Sfoglia per Autore
Synthesis, in vitro, and in vivo biological evaluation and molecular docking simulations of chiral alcohol and ether derivatives of the 1,5-diarylpyrrole scaffold as novel anti-inflammatory and analgesic agents
2008 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Sibilla, Supino; Fabrizio, Manetti; Stefano, Forli; Maurizio, Botta; Lidia, Sautebin; Antonietta, Rossi; Carlo, Pergola; Carla, Ghelardini; Monica, Norcini; Francesco, Makovec; Paola, Anzellotti; Roberto, Cirilli; Rosella, Ferretti; Bruno, Gallinella; F., La Torre; Maurizio, Anzini; Paola, Patrignani
HPLC Enantioseparation and Absolute Configuration of Novel Antiinflammatory Pyrrole Derivatives
2008 Biava, Mariangela; Cirilli, R; Fares, V; Ferretti, R; Gallinella, B; Poce, Giovanna; Porretta, Giulio Cesare; Supino, Sibilla; Villani, Claudio
Design and Synthesis of novel diarylpyrroles as p38 MAP kinase inhibitors
2008 Biava, Mariangela; Porretta, G. C.; Poce, Giovanna; Giordani, A; Menziani, C.
Potent in vitro and in vivo novel 1,5-Diarylpyrrole-3-acetic Esters COX-2 inhibitors.
2009 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Sautebin, L; Patrignani, P; Ghelardini, C; Giordani, A; Anzini, M.
Derivatives of BM 212: synthesis and biological evaluation of new derivatives with improved antimycobacterial activity.
2009 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Pompei, R; DE LOGU, A; Manetti, F; Botta, M.
BM212 and its derivatives: lead optimization of a new class of antimycobacterial agents.
2009 Poce, Giovanna; Porretta, Giulio Cesare; DE LOGU, A; DE ROSSI, E; Manetti, F; Botta, M; Biava, Mariangela
Pyrrole derivatives of BM212 as novel antimycobacterial agents Design, synthesis, biological evaluation and study of their mode of action
2009 Biava, Mariangela; Porretta, Giulio Cesare; Battilocchio, Claudio; Poce, G; Pompei, R; DE LOGU, A; Manetti, F; Botta, M.
New pyrrole derivatives of BM 212: a new class of antimycobacterial agents.Design, synthesis, biological evaluation and study of their mode of action.
2009 Biava, Mariangela; Porretta, G. C.; Poce, G; DE LOGU, A; Manetti, F; Botta, M.
New pyrrole derivatives of BM 212: lead compound optimization strategy, Tuberculosis drug development. Targets, technologies and trials
2009 Poce, Giovanna; Porretta, Giulio Cesare; Borzi, F; DE LOGU, A; DE ROSSI, E; Manetti, F; Botta, M; Biava, Mariangela
1,5-Diaryl-2-ethyl pyrrole derivatives as antimycobacterial agents: design, synthesis, and microbiological evaluation
2009 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; DE LOGU, A; Saddi, M; Meleddu, R; Manetti, F; DE ROSSI, E; Botta, M.
C-9 Alkenylidine bridged macrolides: WO2008061189.
2009 Poce, Giovanna; Porretta, Giulio Cesare; Biava, Mariangela
1,5-Diaryl-Pyrroles as New Generation of Anti-Inflammatory and Analgesic Agents: Design, Synthesis, in vitro and in vivo Evaluation
2010 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Alfonso, S; Battilocchio, Claudio; DE LOGU, A; Manetti, F; Botta, M.
Novel Ester and Acid Derivatives of the 1,5-Diarylpyrrole Scaffold as Anti-inflammatory and Analgesic Agents. Synthesis, in vitro and in vivo Biological Evaluation
2010 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; Manetti, F; Botta, M; Sautebin, L; Rossi, A; Pergola, C; Ghelardini, C; Norcini, M; Makovec, F; Anzellotti, P; Cirilli, R; Ferretti, R; Patrignani, P; Anzini, M.
