ZWERGEL, CLEMENS
ZWERGEL, CLEMENS
DIPARTIMENTO DI CHIMICA E TECNOLOGIE DEL FARMACO
1,4-Dihydropyridines Active on the SIRT1/AMPK Pathway Ameliorate Skin Repair and Mitochondrial Function and Exhibit Inhibition of Proliferation in Cancer Cells
2016 Valente, Sergio; Mellini, Paolo; Spallotta, Francesco; Carafa, Vincenzo; Nebbioso, Angela; Polletta, Lucia; Carnevale, Ilaria; Saladini, Serena; Trisciuoglio, Daniela; Gabellini, Chiara; Tardugno, Maria; Zwergel, Clemens; Cencioni, Chiara; Atlante, Sandra; Moniot, Sébastien; Steegborn, Clemens; Budriesi, Roberta; Tafani, Marco; Del Bufalo, Donatella; Altucci, Lucia; Gaetano, Carlo; Mai, Antonello
A quinoline-based DNA methyltransferase inhibitor as a possible adjuvant in osteosarcoma therapy
2018 Manara, Maria Cristina; Valente, Sergio; Cristalli, Camilla; Nicoletti, Giordano; Landuzzi, Lorena; Zwergel, Clemens; Mazzone, Roberta; Stazi, Giulia; Arimondo, Paola B.; Pasello, Michela; Guerzoni, Clara; Picci, Piero; Nanni, Patrizia; Lollini, Pier-Luigi; Mai, Antonello; Scotlandi, Katia
A xanthine derivative with Nnovel heat shock protein 90-alpha inhibitory and senolytic properties
2025 Atlante, Sandra; Cis, Luca; Pirolli, Davide; Gottardi Zamperla, Michela; Barbi, Veronica; Mai, Antonello; Zwergel, Clemens; Marcozzi, Serena; Giuliani, Maria Elisa; Bigossi, Giorgia; Lai, Giovanni; Orlando, Fiorenza; Giacconi, Robertina; Lattanzio, Fabrizia; Matacchione, Giulia; Giordani, Chiara; Bracci, Massimo; Olivieri, Fabiola; Boschi, Federico; Tabarelli De Fatis, Paola; Ivaldi, Giovanni Battista; Malavolta, Marco; Farsetti, Antonella; De Rosa, Maria Cristina; Gaetano, Carlo
Abstract 2946: Effects of two novel quinoline-based non-nucleoside DNA methyltransferase inhibitors against bone sarcomas
2015 Manara, Maria Cristina; Valente, Sergio; Cristalli, Camilla; Baricordi, Cristina; Zwergel, Clemens; Arimondo, Paola B; Picci, Piero; Mai, Antonello; Scotlandi, Katia
Acute and chronic neurobehavioral effects of the designer drug and bath salt constituent 3,4-methylenedioxypyrovalerone in the rat
2019 ATEHORTUA MARTINEZ, LUISA ALESSANDRA; Masniere, Cyriaque; Campolongo, Patrizia; Chasseigneaux, Stéphanie; Callebert, Jacques; Zwergel, Clemens; Mai, Antonello; Laplanche, Jean-Louis; Chen, Huixiong; Etheve-Quelquejeu, Mélanie; Mégarbane, Bruno; Benturquia, Nadia
Advancements in hydrazide-based HDAC inhibitors. A review of recent developments and therapeutic potential
2025 Raucci, Alessia; Zwergel, Clemens; Valente, Sergio; Mai, Antonello
Amphetamine and the Smart Drug 3,4-Methylenedioxypyrovalerone (MDPV) Induce Generalization of Fear Memory in Rats
2019 Colucci, Paola; Mancini, Giulia Federica; Santori, Alessia; Zwergel, Clemens; Mai, Antonello; Trezza, Viviana; Roozendaal, Benno; Campolongo, Patrizia
Amphetamine modulation of long-term object recognition memory in rats: influence of stress
2021 Colucci, Paola; Santori, Alessia; Romanelli, Luca; Zwergel, Clemens; Mai, Antonello; Scaccianoce, Sergio; Campolongo, Patrizia
Application of small epigenetic modulators in pediatric medulloblastoma
2018 Zwergel, Clemens; Romanelli, Annalisa; Stazi, Giulia; Besharat, Zein Mersini; Catanzaro, Giuseppina; Tafani, Marco; Valente, Sergio; Mai, Antonello
Aurones: Interesting Natural and Synthetic Compounds with Emerging Biological Potential
2012 Zwergel, Clemens; F., Gaascht; Valente, Sergio; M., Diederich; D., Bagrel; G., Kirsch
Beyond antibodies. Reinventing Alzheimer’s treatment for the next decade
2025 Garbo, Sabrina; Raucci, Alessia; Zwergel, Clemens; Handzlik, Jadwiga; Battistelli, Cecilia
