Sfoglia per Autore
Discovery of (Aryloxo propenyl)pyrrolyl Hydroxyamides as Selective Inhibitors of Class IIa Histone Deacetylase Homologue HD1-A
2003 Mai, Antonello; Massa, S.; Pezzi, R.; Rotili, Dante; Loidl, P.; Brosch, G.
Synthesis and evaluation of sirtinol analogues as yeast Sir2 and human SIRT inhibitors
2004 Pezzi, R.; Rotili, D.; Simeoni, S.; Ragno, Rino; Mariotti, FRANCESCA ROMANA; Chiani, Francesco; Camilloni, Giorgio; Massa, S.; Mai, Antonello
A novel Gcn5p inhibitor represses cell growth, gene transcription and histone acetylation in budding yeast
2005 Prisca, Ornaghi; Rotili, Dante; Gianluca, Sbardella; Mai, Antonello; Patrizia, Filetici
Histone Deacetylation in Epigenetics: An Attractive Target for Anticancer Therapy
2005 Mai, Antonello; Massa, S; Rotili, Dante; Cerbara, I; Valente, Sergio; Pezzi, R; Simeoni, S; Ragno, Rino
6-[1-(2,6-difluorophenyl)ethyl]pyrimidinones antagonize cell proliferation and induce cell differentiation by inhibiting (a nontelomeric) endogenous reverse transcriptase
2005 Sara, Bartolini; Mai, Antonello; Artico, Marino; Nicola, Paesano; Rotili, Dante; Corrado, Spadafora; Gianluca, Sbardella
Class II (IIa)-selective histone deacetylase inhibitors. 1. Synthesis and biological evaluation of novel (aryloxopropenyl)pyrrolyl hydroxyamides
2005 Mai, Antonello; Silvio, Massa; Riccardo, Pezzi; Silvia, Simeoni; Rotili, Dante; Angela, Nebbioso; Annamaria, Scognamiglio; Lucia, Altucci; Peter, Loidl; Gerald, Brosch
Exploring the connection unit in the HDAC inhibitor pharmacophore model: Novel uracil-based hydroxamates
2005 Mai, Antonello; Silvio, Massa; Rotili, Dante; Riccardo, Pezzi; Patrizia, Bottoni; Roberto, Scatena; Joachim, Meraner; Gerald, Brosch
Analytical and semipreparative high performance liquid chromatography separation of stereoisomers of novel 3,4-dihydropyrimidin-4(3H)-one derivatives on the immobilised amylose-based Chiralpack IA chiral stationary phase.
2006 Cirilli, R; Ferretti, R; Gallinella, B; LA TORRE, F; Mai, Antonello; Rotili, Dante
Small-Molecule Inhibitors of Histone Acetyltransferase Activity: Identification and Biological Properties
2006 Mai, A; Rotili, D.; Tarantino, D; Ornaghi, P; Tosi, F; Vicidomini, C; Sbardella, G; Nebbioso, A; Miceli, M; Altucci, L; Filetici, P
Synthesis and biological properties of novel, uracil-containing histone deacetylase inhibitors
2006 Mai, Antonello; Silvio, Massa; Rotili, Dante; Silvia, Simeoni; Ragno, Rino; Giorgia, Botta; Angela, Nebbioso; Marco, Miceli; Lucia, Altucci; Gerald, Brosch
One-Pot, High Yielding Synthesis of Novel Dihydrothiazolo[3,2-a]pyrimidinones
2006 Rotili, Dante; Mai, Antonello; Ambrogio, I; G., Fabrizi
Identification of small molecules inhibitors of GCN5 histone acetyltransferase activity
2006 Mai, Antonello; Rotili, Dante; Ornaghi, P; Tosi, F; Vicidomini, C; Sbardella, G; Nebbioso, A; Altucci, L; Filetici, P.
6-Alkylthio-4-[1-(2,6-difluorophenyl)alkyl]-1H-[1,3,5]triazin-2-ones (ADATs): Novel Regulators of Cell Differentiation and Proliferation
2006 Sbardella, G; Bartolini, S; Castellano, S; Artico, Marino; Paesano, N; Rotili, Dante; Spadafora, C; Mai, Antonello
Docking and 3-D QSAR Studies on SIRT2 Inhibitors: A GRID/GOLPE Approach on Different Series of Compounds.
