Sfoglia per Autore
Pyrrole derivatives of BM212 as novel antimycobacterial agents Design, synthesis, biological evaluation and study of their mode of action
2009 Biava, Mariangela; Porretta, Giulio Cesare; Battilocchio, Claudio; Poce, G; Pompei, R; DE LOGU, A; Manetti, F; Botta, M.
Developing New Antiinflammatory and Analgesic Agents: Design, Synthesis, Biological and harmacological Evaluation
2010 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; Alfonso, Salvatore; Botta, M.; Manetti, F.; Sautebin, L; Ghelardini, C; Makovec, F; Giordani, A; Patrignani, P; Anzini, M.
1,5-Diaryl-Pyrroles as New Generation of Anti-Inflammatory and Analgesic Agents: Design, Synthesis, in vitro and in vivo Evaluation
2010 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Alfonso, S; Battilocchio, Claudio; DE LOGU, A; Manetti, F; Botta, M.
Identification of a new Chemical Class of Potent Antimycobacterial Compounds
2010 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Alfonso, Salvatore; Battilocchio, Claudio; De Logu, A; Manetti, F; Botta, M.
BM 579: a novel pyrrole derivative with improved antimycobacterial activity
2010 Biava, Mariangela; Porretta, G. C.; Poce, Giovanna; Alfonso, Salvatore; Battilocchio, Claudio; De Logu, A.; Manetti, F; Botta, M.
New heterocyclic compounds with potential activity against parasitic protozoan: Trypanosoma and Leishmania
2010 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; V., Yardley; Alfonso, Salvatore
Novel Ester and Acid Derivatives of the 1,5-Diarylpyrrole Scaffold as Anti-inflammatory and Analgesic Agents. Synthesis, in vitro and in vivo Biological Evaluation
2010 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; Manetti, F; Botta, M; Sautebin, L; Rossi, A; Pergola, C; Ghelardini, C; Norcini, M; Makovec, F; Anzellotti, P; Cirilli, R; Ferretti, R; Patrignani, P; Anzini, M.
New pyrrole derivatives of BM 212: a new class of antimycobacterial agents. Design, synthesis, biological evaluation and study of their mode of action
2010 Biava, Mariangela; Porretta, G. C.; Poce, Giovanna; Alfonso, Salvatore; Battilocchio, Claudio; De Logu, A.; De Rossi, E.; Manetti, F; Botta, M.
Identification of a novel pyrrole derivative endowed with antimycobacterial activity and protection index comparable to that of the current antitubercular drugs streptomycin and rifampin
2010 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; Alfonso, Salvatore; A., De Logu; Nadia, Serra; Fabrizio, Manetti; Maurizio, Botta
New Pyrrole-based selective COX-2 inhibiting nitric oxide donors: synthesis, in vitro and in vivo evaluation
2011 Battilocchio, Claudio; Porretta, Giulio Cesare; Poce, Giovanna; Alfonso, Salvatore; Giordani, A.; Sautebin, L.; Ghelardini, C.; Calderone, V.; Patrignani, P.; Anzini, M.; Biava, Mariangela
Synthesis and biological evaluation of new heterocyclic derivatives with potential antimycobacterial activity: systematic approach to lead compound optimization
2011 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Alfonso, Salvatore; Battilocchio, Claudio; De Logu, A; Manetti, F; Botta, M.
Pyrrole-based selective COX-2 inhibiting nitric oxide donors: synthesis, in vitro and in vivo evaluation
2011 Battilocchio, Claudio; Porretta, Giulio Cesare; Poce, Giovanna; Alfonso, Salvatore; Calderone, V.; Sautebin, L.; Ghelardini, C.; Giordani, A.; Anzini, M.; Biava, Mariangela
BM212 targets MmpL3, Gordon Research Conference on Tuberculosis Drug Development
2011 Poce, Giovanna; Biava, Mariangela; Porretta, Giulio Cesare; Battilocchio, Claudio; Alfonso, Salvatore; Botta, M.; Javid, B.; Sorrentino, F.; Ioerger, T. R.; Sacchettini, J. R.; Rubin, E.
