BUFANO, MARIANNA
BUFANO, MARIANNA
DIPARTIMENTO DI CHIMICA E TECNOLOGIE DEL FARMACO
Anticancer activity of (S)-5-Chloro-3-((3,5-dimethylphenyl)sulfonyl)-N-(1-oxo-1-((pyridin-4-ylmethyl)amino)propan-2-yl)-1H-indole-2-carboxamide (RS4690), a new dishevelled 1 inhibitor
2022 Coluccia, Antonio; Bufano, Marianna; La Regina, Giuseppe La; Puxeddu, Michela; Toto, Angelo; Paone, Alessio; Bouzidi, Amani; Musto, Giorgia; Badolati, Nadia; Orlando, Viviana; Biagioni, Stefano; Masci, Domiziana; Cantatore, Chiara; Cirilli, Roberto; Cutruzzolà, Francesca; Gianni, Stefano; Stornaiuolo, Mariano; Silvestri, Romano
Anticancer activity of RS4690, a new Dishevelled I inhibitor
2022 Coluccia, A.; Bufano, M.; La Regina, G.; Puxeddu, M.; Silvestri, R.
Application of computer aided drug design techniques for the identification of bioactive compounds
2023 Bufano, Marianna
Design, synthesis and biological evaluation of PDZ1 targeting NHERF1 inhibitors as anticancer agents
2019 La Regina, G.; Naccarato, V.; Masci, D.; Puxeddu, M.; Bufano, M.; Nalli, M.; Coluccia, A.; Orlando, V.; Canettieri, G.; Gianni, S.; Silvestri, R.
Discovery of novel human lactate dehydrogenase inhibitors. Structure-based virtual screening studies and biological assessment
2022 Di Magno, L; Coluccia, A; Bufano, M; Ripa, S; La Regina, G; Nalli, M; Di Pastena, F; Canettieri, G; Silvestri, R; Frati, L
Discovery of pyrrole derivatives for the treatment of glioblastoma and chronic myeloid leukemia
2021 Puxeddu, M.; Shen, H.; Bai, R.; Coluccia, A.; Bufano, M.; Nalli, M.; Sebastiani, J.; Brancaccio, D.; Da Pozzo, E.; Tremolanti, C.; Martini, C.; Orlando, V.; Biagioni, S.; Sinicropi, M. S.; Ceramella, J.; Iacopetta, D.; Coluccia, A. M. L.; Hamel, E.; Liu, T.; Silvestri, R.; La Regina, G.
Evaluation of pharmacophoric models at colchicine binding site by ROC curves
2019 Esposito, Chiara; Bufano, Marianna; Coluccia, Antonio
Exploring CCRL2 chemerin binding using accelerated molecular dynamics
2022 Bufano, M.; Laffranchi, M.; Sozzani, S.; Raimondo, D.; Silvestri, R.; Coluccia, A.
First in class pdz1 targeting NHERF1 inhibitors as anticancer agents
2019 LA REGINA, Giuseppe; Naccarato, Valentina; Puxeddu, Michela; Bufano, Marianna; Nalli, Marianna; Coluccia, Antonio; Silvestri, Romano
Identification of a New FtsZ Inhibitor by Virtual Screening, Mechanistic Insights, and Structure–Activity Relationship Analyses
2025 Scio', Pietro; Scoffone, Viola Camilla; Parisi, Anastasia; Bufano, Marianna; Caneva, Martina; Trespidi, Gabriele; Irudal, Samuele; Barbieri, Giulia; Cariani, Lisa; Orena, Beatrice Silvia; Daccò, Valeria; Imperi, Francesco; Buroni, Silvia; Coluccia, Antonio
Modeling Epac1 interactions with the allosteric inhibitor AM-001 by co-solvent molecular dynamics
2020 Bufano, M.; Laudette, M.; Blondeau, J. -P.; Lezoualc'H, F.; Nalli, M.; Silvestri, R.; Brancale, A.; Coluccia, A.
New pyrrole derivatives for the treatment of glioblastoma and chronic myeloid leukemia
2021 Sebastiani, J.; Puxeddu, M.; Coluccia, A.; Bufano, M.; Hamel, E.; Liu, T.; Silvestri, R.; La Regina, G.
New pyrroles derivatives as anti-glioblastoma and anti-chronic myeloid leukemia agents