One-pot conversions of olefins to cyclic carbonates and secondary allylic and homoallylic amines to cyclic carbamates
2010 Stephen G., Davies; Ai M., Fletcher; Wataru, Kurosawa; James A., Lee; Poce, Giovanna; Paul M., Roberts; James E., Thomson; David M., Williamson
New pyrrole derivatives of BM 212: a new class of antimycobacterial agents. Design, synthesis, biological evaluation and study of their mode of action
2010 Biava, Mariangela; Porretta, G. C.; Poce, Giovanna; Alfonso, Salvatore; Battilocchio, Claudio; De Logu, A.; De Rossi, E.; Manetti, F; Botta, M.
BM 579: a novel pyrrole derivative with improved antimycobacterial activity
2010 Biava, Mariangela; Porretta, G. C.; Poce, Giovanna; Alfonso, Salvatore; Battilocchio, Claudio; De Logu, A.; Manetti, F; Botta, M.
Doubly diastereoselective conjugate addition of enantiopure lithium amides to enantiopure N-enoyl oxazolidin-2-ones: a mechanistic probe
2010 Stephen G., Davies; M. A., Fletcher; Gesine J., Hermann; Poce, Giovanna; Paul M., Roberts; Andrew D., Smith; Miles J., Sweet; James E., Thomson
Identification of a novel pyrrole derivative endowed with antimycobacterial activity and protection index comparable to that of the current antitubercular drugs streptomycin and rifampin
2010 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; Alfonso, Salvatore; A., De Logu; Nadia, Serra; Fabrizio, Manetti; Maurizio, Botta
New heterocyclic compounds with potential activity against parasitic protozoan: Trypanosoma and Leishmania
2010 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; V., Yardley; Alfonso, Salvatore
Developing New Antiinflammatory and Analgesic Agents: Design, Synthesis, Biological and harmacological Evaluation
2010 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; Alfonso, Salvatore; Botta, M.; Manetti, F.; Sautebin, L; Ghelardini, C; Makovec, F; Giordani, A; Patrignani, P; Anzini, M.
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Synthesis, in vitro, and in vivo biological evaluation and molecular docking simulations of chiral alcohol and ether derivatives of the 1,5-diarylpyrrole scaffold as novel anti-inflammatory and analgesic agents | 2008 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Sibilla, Supino; Fabrizio, Manetti; Stefano, Forli; Maurizio, Botta; Lidia, Sautebin; Antonietta, Rossi; Carlo, Pergola; Carla, Ghelardini; Monica, Norcini; Francesco, Makovec; Paola, Anzellotti; Roberto, Cirilli; Rosella, Ferretti; Bruno, Gallinella; F., La Torre; Maurizio, Anzini; Paola, Patrignani | |
| HPLC Enantioseparation and Absolute Configuration of Novel Antiinflammatory Pyrrole Derivatives | 2008 | Biava, Mariangela; Cirilli, R; Fares, V; Ferretti, R; Gallinella, B; Poce, Giovanna; Porretta, Giulio Cesare; Supino, Sibilla; Villani, Claudio | |
| Design and Synthesis of novel diarylpyrroles as p38 MAP kinase inhibitors | 2008 | Biava, Mariangela; Porretta, G. C.; Poce, Giovanna; Giordani, A; Menziani, C. | |
| Potent in vitro and in vivo novel 1,5-Diarylpyrrole-3-acetic Esters COX-2 inhibitors. | 2009 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Sautebin, L; Patrignani, P; Ghelardini, C; Giordani, A; Anzini, M. | |
| Derivatives of BM 212: synthesis and biological evaluation of new derivatives with improved antimycobacterial activity. | 2009 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Pompei, R; DE LOGU, A; Manetti, F; Botta, M. | |
| BM212 and its derivatives: lead optimization of a new class of antimycobacterial agents. | 2009 | Poce, Giovanna; Porretta, Giulio Cesare; DE LOGU, A; DE ROSSI, E; Manetti, F; Botta, M; Biava, Mariangela | |