Cardioprotection through pharmacological activation of Sirtuin 5 in a murine model of acute myocardial infarction
2025 Castiello, Carola; Efentakis, Panagiotis; Nikolaou, Panagiota-Efstathia; Symeonidi, Lydia; Chania, Christina; Barla, Ioanna; Akrani, Ifigeneia; Kostomitsopoulos, Nikolaos; Gikas, Evangelos; Thomaidis, Nikolaos; Mikros, Emmanuel; Kleinbongard, Petra; Fioravanti, Rossella; Zwergel, Clemens; Valente, Sergio; Mai, Antonello; Andreadou, Ioanna
Chemically diverse S. mansoni HDAC8 inhibitors reduced viability in worm larval and adult stages
2023 Noce, Beatrice; Di Bello, Elisabetta; Zwergel, Clemens; Fioravanti, Rossella; Valente, Sergio; Rotili, Dante; Masotti, Andrea; Ansari, Mohammad Salik Zeya; Trisciuoglio, Daniela; Chakrabarti, Alokta; Romier, Christophe; Robaa, Dina; Sippl, Wolfgang; Jung, Manfred; Häberli, Cécile; Keiser, Jennifer; Mai, Antonello
Design of first-in-class dual EZH2/HDAC inhibitor: biochemical activity and biological evaluation in cancer cells
2020 Romanelli, Annalisa; Stazi, Giulia; Fioravanti, Rossella; Zwergel, Clemens; Di Bello, Elisabetta; Pomella, Silvia; Perrone, Clara; Battistelli, Cecilia; Strippoli, Raffaele; Tripodi, Marco; del Bufalo, Donatella; Rota, Rossella; Trisciuoglio, Daniela; Mai, Antonello; Valente, Sergio
Detrimental effects of the 'bath salt' methylenedioxypyrovalerone on social play behavior in male rats
2020 Schiavi, Sara; Melancia, Francesca; Carbone, Emilia; Buzzelli, Valeria; Manduca, Antonia; Peinado, Patricia Jiménez; Zwergel, Clemens; Mai, Antonello; Campolongo, Patrizia; Vanderschuren, Louk J M J; Trezza, Viviana
Development of alkyl glycerone phosphate synthase inhibitors: Structure-activity relationship and effects on ether lipids and epithelial-mesenchymal transition in cancer cells
2019 Stazi, Giulia; Battistelli, Cecilia; Piano, Valentina; Mazzone, Roberta; Marrocco, Biagina; Marchese, Sara; Louie, Sharon M.; Zwergel, Clemens; Antonini, Lorenzo; Patsilinakos, Alexandros; Ragno, Rino; Viviano, Monica; Sbardella, Gianluca; Ciogli, Alessia; Fabrizi, Giancarlo; Cirilli, Roberto; Strippoli, Raffaele; Marchetti, Alessandra; Tripodi, Marco; Nomura, Daniel K.; Mattevi, Andrea; Mai, Antonello; Valente, Sergio
Discovery of First-in-Class Carbonic Anhydrase/Histone Deacetylase Dual Inhibitors with Antiproliferative Activity in Cancer Cells
2025 Bozdag, Murat; Mroweh, Nabil; Raucci, Alessia; Angeli, Andrea; Peppicelli, Silvia; Biagioni, Alessio; Calorini, Lido; Trisciuoglio, Daniela; Ragno, Rino; Astolfi, Roberta; Giuliani, Lidia; Zwergel, Clemens; Valente, Sergio; Andreucci, Elena; Carta, Fabrizio; Mai, Antonello; Supuran, Claudiu T
Discovery of phenylselenoether-hydantoin hybrids as ABCB1 efflux pump modulating agents with cytotoxic and antiproliferative actions in resistant T-lymphoma
2020 Ali, Wesam; Spengler, Gabriella; Kincses, Annamária; Nové, Márta; Battistelli, Cecilia; Latacz, Gniewomir; Starek, Małgorzata; Dąbrowska, Monika; Honkisz-Orzechowska, Ewelina; Romanelli, Annalisa; Rasile, Manuela Monica; Szymańska, Ewa; Jacob, Claus; Zwergel, Clemens; Handzlik, Jadwiga
Discovery of the first human arylsulfatase a reversible inhibitor impairing mouse oocyte fertilization
2020 Caroselli, Silvia; Zwergel, Clemens; Pirolli, Adele; Sabatino, Manuela; Xu, Zhanjie; Kirsch, Gilbert; Mai, Antonello; Colotti, Gianni; Altieri, Fabio; Canipari, Rita; Valente, Sergio; Ragno, Rino
DNA methyltransferases Inhibitors from natural sources
2016 Zwergel, Clemens; Valente, Sergio; Mai, Antonello