2007 Ragno, Rino; Mai, Antonello; Simeoni, Silvia; Caroli, Antonia; Rotili, Dante; Botta, Giorgia
Slow-, tight-binding HIV-1 reverse transcriptase non-nucleoside inhibitors highly active against drug-resistant mutants
2007 Reynel, Cancio; Mai, Antonello; Rotili, Dante; Marino, Artico; Gianluca, Sbardella; Imma Clotet, Codina; José a, Este; Emmanuele, Crespan; Samantha, Zanoli; Ulrich, Hubscher; Silvio, Spadari; Giovanni, Maga
Histone deacetylase inhibitors may reduce pathogenicity and virulence in Candida albicans
2007 Simonetti, Giovanna; Passariello, Claudio; Rotili, Dante; Mai, Antonello; Enrico, Garaci; Palamara, ANNA TERESA
Discovery of uracil-based histone deacetylase inhibitors able to reduce acquired antifungal resistance and trailing growth in Candida albicans
2007 Mai, Antonello; Rotili, Dante; Massa, Silvio; Gerald, Brosch; Simonetti, Giovanna; Passariello, Claudio; Palamara, ANNA TERESA
Novel pyrrole-containing histone deacetylase inhibitors endowed with cytodifferentiation activity
2007 Mai, Antonello; Valente, Sergio; Rotili, Dante; Silvio, Massa; Giorgia, Botta; Gerald, Brosch; Marco, Miceli; Angela, Nebbioso; Lucia, Altucci
Identification of two new synthetic histone deacetylase inhibitors that modulate globin gene expression in erythroid cells from healthy donors and patients with thalassemia
2007 Mai, Antonello; K., Jelicic; Rotili, Dante; A., Di Noia; E., Alfani; Valente, Sergio; L., Altucci; A., Nebbioso; S., Massa; R., Galanello; G., Brosch; A. R., Migliaccio; G., Migliaccio
Synthesis and biological properties of novel 2-aminopyrimidin-4(3H)-ones highly potent against HIV-1 mutant strains
2007 Mai, Antonello; Artico, Marino; Rotili, Dante; Tarantino, Domenico; CLOTET CODINA, I; ARMAND UGÓN, M; Ragno, Rino; Simeoni, S; Sbardella, G; Nawrozkij, M. B.; Samuele, A; Maga, G; Esté, J. A.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Discovery of (Aryloxo propenyl)pyrrolyl Hydroxyamides as Selective Inhibitors of Class IIa Histone Deacetylase Homologue HD1-A | 2003 | Mai, Antonello; Massa, S.; Pezzi, R.; Rotili, Dante; Loidl, P.; Brosch, G. | |
Synthesis and evaluation of sirtinol analogues as yeast Sir2 and human SIRT inhibitors | 2004 | Pezzi, R.; Rotili, D.; Simeoni, S.; Ragno, Rino; Mariotti, FRANCESCA ROMANA; Chiani, Francesco; Camilloni, Giorgio; Massa, S.; Mai, Antonello | |
A novel Gcn5p inhibitor represses cell growth, gene transcription and histone acetylation in budding yeast | 2005 | Prisca, Ornaghi; Rotili, Dante; Gianluca, Sbardella; Mai, Antonello; Patrizia, Filetici | |
Histone Deacetylation in Epigenetics: An Attractive Target for Anticancer Therapy | 2005 | Mai, Antonello; Massa, S; Rotili, Dante; Cerbara, I; Valente, Sergio; Pezzi, R; Simeoni, S; Ragno, Rino | |
6-[1-(2,6-difluorophenyl)ethyl]pyrimidinones antagonize cell proliferation and induce cell differentiation by inhibiting (a nontelomeric) endogenous reverse transcriptase | 2005 | Sara, Bartolini; Mai, Antonello; Artico, Marino; Nicola, Paesano; Rotili, Dante; Corrado, Spadafora; Gianluca, Sbardella | |
Class II (IIa)-selective histone deacetylase inhibitors. 1. Synthesis and biological evaluation of novel (aryloxopropenyl)pyrrolyl hydroxyamides | 2005 | Mai, Antonello; Silvio, Massa; Riccardo, Pezzi; Silvia, Simeoni; Rotili, Dante; Angela, Nebbioso; Annamaria, Scognamiglio; Lucia, Altucci; Peter, Loidl; Gerald, Brosch | |
Exploring the connection unit in the HDAC inhibitor pharmacophore model: Novel uracil-based hydroxamates | 2005 | Mai, Antonello; Silvio, Massa; Rotili, Dante; Riccardo, Pezzi; Patrizia, Bottoni; Roberto, Scatena; Joachim, Meraner; Gerald, Brosch | |
