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Mostrati risultati da 201 a 238 di 238
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Experimental data based machine learning classification models with predictive ability to select in vitro active antiviral and non-toxic essential oils 2020 Sabatino, M.; Fabiani, M.; Božović, M.; Garzoli, S.; Antonini, L.; Marcocci, M. E.; Palamara, A. T.; De Chiara, G.; Ragno, R.
Potent in vitro activity of citrus aurantium essential oil and vitis vinifera hydrolate against gut yeast isolates from irritable bowel syndrome patients—the right mix for potential therapeutic use 2020 Di Vito, M.; Grazia Bellardi, M.; Sanguinetti, M.; Mondello, F.; Girolamo, A.; Barbanti, L.; Garzoli, S.; Sabatino, M.; Ragno, R.; Vitali, A.; Palucci, I.; Posteraro, B.; Gasbarrini, A.; Maria Prati, G.; Aragona, G.; Mattarelli, P.; Bugli, F.
Antimicrobial essential oil formulation: chitosan coated nanoemulsions for nose to brain delivery 2020 Rinaldi, F.; Oliva, A.; Sabatino, M.; Imbriano, A.; Hanieh, P. N.; Garzoli, S.; Mastroianni, C. M.; De Angelis, M.; Miele, M. C.; Arnaut, M.; Di Timoteo, F.; Marianecci, C.; Ragno, R.; Carafa, M.
Essential oils and their main chemical components: the past 20 years of preclinical studies in melanoma 2020 Di Martile, M.; Garzoli, S.; Ragno, R.; Del Bufalo, D.
Teaching and learning computational drug design: student investigations of 3D quantitative structure–activity relationships through web applications 2020 Ragno, Rino; Esposito, Valeria; Di Mario, Martina; Masiello, Stefano; Viscovo, Marco; Cramer, Richard
Essential oils against bacterial isolates from cystic fibrosis patients by means of antimicrobial and unsupervised machine learning approaches 2020 Ragno, Rino; Papa, Rosanna; Patsilinakos, Alexandros; Vrenna, Gianluca; Garzoli, Stefania; Vanessatuccio, ; Fiscarelli, Ersiliavita; Selan, Laura; Artini, Marco
Human Estrogen Receptor α Antagonists. Part 1: 3-D QSAR-Driven Rational Design of Innovative Coumarin-Related Antiestrogens as Breast Cancer Suppressants through Structure-Based and Ligand-Based Studies 2021 Mihović, Nezrina; Tomašević, Nevena; Matić, Sanja; Mitrović, Marina M; Kostić, Danijela A; Sabatino, Manuela; Antonini, Lorenzo; Ragno, Rino; Mladenović, Milan
Anti-virulence properties of Coridothymus capitatus essential oil against Pseudomonas aeruginosa clinical isolates from cystic fibrosis patients 2021 Vrenna, Gianluca; Artini, Marco; Ragno, Rino; Relucenti, Michela; Vita Fiscarelli, Ersilia; Tuccio Guarna Assanti, Vanessa; Papa, Rosanna; Selan, Laura
First-in-Class Inhibitors of the Ribosomal Oxygenase MINA53 2021 Nowak, R. P.; Tumber, A.; Hendrix, E.; Ansari, M. S. Z.; Sabatino, M.; Antonini, L.; Andrijes, R.; Salah, E.; Mautone, N.; Pellegrini, F. R.; Simelis, K.; Kawamura, A.; Johansson, C.; Passeri, D.; Pellicciari, R.; Ciogli, A.; Del Bufalo, D.; Ragno, R.; Coleman, M. L.; Trisciuoglio, D.; Mai, A.; Oppermann, U.; Schofield, C. J.; Rotili, D.
Antitumor effect of Melaleuca alternifolia essential oil and its main component terpinen-4-ol in combination with target therapy in melanoma models 2021 Di Martile, M.; Garzoli, S.; Sabatino, M.; Valentini, E.; D'Aguanno, S.; Ragno, R.; Del Bufalo, D.
