Sfoglia per Autore
Progress in the development of arylthioindoles, potent inhibitors of tubulin polymerization and MCF-7 cell growth.
2008 LA REGINA, Giuseppe; Piscitelli, Francesco; Coluccia, Antonio; Brancale, A.; Hamel, E.; Diaz, J. F.; Scovassi, A. I.; Lavecchia, A.; Novellino, E.; Silvestri, Romano
Docking and Molecular Dynamics Studies of Arylthioindoles.
2008 LA REGINA, Giuseppe; Piscitelli, Francesco; Coluccia, Antonio; Minelli, L.; Brancale, A.; Kandil, S.; Lavecchia, A.; Novellino, E.; Silvestri, Romano
Cdc25B phosphatase inhibitors in cancer therapy: latest developments, trends and medicinal chemistry perspective.
2008 Lavecchia, A; Coluccia, Antonio; DI GIOVANNI, C; Novellino, E.
Indolyl Aryl Sulfones, HIV-1 Non-Nucleoside Reverse Transcriptase Inhibitors: Docking and 3-D QSAR studies
2008 Coluccia, Antonio
Indolylarylsulfones Bearing Natural and Unnatural Amino Acids as Potent HIV-1 NNRTIs.
2009 Piscitelli, Francesco; LA REGINA, Giuseppe; Gatti, Valerio; Coluccia, Antonio; Brancale, A.; Giordano, C.; Balzarini, J.; Maga, G.; Lavecchia, A.; Novellino, E.; Silvestri, Romano
Arylthioindole Bioisosteres as Potent Tubulin Polymerization and MCF-7 Cell Growth Inhibitors
2009 Gatti, Valerio; LA REGINA, Giuseppe; Coluccia, Antonio; Brancale, A.; Hamel, E.; Scovassi, A.; Maresca, B.; Campiglia, P.; Novellino, E.; Silvestri, Romano
Drug Design of New NS3/4A HCV Serine Protease Inhibitors. Structure-Based and Ligand-Based Approaches.
2009 Coluccia, Antonio; LA REGINA, Giuseppe; Giordano, C.; Sansone, A.; Brancale, A.; Neyts, J.; Leyssen, P.; Novellino, E.; Silvestri, Romano
New arylthioindoles and related bioisosteres at the sulfur bridging group. 4. Synthesis, tubulin polymerization, cell growth inhibition, and molecular modeling studies
2009 LA REGINA, Giuseppe; Taradas, Sarkar; Ruoli, Bai; Michael C., Edler; Roberto, Saletti; Coluccia, Antonio; Piscitelli, Francesco; Lara, Minelli; Gatti, Valerio; Carmela, Mazzoccoli; Palermo, Vanessa; Mazzoni, Cristina; Falcone, Claudio; Anna Ivana, Scovassi; Vincenzo, Giansanti; Pietro, Campiglia; Amalia, Porta; Bruno, Maresca; Ernest, Hamel; Andrea, Brancale; Ettore, Novellino; Silvestri, Romano
Molecular Modeling Studies of Arylthioindoles and Related Bioisosteres, Potent Inhibitors of Tubulin Polymerization.
2009 LA REGINA, Giuseppe; Coluccia, Antonio; Gatti, Valerio; Saletti, R.; Brancale, A.; Novellino, E.; Silvestri, Romano
Indolylarylsulfones Bearing Natural and Unnatural Amino Acids are Potent HIV-1 Reverse Transcriptase and Coxsackie B4 Virus Non-Nucleoside Inhibitors.
2009 Piscitelli, Francesco; Coluccia, Antonio; Brancale, A.; LA REGINA, Giuseppe; Sansone, A.; Giordano, C.; Balzarini, J.; Maga, G.; Zanoli, S.; Samuele, A.; Cirilli, R.; LA TORRE, F.; Lavecchia, A.; Novellino, E.; Silvestri, Romano
Molecular Modeling applications studies on the Indolyl Aryl Sulphones (IASs) as HIV-1 Non-Nucleotidic Reverse transcriptase inhibitors.
2009 Coluccia, Antonio; Brancale, A.; LA REGINA, Giuseppe; Lavecchia, A.; Silvestri, Romano
Indolyl Aryl Sulfones bearing Natural and Unnatural Aminoacids. Discovery of Potent Inhibitors of both HIV-1 Non-Nucleoside Wild Type and Resistant Mutant Strains Reverse Transcriptase, and Coxsackie B4 Virus.
