DE MONTE, CELESTE
DE MONTE, CELESTE
DIPARTIMENTO DI CHIMICA E TECNOLOGIE DEL FARMACO
(Thiazol-2-yl)hydrazone derivatives from acetylpyridines as dual inhibitors of MAO and AChE: synthesis, biological evaluation and molecular modeling studies
2015 D’Ascenzio, M; Chimenti, Paola; Gidaro, Mc; DE MONTE, Celeste; DE VITA, Daniela; Granese, Arianna; Scipione, Luigi; DI SANTO, Roberto; Costa, G; Alcaro, S; Yáñez, M; Carradori, S.
A novel library of saccharin and acesulfame derivatives as potent and selective inhibitors of carbonic anhydrase IX and XII isoforms
2016 Carradori, Simone; Secci, Daniela; DE MONTE, Celeste; Mollica, Adriano; Ceruso, Mariangela; Akdemir, Atilla; Sobolev, Anatoly P; Codispoti, Rossella; DE COSMI, Federica; Guglielmi, Paolo; Supuran, Claudiu T.
Anti-Candida activity and cytotoxicity of a large library of new N-substituted-1,3-thiazolidin-4-one derivatives
2016 DE MONTE, Celeste; Carradori, Simone; Bizzarri, Bruna; Bolasco, Adriana; Caprara, Federica; Mollica, Adriano; Rivanera, Daniela; Mari, Emanuela; Zicari, Alessandra; Akdemir, Atilla; Secci, Daniela
Bioactive compounds of Crocus sativus L. and their semisynthetic derivatives as promising anti-Helicobacter pylori, anti-malarial and anti-leishmanial agents
2015 DE MONTE, Celeste; Bizzarri, Bruna; Gidaro, Maria Concetta; Carradori, Simone; Mollica, Adriano; Luisi, Grazia; Granese, Arianna; Alcaro, Stefano; Costa, Giosuè; Basilico, Nicoletta; Parapini, Silvia; Scaltrito, Maria Maddalena; Masia, Carla; Sisto, Francesca
Bladder cancer: Innovative approaches beyond the diagnosis
2014 Piergentili, Roberto; Carradori, Simone; Gulia, Caterina; DE MONTE, Celeste; Cristini, Cristiano; Grande, Pietro; Santini, Edoardo; Gentile, Vincenzo; DI PIERRO, GIOVANNI BATTISTA
Computational investigation of the selectivity of salen and tetrahydrosalen compounds towards the tumor-associated hCA XII isozyme
2015 Atilla, Akdemir; DE MONTE, Celeste; Simone, Carradori; Claudiu T., Supuran
Cyclic tertiary sulfamates: Selective inhibition of the tumor-associated carbonic anhydrases IX and XII by N- and O-substituted acesulfame derivatives
2014 DE MONTE, Celeste; Carradori, Simone; Secci, Daniela; D'Ascenzio, Melissa; Vullo, D; Ceruso, M; Supuran, Ct
Design, synthesis and biochemical evaluation of novel multi-target inhibitors as potential anti-Parkinson agents
2018 Carradori, Simone; Ottuso, Francesco; Petzer, Anèl; Bagetta, Donatella; DE MONTE, Celeste; Secci, Daniela; DE VITA, Daniela; Guglielmi, Paolo; Zengin, Gokhan; Aktumsek, Abdurrahman; Alcaro, Stefano; Petzer, Jacobus P.
Design, synthesis and biological activity of selective hCAs inhibitors based on 2-(benzylsulfinyl)benzoic acid scaffold
2019 Rotondi, G.; Guglielmi, P.; Carradori, S.; Secci, D.; De Monte, C.; De Filippis, B.; Maccallini, C.; Amoroso, R.; Cirilli, R.; Akdemir, A.; Angeli, A.; Supuran, C. T.