Analytical and semipreparative high performance liquid chromatography separation of stereoisomers of novel 3,4-dihydropyrimidin-4(3H)-one derivatives on the immobilised amylose-based Chiralpack IA chiral stationary phase. | 2006 | Cirilli, R; Ferretti, R; Gallinella, B; LA TORRE, F; Mai, Antonello; Rotili, Dante | |
Small-Molecule Inhibitors of Histone Acetyltransferase Activity: Identification and Biological Properties | 2006 | Mai, A; Rotili, D.; Tarantino, D; Ornaghi, P; Tosi, F; Vicidomini, C; Sbardella, G; Nebbioso, A; Miceli, M; Altucci, L; Filetici, P | |
Synthesis and biological properties of novel, uracil-containing histone deacetylase inhibitors | 2006 | Mai, Antonello; Silvio, Massa; Rotili, Dante; Silvia, Simeoni; Ragno, Rino; Giorgia, Botta; Angela, Nebbioso; Marco, Miceli; Lucia, Altucci; Gerald, Brosch | |
One-Pot, High Yielding Synthesis of Novel Dihydrothiazolo[3,2-a]pyrimidinones | 2006 | Rotili, Dante; Mai, Antonello; Ambrogio, I; G., Fabrizi | |
Identification of small molecules inhibitors of GCN5 histone acetyltransferase activity | 2006 | Mai, Antonello; Rotili, Dante; Ornaghi, P; Tosi, F; Vicidomini, C; Sbardella, G; Nebbioso, A; Altucci, L; Filetici, P. | |
6-Alkylthio-4-[1-(2,6-difluorophenyl)alkyl]-1H-[1,3,5]triazin-2-ones (ADATs): Novel Regulators of Cell Differentiation and Proliferation | 2006 | Sbardella, G; Bartolini, S; Castellano, S; Artico, Marino; Paesano, N; Rotili, Dante; Spadafora, C; Mai, Antonello | |
Docking and 3-D QSAR Studies on SIRT2 Inhibitors: A GRID/GOLPE Approach on Different Series of Compounds. | 2007 | Ragno, Rino; Mai, Antonello; Simeoni, Silvia; Caroli, Antonia; Rotili, Dante; Botta, Giorgia | |
Slow-, tight-binding HIV-1 reverse transcriptase non-nucleoside inhibitors highly active against drug-resistant mutants | 2007 | Reynel, Cancio; Mai, Antonello; Rotili, Dante; Marino, Artico; Gianluca, Sbardella; Imma Clotet, Codina; José a, Este; Emmanuele, Crespan; Samantha, Zanoli; Ulrich, Hubscher; Silvio, Spadari; Giovanni, Maga | |
Histone deacetylase inhibitors may reduce pathogenicity and virulence in Candida albicans | 2007 | Simonetti, Giovanna; Passariello, Claudio; Rotili, Dante; Mai, Antonello; Enrico, Garaci; Palamara, ANNA TERESA | |
Discovery of uracil-based histone deacetylase inhibitors able to reduce acquired antifungal resistance and trailing growth in Candida albicans | 2007 | Mai, Antonello; Rotili, Dante; Massa, Silvio; Gerald, Brosch; Simonetti, Giovanna; Passariello, Claudio; Palamara, ANNA TERESA | |
Novel pyrrole-containing histone deacetylase inhibitors endowed with cytodifferentiation activity | 2007 | Mai, Antonello; Valente, Sergio; Rotili, Dante; Silvio, Massa; Giorgia, Botta; Gerald, Brosch; Marco, Miceli; Angela, Nebbioso; Lucia, Altucci | |
Identification of two new synthetic histone deacetylase inhibitors that modulate globin gene expression in erythroid cells from healthy donors and patients with thalassemia | 2007 | Mai, Antonello; K., Jelicic; Rotili, Dante; A., Di Noia; E., Alfani; Valente, Sergio; L., Altucci; A., Nebbioso; S., Massa; R., Galanello; G., Brosch; A. R., Migliaccio; G., Migliaccio | |
Synthesis and biological properties of novel 2-aminopyrimidin-4(3H)-ones highly potent against HIV-1 mutant strains | 2007 | Mai, Antonello; Artico, Marino; Rotili, Dante; Tarantino, Domenico; CLOTET CODINA, I; ARMAND UGÓN, M; Ragno, Rino; Simeoni, S; Sbardella, G; Nawrozkij, M. B.; Samuele, A; Maga, G; Esté, J. A. |
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