Sfoglia per Autore
Benzo[b]tiophen-3-ol derivatives as effective inhibitors of human monoamine oxidase: design, synthesis, and biological activity
2019 Guglielmi, Paolo; Secci, Daniela; Petzer, Anél; Bagetta, Donatella; Chimenti, Paola; Rotondi, Giulia; Ferrante, Claudio; Recinella, Lucia; Leone, Sheila; Alcaro, Stefano; Zengin, Gokhan; Petzer, Jacobus P; Ortuso, Francesco; Carradori, Simone
Novel therapies for glaucoma: a patent review (2013-2019)
2019 Guglielmi, Paolo; Carradori, Simone; Campestre, Cristina; Poce, Giovanna
Design, synthesis, docking studies and monoamine oxidase inhibition of a small library of 1-acetyl- and 1-thiocarbamoyl-3,5-diphenyl-4,5-dihydro-(1h)-pyrazoles
2019 Guglielmi, Paolo; Carradori, Simone; Poli, Giulio; Secci, Daniela; Cirilli, Roberto; Rotondi, Giulia; Chimenti, Paola; Petzer, Anél; Petzer, Jacobus P.
Chalcones: Unearthing their therapeutic possibility as monoamine oxidase B inhibitors
2020 Guglielmi, Paolo; Mathew, Bijo; Secci, Daniela; Carradori, Simone
Innovative pH-interfering agents in association with anticancer agents
2020 Secci, D.; Guglielmi, P.
Antimalarial agents from medicinal plant and fungal sources
2020 Luisi, Grazia; Carradori, Simone; Grande, Rossella; Secci, Daniela; Guglielmi, Paolo
1,3-Dipolar Cycloaddition, HPLC Enantioseparation, and Docking Studies of Saccharin/Isoxazole and Saccharin/Isoxazoline Derivatives as Selective Carbonic Anhydrase IX and XII Inhibitors
2020 D'Ascenzio, M.; Secci, D.; Carradori, S.; Zara, S.; Guglielmi, P.; Cirilli, R.; Pierini, M.; Poli, G.; Tuccinardi, T.; Angeli, A.; Supuran, C. T.
High-performance liquid chromatography enantioseparation of chiral 2-(benzylsulfinyl)benzamide derivatives on cellulose tris(3,5-dichlorophenylcarbamate) chiral stationary phase
2020 Carradori, S.; Secci, D.; Guglielmi, P.; Pierini, M.; Cirilli, R.
Novel insights on saccharin- and acesulfame-based carbonic anhydrase inhibitors: design, synthesis, modelling investigations and biological activity evaluation
2020 Guglielmi, P.; Rotondi, G.; Secci, D.; Angeli, A.; Chimenti, P.; Nocentini, A.; Bonardi, A.; Gratteri, P.; Carradori, S.; Supuran, C. T.
Natural compounds and extracts as novel antimicrobial agents
2020 Guglielmi, P.; Pontecorvi, V.; Rotondi, G.
Synthesis and evaluation of a large library of nitroxoline derivatives as pancreatic cancer antiproliferative agents
2020 Veschi, Serena; Carradori, Simone; De Lellis, Laura; Florio, Rosalba; Brocco, Davide; Secci, Daniela; Guglielmi, Paolo; Spano, Mattia; Sobolev, Anatoly P.; Cama, Alessandro
Synthesis and biological evaluation of carvacrol-based derivatives as dual inhibitors of H. Pylori strains and ags cell proliferation
2020 Sisto, F.; Carradori, S.; Guglielmi, P.; Traversi, C. B.; Spano, M.; Sobolev, A. P.; Secci, D.; Di Marcantonio, M. C.; Haloci, E.; Grande, R.; Mincione, G.
Dual carbonic anhydrase ix/xii inhibitors and carbon monoxide releasing molecules modulate LPS-mediated inflammation in mouse macrophages
2021 Berrino, E.; Carradori, S.; Angeli, A.; Carta, F.; Supuran, C. T.; Guglielmi, P.; Coletti, C.; Paciotti, R.; Schweikl, H.; Maestrelli, F.; Cerbai, E.; Gallorini, M.