Novel Analgesic/Anti-Inflammatory Agents: Diarylpyrrole Acetic Esters Endowed with Nitric Oxide Releasing Properties
2011 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; Alfonso, Salvatore; Michele, Rovini; Salvatore, Valenti; Gianluca, Giorgi; Vincenzo, Calderone; Alma, Martelli; Lara, Testai; Lidia, Sautebin; Antonietta, Rossi; Giuseppina, Papa; Carla, Ghelardini; Lorenzo Di Cesare, Mannelli; Antonio, Giordani; Paola, Anzellotti; Annalisa, Bruno; Paola, Patrignani; Anzini,
Developing Pyrrole-Derived Antimycobacterial Agents: a Rational Lead Optimization Approach
2011 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; Alfonso, Salvatore; A., De Logu; Fabrizio, Manetti; Maurizio, Botta
Enlarging the NSAIDs Family: Ether, Ester and Acid Derivatives of the 1,5-Diarylpyrrole Scaffold as Novel Anti-Inflammatory and Analgesic Agents
2011 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; Botta, M; Manetti, F; Rovini, M; Cappelli, A; Sautebin, L; Rossi, A; Pergola, C; Ghelardini, C; Galeotti, N; Makovec, F; Giordani, A; Anzellotti, P; Tacconelli, S; Patrignani, P; Anzini, M.
New 1,5-diphenyl pyrrole derivatives as anti-inflammatory COX-2 selective compounds and their use as potential antitumoral agents.
2012 Consalvi, Sara; Battilocchio, Claudio; Poce, Giovanna; Alfonso, Salvatore; Porretta, Giulio Cesare; M., Anzini; L., Sautebin; C., Ghelardini; A., Giordani; P., Patrignani; V., Calderone; Biava, Mariangela
New Pyrrole Derivatives as Anti-inflammatory and Analgesic Agents: Design, Synthesis and Biological Evaluation
2012 Biava, Mariangela; Consalvi, Sara; Poce, Giovanna; Battilocchio, Claudio; Alfonso, Salvatore; Ghelardini, C.; Sautebin, L.
Flow Based Synthesis of 2-aminoadamantane-2-carboxylic acid
2012 Battilocchio, Claudio; Baxendale, I. R.; Biava, Mariangela; Kitching, Mo; Ley, S. V.
New 1,5 diarylpyrrole derivatives as antimycobacterial agents: Design, synthesis, biological evaluation and study of their mode of action
2012 Alfonso, Salvatore; Poce, Giovanna; Porretta, Giulio Cesare; Battilocchio, Claudio; Rubin, E. J.; De Rossi, E.; De Logu, A.; Franzblau, S. C.; Botta, M.; Biava, Mariangela
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Pyrrole derivatives of BM212 as novel antimycobacterial agents Design, synthesis, biological evaluation and study of their mode of action | 2009 | Biava, Mariangela; Porretta, Giulio Cesare; Battilocchio, Claudio; Poce, G; Pompei, R; DE LOGU, A; Manetti, F; Botta, M. | |
Developing New Antiinflammatory and Analgesic Agents: Design, Synthesis, Biological and harmacological Evaluation | 2010 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; Alfonso, Salvatore; Botta, M.; Manetti, F.; Sautebin, L; Ghelardini, C; Makovec, F; Giordani, A; Patrignani, P; Anzini, M. | |
1,5-Diaryl-Pyrroles as New Generation of Anti-Inflammatory and Analgesic Agents: Design, Synthesis, in vitro and in vivo Evaluation | 2010 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Alfonso, S; Battilocchio, Claudio; DE LOGU, A; Manetti, F; Botta, M. | |
Identification of a new Chemical Class of Potent Antimycobacterial Compounds | 2010 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Alfonso, Salvatore; Battilocchio, Claudio; De Logu, A; Manetti, F; Botta, M. | |
BM 579: a novel pyrrole derivative with improved antimycobacterial activity | 2010 | Biava, Mariangela; Porretta, G. C.; Poce, Giovanna; Alfonso, Salvatore; Battilocchio, Claudio; De Logu, A.; Manetti, F; Botta, M. | |
New heterocyclic compounds with potential activity against parasitic protozoan: Trypanosoma and Leishmania | 2010 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; V., Yardley; Alfonso, Salvatore | |
Novel Ester and Acid Derivatives of the 1,5-Diarylpyrrole Scaffold as Anti-inflammatory and Analgesic Agents. Synthesis, in vitro and in vivo Biological Evaluation | 2010 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; Manetti, F; Botta, M; Sautebin, L; Rossi, A; Pergola, C; Ghelardini, C; Norcini, M; Makovec, F; Anzellotti, P; Cirilli, R; Ferretti, R; Patrignani, P; Anzini, M. | |