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| 1,4-Dihydropyridines Active on the SIRT1/AMPK Pathway Ameliorate Skin Repair and Mitochondrial Function and Exhibit Inhibition of Proliferation in Cancer Cells | 2016 | Valente, Sergio; Mellini, Paolo; Spallotta, Francesco; Carafa, Vincenzo; Nebbioso, Angela; Polletta, Lucia; Carnevale, Ilaria; Saladini, Serena; Trisciuoglio, Daniela; Gabellini, Chiara; Tardugno, Maria; Zwergel, Clemens; Cencioni, Chiara; Atlante, Sandra; Moniot, Sébastien; Steegborn, Clemens; Budriesi, Roberta; Tafani, Marco; Del Bufalo, Donatella; Altucci, Lucia; Gaetano, Carlo; Mai, Antonello | |
| A quinoline-based DNA methyltransferase inhibitor as a possible adjuvant in osteosarcoma therapy | 2018 | Manara, Maria Cristina; Valente, Sergio; Cristalli, Camilla; Nicoletti, Giordano; Landuzzi, Lorena; Zwergel, Clemens; Mazzone, Roberta; Stazi, Giulia; Arimondo, Paola B.; Pasello, Michela; Guerzoni, Clara; Picci, Piero; Nanni, Patrizia; Lollini, Pier-Luigi; Mai, Antonello; Scotlandi, Katia | |
| A xanthine derivative with Nnovel heat shock protein 90-alpha inhibitory and senolytic properties | 2025 | Atlante, Sandra; Cis, Luca; Pirolli, Davide; Gottardi Zamperla, Michela; Barbi, Veronica; Mai, Antonello; Zwergel, Clemens; Marcozzi, Serena; Giuliani, Maria Elisa; Bigossi, Giorgia; Lai, Giovanni; Orlando, Fiorenza; Giacconi, Robertina; Lattanzio, Fabrizia; Matacchione, Giulia; Giordani, Chiara; Bracci, Massimo; Olivieri, Fabiola; Boschi, Federico; Tabarelli De Fatis, Paola; Ivaldi, Giovanni Battista; Malavolta, Marco; Farsetti, Antonella; De Rosa, Maria Cristina; Gaetano, Carlo | |
| Abstract 2946: Effects of two novel quinoline-based non-nucleoside DNA methyltransferase inhibitors against bone sarcomas | 2015 | Manara, Maria Cristina; Valente, Sergio; Cristalli, Camilla; Baricordi, Cristina; Zwergel, Clemens; Arimondo, Paola B; Picci, Piero; Mai, Antonello; Scotlandi, Katia | |
| Acute and chronic neurobehavioral effects of the designer drug and bath salt constituent 3,4-methylenedioxypyrovalerone in the rat | 2019 | ATEHORTUA MARTINEZ, LUISA ALESSANDRA; Masniere, Cyriaque; Campolongo, Patrizia; Chasseigneaux, Stéphanie; Callebert, Jacques; Zwergel, Clemens; Mai, Antonello; Laplanche, Jean-Louis; Chen, Huixiong; Etheve-Quelquejeu, Mélanie; Mégarbane, Bruno; Benturquia, Nadia | |
| Advancements in hydrazide-based HDAC inhibitors. A review of recent developments and therapeutic potential | 2025 | Raucci, Alessia; Zwergel, Clemens; Valente, Sergio; Mai, Antonello | |
| Amphetamine and the Smart Drug 3,4-Methylenedioxypyrovalerone (MDPV) Induce Generalization of Fear Memory in Rats | 2019 | Colucci, Paola; Mancini, Giulia Federica; Santori, Alessia; Zwergel, Clemens; Mai, Antonello; Trezza, Viviana; Roozendaal, Benno; Campolongo, Patrizia | |
| Amphetamine modulation of long-term object recognition memory in rats: influence of stress | 2021 | Colucci, Paola; Santori, Alessia; Romanelli, Luca; Zwergel, Clemens; Mai, Antonello; Scaccianoce, Sergio; Campolongo, Patrizia | |
| Application of small epigenetic modulators in pediatric medulloblastoma | 2018 | Zwergel, Clemens; Romanelli, Annalisa; Stazi, Giulia; Besharat, Zein Mersini; Catanzaro, Giuseppina; Tafani, Marco; Valente, Sergio; Mai, Antonello | |
| Aurones: Interesting Natural and Synthetic Compounds with Emerging Biological Potential | 2012 | Zwergel, Clemens; F., Gaascht; Valente, Sergio; M., Diederich; D., Bagrel; G., Kirsch | |
| Beyond antibodies. Reinventing Alzheimer’s treatment for the next decade | 2025 | Garbo, Sabrina; Raucci, Alessia; Zwergel, Clemens; Handzlik, Jadwiga; Battistelli, Cecilia | |
