SUPURAN, CLAUDIU TRANDAFIR
SUPURAN, CLAUDIU TRANDAFIR
DIPARTIMENTO DI CHIMICA E TECNOLOGIE DEL FARMACO
4-(3-Phenyl-4-(3,4,5-trimethoxybenzoyl)-1H-pyrrol-1-yl)benzenesulfonamide, a novel carbonic anhydrase and Wnt/β-Catenin signaling pathway dual-targeting inhibitor with potent activity against multidrug resistant cancer cells
2023 Masci, Domiziana; Puxeddu, Michela; Di Magno, Laura; D'Ambrosio, Michele; Parisi, Anastasia; Nalli, Marianna; Bai, Ruoli; Coluccia, Antonio; Sciò, Pietro; Orlando, Viviana; D'Angelo, Sara; Biagioni, Stefano; Urbani, Andrea; Hamel, Ernest; Nocentini, Alessio; Filiberti, Serena; Turati, Marta; Ronca, Roberto; Kopecka, Joanna; Riganti, Chiara; Fionda, Cinzia; Bordone, Rosa; Della Rocca, Giorgia; Canettieri, Gianluca; Supuran, Claudiu T; Silvestri, Romano; La Regina, Giuseppe
A novel inhibitor of carbonic anhydrases prevents hypoxia-induced tnbc cell plasticity
2020 Sarnella, A.; D'Avino, G.; Hill, B. S.; Alterio, V.; Winum, J. -Y.; Supuran, C. T.; De Simone, G.; Zannetti, A.
Amine-and amino acid-based compounds as carbonic anhydrase activators
2021 Angeli, A.; Berrino, E.; Carradori, S.; Supuran, C. T.; Cirri, M.; Carta, F.; Costantino, G.
An innovative spectroscopic approach for qualitative and quantitative evaluation of Mb-CO from myoglobin carbonylation reaction through chemometrics methods
2021 Mansoldo, F. R. P.; Berrino, E.; Guglielmi, P.; Carradori, S.; Carta, F.; Secci, D.; Supuran, C. T.; Vermelho, A. B.
Azidothymidine "clicked" into 1,2,3-Triazoles: First Report on Carbonic Anhydrase-Telomerase Dual-Hybrid Inhibitors
2020 Berrino, E.; Angeli, A.; Zhdanov, D. D.; Kiryukhina, A. P.; Milaneschi, A.; De Luca, A.; Bozdag, M.; Carradori, S.; Selleri, S.; Bartolucci, G.; Peat, T. S.; Ferraroni, M.; Supuran, C. T.; Carta, F.
Carbon Monoxide Release from Aryl-Propargyl Dicobalt(0)Hexacarbonyl Derivatives: A Computational and Experimental Study
2024 Paciotti, Roberto; Coletti, Cecilia; Berrino, Emanuela; Arrighi, Francesca; Maccelli, Alessandro; Lasalvia, Alba; Crestoni, Maria Elisa; Secci, Daniela; Carradori, Simone; Supuran, Claudiu; Carta, Fabrizio
Carbonic anhydrase inhibitors of different structures dilate pre-contracted porcine retinal arteries
2019 Eysteinsson, T.; Gudmundsdottir, H.; Hardarson, A. O.; Berrino, E.; Selleri, S.; Supuran, C. T.; Carta, F.
Design, synthesis, molecular modelling investigation and biological studies of novel human carbonic anhydrase inhibitors based on coumalic acid
2025 Pontecorvi, Virginia; Angeli, Andrea; Cutarella, Luigi; Mori, Mattia; Secci, Daniela; Coluccia, Michele; Carradori, Simone; Troiani, Anna; Pepi, Federico; Salvitti, Chiara; DI NOI, Alessia; Spano, Mattia; Arrighi, Francesca; DE FALCO, Elena; Bordin, Antonella; Berrino, Emanuela; Granese, Arianna; Chimenti, Paola; Guglielmi, Paolo; Supuran, Claudiu T.
Dual carbonic anhydrase ix/xii inhibitors and carbon monoxide releasing molecules modulate LPS-mediated inflammation in mouse macrophages
2021 Berrino, E.; Carradori, S.; Angeli, A.; Carta, F.; Supuran, C. T.; Guglielmi, P.; Coletti, C.; Paciotti, R.; Schweikl, H.; Maestrelli, F.; Cerbai, E.; Gallorini, M.
