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Titolo Data di pubblicazione Autore(i) File
Epi-drugs in combination with immunotherapy: a new avenue to improve anticancer efficacy 2017 Mazzone, Roberta; Zwergel, Clemens; Mai, Antonello; Valente, Sergio
Towards the development of activity-based probes for detection of lysine-specific demethylase-1 activity. 2017 Ourailidou, Me; Lenoci, A; Zwergel, Clemens; Rotili, Dante; Mai, Antonello; Dekker, F. j. 4.
Pyrazole-based inhibitors of enhancer of zeste homologue 2 induce apoptosis and autophagy in cancer cells 2018 Mellini, Paolo; Marrocco, Biagina; Borovika, Diana; Polletta, Lucia; Carnevale, Ilaria; Saladini, Serena; Stazi, Giulia; Zwergel, Clemens; Trapencieris, Peteris; Ferretti, Elisabetta; Tafani, Marco; Valente, Sergio; Mai, Antonello
Application of small epigenetic modulators in pediatric medulloblastoma 2018 Zwergel, Clemens; Romanelli, Annalisa; Stazi, Giulia; Besharat, Zein Mersini; Catanzaro, Giuseppina; Tafani, Marco; Valente, Sergio; Mai, Antonello
Nucleocytoplasmic export of HDAC5 and SIRT2 downregulation: two epigenetic mechanisms by which antidepressants enhance synaptic plasticity markers 2018 Muñoz-Cobo, I.; Erburu, M. M.; Zwergel, C.; Cirilli, Raffaela; Mai, A.; Valente, S.; Puerta, E.; Tordera, Rosa M.
HDAC1 inhibition by MS-275 in mesothelial cells limits cellular invasion and promotes MMT reversal 2018 Rossi, Lucia; Battistelli, Cecilia; DE TURRIS, Valeria; Noce, Valeria; Zwergel, Clemens; Valente, Sergio; Moioli, Alessandra; Manzione, Andrea; Palladino, Marco; Bordoni, Veronica; Domenici, Alessandro; Mene', Paolo; Mai, Antonello; Tripodi, Marco; Strippoli, Raffaele
Trends of LSD1 inhibitors in viral infections 2018 Zwergel, Clemens; Stazi, Giulia; Mai, Antonello; Valente, Sergio
Effects of class II-selective histone deacetylase inhibitor on neuromuscular function and disease progression in SOD1-ALS mice 2018 Buonvicino, Daniela; Felici, Roberta; Ranieri, GIUSEPPE ANTONIO; Caramelli, Riccardo; Lapucci, Andrea; Cavone, Leonardo; Muzzi, Mirko; Di Pietro, Lorena; Bernardini, Camilla; Zwergel, Clemens; Valente, Sergio; Mai, Antonello; Chiarugi, Alberto
Six years (2012-2018) of researches on catalytic EZH2 inhibitors: the boom of the 2-pyridone compounds 2018 Fioravanti, R; Stazi, G; Zwergel, C; Valente, S; Mai, A.
A quinoline-based DNA methyltransferase inhibitor as a possible adjuvant in osteosarcoma therapy 2018 Manara, Maria Cristina; Valente, Sergio; Cristalli, Camilla; Nicoletti, Giordano; Landuzzi, Lorena; Zwergel, Clemens; Mazzone, Roberta; Stazi, Giulia; Arimondo, Paola B.; Pasello, Michela; Guerzoni, Clara; Picci, Piero; Nanni, Patrizia; Lollini, Pier-Luigi; Mai, Antonello; Scotlandi, Katia
Sirtuins as drug targets 2019 Zwergel, Clemens; Rotili, Dante; Valente, Sergio; Mai, Antonello
Lysine methyltransferases and their inhibitors 2019 Stazi, Giulia; Zwergel, Clemens; Valente, Sergio
Identification of a novel quinoline-based DNA demethylating compound highly potent in cancer cells 2019 Zwergel, Clemens; Schnekenburger, Michael; Sarno, Federica; Battistelli, Cecilia; Manara, Maria Cristina; Stazi, Giulia; Mazzone, Roberta; Fioravanti, Rossella; Gros, Christina; Ausseil, Frédéric; Florean, Cristina; Nebbioso, Angela; Strippoli, Raffaele; Ushijima, Toshikazu; Scotlandi, Katia; Tripodi, Marco; Arimondo, Paola B.; Altucci, Lucia; Diederich, Marc; Mai, Antonello; Valente, Sergio
Acute and chronic neurobehavioral effects of the designer drug and bath salt constituent 3,4-methylenedioxypyrovalerone in the rat 2019 ATEHORTUA MARTINEZ, LUISA ALESSANDRA; Masniere, Cyriaque; Campolongo, Patrizia; Chasseigneaux, Stéphanie; Callebert, Jacques; Zwergel, Clemens; Mai, Antonello; Laplanche, Jean-Louis; Chen, Huixiong; Etheve-Quelquejeu, Mélanie; Mégarbane, Bruno; Benturquia, Nadia
Development of alkyl glycerone phosphate synthase inhibitors: Structure-activity relationship and effects on ether lipids and epithelial-mesenchymal transition in cancer cells 2019 Stazi, Giulia; Battistelli, Cecilia; Piano, Valentina; Mazzone, Roberta; Marrocco, Biagina; Marchese, Sara; Louie, Sharon M.; Zwergel, Clemens; Antonini, Lorenzo; Patsilinakos, Alexandros; Ragno, Rino; Viviano, Monica; Sbardella, Gianluca; Ciogli, Alessia; Fabrizi, Giancarlo; Cirilli, Roberto; Strippoli, Raffaele; Marchetti, Alessandra; Tripodi, Marco; Nomura, Daniel K.; Mattevi, Andrea; Mai, Antonello; Valente, Sergio
Epigenetic Pharmacology in Regenerative Medicine (Epi-Drugs) 2019 Stazi, Giulia; Zwergel, Clemens; Valente, Sergio; Mai, Antonello
Amphetamine and the Smart Drug 3,4-Methylenedioxypyrovalerone (MDPV) Induce Generalization of Fear Memory in Rats 2019 Colucci, Paola; Mancini, Giulia Federica; Santori, Alessia; Zwergel, Clemens; Mai, Antonello; Trezza, Viviana; Roozendaal, Benno; Campolongo, Patrizia
The emerging role of epigenetics in human autoimmune disorders 2019 Mazzone, Roberta; Zwergel, Clemens; Artico, Marco; Taurone, Samanta; Ralli, Massimo; Greco, Antonio; Mai, Antonello
Editorial: chemical innovative approaches in cancer molecular medicine and translational clinical research 2020 Benedetti, Rosaria; Conte, Mariarosaria; Dell'Aversana, Carmela; Hansen, Finn K.; Zwergel, Clemens
Design of first-in-class dual EZH2/HDAC inhibitor: biochemical activity and biological evaluation in cancer cells 2020 Romanelli, Annalisa; Stazi, Giulia; Fioravanti, Rossella; Zwergel, Clemens; Di Bello, Elisabetta; Pomella, Silvia; Perrone, Clara; Battistelli, Cecilia; Strippoli, Raffaele; Tripodi, Marco; del Bufalo, Donatella; Rota, Rossella; Trisciuoglio, Daniela; Mai, Antonello; Valente, Sergio
Mostrati risultati da 21 a 40 di 75
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