Design, synthesis and biological characterization of thiazolidin-4-one derivatives as promising inhibitors of Toxoplasma gondii
2014 D'Ascenzio, Melissa; Bizzarri, Bruna; DE MONTE, Celeste; Carradori, S; Bolasco, Adriana; Secci, Daniela; Rivanera, Daniela; Faulhaber, N; Bordon, C; Jones Brando, L.
Design, synthesis and evaluation of N-substituted saccharin derivatives as selective inhibitors of tumor-associated carbonic anhydrase XII
2014 D'Ascenzio, M; Carradori, S; DE MONTE, Celeste; Secci, Daniela; Ceruso, M; Supuran, Ct
Dual Cyclooxygenase and Carbonic Anhydrase Inhibition by Nonsteroidal Anti-Inflammatory Drugs for the Treatment of Cancer
2015 DE MONTE, Celeste; Carradori, Simone; Gentili, Andrea; Mollica, Adriano; Trisciuoglio, Daniela; Supuran, Claudiu T.
Evaluation of a large library of (thiazol-2-yl)hydrazones and analogues as histone acetyltransferase inhibitors: Enzyme and cellular studies.
2014 Carradori, S; Rotili, Dante; DE MONTE, Celeste; Lenoci, A; D'Ascenzio, M; Rodriguez, V; Filetici, Patrizia; Miceli, M; Nebbioso, A; Altucci, L; Secci, Daniela; Mai, Antonello
Geographical characterization by MAE-HPLC and NIR methodologies and carbonic anhydrase inhibition of Saffron components
2017 Nescatelli, Riccardo; Carradori, Simone; Marini, Federico; Caponigro, Vicky; Bucci, Remo; DE MONTE, Celeste; Mollica, Adriano; Mannina, Luisa; Ceruso, Mariangela; Supuran, CLAUDIU TRANDAFIR; Secci, Daniela
Identification of the stereochemical requirements in the 4-aryl-2-cycloalkylidenhydrazinylthiazole scaffold for the design of selective human monoamine oxidase B inhibitors
2014 D'Ascenzio, M; Carradori, S; Secci, Daniela; Mannina, Luisa; Sobolev, Ap; DE MONTE, Celeste; Cirilli, R; Yanez, M; Alcaro, S; Ortuso, F.
Metal-chelating salens and tetrahydrosalens and N- and O-substituted acesulfame and saccharin derivatives as selective inhibitors of the cancer-related carbonic anhydrases IX and XII
2015 DE MONTE, Celeste; Secci, Daniela; Simone, Carradori; Melissa, D’Ascenzio; Mariana, Farella; Claudiu T., Supuran
Modern extraction techniques and their impact on the pharmacological profile of Serenoa repens extracts for the treatment of lower urinary tract symptoms.
2014 DE MONTE, Celeste; S., Carradori; Granese, Arianna; DI PIERRO, GIOVANNI BATTISTA; Leonardo, Costantino; DE NUNZIO, Cosimo
New amide derivatives of Probenecid as selective inhibitors of carbonic anhydrase IX and XII: Biological evaluation and molecular modelling studies
2015 Carradori, Simone; Mollica, Adriano; Ceruso, Mariangela; D'Ascenzio, Melissa; DE MONTE, Celeste; Chimenti, Paola; Sabia, Rocchina; Akdemir, Atilla; Supuran, Claudiu T.
