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Antifungal estrogen-like imidazoles. Synthesis and antifungal activities of thienyl and 1H-pyrrolyl derivatives of 1-aryl-2-(1H-imidazol-1-yl)ethane. 1997 DI SANTO, Roberto; Costi, Roberta; Artico, Marino; Massa, S.; Musiu, C.; Scintu, F.; Putzolu, M.; LA COLLA, P.
Arylketotetramethylene analogues of disoxaril with anti-human rhinovirus 14 activity 1997 Mai, A.; Artico, M.; Sbardella, G.; Massa, S.; DE MONTIS, Andrea; Puddu, I.; Musiu, C.; La Colla, P.
Pyrrolnitrin and Related Pyrroles Endowed with Antibacterial Activities against Mycobacterium Tuberculosis. 1998 DI SANTO, Roberto; Costi, Roberta; Artico, Marino; Massa, S.; Lampis, G.; Deidda, D.; Pompei, R.
N-[4-(1,1'-Biphenyl)methyl]-4-(4-thiomorpholinylmethyl)benzenamines as non-oxazolidinone analogues of antimycobacterial U-100480. 1998 Artico, Marino; Mai, Antonello; Sbardella, G; Massa, S; Lampis, G; Deidda, D; Pompei, R.
CRYSTAL STRUCTURE OF 2-[5-(4-CARBETOXYPHENOXY)PENTANOYL]-5-CHLOROTHIOPHENE, C18H19O4ClS 1998 A., Ettorre; Artico, Marino; Mai, Antonello; Ragno, Rino; Porretta, Giulio Cesare; S., Massa
Geometrically and Conformationally Restrained Cinnamoyl-Compounds as Inhibitors of HIV-1 Integrase: Synthesis, Biological Evaluation and Molecular Modeling 1998 Artico, Marino; DI SANTO, Roberto; Costi, Roberta; Novellino, E.; Greco, G.; Massa, S.; Tramontano, E.; Marongiu, M. E.; DE MONTIS, A.; LA COLLA, P:
N-[4-(1,1'-Biphenylyl)methyl]-4-(4-thiomorpholinylmethyl)benzenamines, a New Class of Synthetic Antituberculosis Agents Active Against Mycobacterium Avium. 1999 Mai, Antonello; Sbardella, G.; Artico, Marino; Massa, S.; Lampis, G.; Deidda, D.; Pompei, R.
Nitroquinolones with Broad-Spectrum Antimycobacterial Activity in Vitro. 1999 Artico, Marino; Mai, Antonello; Sbardella, G; Massa, S; Musiu, C; Lostia, S; Demontis, F; LA COLLA, P.
Pyridinylpyrrolyl Analogs of Isoniazid: Synthesis and Antimycobacterial Activities. 1999 Costi, Roberta; Artico, Marino; DI SANTO, Roberto; DE MARTINO, G.; Massa, S.; Deidda, D.; Lampis, G.; Pompei, R.
5-alkyl-2-(alkylthio)-6-(2,6-dihalophenylmethyl)-3,4-dihydropyrimidin-4(3h)-ones: novel potent and selective dihydro-alkoxy-benzyl-oxopyrimidine derivatives 1999 Mai, Antonello; Artico, Marino; Sbardella, G.; Massa, S.; Novellino, E.; Greco, G.; Loi, A. G.; Tramontano, E.; Marongiu, M. E.; LA COLLA, P.
Structure-activity relationship studies on potential non-nucleoside DABO-like inhibitors of HIV-1 reverse transcriptase. 2000 Costi, Roberta; DI SANTO, Roberto; Artico, Marino; Massa, S.; LA VECCHIA, A.; Marceddu, T.; Sanna, L.; LA COLLA, P.; Marongiu, M. E.
Derivati del 2H-pirrolo[3,4-c]chinolin-4(5H)-one: Nuovi Potenziali Agonisti dei Recettori 5-HT3 2000 Costi, Roberta; DI SANTO, Roberto; Artico, Marino; Massa, Silvio; DE MARTINO, G.; Saturnino, C.
Structure based design, synthesis and biological evaluation of novel pyrrolyl aryl sulfones (PASs) active at nanomolar concentration as HIV-1 non nucleoside reverse transcriptase inhibitors. 2000 Artico, Marino; Silvestri, Romano; Pagnozzi, E.; Bruno, B.; Novellino, E.; Greco, G.; Massa, S.; Ettorre, A.; Loi, A. G.; Scintu, F.; LA COLLA, P.
Does the 2-methylthiomethyl substituent really confer high anti-HIV-1 activity to S-DABOs ? 2000 Sbardella, G; Mai, Antonello; Artico, Marino; Massa, S; Marceddu, T; Vargiu, L; MARONGIU M., E; LA COLLA, P.
Antimycobacterial Pyrroles: Synthesis, Anti-Mycobacterium tuberculosis Activity and QSAR Studies. 2000 Ragno, Rino; Marshall, G. R.; DI SANTO, Roberto; Costi, Roberta; Massa, S.; Pompei, R.; Artico, Marino
3,4-Dihydro-2-alkoxy-6-benzyl-oxopyrimidines (DABOs): Development of a Potent Class of Non-nucleoside Reverse Transcriptase Inhibitors 2001 Marongiu, M. E.; Pani, A.; Musiu, C.; LA COLLA, P.; Mai, Antonello; Sbardella, G.; Massa, S.; Artico, M.
Structure-Based Design, Synthesis and Biological Evaluation of Conformationally Restricted Novel 2-Alkylthio-6-[1-(2,6-difluorophenyl)alkyl]-3,4-dihydro-5-alkylpyrimidin-4(3H)-ones as Non-nucleoside Inhibitors of HIV-1 Reverse Transcriptase 2001 Mai, Antonello; Sbardella, G; Artico, Marino; Ragno, Rino; Massa, S; Novellino, E; Greco, G; Lavecchia, A; Musiu, C; LA COLLA, M; Murgioni, C; LA COLLA, P.
Chiral resolution and molecular modeling investigation of rac-2-cyclopentylthio-6-[1-(2,6-difluorophenyl)ethyl]-3,4-dihydro-5- methylpyrimidin-4(3H)-one (MC-1047), a potent anti-HIV-1 reverse transcriptase agent of the DABO class. 2001 Quaglia, M. G.; Mai, Antonello; Sbardella, G.; Artico, Marino; Ragno, Rino; Massa, S.; DEL PIANO, D.; Setzu, G.; Doratiotto, S.; Cotichini, V.
1-[4-(4-Chlorophenyl)-1H-pyrrol-3-yl](2,4-dichlorophenyl)methyl-1H-imidazole (RDS 416) 2001 Camalli, M.; Pifferi, A.; Costi, Roberta; DI SANTO, Roberto; Massa, S.; Artico, Marino
Anti-HIV-1 NNRT Agents: Acylamino Pyrryl Aryl Sulfones (APASs) as Truncated Analogues of Tricyclic PBTDs. 2002 Silvestri, Romano; DE MARTINO, G.; LA REGINA, Giuseppe; Artico, Marino; Ragno, Rino; LA COLLA, P.; Marongiu, M. E.; Pani, A.
Mostrati risultati da 21 a 40 di 129
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