RAUCCI, ALESSIA
RAUCCI, ALESSIA
DIPARTIMENTO DI SCIENZE BIOCHIMICHE "ALESSANDRO ROSSI FANELLI"
Advancements in hydrazide-based HDAC inhibitors. A review of recent developments and therapeutic potential
2025 Raucci, Alessia; Zwergel, Clemens; Valente, Sergio; Mai, Antonello
Beyond antibodies. Reinventing Alzheimer’s treatment for the next decade
2025 Garbo, Sabrina; Raucci, Alessia; Zwergel, Clemens; Handzlik, Jadwiga; Battistelli, Cecilia
Design of Benzyl-triazolopyrimidine-Based NADPH Oxidase Inhibitors Leads to the Discovery of a Potent Dual Covalent NOX2/MAOB Inhibitor
2025 Noce, Beatrice; Marchese, Sara; Massari, Marta; Lambona, Chiara; Reis, Joana; Fiorentino, Francesco; Raucci, Alessia; Fioravanti, Rossella; Castelôa, Mariana; Mormino, Alessandro; Garofalo, Stefano; Limatola, Cristina; Basile, Lorenzo; Gottinger, Andrea; Binda, Claudia; Mattevi, Andrea; Mai, Antonello; Valente, Sergio
Discovery of First-in-Class Carbonic Anhydrase/Histone Deacetylase Dual Inhibitors with Antiproliferative Activity in Cancer Cells
2025 Bozdag, Murat; Mroweh, Nabil; Raucci, Alessia; Angeli, Andrea; Peppicelli, Silvia; Biagioni, Alessio; Calorini, Lido; Trisciuoglio, Daniela; Ragno, Rino; Astolfi, Roberta; Giuliani, Lidia; Zwergel, Clemens; Valente, Sergio; Andreucci, Elena; Carta, Fabrizio; Mai, Antonello; Supuran, Claudiu T
Heterocycles-containing HDAC inhibitors active in cancer. An overview of the last fifteen years
2024 Raucci, Alessia; Castiello, Carola; Mai, Antonello; Zwergel, Clemens; Valente, Sergio
Procognitive Potential of Neuroprotective Triazine 5-HT6 Receptor Antagonists Tested on Chronic Activity In Vivo in Rats: Computer-Aided Insight into the Role of Chalcogen-Differences on the Pharmacological Profile
2025 Jastrzębska-Więsek, Magdalena; Garbo, Sabrina; Cios, Agnieszka; Wilczyńska-Zawal, Natalia; Partyka, Anna; Honkisz-Orzechowska, Ewelina; Żesławska, Ewa; Handzlik, Jarosław; Mordyl, Barbara; Głuch-Lutwin, Monika; Raucci, Alessia; Hittinger, Marius; Starek, Małgorzata; Dąbrowska, Monika; Nitek, Wojciech; Karcz, Tadeusz; Skórkowska, Alicja; Gdula-Argasińska, Joanna; Czarnota-Łydka, Kinga; Pyka, Patryk; Szymańska, Ewa; Kucwaj-Brysz, Katarzyna; Zwergel, Clemens; Wesołowska, Anna; Battistelli, Cecilia; Handzlik, Jadwiga
Quinoline-Based DNA Methyltransferase Inhibitors Featuring Basic Side Chains: Design, Synthesis, and Insight in Biochemical and Anticancer Cell Properties
2025 Zwergel, Clemens; Lambona, Chiara; Fioravanti, Rossella; Raucci, Alessia; Fiorentino, Francesco; Nchugoua Tchieh, Guilaine; Jallet, Corinne; Lacroix, Laurent; Pierrettori, Michela; Pellegrini, Francesca Romana; Xiong, Yan; Jin, Jian; Arimondo, Paola; Trisciuoglio, Daniela; Mai, Antonello; Valente, Sergio
Unlocking the potential of higher-molecular-weight 5-HT7R ligands. Synthesis, affinity, and ADMET examination
2024 Pyka, Patryk; Garbo, Sabrina; Murzyn, Aleksandra; Satała, Grzegorz; Janusz, Artur; Górka, Michał; Pietruś, Wojciech; Mituła, Filip; Popiel, Delfina; Wieczorek, Maciej; Palmisano, Biagio; Raucci, Alessia; Bojarski, Andrzej J.; Zwergel, Clemens; Szymańska, Ewa; Kucwaj-Brysz, Katarzyna; Battistelli, Cecilia; Handzlik, Jadwiga; Podlewska, Sabina
Uracil- and Pyridine-containing HDAC inhibitors displayed cytotoxicity in colorectal and glioblastoma cancer stem cells
2024 Fiorentino, Francesco; Fabbrizi, Emanuele; Raucci, Alessia; Noce, Beatrice; Fioravanti, Rossella; Valente, Sergio; Paolini, Chantal; De Maria, Ruggero; Steinkühler, Christian; Gallinari, Paola; Rotili, Dante; Mai, Antonello