A comparative analysis of punicalagin interaction with PDIA1 and PDIA3 by biochemical and computational approaches 2021 Paglia, G.; Antonini, L.; Cervoni, L.; Ragno, R.; Sabatino, M.; Minacori, M.; Rubini, E.; Altieri, F.
Ligand-based and structure-based studies to develop predictive models for {SARS}-{CoV}-2 main protease inhibitors through the 3d-qsar.com portal 2022 Proia, Eleonora; Ragno, Alessio; Antonini, Lorenzo; Sabatino, Manuela; Mladenović, Milan; Capobianco, Roberto; Ragno, Rino
Inhibition of PKCθ Improves Dystrophic Heart Phenotype and Function in a Novel Model of DMD Cardiomyopathy 2022 Morroni, Jacopo; Schirone, Leonardo; Valenti, Valentina; Zwergel, Clemens; Riera, Carles Sánchez; Valente, Sergio; Vecchio, Daniele; Schiavon, Sonia; Ragno, Rino; Mai, Antonello; Sciarretta, Sebastiano; Lozanoska-Ochser, Biliana; Bouchè, Marina
Essential oils biofilm modulation activity and machine learning analysis on Pseudomonas aeruginosa isolates from cystic fibrosis patients 2022 Artini, M.; Papa, R.; Sapienza, F.; Božovic ́, M.; Vrenna, G.; Tuccio Guarna Assanti, V.; Sabatino, M.; Garzoli, S.; Fiscarelli, E. V.; Ragno, R.; Selan, L.
Targeting the anti-apoptotic Bcl-2 family proteins: Machine learning virtual screening and biological evaluation of new small molecules 2022 Valentini, E.; D'Aguanno, S.; Di Martile, M.; Montesano, C.; Ferraresi, V.; Patsilinakos, A.; Sabatino, M.; Antonini, L.; Chiacchiarini, M.; Valente, S.; Mai, A.; Colotti, G.; Ragno, R.; Trisciuoglio, D.; Del Bufalo, D.
Bovine serum amine oxidase and polyamine analogues: chemical synthesis and biological evaluation integrated with molecular docking and 3-D QSAR studies 2022 Ragno, Rino; Anna, Minarini; Proia, Eleonora; Antonini, Lorenzo; Andrea, Milelli; Vincenzo, Tumiatti; Marco, Fiore; Fino, Pasquale; Rutigliano, Lavinia; Fioravanti, Rossella; Tahara, Tomoaki; Pacella, Elena; Greco, Antonio; Canettieri, Gianluca; Maria Luisa Di Paolo, ; Agostinelli, Enzo
Human Estrogen Receptor Alpha Antagonists, Part 3: 3-D Pharmacophore and 3-D QSAR Guided Brefeldin A Hit-to-Lead Optimization toward New Breast Cancer Suppressants 2022 Kurtanović, Nezrina; Tomašević, Nevena; Matić, Sanja; Proia, Elenora; Sabatino, Manuela; Antonini, Lorenzo; Mladenović, Milan; Ragno, Rino
Development of eco-friendly biocides based on Calamintha nepeta – loaded chitosan nanoparticles to be employed in the conservation of biocolonized cultural heritage materials. 2022 Genova, C.; Lazzara, A.; Ciccola, A.; Ragno, R.; Sapienza, F.; Montesano, C.; Favero, G.; Curini, R.; Masi, A.
Effetto di metaboliti naturali su crescita e sintesi di aflatossine in Aspergillus flavus 2022 Beccaccioli, Marzia; Cecchetti, Valentina; Fratini, ROSITA SILVANA; Ragno, Rino; Reverberi, Massimo
In vivo Antiphytoviral Activity of Essential Oils and Hydrosols From Origanum vulgare, Thymus vulgaris, and Rosmarinus officinalis to Control Zucchini Yellow Mosaic Virus and Tomato Leaf Curl New Delhi Virus in Cucurbita pepo L 2022 Taglienti, A.; Donati, L.; Ferretti, L.; Tomassoli, L.; Sapienza, F.; Sabatino, M.; Di Massimo, G.; Fiorentino, S.; Vecchiarelli, V.; Nota, P.; Ragno, R.