| Pyrrole derivatives of BM212 as novel antimycobacterial agents Design, synthesis, biological evaluation and study of their mode of action | 2009 | Biava, Mariangela; Porretta, Giulio Cesare; Battilocchio, Claudio; Poce, G; Pompei, R; DE LOGU, A; Manetti, F; Botta, M. | |
| New pyrrole derivatives of BM 212: a new class of antimycobacterial agents.Design, synthesis, biological evaluation and study of their mode of action. | 2009 | Biava, Mariangela; Porretta, G. C.; Poce, G; DE LOGU, A; Manetti, F; Botta, M. | |
| New pyrrole derivatives of BM 212: lead compound optimization strategy, Tuberculosis drug development. Targets, technologies and trials | 2009 | Poce, Giovanna; Porretta, Giulio Cesare; Borzi, F; DE LOGU, A; DE ROSSI, E; Manetti, F; Botta, M; Biava, Mariangela | |
| 1,5-Diaryl-2-ethyl pyrrole derivatives as antimycobacterial agents: design, synthesis, and microbiological evaluation | 2009 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; DE LOGU, A; Saddi, M; Meleddu, R; Manetti, F; DE ROSSI, E; Botta, M. | |
| C-9 Alkenylidine bridged macrolides: WO2008061189. | 2009 | Poce, Giovanna; Porretta, Giulio Cesare; Biava, Mariangela | |
| 1,5-Diaryl-Pyrroles as New Generation of Anti-Inflammatory and Analgesic Agents: Design, Synthesis, in vitro and in vivo Evaluation | 2010 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Alfonso, S; Battilocchio, Claudio; DE LOGU, A; Manetti, F; Botta, M. | |
| Novel Ester and Acid Derivatives of the 1,5-Diarylpyrrole Scaffold as Anti-inflammatory and Analgesic Agents. Synthesis, in vitro and in vivo Biological Evaluation | 2010 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; Manetti, F; Botta, M; Sautebin, L; Rossi, A; Pergola, C; Ghelardini, C; Norcini, M; Makovec, F; Anzellotti, P; Cirilli, R; Ferretti, R; Patrignani, P; Anzini, M. | |
| One-pot conversions of olefins to cyclic carbonates and secondary allylic and homoallylic amines to cyclic carbamates | 2010 | Stephen G., Davies; Ai M., Fletcher; Wataru, Kurosawa; James A., Lee; Poce, Giovanna; Paul M., Roberts; James E., Thomson; David M., Williamson | |
| New pyrrole derivatives of BM 212: a new class of antimycobacterial agents. Design, synthesis, biological evaluation and study of their mode of action | 2010 | Biava, Mariangela; Porretta, G. C.; Poce, Giovanna; Alfonso, Salvatore; Battilocchio, Claudio; De Logu, A.; De Rossi, E.; Manetti, F; Botta, M. | |
| BM 579: a novel pyrrole derivative with improved antimycobacterial activity | 2010 | Biava, Mariangela; Porretta, G. C.; Poce, Giovanna; Alfonso, Salvatore; Battilocchio, Claudio; De Logu, A.; Manetti, F; Botta, M. | |
| Doubly diastereoselective conjugate addition of enantiopure lithium amides to enantiopure N-enoyl oxazolidin-2-ones: a mechanistic probe | 2010 | Stephen G., Davies; M. A., Fletcher; Gesine J., Hermann; Poce, Giovanna; Paul M., Roberts; Andrew D., Smith; Miles J., Sweet; James E., Thomson | |
| Identification of a novel pyrrole derivative endowed with antimycobacterial activity and protection index comparable to that of the current antitubercular drugs streptomycin and rifampin | 2010 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; Alfonso, Salvatore; A., De Logu; Nadia, Serra; Fabrizio, Manetti; Maurizio, Botta | |
| New heterocyclic compounds with potential activity against parasitic protozoan: Trypanosoma and Leishmania | 2010 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; V., Yardley; Alfonso, Salvatore | |
| Developing New Antiinflammatory and Analgesic Agents: Design, Synthesis, Biological and harmacological Evaluation | 2010 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; Alfonso, Salvatore; Botta, M.; Manetti, F.; Sautebin, L; Ghelardini, C; Makovec, F; Giordani, A; Patrignani, P; Anzini, M. |
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