New insights into the biological properties of Crocus sativus L.: chemical modifications, human monoamine oxidases inhibition and molecular modeling studies
2014 DE MONTE, Celeste; Carradori, Simone; Chimenti, Paola; Secci, Daniela; Mannina, Luisa; Alcaro, F; Petzer, A; N'Da, Ci; Gidaro, Mc; Costa, G; Alcaro, S; Petzer, Jp
New thiadiazoline and thiadiazole analogues of K858: antiproliferative activity in a model of prostate carcinoma
2013 DE MONTE, Celeste; Carradori, S.; D’Ascenzio, M.; Chimenti, Paola; Secci, Daniela; Bolasco, Adriana; Nicolazzo, Chiara; Silvestri, Ida
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| (Thiazol-2-yl)hydrazone derivatives from acetylpyridines as dual inhibitors of MAO and AChE: synthesis, biological evaluation and molecular modeling studies | 2015 | D’Ascenzio, M; Chimenti, Paola; Gidaro, Mc; DE MONTE, Celeste; DE VITA, Daniela; Granese, Arianna; Scipione, Luigi; DI SANTO, Roberto; Costa, G; Alcaro, S; Yáñez, M; Carradori, S. | |
| A novel library of saccharin and acesulfame derivatives as potent and selective inhibitors of carbonic anhydrase IX and XII isoforms | 2016 | Carradori, Simone; Secci, Daniela; DE MONTE, Celeste; Mollica, Adriano; Ceruso, Mariangela; Akdemir, Atilla; Sobolev, Anatoly P; Codispoti, Rossella; DE COSMI, Federica; Guglielmi, Paolo; Supuran, Claudiu T. | |
| Anti-Candida activity and cytotoxicity of a large library of new N-substituted-1,3-thiazolidin-4-one derivatives | 2016 | DE MONTE, Celeste; Carradori, Simone; Bizzarri, Bruna; Bolasco, Adriana; Caprara, Federica; Mollica, Adriano; Rivanera, Daniela; Mari, Emanuela; Zicari, Alessandra; Akdemir, Atilla; Secci, Daniela | |
| Bioactive compounds of Crocus sativus L. and their semisynthetic derivatives as promising anti-Helicobacter pylori, anti-malarial and anti-leishmanial agents | 2015 | DE MONTE, Celeste; Bizzarri, Bruna; Gidaro, Maria Concetta; Carradori, Simone; Mollica, Adriano; Luisi, Grazia; Granese, Arianna; Alcaro, Stefano; Costa, Giosuè; Basilico, Nicoletta; Parapini, Silvia; Scaltrito, Maria Maddalena; Masia, Carla; Sisto, Francesca | |
| Bladder cancer: Innovative approaches beyond the diagnosis | 2014 | Piergentili, Roberto; Carradori, Simone; Gulia, Caterina; DE MONTE, Celeste; Cristini, Cristiano; Grande, Pietro; Santini, Edoardo; Gentile, Vincenzo; DI PIERRO, GIOVANNI BATTISTA | |
| Computational investigation of the selectivity of salen and tetrahydrosalen compounds towards the tumor-associated hCA XII isozyme | 2015 | Atilla, Akdemir; DE MONTE, Celeste; Simone, Carradori; Claudiu T., Supuran | |
| Cyclic tertiary sulfamates: Selective inhibition of the tumor-associated carbonic anhydrases IX and XII by N- and O-substituted acesulfame derivatives | 2014 | DE MONTE, Celeste; Carradori, Simone; Secci, Daniela; D'Ascenzio, Melissa; Vullo, D; Ceruso, M; Supuran, Ct | |
| Design, synthesis and biochemical evaluation of novel multi-target inhibitors as potential anti-Parkinson agents | 2018 | Carradori, Simone; Ottuso, Francesco; Petzer, Anèl; Bagetta, Donatella; DE MONTE, Celeste; Secci, Daniela; DE VITA, Daniela; Guglielmi, Paolo; Zengin, Gokhan; Aktumsek, Abdurrahman; Alcaro, Stefano; Petzer, Jacobus P. | |
| Design, synthesis and biological activity of selective hCAs inhibitors based on 2-(benzylsulfinyl)benzoic acid scaffold | 2019 | Rotondi, G.; Guglielmi, P.; Carradori, S.; Secci, D.; De Monte, C.; De Filippis, B.; Maccallini, C.; Amoroso, R.; Cirilli, R.; Akdemir, A.; Angeli, A.; Supuran, C. T. | |