Geographical characterization by MAE-HPLC and NIR methodologies and carbonic anhydrase inhibition of Saffron components
2017 Nescatelli, Riccardo; Carradori, Simone; Marini, Federico; Caponigro, Vicky; Bucci, Remo; DE MONTE, Celeste; Mollica, Adriano; Mannina, Luisa; Ceruso, Mariangela; Supuran, CLAUDIU TRANDAFIR; Secci, Daniela
In silico identification and biological evaluation of antioxidant food components endowed with IX and XII hCA inhibition
2020 Costa, G.; Maruca, A.; Rocca, R.; Ambrosio, F. A.; Berrino, E.; Carta, F.; Mesiti, F.; Salatino, A.; Lanzillotta, D.; Trapasso, F.; Artese, A.; Alcaro, S.; Supuran, C. T.
Mechanisms of the Antiproliferative and Antitumor Activity of Novel Telomerase-Carbonic Anhydrase Dual-Hybrid Inhibitors
2021 Plyasova, A. A.; Berrino, E.; Khan, I. I.; Veselovsky, A. V.; Pokrovsky, V. S.; Angeli, A.; Ferraroni, M.; Supuran, C. T.; Pokrovskaya, M. V.; Alexandrova, S. S.; Gladilina, Y. A.; Sokolov, N. N.; Hilal, A.; Carta, F.; Zhdanov, D. D.
N-aryl-N′-ureido-O-sulfamates as potent and selective inhibitors of hCA VB over hCA VA: Deciphering the binding mode of new potential agents in mitochondrial dysfunctions
2020 Poli, G.; Bozdag, M.; Berrino, E.; Angeli, A.; Tuccinardi, T.; Carta, F.; Supuran, C. T.
New 1 H ‐indole‐2,3‐dione 3‐thiosemicarbazones with 3‐sulfamoylphenyl moiety as selective carbonic anhydrase inhibitors
2022 Eraslan‐elma, Pınar; Akdemir, Atilla; Berrino, Emanuela; Bozdağ, Murat; Supuran, Claudiu T.; Karalı, Nilgün
Novel Insights on CAI–CORM hybrids. Evaluation of the CO releasing properties and pain-relieving activity of differently substituted coumarins for the treatment of rheumatoid arthritis
2023 Berrino, Emanuela; Micheli, Laura; Carradori, Simone; di Cesare Mannelli, Lorenzo; Guglielmi, Paolo; De Luca, Alessandro; Carta, Fabrizio; Ghelardini, Carla; Secci, Daniela; Supuran, Claudiu T.
Novel sulfamide-containing compounds as selective carbonic anhydrase i inhibitors
2017 Berrino, Emanuela; Bua, Silvia; Mori, Mattia; Botta, Maurizio; Murthy, Vallabhaneni S.; Vijayakumar, Vijayaparthasarathi; Tamboli, Yasinalli; Bartolucci, GIAN LUCA; Mugelli, Alessandro; Cerbai, Elisabetta; Supuran, CLAUDIU TRANDAFIR; Carta, Fabrizio
Plasmatic exosomes from prostate cancer patients show increased carbonic anhydrase IX expression and activity and low ph
2020 Logozzi, Mariantonia; Mizzoni, Davide; Capasso, Clemente; Del Prete, Sonia; Di Raimo, Rossella; Falchi, Mario; Angelini, Daniela F; Sciarra, Alessandro; Maggi, Martina; Supuran, Claudiu T; Fais, Stefano
Pyrrolyl and indolyl α-γ-diketo acid derivatives acting as selective inhibitors of human carbonic anhydrases IX and XII
2023 Ialongo, Davide; Messore, Antonella; Madia, VALENTINA NOEMI; Tudino, Valeria; Nocentini, Alessio; Gratteri, Paola; Giovannuzzi, Simone; Supuran, Claudiu T.; Nicolai, Alice; Scarpa, Susanna; Taurone, Samanta; Camarda, Michele; Artico, Marco; Papa, Veronica; Saccoliti, Francesco; Scipione, Luigi; DI SANTO, Roberto; Costi, Roberta
State of the art of carbonic anhydrase activators
2023 Fiorentino, Francesco; Carta, Fabrizio; Rotili, Dante; Mai, Antonello; Supuran, Claudiu T
Synthesis and carbonic anhydrase inhibitory properties of novel 4-(2-aminoethyl)benzenesulfonamide-dipeptide conjugates
2019 Küçükbay, Hasan; Buğday, Nesrin; Küçükbay, F. Zehra; Berrino, Emanuela; Bartolucci, Gian Luca; Del Prete, Sonia; Capasso, Clemente; Supuran, Claudiu T.
