TOMASELLI, DANIELA
TOMASELLI, DANIELA
DIPARTIMENTO DI MEDICINA MOLECOLARE
Different strategies to target the epigenome
2020 Tomaselli, Daniela
Disruptor of telomeric silencing 1-like (DOT1L): disclosing a new class of non-nucleoside inhibitors by means of ligand-based and structure-based approaches
2018 Sabatino, Manuela; Rotili, Dante; Patsilinakos, Alexandros; Forgione, Mariantonietta; Tomaselli, Daniela; Alby, Fréderic; Arimondo, Paola B.; Mai, Antonello; Ragno, Rino
DNA Methylation: Biological Implications and Modulation of Its Aberrant Dysregulation
2019 Lucidi, Alessia; Tomaselli, Daniela; Rotili, Dante; Mai, Antonello
Effect of α-methoxy substitution on the anti-HIV activity of dihydropyrimidin-4(3 H)-ones
2019 Nawrozkij, Maxim B.; Forgione, Mariantonietta; Yablokov, Alexandre S.; Lucidi, Alessia; Tomaselli, Daniela; Patsilinakos, Alexandros; Panella, Cristina; Hailu, Gebremedhin S.; Kirillov, Ivan A.; Badia, Roger; Riveira-Munoz, Eva; Crespan, Emmanuele; Armijos Rivera, Jorge I.; Cirilli, Roberto; Ragno, Rino; Esté, José A.; Maga, Giovanni; Mai, Antonello; Rotili, Dante
Epigenetic metalloenzymes
2018 Blanquart, Christophe; Linot, Camille; Cartron, Pierre-Francois; Tomaselli, Daniela; Mai, Antonello; Bertrand, Philippe
Epigenetic polypharmacology: a new frontier for epi-drug discovery
2019 Tomaselli, Daniela; Lucidi, Alessia; Rotili, Dante; Mai, Antonello
Novel polyamine-based Histone deacetylases-Lysine demethylase 1 dual binding inhibitors
2018 Milelli, Andrea; Marchetti, Chiara; Turrini, Eleonora; Catanzaro, Elena; Mazzone, Roberta; Tomaselli, Daniela; Fimognari, Carmela; Tumiatti, Vincenzo; Minarini, Anna
Recent advances in epigenetic proteolysis targeting chimeras (Epi-PROTACs)
2020 Tomaselli, D.; Mautone, N.; Mai, A.; Rotili, D.
Sirt4: a multifaceted enzyme at the crossroads of mitochondrial metabolism and cancer
2020 Tomaselli, D.; Steegborn, C.; Mai, A.; Rotili, D.
Sirtuins
2021 Zwergel, Clemens; Tomaselli, Daniela; Mai, Antonello
Specific inhibitors of mitochondrial deacylase sirtuin 4 endowed with cellular activity
2024 Pannek, M.; Alhalabi, Z.; Tomaselli, D.; Menna, M.; Fiorentino, F.; Robaa, D.; Weyand, M.; Puhlmann, M.; Tomassi, S.; Barreca, F.; Tafani, M.; Zaganjor, E.; Haigis, M. C.; Sippl, W.; Rotili, D.; Mai, A.; Steegborn, C.
Structure-reactivity relationships on substrates and inhibitors of the lysine deacylase sirtuin 2 from schistosoma mansoni (SmSirt2)
2019 Monaldi, Daria; Rotili, Dante; Julien Lancelot, ‡; Martin Marek, §; Nathalie Wössner, ∥; Lucidi, Alessia; Tomaselli, Daniela; Elizabeth Ramos-Morales, ‡; Christophe Romier, ∥; Pierce, ∥ Raymond J.; Mai, Antonello; and Manfred Jung, ‡
α,γ-Diketocarboxylic acids and their esters act as carbonic anhydrase IX and XII selective inhibitors
2019 Nocentini, Alessio; Lucidi, Alessia; Perut, Francesca; Massa, Annamaria; Tomaselli, Daniela; Gratteri, Paola; Baldini, Nicola; Rotili, Dante; Mai, Antonello; Supuran, Claudiu T.