Synthesis and evaluation of thymol-based synthetic derivatives as dual-action inhibitors against different strains of h. pylori and AGS cell line
2021 Sisto, F.; Carradori, S.; Guglielmi, P.; Spano, M.; Secci, D.; Granese, A.; Sobolev, A. P.; Grande, R.; Campestre, C.; Di Marcantonio, M. C.; Mincione, G.
An innovative spectroscopic approach for qualitative and quantitative evaluation of Mb-CO from myoglobin carbonylation reaction through chemometrics methods
2021 Mansoldo, F. R. P.; Berrino, E.; Guglielmi, P.; Carradori, S.; Carta, F.; Secci, D.; Supuran, C. T.; Vermelho, A. B.
New aspects of monoamine oxidase b inhibitors: The key role of halogens to open the golden door
2021 Mathew, B.; Carradori, S.; Guglielmi, P.; Uddin, M. D.; Kim, H.
An updated patent review on monoamine oxidase (MAO) inhibitors
2022 Guglielmi, Paolo; Carradori, Simone; D'Agostino, Ilaria; Campestre, Cristina; Petzer, Jacobus P
Aurone Scaffold and Structural Analogues for the Development of Monoamine Oxidase (MAO) Inhibitors
2022 Guglielmi, Paolo; Pontecorvi, Virginia; Akdemir, Atilla
Novel Insights on Human Carbonic Anhydrase Inhibitors Based on Coumalic Acid: Design, Synthesis, Molecular Modeling Investigation, and Biological Studies
2022 Pontecorvi, Virginia; Mori, Mattia; Picarazzi, Francesca; Zara, Susi; Carradori, Simone; Cataldi, Amelia; Angeli, Andrea; Berrino, Emanuela; Chimenti, Paola; Ciogli, Alessia; Secci, Daniela; Guglielmi, Paolo; Supuran, Claudiu T.
Treatment of Toxoplasmosis: An Insight on Epigenetic Drugs
2022 Guglielmi, P.; Secci, D.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Benzo[b]tiophen-3-ol derivatives as effective inhibitors of human monoamine oxidase: design, synthesis, and biological activity | 2019 | Guglielmi, Paolo; Secci, Daniela; Petzer, Anél; Bagetta, Donatella; Chimenti, Paola; Rotondi, Giulia; Ferrante, Claudio; Recinella, Lucia; Leone, Sheila; Alcaro, Stefano; Zengin, Gokhan; Petzer, Jacobus P; Ortuso, Francesco; Carradori, Simone | |
Novel therapies for glaucoma: a patent review (2013-2019) | 2019 | Guglielmi, Paolo; Carradori, Simone; Campestre, Cristina; Poce, Giovanna | |
Design, synthesis, docking studies and monoamine oxidase inhibition of a small library of 1-acetyl- and 1-thiocarbamoyl-3,5-diphenyl-4,5-dihydro-(1h)-pyrazoles | 2019 | Guglielmi, Paolo; Carradori, Simone; Poli, Giulio; Secci, Daniela; Cirilli, Roberto; Rotondi, Giulia; Chimenti, Paola; Petzer, Anél; Petzer, Jacobus P. | |
Chalcones: Unearthing their therapeutic possibility as monoamine oxidase B inhibitors | 2020 | Guglielmi, Paolo; Mathew, Bijo; Secci, Daniela; Carradori, Simone | |
Innovative pH-interfering agents in association with anticancer agents | 2020 | Secci, D.; Guglielmi, P. | |
Antimalarial agents from medicinal plant and fungal sources | 2020 | Luisi, Grazia; Carradori, Simone; Grande, Rossella; Secci, Daniela; Guglielmi, Paolo | |
1,3-Dipolar Cycloaddition, HPLC Enantioseparation, and Docking Studies of Saccharin/Isoxazole and Saccharin/Isoxazoline Derivatives as Selective Carbonic Anhydrase IX and XII Inhibitors | 2020 | D'Ascenzio, M.; Secci, D.; Carradori, S.; Zara, S.; Guglielmi, P.; Cirilli, R.; Pierini, M.; Poli, G.; Tuccinardi, T.; Angeli, A.; Supuran, C. T. | |