Pinus mugo Essential Oil Impairs STAT3 Activation through Oxidative Stress and Induces Apoptosis in Prostate Cancer Cells 2022 Ashiq Thalappil, Muhammed; Butturini, Elena; Carcereri de Prati, Alessandra; Bettin, Ilaria; Antonini, Lorenzo; Sapienza, FILIPPO UMBERTO; Garzoli, Stefania; Ragno, Rino; Mariotto, Sofia
Human estrogen receptor α antagonists, part 2: Synthesis driven by rational design, in vitro antiproliferative, and in vivo anticancer evaluation of innovative coumarin-related antiestrogens as breast cancer suppressants 2022 Kurtanovic, N.; Tomasevic, N.; Matic, S.; Mitrovic, M. M.; Kostic, D. A.; Sabatino, M.; Antonini, L.; Ragno, R.; Mladenovic, M.
Py-Graph: An Easy-To-Use Interface for Building Graph-Based QSAR Models 2022 Ragno, Alessio; Capobianco, Roberto; Ragno, Rino
Chemical Composition of Various Nepeta cataria Plant Organs’ Methanol Extracts Associated with In Vivo Hepatoprotective and Antigenotoxic Features as well as Molecular Modeling Investigations 2022 Vukić, Milena D.; Vuković, Nenad L.; Mladenović, Milan; Tomašević, Nevena; Matić, Sanja; Stanić, Snežana; Sapienza, FILIPPO UMBERTO; Ragno, Rino; Božović, Mijat; Kačániová, Miroslava
Foeniculum vulgare miller, a new chemotype from Montenegro 2022 Bozovic, M.; Garzoli, S.; Vujovic, S.; Sapienza, F.; Ragno, R.
Transcriptomic and genomic studies classify NKL54 as a histone deacetylase inhibitor with indirect influence on MEF2-dependent transcription 2022 Minisini, Martina; Di Giorgio, Eros; Kerschbamer, Emanuela; Dalla, Emiliano; Faggiani, Massimo; Franforte, Elisa; Meyer-Almes, Franz-Josef; Ragno, Rino; Antonini, Lorenzo; Mai, Antonello; Fiorentino, Francesco; Rotili, Dante; Chinellato, Monica; Perin, Stefano; Cendron, Laura; Weichenberger, Christian X; Angelini, Alessandro; Brancolini, Claudio
Application of Machine Learning algorithms to essential oils to develop classification models of quantitative composition-activity relationship (QCAR) 2023 Astolfi, Roberta; Oliva, Alessandra; Sapienza, Filippo; Ragno, Rino
Sviluppo di nanosistemi sostenibili per l’incapsulamento di oli essenziali e dei loro principi attivi per la conservazione dei beni culturali di origine lignea 2023 Genova, C.; Beccaccioli, M.; Sapienza, F.; Ragno, R.; Reverberi, M.; Favero, G.; Masi, A.