2021 Puxeddu, M.; Sebastiani, J.; Coluccia, A.; Bufano, M.; Hamel, E.; Liu, T.; Silvestri, R.; La Regina, G.
Retrospective Benchmarking and Novel Shape-Pharmacophore Based Implementation of the MORLD Method for the Autonomous Optimization of 3-Aroyl-1,4-diarylpyrroles (ARDAP)
2025 Scio', Pietro; Bufano, Marianna; Silvestri, Romano; Coluccia, Antonio
Structure-function relationship of the Pseudomonas aeruginosa AsmA-like proteins YhdP and YdbH involved in outer membrane biogenesis
2025 Sposato, Davide; Pederzoli, Camilla; Bufano, Marianna; Scio', Pietro; Rossi, Ludovica; Leoni, Livia; Rampioni, Giordano; Visca, Paolo; Coluccia, Antonio; Imperi, Francesco
Targeting PDZ domains as potential treatment for viral infections, neurodegeneration and cancer
2021 Nardella, Caterina; Visconti, Lorenzo; Malagrinò, Francesca; Pagano, Livia; Bufano, Marianna; Nalli, Marianna; Coluccia, Antonio; La Regina, Giuseppe; Silvestri, Romano; Gianni, Stefano; Toto, Angelo
Targeting the Grb2 cSH3 domain: design, synthesis and biological evaluation of the first series of modulators
2023 Bufano, Marianna; Puxeddu, Michela; Nalli, Marianna; La Regina, Giuseppe; Toto, Angelo; Liberati, Francesca Romana; Paone, Alessio; Cutruzzolà, Francesca; Masci, Domiziana; Bigogno, Chiara; Dondio, Giulio; Silvestri, Romano; Gianni, Stefano; Coluccia, Antonio
Targeting the interaction between the SH3 domain of Grb2 and Gab2
2020 Malagrinò, Francesca; Coluccia, Antonio; Bufano, Marianna; La Regina, Giuseppe; Puxeddu, Michela; Toto, Angelo; Visconti, Lorenzo; Paone, Alessio; Magnifico, Maria Chiara; Troilo, Francesca; Cutruzzolà, Francesca; Silvestri, Romano; Gianni, Stefano
Toll-like receptor 4-dependent platelet-related thrombosis in SARS-CoV-2 infection
2023 Carnevale, Roberto; Cammisotto, Vittoria; Bartimoccia, Simona; Nocella, Cristina; Castellani, Valentina; Bufano, Marianna; Loffredo, Lorenzo; Sciarretta, Sebastiano; Frati, Giacomo; Coluccia, Antonio; Silvestri, Romano; Ceccarelli, Giancarlo; Oliva, Alessandra; Venditti, Mario; Pugliese, Francesco; Maria Mastroianni, Claudio; Turriziani, Ombretta; Leopizzi, Martina; D'Amati, Giulia; Pignatelli, Pasquale; Violi, Francesco
Unveiling an unexpected redox regulation of the folding, function and inhibition in the phosphotyrosine binding domain of FRS2
2025 Pennacchietti, Valeria; Pagano, Livia; Di Felice, Mariana; Toso, Julian; Bufano, Marianna; Coluccia, Antonio; Silvestri, Romano; Capelli, Riccardo; Camilloni, Carlo; Malagrinò, Francesca; Toto, Angelo; Gianni, Stefano
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Anticancer activity of (S)-5-Chloro-3-((3,5-dimethylphenyl)sulfonyl)-N-(1-oxo-1-((pyridin-4-ylmethyl)amino)propan-2-yl)-1H-indole-2-carboxamide (RS4690), a new dishevelled 1 inhibitor | 2022 | Coluccia, Antonio; Bufano, Marianna; La Regina, Giuseppe La; Puxeddu, Michela; Toto, Angelo; Paone, Alessio; Bouzidi, Amani; Musto, Giorgia; Badolati, Nadia; Orlando, Viviana; Biagioni, Stefano; Masci, Domiziana; Cantatore, Chiara; Cirilli, Roberto; Cutruzzolà, Francesca; Gianni, Stefano; Stornaiuolo, Mariano; Silvestri, Romano | |
| Anticancer activity of RS4690, a new Dishevelled I inhibitor | 2022 | Coluccia, A.; Bufano, M.; La Regina, G.; Puxeddu, M.; Silvestri, R. | |
| Application of computer aided drug design techniques for the identification of bioactive compounds | 2023 | Bufano, Marianna | |
| Design, synthesis and biological evaluation of PDZ1 targeting NHERF1 inhibitors as anticancer agents | 2019 | La Regina, G.; Naccarato, V.; Masci, D.; Puxeddu, M.; Bufano, M.; Nalli, M.; Coluccia, A.; Orlando, V.; Canettieri, G.; Gianni, S.; Silvestri, R. | |
| Discovery of novel human lactate dehydrogenase inhibitors. Structure-based virtual screening studies and biological assessment | 2022 | Di Magno, L; Coluccia, A; Bufano, M; Ripa, S; La Regina, G; Nalli, M; Di Pastena, F; Canettieri, G; Silvestri, R; Frati, L | |
| Discovery of pyrrole derivatives for the treatment of glioblastoma and chronic myeloid leukemia | 2021 | Puxeddu, M.; Shen, H.; Bai, R.; Coluccia, A.; Bufano, M.; Nalli, M.; Sebastiani, J.; Brancaccio, D.; Da Pozzo, E.; Tremolanti, C.; Martini, C.; Orlando, V.; Biagioni, S.; Sinicropi, M. S.; Ceramella, J.; Iacopetta, D.; Coluccia, A. M. L.; Hamel, E.; Liu, T.; Silvestri, R.; La Regina, G. | |