High-performance liquid chromatography enantioseparation of chiral 2-(benzylsulfinyl)benzamide derivatives on cellulose tris(3,5-dichlorophenylcarbamate) chiral stationary phase | 2020 | Carradori, S.; Secci, D.; Guglielmi, P.; Pierini, M.; Cirilli, R. | |
Novel insights on saccharin- and acesulfame-based carbonic anhydrase inhibitors: design, synthesis, modelling investigations and biological activity evaluation | 2020 | Guglielmi, P.; Rotondi, G.; Secci, D.; Angeli, A.; Chimenti, P.; Nocentini, A.; Bonardi, A.; Gratteri, P.; Carradori, S.; Supuran, C. T. | |
Natural compounds and extracts as novel antimicrobial agents | 2020 | Guglielmi, P.; Pontecorvi, V.; Rotondi, G. | |
Synthesis and evaluation of a large library of nitroxoline derivatives as pancreatic cancer antiproliferative agents | 2020 | Veschi, Serena; Carradori, Simone; De Lellis, Laura; Florio, Rosalba; Brocco, Davide; Secci, Daniela; Guglielmi, Paolo; Spano, Mattia; Sobolev, Anatoly P.; Cama, Alessandro | |
Synthesis and biological evaluation of carvacrol-based derivatives as dual inhibitors of H. Pylori strains and ags cell proliferation | 2020 | Sisto, F.; Carradori, S.; Guglielmi, P.; Traversi, C. B.; Spano, M.; Sobolev, A. P.; Secci, D.; Di Marcantonio, M. C.; Haloci, E.; Grande, R.; Mincione, G. | |
Dual carbonic anhydrase ix/xii inhibitors and carbon monoxide releasing molecules modulate LPS-mediated inflammation in mouse macrophages | 2021 | Berrino, E.; Carradori, S.; Angeli, A.; Carta, F.; Supuran, C. T.; Guglielmi, P.; Coletti, C.; Paciotti, R.; Schweikl, H.; Maestrelli, F.; Cerbai, E.; Gallorini, M. | |
Synthesis and evaluation of thymol-based synthetic derivatives as dual-action inhibitors against different strains of h. pylori and AGS cell line | 2021 | Sisto, F.; Carradori, S.; Guglielmi, P.; Spano, M.; Secci, D.; Granese, A.; Sobolev, A. P.; Grande, R.; Campestre, C.; Di Marcantonio, M. C.; Mincione, G. | |
An innovative spectroscopic approach for qualitative and quantitative evaluation of Mb-CO from myoglobin carbonylation reaction through chemometrics methods | 2021 | Mansoldo, F. R. P.; Berrino, E.; Guglielmi, P.; Carradori, S.; Carta, F.; Secci, D.; Supuran, C. T.; Vermelho, A. B. | |
New aspects of monoamine oxidase b inhibitors: The key role of halogens to open the golden door | 2021 | Mathew, B.; Carradori, S.; Guglielmi, P.; Uddin, M. D.; Kim, H. | |
An updated patent review on monoamine oxidase (MAO) inhibitors | 2022 | Guglielmi, Paolo; Carradori, Simone; D'Agostino, Ilaria; Campestre, Cristina; Petzer, Jacobus P | |
Aurone Scaffold and Structural Analogues for the Development of Monoamine Oxidase (MAO) Inhibitors | 2022 | Guglielmi, Paolo; Pontecorvi, Virginia; Akdemir, Atilla | |
Novel Insights on Human Carbonic Anhydrase Inhibitors Based on Coumalic Acid: Design, Synthesis, Molecular Modeling Investigation, and Biological Studies | 2022 | Pontecorvi, Virginia; Mori, Mattia; Picarazzi, Francesca; Zara, Susi; Carradori, Simone; Cataldi, Amelia; Angeli, Andrea; Berrino, Emanuela; Chimenti, Paola; Ciogli, Alessia; Secci, Daniela; Guglielmi, Paolo; Supuran, Claudiu T. | |
Treatment of Toxoplasmosis: An Insight on Epigenetic Drugs | 2022 | Guglielmi, P.; Secci, D. |
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