CIANNI, LORENZO

CIANNI, LORENZO  

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Titolo Data di pubblicazione Autore(i) File
A comparative study of warheads for design of cysteine protease inhibitors 2017 Silva, Daniel G; Ribeiro, Jean F R; De Vita, Daniela; Cianni, Lorenzo; Franco, Caio Haddad; Freitas-Junior, Lucio H; Moraes, Carolina Borsoi; Rocha, Josmar R; Burtoloso, Antonio C B; Kenny, Peter W; Leitão, Andrei; Montanari, Carlos A
Experimental study and computational modelling of cruzain cysteine protease inhibition by dipeptidyl nitriles 2018 Dos Santos, Alberto Monteiro; Cianni, Lorenzo; De Vita, Daniela; Rosini, Fabiana; Leitão, Andrei; Laughton, Charles A; Lameira, Jerônimo; Montanari, Carlos A
Leveraging the cruzain S3 subsite to increase affinity for reversible covalent inhibitors 2018 Cianni, Lorenzo; Sartori, Geraldo; Rosini, Fabiana; De Vita, Daniela; Pires, Gabriel; Lopes, Bianca Rebelo; Leitão, Andrei; Burtoloso, Antonio C B; Montanari, Carlos A
Perylene and coronene derivatives binding to G-rich promoter oncogene sequences efficiently reduce their expression in cancer cells 2016 Micheli, Emanuela; Altieri, Alessandro; Cianni, Lorenzo; Cingolani, Chiara; Iachettini, Sara; Bianco, Armandodoriano; Leonetti, Carlo; Cacchione, Stefano; Biroccio, Annamaria; Franceschin, Marco; Rizzo, Angela
Synthesis and structure-activity relationship of nitrile-based cruzain inhibitors incorporating a trifluoroethylamine-based P2 amide replacement 2019 Gomes, Juliana C; Cianni, Lorenzo; Ribeiro, Jean; Dos Reis Rocho, Fernanda; da Costa Martins Silva, Samelyn; Batista, Pedro Henrique Jatai; Moraes, Carolina Borsoi; Franco, Caio Haddad; Freitas-Junior, Lucio H G; Kenny, Peter W; Leitão, Andrei; Burtoloso, Antonio C B; de Vita, Daniela; Montanari, Carlos A