| Evaluation of pharmacophoric models at colchicine binding site by ROC curves | 2019 | Esposito, Chiara; Bufano, Marianna; Coluccia, Antonio | |
| Exploring CCRL2 chemerin binding using accelerated molecular dynamics | 2022 | Bufano, M.; Laffranchi, M.; Sozzani, S.; Raimondo, D.; Silvestri, R.; Coluccia, A. | |
| First in class pdz1 targeting NHERF1 inhibitors as anticancer agents | 2019 | LA REGINA, Giuseppe; Naccarato, Valentina; Puxeddu, Michela; Bufano, Marianna; Nalli, Marianna; Coluccia, Antonio; Silvestri, Romano | |
| Identification of a New FtsZ Inhibitor by Virtual Screening, Mechanistic Insights, and Structure–Activity Relationship Analyses | 2025 | Scio', Pietro; Scoffone, Viola Camilla; Parisi, Anastasia; Bufano, Marianna; Caneva, Martina; Trespidi, Gabriele; Irudal, Samuele; Barbieri, Giulia; Cariani, Lisa; Orena, Beatrice Silvia; Daccò, Valeria; Imperi, Francesco; Buroni, Silvia; Coluccia, Antonio | |
| Modeling Epac1 interactions with the allosteric inhibitor AM-001 by co-solvent molecular dynamics | 2020 | Bufano, M.; Laudette, M.; Blondeau, J. -P.; Lezoualc'H, F.; Nalli, M.; Silvestri, R.; Brancale, A.; Coluccia, A. | |
| New pyrrole derivatives for the treatment of glioblastoma and chronic myeloid leukemia | 2021 | Sebastiani, J.; Puxeddu, M.; Coluccia, A.; Bufano, M.; Hamel, E.; Liu, T.; Silvestri, R.; La Regina, G. | |
| New pyrroles derivatives as anti-glioblastoma and anti-chronic myeloid leukemia agents | 2021 | Puxeddu, M.; Sebastiani, J.; Coluccia, A.; Bufano, M.; Hamel, E.; Liu, T.; Silvestri, R.; La Regina, G. | |
| Retrospective Benchmarking and Novel Shape-Pharmacophore Based Implementation of the MORLD Method for the Autonomous Optimization of 3-Aroyl-1,4-diarylpyrroles (ARDAP) | 2025 | Scio', Pietro; Bufano, Marianna; Silvestri, Romano; Coluccia, Antonio | |
| Structure-function relationship of the Pseudomonas aeruginosa AsmA-like proteins YhdP and YdbH involved in outer membrane biogenesis | 2025 | Sposato, Davide; Pederzoli, Camilla; Bufano, Marianna; Scio', Pietro; Rossi, Ludovica; Leoni, Livia; Rampioni, Giordano; Visca, Paolo; Coluccia, Antonio; Imperi, Francesco | |
| Targeting PDZ domains as potential treatment for viral infections, neurodegeneration and cancer | 2021 | Nardella, Caterina; Visconti, Lorenzo; Malagrinò, Francesca; Pagano, Livia; Bufano, Marianna; Nalli, Marianna; Coluccia, Antonio; La Regina, Giuseppe; Silvestri, Romano; Gianni, Stefano; Toto, Angelo | |
| Targeting the Grb2 cSH3 domain: design, synthesis and biological evaluation of the first series of modulators | 2023 | Bufano, Marianna; Puxeddu, Michela; Nalli, Marianna; La Regina, Giuseppe; Toto, Angelo; Liberati, Francesca Romana; Paone, Alessio; Cutruzzolà, Francesca; Masci, Domiziana; Bigogno, Chiara; Dondio, Giulio; Silvestri, Romano; Gianni, Stefano; Coluccia, Antonio | |
| Targeting the interaction between the SH3 domain of Grb2 and Gab2 | 2020 | Malagrinò, Francesca; Coluccia, Antonio; Bufano, Marianna; La Regina, Giuseppe; Puxeddu, Michela; Toto, Angelo; Visconti, Lorenzo; Paone, Alessio; Magnifico, Maria Chiara; Troilo, Francesca; Cutruzzolà, Francesca; Silvestri, Romano; Gianni, Stefano | |
| Toll-like receptor 4-dependent platelet-related thrombosis in SARS-CoV-2 infection | 2023 | Carnevale, Roberto; Cammisotto, Vittoria; Bartimoccia, Simona; Nocella, Cristina; Castellani, Valentina; Bufano, Marianna; Loffredo, Lorenzo; Sciarretta, Sebastiano; Frati, Giacomo; Coluccia, Antonio; Silvestri, Romano; Ceccarelli, Giancarlo; Oliva, Alessandra; Venditti, Mario; Pugliese, Francesco; Maria Mastroianni, Claudio; Turriziani, Ombretta; Leopizzi, Martina; D'Amati, Giulia; Pignatelli, Pasquale; Violi, Francesco | |
| Unveiling an unexpected redox regulation of the folding, function and inhibition in the phosphotyrosine binding domain of FRS2 | 2025 | Pennacchietti, Valeria; Pagano, Livia; Di Felice, Mariana; Toso, Julian; Bufano, Marianna; Coluccia, Antonio; Silvestri, Romano; Capelli, Riccardo; Camilloni, Carlo; Malagrinò, Francesca; Toto, Angelo; Gianni, Stefano |