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| 4-(3-Phenyl-4-(3,4,5-trimethoxybenzoyl)-1H-pyrrol-1-yl)benzenesulfonamide, a novel carbonic anhydrase and Wnt/β-Catenin signaling pathway dual-targeting inhibitor with potent activity against multidrug resistant cancer cells | 2023 | Masci, Domiziana; Puxeddu, Michela; Di Magno, Laura; D'Ambrosio, Michele; Parisi, Anastasia; Nalli, Marianna; Bai, Ruoli; Coluccia, Antonio; Sciò, Pietro; Orlando, Viviana; D'Angelo, Sara; Biagioni, Stefano; Urbani, Andrea; Hamel, Ernest; Nocentini, Alessio; Filiberti, Serena; Turati, Marta; Ronca, Roberto; Kopecka, Joanna; Riganti, Chiara; Fionda, Cinzia; Bordone, Rosa; Della Rocca, Giorgia; Canettieri, Gianluca; Supuran, Claudiu T; Silvestri, Romano; La Regina, Giuseppe | |
| A novel inhibitor of carbonic anhydrases prevents hypoxia-induced tnbc cell plasticity | 2020 | Sarnella, A.; D'Avino, G.; Hill, B. S.; Alterio, V.; Winum, J. -Y.; Supuran, C. T.; De Simone, G.; Zannetti, A. | |
| Amine-and amino acid-based compounds as carbonic anhydrase activators | 2021 | Angeli, A.; Berrino, E.; Carradori, S.; Supuran, C. T.; Cirri, M.; Carta, F.; Costantino, G. | |
| An innovative spectroscopic approach for qualitative and quantitative evaluation of Mb-CO from myoglobin carbonylation reaction through chemometrics methods | 2021 | Mansoldo, F. R. P.; Berrino, E.; Guglielmi, P.; Carradori, S.; Carta, F.; Secci, D.; Supuran, C. T.; Vermelho, A. B. | |
| Azidothymidine "clicked" into 1,2,3-Triazoles: First Report on Carbonic Anhydrase-Telomerase Dual-Hybrid Inhibitors | 2020 | Berrino, E.; Angeli, A.; Zhdanov, D. D.; Kiryukhina, A. P.; Milaneschi, A.; De Luca, A.; Bozdag, M.; Carradori, S.; Selleri, S.; Bartolucci, G.; Peat, T. S.; Ferraroni, M.; Supuran, C. T.; Carta, F. | |
| Carbon Monoxide Release from Aryl-Propargyl Dicobalt(0)Hexacarbonyl Derivatives: A Computational and Experimental Study | 2024 | Paciotti, Roberto; Coletti, Cecilia; Berrino, Emanuela; Arrighi, Francesca; Maccelli, Alessandro; Lasalvia, Alba; Crestoni, Maria Elisa; Secci, Daniela; Carradori, Simone; Supuran, Claudiu; Carta, Fabrizio | |
| Carbonic anhydrase inhibitors of different structures dilate pre-contracted porcine retinal arteries | 2019 | Eysteinsson, T.; Gudmundsdottir, H.; Hardarson, A. O.; Berrino, E.; Selleri, S.; Supuran, C. T.; Carta, F. | |
| Design, synthesis, molecular modelling investigation and biological studies of novel human carbonic anhydrase inhibitors based on coumalic acid | 2025 | Pontecorvi, Virginia; Angeli, Andrea; Cutarella, Luigi; Mori, Mattia; Secci, Daniela; Coluccia, Michele; Carradori, Simone; Troiani, Anna; Pepi, Federico; Salvitti, Chiara; DI NOI, Alessia; Spano, Mattia; Arrighi, Francesca; DE FALCO, Elena; Bordin, Antonella; Berrino, Emanuela; Granese, Arianna; Chimenti, Paola; Guglielmi, Paolo; Supuran, Claudiu T. | |
| Dual carbonic anhydrase ix/xii inhibitors and carbon monoxide releasing molecules modulate LPS-mediated inflammation in mouse macrophages | 2021 | Berrino, E.; Carradori, S.; Angeli, A.; Carta, F.; Supuran, C. T.; Guglielmi, P.; Coletti, C.; Paciotti, R.; Schweikl, H.; Maestrelli, F.; Cerbai, E.; Gallorini, M. | |
| Geographical characterization by MAE-HPLC and NIR methodologies and carbonic anhydrase inhibition of Saffron components | 2017 | Nescatelli, Riccardo; Carradori, Simone; Marini, Federico; Caponigro, Vicky; Bucci, Remo; DE MONTE, Celeste; Mollica, Adriano; Mannina, Luisa; Ceruso, Mariangela; Supuran, CLAUDIU TRANDAFIR; Secci, Daniela | |