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Different strategies to target the epigenome | 2020 | Tomaselli, Daniela | |
| Disruptor of telomeric silencing 1-like (DOT1L): disclosing a new class of non-nucleoside inhibitors by means of ligand-based and structure-based approaches | 2018 | Sabatino, Manuela; Rotili, Dante; Patsilinakos, Alexandros; Forgione, Mariantonietta; Tomaselli, Daniela; Alby, Fréderic; Arimondo, Paola B.; Mai, Antonello; Ragno, Rino | |
| DNA Methylation: Biological Implications and Modulation of Its Aberrant Dysregulation | 2019 | Lucidi, Alessia; Tomaselli, Daniela; Rotili, Dante; Mai, Antonello | |
| Effect of α-methoxy substitution on the anti-HIV activity of dihydropyrimidin-4(3 H)-ones | 2019 | Nawrozkij, Maxim B.; Forgione, Mariantonietta; Yablokov, Alexandre S.; Lucidi, Alessia; Tomaselli, Daniela; Patsilinakos, Alexandros; Panella, Cristina; Hailu, Gebremedhin S.; Kirillov, Ivan A.; Badia, Roger; Riveira-Munoz, Eva; Crespan, Emmanuele; Armijos Rivera, Jorge I.; Cirilli, Roberto; Ragno, Rino; Esté, José A.; Maga, Giovanni; Mai, Antonello; Rotili, Dante | |
| Epigenetic metalloenzymes | 2018 | Blanquart, Christophe; Linot, Camille; Cartron, Pierre-Francois; Tomaselli, Daniela; Mai, Antonello; Bertrand, Philippe | |
| Epigenetic polypharmacology: a new frontier for epi-drug discovery | 2019 | Tomaselli, Daniela; Lucidi, Alessia; Rotili, Dante; Mai, Antonello | |
| Novel polyamine-based Histone deacetylases-Lysine demethylase 1 dual binding inhibitors | 2018 | Milelli, Andrea; Marchetti, Chiara; Turrini, Eleonora; Catanzaro, Elena; Mazzone, Roberta; Tomaselli, Daniela; Fimognari, Carmela; Tumiatti, Vincenzo; Minarini, Anna | |
| Recent advances in epigenetic proteolysis targeting chimeras (Epi-PROTACs) | 2020 | Tomaselli, D.; Mautone, N.; Mai, A.; Rotili, D. | |
| Sirt4: a multifaceted enzyme at the crossroads of mitochondrial metabolism and cancer | 2020 | Tomaselli, D.; Steegborn, C.; Mai, A.; Rotili, D. | |
| Sirtuins | 2021 | Zwergel, Clemens; Tomaselli, Daniela; Mai, Antonello | |
| Specific inhibitors of mitochondrial deacylase sirtuin 4 endowed with cellular activity | 2024 | Pannek, M.; Alhalabi, Z.; Tomaselli, D.; Menna, M.; Fiorentino, F.; Robaa, D.; Weyand, M.; Puhlmann, M.; Tomassi, S.; Barreca, F.; Tafani, M.; Zaganjor, E.; Haigis, M. C.; Sippl, W.; Rotili, D.; Mai, A.; Steegborn, C. | |
| Structure-reactivity relationships on substrates and inhibitors of the lysine deacylase sirtuin 2 from schistosoma mansoni (SmSirt2) | 2019 | Monaldi, Daria; Rotili, Dante; Julien Lancelot, ‡; Martin Marek, §; Nathalie Wössner, ∥; Lucidi, Alessia; Tomaselli, Daniela; Elizabeth Ramos-Morales, ‡; Christophe Romier, ∥; Pierce, ∥ Raymond J.; Mai, Antonello; and Manfred Jung, ‡ | |
| α,γ-Diketocarboxylic acids and their esters act as carbonic anhydrase IX and XII selective inhibitors | 2019 | Nocentini, Alessio; Lucidi, Alessia; Perut, Francesca; Massa, Annamaria; Tomaselli, Daniela; Gratteri, Paola; Baldini, Nicola; Rotili, Dante; Mai, Antonello; Supuran, Claudiu T. |