New pyrrole derivatives of BM 212: a new class of antimycobacterial agents. Design, synthesis, biological evaluation and study of their mode of action | 2010 | Biava, Mariangela; Porretta, G. C.; Poce, Giovanna; Alfonso, Salvatore; Battilocchio, Claudio; De Logu, A.; De Rossi, E.; Manetti, F; Botta, M. | |
Identification of a novel pyrrole derivative endowed with antimycobacterial activity and protection index comparable to that of the current antitubercular drugs streptomycin and rifampin | 2010 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; Alfonso, Salvatore; A., De Logu; Nadia, Serra; Fabrizio, Manetti; Maurizio, Botta | |
New Pyrrole-based selective COX-2 inhibiting nitric oxide donors: synthesis, in vitro and in vivo evaluation | 2011 | Battilocchio, Claudio; Porretta, Giulio Cesare; Poce, Giovanna; Alfonso, Salvatore; Giordani, A.; Sautebin, L.; Ghelardini, C.; Calderone, V.; Patrignani, P.; Anzini, M.; Biava, Mariangela | |
Synthesis and biological evaluation of new heterocyclic derivatives with potential antimycobacterial activity: systematic approach to lead compound optimization | 2011 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Alfonso, Salvatore; Battilocchio, Claudio; De Logu, A; Manetti, F; Botta, M. | |
Pyrrole-based selective COX-2 inhibiting nitric oxide donors: synthesis, in vitro and in vivo evaluation | 2011 | Battilocchio, Claudio; Porretta, Giulio Cesare; Poce, Giovanna; Alfonso, Salvatore; Calderone, V.; Sautebin, L.; Ghelardini, C.; Giordani, A.; Anzini, M.; Biava, Mariangela | |
BM212 targets MmpL3, Gordon Research Conference on Tuberculosis Drug Development | 2011 | Poce, Giovanna; Biava, Mariangela; Porretta, Giulio Cesare; Battilocchio, Claudio; Alfonso, Salvatore; Botta, M.; Javid, B.; Sorrentino, F.; Ioerger, T. R.; Sacchettini, J. R.; Rubin, E. | |
Novel Analgesic/Anti-Inflammatory Agents: Diarylpyrrole Acetic Esters Endowed with Nitric Oxide Releasing Properties | 2011 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; Alfonso, Salvatore; Michele, Rovini; Salvatore, Valenti; Gianluca, Giorgi; Vincenzo, Calderone; Alma, Martelli; Lara, Testai; Lidia, Sautebin; Antonietta, Rossi; Giuseppina, Papa; Carla, Ghelardini; Lorenzo Di Cesare, Mannelli; Antonio, Giordani; Paola, Anzellotti; Annalisa, Bruno; Paola, Patrignani; Anzini, | |
Developing Pyrrole-Derived Antimycobacterial Agents: a Rational Lead Optimization Approach | 2011 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; Alfonso, Salvatore; A., De Logu; Fabrizio, Manetti; Maurizio, Botta | |
Enlarging the NSAIDs Family: Ether, Ester and Acid Derivatives of the 1,5-Diarylpyrrole Scaffold as Novel Anti-Inflammatory and Analgesic Agents | 2011 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; Botta, M; Manetti, F; Rovini, M; Cappelli, A; Sautebin, L; Rossi, A; Pergola, C; Ghelardini, C; Galeotti, N; Makovec, F; Giordani, A; Anzellotti, P; Tacconelli, S; Patrignani, P; Anzini, M. | |
New 1,5-diphenyl pyrrole derivatives as anti-inflammatory COX-2 selective compounds and their use as potential antitumoral agents. | 2012 | Consalvi, Sara; Battilocchio, Claudio; Poce, Giovanna; Alfonso, Salvatore; Porretta, Giulio Cesare; M., Anzini; L., Sautebin; C., Ghelardini; A., Giordani; P., Patrignani; V., Calderone; Biava, Mariangela | |
New Pyrrole Derivatives as Anti-inflammatory and Analgesic Agents: Design, Synthesis and Biological Evaluation | 2012 | Biava, Mariangela; Consalvi, Sara; Poce, Giovanna; Battilocchio, Claudio; Alfonso, Salvatore; Ghelardini, C.; Sautebin, L. | |
Flow Based Synthesis of 2-aminoadamantane-2-carboxylic acid | 2012 | Battilocchio, Claudio; Baxendale, I. R.; Biava, Mariangela; Kitching, Mo; Ley, S. V. | |
New 1,5 diarylpyrrole derivatives as antimycobacterial agents: Design, synthesis, biological evaluation and study of their mode of action | 2012 | Alfonso, Salvatore; Poce, Giovanna; Porretta, Giulio Cesare; Battilocchio, Claudio; Rubin, E. J.; De Rossi, E.; De Logu, A.; Franzblau, S. C.; Botta, M.; Biava, Mariangela |
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