2009 Piscitelli, Francesco; Coluccia, Antonio; Brancale, A.; LA REGINA, Giuseppe; Sansone, A.; Giordano, C.; Balzarini, J.; Maga, G.; Zanoli, S.; Samuele, A.; Cirilli, R.; LA TORRE, F.; Lavecchia, A.; Novellino, E.; Silvestri, Romano
Discovery of a novel HCV helicase inhibitor by a de novo drug design approach
2009 Kandil, S; Biondaro, S; Vlachakis, D; Cummins, Ac; Coluccia, Antonio; Berry, C; Leyssen, P; Neyts, J; Brancale, A.
Molecular dynamic studies of arylthioindoles, potent inhibitors of tubulin polymerization
2010 Coluccia, A; Brancale, A; Silvestri, Romano
Indolylarylsulfones bearing natural and unnatural amino acids as inhibitors of HIV-1 reverse transcriptase and Coxsackie B4 virus.
2010 Gatti, Valerio; LA REGINA, Giuseppe; Coluccia, Antonio; Piscitelli, Francesco; C., Giordano; A., Brancale; J., Balzarini; G., Maga; E., Novellino; Silvestri, Romano
Advanced in silico approaches in antiviral research
2010 Zonta, N; Coluccia, Antonio; Brancale, A.
Discovery of a novel hcv helicase inhibitors by a de novo design approach.
2010 Coluccia, A; Leyssen, P; Neyts, J; Kandil, S; Brancale, A; Silvestri, Romano
Looking for an active conformation of the future HIV type-1 non-nucleoside reverse transcriptase inhibitors
2010 LA REGINA, Giuseppe; Coluccia, Antonio; Silvestri, Romano
Indolylarylsulfones as HIV-1 Non-Nucleoside Reverse Transcriptase Inhibitors. New Cyclic Substituents at the Indole-2-carboxamide.
2011 Coluccia, Antonio; LA REGINA, Giuseppe; Gatti, Valerio; Piscitelli, Francesco; Famiglini, V.; Brancale, A.; Maga, G.; Balzarini, J.; Novellino, E.; Silvestri, Romano
Molecular modelling studies on Arylthioindoles as potent inhibitors of tubulin polymerization
2011 Coluccia, Antonio; Sabbadin, Davide; Brancale, Andrea
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Progress in the development of arylthioindoles, potent inhibitors of tubulin polymerization and MCF-7 cell growth. | 2008 | LA REGINA, Giuseppe; Piscitelli, Francesco; Coluccia, Antonio; Brancale, A.; Hamel, E.; Diaz, J. F.; Scovassi, A. I.; Lavecchia, A.; Novellino, E.; Silvestri, Romano | |
Docking and Molecular Dynamics Studies of Arylthioindoles. | 2008 | LA REGINA, Giuseppe; Piscitelli, Francesco; Coluccia, Antonio; Minelli, L.; Brancale, A.; Kandil, S.; Lavecchia, A.; Novellino, E.; Silvestri, Romano | |
Cdc25B phosphatase inhibitors in cancer therapy: latest developments, trends and medicinal chemistry perspective. | 2008 | Lavecchia, A; Coluccia, Antonio; DI GIOVANNI, C; Novellino, E. | |
Indolyl Aryl Sulfones, HIV-1 Non-Nucleoside Reverse Transcriptase Inhibitors: Docking and 3-D QSAR studies | 2008 | Coluccia, Antonio | |
Indolylarylsulfones Bearing Natural and Unnatural Amino Acids as Potent HIV-1 NNRTIs. | 2009 | Piscitelli, Francesco; LA REGINA, Giuseppe; Gatti, Valerio; Coluccia, Antonio; Brancale, A.; Giordano, C.; Balzarini, J.; Maga, G.; Lavecchia, A.; Novellino, E.; Silvestri, Romano | |
Arylthioindole Bioisosteres as Potent Tubulin Polymerization and MCF-7 Cell Growth Inhibitors | 2009 | Gatti, Valerio; LA REGINA, Giuseppe; Coluccia, Antonio; Brancale, A.; Hamel, E.; Scovassi, A.; Maresca, B.; Campiglia, P.; Novellino, E.; Silvestri, Romano | |
Drug Design of New NS3/4A HCV Serine Protease Inhibitors. Structure-Based and Ligand-Based Approaches. | 2009 | Coluccia, Antonio; LA REGINA, Giuseppe; Giordano, C.; Sansone, A.; Brancale, A.; Neyts, J.; Leyssen, P.; Novellino, E.; Silvestri, Romano | |
