristina; Petzer, Jacobus P | |
| Analysis of imidazoles and triazoles in biological samples after MicroExtraction by packed sorbent | 2017 | Campestre, Cristina; Locatelli, Marcello; Guglielmi, Paolo; De Luca, Elisa; Bellagamba, Giuseppe; Menta, Sergio; Zengin, Gokhan; Celia, Christian; Di Marzio, Luisa; Carradori, Simone | |
| Antimalarial agents from medicinal plant and fungal sources | 2020 | Luisi, Grazia; Carradori, Simone; Grande, Rossella; Secci, Daniela; Guglielmi, Paolo | |
| Aurone Scaffold and Structural Analogues for the Development of Monoamine Oxidase (MAO) Inhibitors | 2022 | Guglielmi, Paolo; Pontecorvi, Virginia; Akdemir, Atilla | |
| Benzo[b]tiophen-3-ol derivatives as effective inhibitors of human monoamine oxidase: design, synthesis, and biological activity | 2019 | Guglielmi, Paolo; Secci, Daniela; Petzer, Anél; Bagetta, Donatella; Chimenti, Paola; Rotondi, Giulia; Ferrante, Claudio; Recinella, Lucia; Leone, Sheila; Alcaro, Stefano; Zengin, Gokhan; Petzer, Jacobus P; Ortuso, Francesco; Carradori, Simone | |
| Chalcones: Unearthing their therapeutic possibility as monoamine oxidase B inhibitors | 2020 | Guglielmi, Paolo; Mathew, Bijo; Secci, Daniela; Carradori, Simone | |
| Chiral hydroxy metabolite of Mebendazole. Analytical and semi-preparative high-performance liquid chromatography resolution and chiroptical properties | 2024 | Guglielmi, Paolo; Pulitelli, Gaia; Arrighi, Francesca; Secci, Daniela; Pierini, Marco; Cirilli, Roberto | |
| Crystal structure of the Eg5 - K858 complex and implications for structure-based design of thiadiazole-containing inhibitors | 2018 | Talapatra, Sandeep K.; Tham, Chuin Lean; Guglielmi, Paolo; Cirilli, Roberto; Chandrasekaran, Balakumar; Karpoormath, Rajshekhar; Carradori, Simone; Kozielski, Frank | |
| Design, synthesis and biochemical evaluation of novel multi-target inhibitors as potential anti-Parkinson agents | 2018 | Carradori, Simone; Ottuso, Francesco; Petzer, Anèl; Bagetta, Donatella; DE MONTE, Celeste; Secci, Daniela; DE VITA, Daniela; Guglielmi, Paolo; Zengin, Gokhan; Aktumsek, Abdurrahman; Alcaro, Stefano; Petzer, Jacobus P. | |
| Design, synthesis and biological activity of selective hCAs inhibitors based on 2-(benzylsulfinyl)benzoic acid scaffold | 2019 | Rotondi, G.; Guglielmi, P.; Carradori, S.; Secci, D.; De Monte, C.; De Filippis, B.; Maccallini, C.; Amoroso, R.; Cirilli, R.; Akdemir, A.; Angeli, A.; Supuran, C. T. | |
| Design, synthesis, docking studies and monoamine oxidase inhibition of a small library of 1-acetyl- and 1-thiocarbamoyl-3,5-diphenyl-4,5-dihydro-(1h)-pyrazoles | 2019 | Guglielmi, Paolo; Carradori, Simone; Poli, Giulio; Secci, Daniela; Cirilli, Roberto; Rotondi, Giulia; Chimenti, Paola; Petzer, Anél; Petzer, Jacobus P. | |
| Dual carbonic anhydrase ix/xii inhibitors and carbon monoxide releasing molecules modulate LPS-mediated inflammation in mouse macrophages | 2021 | Berrino, E.; Carradori, S.; Angeli, A.; Carta, F.; Supuran, C. T.; Guglielmi, P.; Coletti, C.; Paciotti, R.; Schweikl, H.; Maestrelli, F.; Cerbai, E.; Gallorini, M. | |
| Enantiomers of triclabendazole sulfoxide: analytical and semipreparative HPLC separation, absolute configuration assignment, and transformation into sodium salt | 2017 | Ferretti, Rosella; Carradori, Simone; Guglielmi, Paolo; Pierini, Marco; Casulli, Adriano; Cirilli, Roberto | |
| High-performance liquid chromatography enantioseparation of chiral 2-(benzylsulfinyl)benzamide derivatives on cellulose tris(3,5-dichlorophenylcarbamate) chiral stationary phase | 2020 | Carradori, S.; Secci, D.; Guglielmi, P.; Pierini, M.; Cirilli, R. | |
| Indoleamine 2,3-dioxygenase | 2023 | Coluccia, Michele; Secci, Daniela; Guglielmi, Paolo |