HAILU, GEBREMEDHIN SOLOMON
HAILU, GEBREMEDHIN SOLOMON
DIPARTIMENTO DI CHIMICA E TECNOLOGIE DEL FARMACO
Design, synthesis and biological evaluation of novel epigenetic modulators for parasitic diseases
2017 Hailu, GEBREMEDHIN SOLOMON
Development of 1,2,4-oxadiazoles as potent and selective inhibitors of the human deacetylase sirtuin 2: structure-activity relationship, X-ray crystal structure, and anticancer activity
2017 Moniot, S; Forgione, M; Lucidi, Alessia; Hailu, GEBREMEDHIN SOLOMON; Nebbioso, A; Carafa, V; Baratta, F; Altucci, L; Giacché, N; Passeri, D; Pellicciari, R; Mai, Antonello; Steegborn, C; Rotili, Dante
Effect of α-methoxy substitution on the anti-HIV activity of dihydropyrimidin-4(3 H)-ones
2019 Nawrozkij, Maxim B.; Forgione, Mariantonietta; Yablokov, Alexandre S.; Lucidi, Alessia; Tomaselli, Daniela; Patsilinakos, Alexandros; Panella, Cristina; Hailu, Gebremedhin S.; Kirillov, Ivan A.; Badia, Roger; Riveira-Munoz, Eva; Crespan, Emmanuele; Armijos Rivera, Jorge I.; Cirilli, Roberto; Ragno, Rino; Esté, José A.; Maga, Giovanni; Mai, Antonello; Rotili, Dante
Lysine deacetylase inhibitors in parasites: past, present, and future perspectives.
2017 Hailu, Gs; Robaa, D; Forgione, M; Sippl, W; Rotili, D; Mai, A.
Sirtuin functions and modulation: from chemistry to the clinic
2016 Carafa, Vincenzo; Rotili, Dante; Forgione, Mariantonietta; Cuomo, Francesca; Serretiello, Enrica; Hailu, GEBREMEDHIN SOLOMON; Jarho, Elina; Lahtela Kakkonen, Maija; Mai, Antonello; Altucci, Lucia
The relevance of Ki calculation for bi-substrate enzymes illustrated by kinetic evaluation of a novel lysine (K) acetyltransferase 8 inhibitor.
2017 Wapenaar, H; van den Bosch, T; Leus, Ngj; van der Wouden, Pe; Eleftheriadis, N; Hermans, J; Hailu, Gs; Rotili, D; Mai, A; Dömling, A; Bischoff, R; Haisma, Hj; Dekker, F. J.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Design, synthesis and biological evaluation of novel epigenetic modulators for parasitic diseases | 2017 | Hailu, GEBREMEDHIN SOLOMON | |
Development of 1,2,4-oxadiazoles as potent and selective inhibitors of the human deacetylase sirtuin 2: structure-activity relationship, X-ray crystal structure, and anticancer activity | 2017 | Moniot, S; Forgione, M; Lucidi, Alessia; Hailu, GEBREMEDHIN SOLOMON; Nebbioso, A; Carafa, V; Baratta, F; Altucci, L; Giacché, N; Passeri, D; Pellicciari, R; Mai, Antonello; Steegborn, C; Rotili, Dante | |
Effect of α-methoxy substitution on the anti-HIV activity of dihydropyrimidin-4(3 H)-ones | 2019 | Nawrozkij, Maxim B.; Forgione, Mariantonietta; Yablokov, Alexandre S.; Lucidi, Alessia; Tomaselli, Daniela; Patsilinakos, Alexandros; Panella, Cristina; Hailu, Gebremedhin S.; Kirillov, Ivan A.; Badia, Roger; Riveira-Munoz, Eva; Crespan, Emmanuele; Armijos Rivera, Jorge I.; Cirilli, Roberto; Ragno, Rino; Esté, José A.; Maga, Giovanni; Mai, Antonello; Rotili, Dante | |
Lysine deacetylase inhibitors in parasites: past, present, and future perspectives. | 2017 | Hailu, Gs; Robaa, D; Forgione, M; Sippl, W; Rotili, D; Mai, A. | |
Sirtuin functions and modulation: from chemistry to the clinic | 2016 | Carafa, Vincenzo; Rotili, Dante; Forgione, Mariantonietta; Cuomo, Francesca; Serretiello, Enrica; Hailu, GEBREMEDHIN SOLOMON; Jarho, Elina; Lahtela Kakkonen, Maija; Mai, Antonello; Altucci, Lucia | |
The relevance of Ki calculation for bi-substrate enzymes illustrated by kinetic evaluation of a novel lysine (K) acetyltransferase 8 inhibitor. | 2017 | Wapenaar, H; van den Bosch, T; Leus, Ngj; van der Wouden, Pe; Eleftheriadis, N; Hermans, J; Hailu, Gs; Rotili, D; Mai, A; Dömling, A; Bischoff, R; Haisma, Hj; Dekker, F. J. |