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Advancements in hydrazide-based HDAC inhibitors. A review of recent developments and therapeutic potential | 2025 | Raucci, Alessia; Zwergel, Clemens; Valente, Sergio; Mai, Antonello | |
| Beyond antibodies. Reinventing Alzheimer’s treatment for the next decade | 2025 | Garbo, Sabrina; Raucci, Alessia; Zwergel, Clemens; Handzlik, Jadwiga; Battistelli, Cecilia | |
| Design of Benzyl-triazolopyrimidine-Based NADPH Oxidase Inhibitors Leads to the Discovery of a Potent Dual Covalent NOX2/MAOB Inhibitor | 2025 | Noce, Beatrice; Marchese, Sara; Massari, Marta; Lambona, Chiara; Reis, Joana; Fiorentino, Francesco; Raucci, Alessia; Fioravanti, Rossella; Castelôa, Mariana; Mormino, Alessandro; Garofalo, Stefano; Limatola, Cristina; Basile, Lorenzo; Gottinger, Andrea; Binda, Claudia; Mattevi, Andrea; Mai, Antonello; Valente, Sergio | |
| Discovery of First-in-Class Carbonic Anhydrase/Histone Deacetylase Dual Inhibitors with Antiproliferative Activity in Cancer Cells | 2025 | Bozdag, Murat; Mroweh, Nabil; Raucci, Alessia; Angeli, Andrea; Peppicelli, Silvia; Biagioni, Alessio; Calorini, Lido; Trisciuoglio, Daniela; Ragno, Rino; Astolfi, Roberta; Giuliani, Lidia; Zwergel, Clemens; Valente, Sergio; Andreucci, Elena; Carta, Fabrizio; Mai, Antonello; Supuran, Claudiu T | |
| Heterocycles-containing HDAC inhibitors active in cancer. An overview of the last fifteen years | 2024 | Raucci, Alessia; Castiello, Carola; Mai, Antonello; Zwergel, Clemens; Valente, Sergio | |
| Procognitive Potential of Neuroprotective Triazine 5-HT6 Receptor Antagonists Tested on Chronic Activity In Vivo in Rats: Computer-Aided Insight into the Role of Chalcogen-Differences on the Pharmacological Profile | 2025 | Jastrzębska-Więsek, Magdalena; Garbo, Sabrina; Cios, Agnieszka; Wilczyńska-Zawal, Natalia; Partyka, Anna; Honkisz-Orzechowska, Ewelina; Żesławska, Ewa; Handzlik, Jarosław; Mordyl, Barbara; Głuch-Lutwin, Monika; Raucci, Alessia; Hittinger, Marius; Starek, Małgorzata; Dąbrowska, Monika; Nitek, Wojciech; Karcz, Tadeusz; Skórkowska, Alicja; Gdula-Argasińska, Joanna; Czarnota-Łydka, Kinga; Pyka, Patryk; Szymańska, Ewa; Kucwaj-Brysz, Katarzyna; Zwergel, Clemens; Wesołowska, Anna; Battistelli, Cecilia; Handzlik, Jadwiga | |
| Quinoline-Based DNA Methyltransferase Inhibitors Featuring Basic Side Chains: Design, Synthesis, and Insight in Biochemical and Anticancer Cell Properties | 2025 | Zwergel, Clemens; Lambona, Chiara; Fioravanti, Rossella; Raucci, Alessia; Fiorentino, Francesco; Nchugoua Tchieh, Guilaine; Jallet, Corinne; Lacroix, Laurent; Pierrettori, Michela; Pellegrini, Francesca Romana; Xiong, Yan; Jin, Jian; Arimondo, Paola; Trisciuoglio, Daniela; Mai, Antonello; Valente, Sergio | |
| Unlocking the potential of higher-molecular-weight 5-HT7R ligands. Synthesis, affinity, and ADMET examination | 2024 | Pyka, Patryk; Garbo, Sabrina; Murzyn, Aleksandra; Satała, Grzegorz; Janusz, Artur; Górka, Michał; Pietruś, Wojciech; Mituła, Filip; Popiel, Delfina; Wieczorek, Maciej; Palmisano, Biagio; Raucci, Alessia; Bojarski, Andrzej J.; Zwergel, Clemens; Szymańska, Ewa; Kucwaj-Brysz, Katarzyna; Battistelli, Cecilia; Handzlik, Jadwiga; Podlewska, Sabina | |
| Uracil- and Pyridine-containing HDAC inhibitors displayed cytotoxicity in colorectal and glioblastoma cancer stem cells | 2024 | Fiorentino, Francesco; Fabbrizi, Emanuele; Raucci, Alessia; Noce, Beatrice; Fioravanti, Rossella; Valente, Sergio; Paolini, Chantal; De Maria, Ruggero; Steinkühler, Christian; Gallinari, Paola; Rotili, Dante; Mai, Antonello |