| In silico identification and biological evaluation of antioxidant food components endowed with IX and XII hCA inhibition | 2020 | Costa, G.; Maruca, A.; Rocca, R.; Ambrosio, F. A.; Berrino, E.; Carta, F.; Mesiti, F.; Salatino, A.; Lanzillotta, D.; Trapasso, F.; Artese, A.; Alcaro, S.; Supuran, C. T. | |
| Mechanisms of the Antiproliferative and Antitumor Activity of Novel Telomerase-Carbonic Anhydrase Dual-Hybrid Inhibitors | 2021 | Plyasova, A. A.; Berrino, E.; Khan, I. I.; Veselovsky, A. V.; Pokrovsky, V. S.; Angeli, A.; Ferraroni, M.; Supuran, C. T.; Pokrovskaya, M. V.; Alexandrova, S. S.; Gladilina, Y. A.; Sokolov, N. N.; Hilal, A.; Carta, F.; Zhdanov, D. D. | |
| N-aryl-N′-ureido-O-sulfamates as potent and selective inhibitors of hCA VB over hCA VA: Deciphering the binding mode of new potential agents in mitochondrial dysfunctions | 2020 | Poli, G.; Bozdag, M.; Berrino, E.; Angeli, A.; Tuccinardi, T.; Carta, F.; Supuran, C. T. | |
| New 1 H ‐indole‐2,3‐dione 3‐thiosemicarbazones with 3‐sulfamoylphenyl moiety as selective carbonic anhydrase inhibitors | 2022 | Eraslan‐elma, Pınar; Akdemir, Atilla; Berrino, Emanuela; Bozdağ, Murat; Supuran, Claudiu T.; Karalı, Nilgün | |
| Novel Insights on CAI–CORM hybrids. Evaluation of the CO releasing properties and pain-relieving activity of differently substituted coumarins for the treatment of rheumatoid arthritis | 2023 | Berrino, Emanuela; Micheli, Laura; Carradori, Simone; di Cesare Mannelli, Lorenzo; Guglielmi, Paolo; De Luca, Alessandro; Carta, Fabrizio; Ghelardini, Carla; Secci, Daniela; Supuran, Claudiu T. | |
| Novel sulfamide-containing compounds as selective carbonic anhydrase i inhibitors | 2017 | Berrino, Emanuela; Bua, Silvia; Mori, Mattia; Botta, Maurizio; Murthy, Vallabhaneni S.; Vijayakumar, Vijayaparthasarathi; Tamboli, Yasinalli; Bartolucci, GIAN LUCA; Mugelli, Alessandro; Cerbai, Elisabetta; Supuran, CLAUDIU TRANDAFIR; Carta, Fabrizio | |
| Plasmatic exosomes from prostate cancer patients show increased carbonic anhydrase IX expression and activity and low ph | 2020 | Logozzi, Mariantonia; Mizzoni, Davide; Capasso, Clemente; Del Prete, Sonia; Di Raimo, Rossella; Falchi, Mario; Angelini, Daniela F; Sciarra, Alessandro; Maggi, Martina; Supuran, Claudiu T; Fais, Stefano | |
| Pyrrolyl and indolyl α-γ-diketo acid derivatives acting as selective inhibitors of human carbonic anhydrases IX and XII | 2023 | Ialongo, Davide; Messore, Antonella; Madia, VALENTINA NOEMI; Tudino, Valeria; Nocentini, Alessio; Gratteri, Paola; Giovannuzzi, Simone; Supuran, Claudiu T.; Nicolai, Alice; Scarpa, Susanna; Taurone, Samanta; Camarda, Michele; Artico, Marco; Papa, Veronica; Saccoliti, Francesco; Scipione, Luigi; DI SANTO, Roberto; Costi, Roberta | |
| State of the art of carbonic anhydrase activators | 2023 | Fiorentino, Francesco; Carta, Fabrizio; Rotili, Dante; Mai, Antonello; Supuran, Claudiu T | |
| Synthesis and carbonic anhydrase inhibitory properties of novel 4-(2-aminoethyl)benzenesulfonamide-dipeptide conjugates | 2019 | Küçükbay, Hasan; Buğday, Nesrin; Küçükbay, F. Zehra; Berrino, Emanuela; Bartolucci, Gian Luca; Del Prete, Sonia; Capasso, Clemente; Supuran, Claudiu T. |