| Cardioprotection through pharmacological activation of Sirtuin 5 in a murine model of acute myocardial infarction | 2025 | Castiello, Carola; Efentakis, Panagiotis; Nikolaou, Panagiota-Efstathia; Symeonidi, Lydia; Chania, Christina; Barla, Ioanna; Akrani, Ifigeneia; Kostomitsopoulos, Nikolaos; Gikas, Evangelos; Thomaidis, Nikolaos; Mikros, Emmanuel; Kleinbongard, Petra; Fioravanti, Rossella; Zwergel, Clemens; Valente, Sergio; Mai, Antonello; Andreadou, Ioanna | |
| Chemically diverse S. mansoni HDAC8 inhibitors reduced viability in worm larval and adult stages | 2023 | Noce, Beatrice; Di Bello, Elisabetta; Zwergel, Clemens; Fioravanti, Rossella; Valente, Sergio; Rotili, Dante; Masotti, Andrea; Ansari, Mohammad Salik Zeya; Trisciuoglio, Daniela; Chakrabarti, Alokta; Romier, Christophe; Robaa, Dina; Sippl, Wolfgang; Jung, Manfred; Häberli, Cécile; Keiser, Jennifer; Mai, Antonello | |
| Design of first-in-class dual EZH2/HDAC inhibitor: biochemical activity and biological evaluation in cancer cells | 2020 | Romanelli, Annalisa; Stazi, Giulia; Fioravanti, Rossella; Zwergel, Clemens; Di Bello, Elisabetta; Pomella, Silvia; Perrone, Clara; Battistelli, Cecilia; Strippoli, Raffaele; Tripodi, Marco; del Bufalo, Donatella; Rota, Rossella; Trisciuoglio, Daniela; Mai, Antonello; Valente, Sergio | |
| Detrimental effects of the 'bath salt' methylenedioxypyrovalerone on social play behavior in male rats | 2020 | Schiavi, Sara; Melancia, Francesca; Carbone, Emilia; Buzzelli, Valeria; Manduca, Antonia; Peinado, Patricia Jiménez; Zwergel, Clemens; Mai, Antonello; Campolongo, Patrizia; Vanderschuren, Louk J M J; Trezza, Viviana | |
| Development of alkyl glycerone phosphate synthase inhibitors: Structure-activity relationship and effects on ether lipids and epithelial-mesenchymal transition in cancer cells | 2019 | Stazi, Giulia; Battistelli, Cecilia; Piano, Valentina; Mazzone, Roberta; Marrocco, Biagina; Marchese, Sara; Louie, Sharon M.; Zwergel, Clemens; Antonini, Lorenzo; Patsilinakos, Alexandros; Ragno, Rino; Viviano, Monica; Sbardella, Gianluca; Ciogli, Alessia; Fabrizi, Giancarlo; Cirilli, Roberto; Strippoli, Raffaele; Marchetti, Alessandra; Tripodi, Marco; Nomura, Daniel K.; Mattevi, Andrea; Mai, Antonello; Valente, Sergio | |
| Discovery of First-in-Class Carbonic Anhydrase/Histone Deacetylase Dual Inhibitors with Antiproliferative Activity in Cancer Cells | 2025 | Bozdag, Murat; Mroweh, Nabil; Raucci, Alessia; Angeli, Andrea; Peppicelli, Silvia; Biagioni, Alessio; Calorini, Lido; Trisciuoglio, Daniela; Ragno, Rino; Astolfi, Roberta; Giuliani, Lidia; Zwergel, Clemens; Valente, Sergio; Andreucci, Elena; Carta, Fabrizio; Mai, Antonello; Supuran, Claudiu T | |
| Discovery of phenylselenoether-hydantoin hybrids as ABCB1 efflux pump modulating agents with cytotoxic and antiproliferative actions in resistant T-lymphoma | 2020 | Ali, Wesam; Spengler, Gabriella; Kincses, Annamária; Nové, Márta; Battistelli, Cecilia; Latacz, Gniewomir; Starek, Małgorzata; Dąbrowska, Monika; Honkisz-Orzechowska, Ewelina; Romanelli, Annalisa; Rasile, Manuela Monica; Szymańska, Ewa; Jacob, Claus; Zwergel, Clemens; Handzlik, Jadwiga | |
| Discovery of the first human arylsulfatase a reversible inhibitor impairing mouse oocyte fertilization | 2020 | Caroselli, Silvia; Zwergel, Clemens; Pirolli, Adele; Sabatino, Manuela; Xu, Zhanjie; Kirsch, Gilbert; Mai, Antonello; Colotti, Gianni; Altieri, Fabio; Canipari, Rita; Valente, Sergio; Ragno, Rino | |
| DNA methyltransferases Inhibitors from natural sources | 2016 | Zwergel, Clemens; Valente, Sergio; Mai, Antonello |