An Undefined Interaction between Polyamines and Heat Shock Proteins Leads to Cellular Protection in Plasmodium falciparum and Proliferating Cells in Various Organisms 2023 Makhoba, Xolani H.; Ragno, Rino; Kaiser, Annette; Agostinelli, Enzo
Molecular Docking Assessment of Cathinones as 5-HT2AR Ligands: Developing of Predictive Structure-Based Bioactive Conformations and Three-Dimensional Structure-Activity Relationships Models for Future Recognition of Abuse Drugs 2023 Tomašević, Nevena; Vujović, Maja; Kostić, Emilija; Ragavendran, Venkatesan; Arsić, Biljana; Matić, Sanja Lj.; Božović, Mijat; Fioravanti, Rossella; Proia, Eleonora; Ragno, Rino; Mladenović, Milan
Essential Oils from Mediterranean Plants Inhibit In Vitro Monocyte Adhesion to Endothelial Cells from Umbilical Cords of Females with Gestational Diabetes Mellitus 2023 Schiavone, Valeria; Tea, Romasco; Di Pietrantonio, Nadia; Garzoli, Stefania; Palmerini, Carola; DI TOMO, Pamela; Pipino, Caterina; Mandatori, Domitilla; Fioravanti, Rossella; Butturini, Elena; Sabatino, Manuela; Pompea Antonia Baldassarre, Maria; Ragno, Rino; Pandolfi, Assunta; Di Pietro, Natalia
Bcl-2 family inhibitors sensitize human cancer models to therapy 2023 Valentini, Elisabetta; Di Martile, Marta; Brignone, Matteo; Di Caprio, Marica; Manni, Isabella; Chiappa, Michela; Sergio, Ilaria; Chiacchiarini, Martina; Bazzichetto, Chiara; Conciatori, Fabiana; D'Aguanno, Simona; D'Angelo, Carmen; Ragno, Rino; Russillo, Michelangelo; Colotti, Gianni; Marchesi, Francesco; Bellone, Maria Laura; Dal Piaz, Fabrizio; Felli, Maria Pia; Damia, Giovanna; Del Bufalo, Donatella
Explainable AI in drug discovery: self-interpretable graph neural network for molecular property prediction using concept whitening 2023 Proietti, Michela; Ragno, Alessio; Rosa, Biagio La; Ragno, Rino; Capobianco, Roberto
In vivo antiphytoviral and aphid repellency activity of essential oils and hydrosols from Mentha suaveolens and Foeniculum vulgare to control zucchini yellow mosaic virus and its vector Aphis gossypii 2023 Taglienti, A.; Donati, L.; Dragone, I.; Ferretti, L.; Gentili, A.; Araniti, F.; Sapienza, F.; Astolfi, R.; Fiorentino, S.; Vecchiarelli, V.; Papalini, C.; Ragno, R.; Bertin, S.
Effect of different soil treatments on production and chemical composition of essential oils extracted from Foeniculum vulgare Mill., Origanum vulgare L. and Thymus vulgaris L 2023 Raffo, Antonio; Sapienza, FILIPPO UMBERTO; Astolfi, Roberta; Lombardi, Gabriele; Fraschetti, Caterina; Božović, Mijat; Artini, Marco; Papa, Rosanna; Trecca, Marika; Fiorentino, Simona; Vechiarelli, Valerio; Papalini, Claudia; Selan, Laura; Ragno, Rino
Pyrimidine thioethers: A novel class of antidepressant agents, endowed with anxiolytic, performance enhancing and nootropic activity 2023 Fioravanti, Rossella; Proia, Eleonora; Tyurenkov, Ivan N; Kurkin, Denis V; Bakulin, Dmitry A; Kovalev, Nikolay S; Sheikin, Dmitry S; Kirillov, Ivan A; Nawrozkij, Maxim B; Vernigora, Andrey A; Brunilina, Leila L; Fiorentino, Francesco; Mladenović, Milan; Rotili, Dante; Ragno, Rino
In Vitro Antioxidant and In Vivo Antigenotoxic Features of a Series of 61 Essential Oils and Quantitative Composition–Activity Relationships Modeled through Machine Learning Algorithms 2023 Mladenovic, Milan; Astolfi, Roberta; Tomasevic, Nevena; Matic, Sanja; Bozovic, Mijat; Sapienza, FILIPPO UMBERTO; Ragno, Rino
Chemical Composition and Anti-Candida Activity of Mentha suaveolens Ehrh. Essential Oils Obtained by Different Distillation Processes 2023 Tadic, V.; Bozovic, M.; Sapienza, F.; Astolfi, R.; Mladenovic, M.; Zaka, M. C.; Del Bove, F.; Borzacchi, F.; Fraschetti, C.; Rossi, C.; Vertuani, S.; Baldisserotto, A.; Manfredini, S.; Ragno, R.
Mostrati risultati da 201 a 238 di 238
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