| Design, synthesis and biological characterization of thiazolidin-4-one derivatives as promising inhibitors of Toxoplasma gondii | 2014 | D'Ascenzio, Melissa; Bizzarri, Bruna; DE MONTE, Celeste; Carradori, S; Bolasco, Adriana; Secci, Daniela; Rivanera, Daniela; Faulhaber, N; Bordon, C; Jones Brando, L. | |
| Design, synthesis and evaluation of N-substituted saccharin derivatives as selective inhibitors of tumor-associated carbonic anhydrase XII | 2014 | D'Ascenzio, M; Carradori, S; DE MONTE, Celeste; Secci, Daniela; Ceruso, M; Supuran, Ct | |
| Dual Cyclooxygenase and Carbonic Anhydrase Inhibition by Nonsteroidal Anti-Inflammatory Drugs for the Treatment of Cancer | 2015 | DE MONTE, Celeste; Carradori, Simone; Gentili, Andrea; Mollica, Adriano; Trisciuoglio, Daniela; Supuran, Claudiu T. | |
| Evaluation of a large library of (thiazol-2-yl)hydrazones and analogues as histone acetyltransferase inhibitors: Enzyme and cellular studies. | 2014 | Carradori, S; Rotili, Dante; DE MONTE, Celeste; Lenoci, A; D'Ascenzio, M; Rodriguez, V; Filetici, Patrizia; Miceli, M; Nebbioso, A; Altucci, L; Secci, Daniela; Mai, Antonello | |
| Geographical characterization by MAE-HPLC and NIR methodologies and carbonic anhydrase inhibition of Saffron components | 2017 | Nescatelli, Riccardo; Carradori, Simone; Marini, Federico; Caponigro, Vicky; Bucci, Remo; DE MONTE, Celeste; Mollica, Adriano; Mannina, Luisa; Ceruso, Mariangela; Supuran, CLAUDIU TRANDAFIR; Secci, Daniela | |
| Identification of the stereochemical requirements in the 4-aryl-2-cycloalkylidenhydrazinylthiazole scaffold for the design of selective human monoamine oxidase B inhibitors | 2014 | D'Ascenzio, M; Carradori, S; Secci, Daniela; Mannina, Luisa; Sobolev, Ap; DE MONTE, Celeste; Cirilli, R; Yanez, M; Alcaro, S; Ortuso, F. | |
| Metal-chelating salens and tetrahydrosalens and N- and O-substituted acesulfame and saccharin derivatives as selective inhibitors of the cancer-related carbonic anhydrases IX and XII | 2015 | DE MONTE, Celeste; Secci, Daniela; Simone, Carradori; Melissa, D’Ascenzio; Mariana, Farella; Claudiu T., Supuran | |
| Modern extraction techniques and their impact on the pharmacological profile of Serenoa repens extracts for the treatment of lower urinary tract symptoms. | 2014 | DE MONTE, Celeste; S., Carradori; Granese, Arianna; DI PIERRO, GIOVANNI BATTISTA; Leonardo, Costantino; DE NUNZIO, Cosimo | |
| New amide derivatives of Probenecid as selective inhibitors of carbonic anhydrase IX and XII: Biological evaluation and molecular modelling studies | 2015 | Carradori, Simone; Mollica, Adriano; Ceruso, Mariangela; D'Ascenzio, Melissa; DE MONTE, Celeste; Chimenti, Paola; Sabia, Rocchina; Akdemir, Atilla; Supuran, Claudiu T. | |
| New insights into the biological properties of Crocus sativus L.: chemical modifications, human monoamine oxidases inhibition and molecular modeling studies | 2014 | DE MONTE, Celeste; Carradori, Simone; Chimenti, Paola; Secci, Daniela; Mannina, Luisa; Alcaro, F; Petzer, A; N'Da, Ci; Gidaro, Mc; Costa, G; Alcaro, S; Petzer, Jp | |
| New thiadiazoline and thiadiazole analogues of K858: antiproliferative activity in a model of prostate carcinoma | 2013 | DE MONTE, Celeste; Carradori, S.; D’Ascenzio, M.; Chimenti, Paola; Secci, Daniela; Bolasco, Adriana; Nicolazzo, Chiara; Silvestri, Ida |