New arylthioindoles and related bioisosteres at the sulfur bridging group. 4. Synthesis, tubulin polymerization, cell growth inhibition, and molecular modeling studies | 2009 | LA REGINA, Giuseppe; Taradas, Sarkar; Ruoli, Bai; Michael C., Edler; Roberto, Saletti; Coluccia, Antonio; Piscitelli, Francesco; Lara, Minelli; Gatti, Valerio; Carmela, Mazzoccoli; Palermo, Vanessa; Mazzoni, Cristina; Falcone, Claudio; Anna Ivana, Scovassi; Vincenzo, Giansanti; Pietro, Campiglia; Amalia, Porta; Bruno, Maresca; Ernest, Hamel; Andrea, Brancale; Ettore, Novellino; Silvestri, Romano | |
Molecular Modeling Studies of Arylthioindoles and Related Bioisosteres, Potent Inhibitors of Tubulin Polymerization. | 2009 | LA REGINA, Giuseppe; Coluccia, Antonio; Gatti, Valerio; Saletti, R.; Brancale, A.; Novellino, E.; Silvestri, Romano | |
Indolylarylsulfones Bearing Natural and Unnatural Amino Acids are Potent HIV-1 Reverse Transcriptase and Coxsackie B4 Virus Non-Nucleoside Inhibitors. | 2009 | Piscitelli, Francesco; Coluccia, Antonio; Brancale, A.; LA REGINA, Giuseppe; Sansone, A.; Giordano, C.; Balzarini, J.; Maga, G.; Zanoli, S.; Samuele, A.; Cirilli, R.; LA TORRE, F.; Lavecchia, A.; Novellino, E.; Silvestri, Romano | |
Molecular Modeling applications studies on the Indolyl Aryl Sulphones (IASs) as HIV-1 Non-Nucleotidic Reverse transcriptase inhibitors. | 2009 | Coluccia, Antonio; Brancale, A.; LA REGINA, Giuseppe; Lavecchia, A.; Silvestri, Romano | |
Indolyl Aryl Sulfones bearing Natural and Unnatural Aminoacids. Discovery of Potent Inhibitors of both HIV-1 Non-Nucleoside Wild Type and Resistant Mutant Strains Reverse Transcriptase, and Coxsackie B4 Virus. | 2009 | Piscitelli, Francesco; Coluccia, Antonio; Brancale, A.; LA REGINA, Giuseppe; Sansone, A.; Giordano, C.; Balzarini, J.; Maga, G.; Zanoli, S.; Samuele, A.; Cirilli, R.; LA TORRE, F.; Lavecchia, A.; Novellino, E.; Silvestri, Romano | |
Discovery of a novel HCV helicase inhibitor by a de novo drug design approach | 2009 | Kandil, S; Biondaro, S; Vlachakis, D; Cummins, Ac; Coluccia, Antonio; Berry, C; Leyssen, P; Neyts, J; Brancale, A. | |
Molecular dynamic studies of arylthioindoles, potent inhibitors of tubulin polymerization | 2010 | Coluccia, A; Brancale, A; Silvestri, Romano | |
Indolylarylsulfones bearing natural and unnatural amino acids as inhibitors of HIV-1 reverse transcriptase and Coxsackie B4 virus. | 2010 | Gatti, Valerio; LA REGINA, Giuseppe; Coluccia, Antonio; Piscitelli, Francesco; C., Giordano; A., Brancale; J., Balzarini; G., Maga; E., Novellino; Silvestri, Romano | |
Advanced in silico approaches in antiviral research | 2010 | Zonta, N; Coluccia, Antonio; Brancale, A. | |
Discovery of a novel hcv helicase inhibitors by a de novo design approach. | 2010 | Coluccia, A; Leyssen, P; Neyts, J; Kandil, S; Brancale, A; Silvestri, Romano | |
Looking for an active conformation of the future HIV type-1 non-nucleoside reverse transcriptase inhibitors | 2010 | LA REGINA, Giuseppe; Coluccia, Antonio; Silvestri, Romano | |
Indolylarylsulfones as HIV-1 Non-Nucleoside Reverse Transcriptase Inhibitors. New Cyclic Substituents at the Indole-2-carboxamide. | 2011 | Coluccia, Antonio; LA REGINA, Giuseppe; Gatti, Valerio; Piscitelli, Francesco; Famiglini, V.; Brancale, A.; Maga, G.; Balzarini, J.; Novellino, E.; Silvestri, Romano | |
Molecular modelling studies on Arylthioindoles as potent inhibitors of tubulin polymerization | 2011 | Coluccia, Antonio; Sabbadin, Davide; Brancale, Andrea |
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