Sfoglia per Autore BIAVA, Mariangela
Direct-Acting Antivirals and Host-Targeting Approaches against Enterovirus B Infections: Recent Advances
2023 Tammaro, Chiara; Guida, Michela; Appetecchia, Federico; Biava, Mariangela; Consalvi, Sara; Poce, Giovanna
Antiviral Mechanisms of N-Phenyl Benzamides on Coxsackie Virus A9
2023 Laajala, Mira; Kalander, Kerttu; Consalvi, Sara; Sheik Amamuddy, Olivier; Tastan Bishop, Özlem; Biava, Mariangela; Poce, Giovanna; Marjomäki, Varpu
Malaria transmission blocking compounds: a patent review
2022 Consalvi, Sara; Tammaro, Chiara; Appetecchia, Federico; Biava, Mariangela; Poce, Giovanna
Nano-Based Drug Delivery Systems of Potent MmpL3 Inhibitors for Tuberculosis Treatment
2022 Hanieh, P. N.; Consalvi, S.; Forte, J.; Cabiddu, G.; De Logu, A.; Poce, G.; Rinaldi, F.; Biava, M.; Carafa, M.; Marianecci, C.
Therapeutic potential for coxibs-nitric oxide releasing hybrids in cystic fibrosis
2021 Consalvi, S.; Poce, G.; Ghelardini, C.; Di Cesare Mannelli, L.; Patrignani, P.; Bruno, A.; Anzini, M.; Calderone, V.; Martelli, A.; Testai, L.; Giordani, A.; Biava, M.
Dietary flavonoids: Nano delivery and nanoparticles for cancer therapy
2021 Aiello, Paola; Consalvi, Sara; Poce, Giovanna; Raguzzini, Anna; Toti, Elisabetta; Palmery, Maura; Biava, Mariangela; Bernardi, Marco; Kamale, Mohammad A.; Perry, George; Peluso, Ilaria
6-Fluorophenylbenzohydrazides inhibit Mycobacterium tuberculosis growth through alteration of tryptophan biosynthesis
2021 Consalvi, S.; Venditti, G.; Zhu, J.; Boshoff, H. I.; Arora, K.; De Logu, A.; Ioerger, T. R.; Rubin, E. J.; Biava, M.; Poce, G.
Metabolomic profiling of fresh goji (Lycium barbarum l.) berries from two cultivars grown in central italy: A multi-methodological approach
2021 Spano, M.; Maccelli, A.; Di Matteo, G.; Ingallina, C.; Biava, M.; Crestoni, M. E.; Bardaud, J. -X.; Giusti, A. M.; Mariano, A.; Scotto D'abusco, A.; Sobolev, A. P.; Lasalvia, A.; Fornarini, S.; Mannina, L.
A novel class of dual-acting DCH-CORMs counteracts oxidative stress-induced inflammation in human primary tenocytes
2021 Appetecchia, F.; Consalvi, S.; Berrino, E.; Gallorini, M.; Granese, A.; Campestre, C.; Carradori, S.; Biava, M.; Poce, G.
Overcoming drug resistance in TB: an update
2020 Consalvi, S.; Poce, G.; Scarpecci, C.; Biava, M.
Sar analysis of small molecules interfering with energy-metabolism in mycobacterium tuberculosis
2020 Appetecchia, F.; Consalvi, S.; Scarpecci, C.; Biava, M.; Poce, G.
Novel pyrazole-containing compounds active against mycobacterium tuberculosis
2019 Poce, Giovanna; Consalvi, Sara; Venditti, Giulia; Alfonso, Salvatore; Desideri, Nicoletta; Fernandez-Menendez, Raquel; Bates, Robert H.; Ballell, Lluis; Barros Aguirre, David; Rullas, Joaquin; De Logu, Alessandro; Gardner, Michelle; Ioerger, Thomas R.; Rubin, Eric J.; Biava, Mariangela
Development of MmpL3 inhibitors for tuberculosis treatment
2019 Poce, Giovanna; Consalvi, Sara; Venditti, Giulia; Scarpecci, Cristina; Biava, Mariangela
Neutrophil-to-lymphocyte ratio, mediterranean diet, and bone health in coeliac disease patients: a pilot Study
2019 Palmacci, Francesca; Toti, Elisabetta; Raguzzini, Anna; Catasta, Giovina; Aiello, Paola; Peluso, Ilaria; Biava, Mariangela; Palmery, Maura
Chocolate consumers and lymphocyte-to-monocyte ratio: a working hypothesis from a preliminary report of a pilot study in celiac subjects
2019 Raguzzini, A; Poce, G; Consalvi, S; Toti, E; Palmacci, F; Biava, M; Peluso, I
Mycobacterial tryptophan biosynthesis: a promising target for tuberculosis drug development?
2019 Consalvi, Sara; Scarpecci, Cristina; Biava, Mariangela; Poce, Giovanna
Introduction to COX inhibitors
2018 Biava, Mariangela
In vitro comprehensive analysis of VA692 a new chemical entity for the treatment of osteoarthritis
2018 Cheleschi, Sara; Calamia, Valentina; Fernandez-Moreno, Mercedes; Biava, Mariangela; Giordani, Antonio; Fioravanti, Antonella; Anzini, Maurizio; Blanco, Francisco
In vivo potent BM635 analogue with improved drug-like properties
2018 Poce, Giovanna; Cocozza, Martina; Alfonso, Salvatore; Consalvi, Sara; Venditti, Giulia; Fernandez-Menendez, Raquel; Bates, Robert H.; Barros Aguirre, David; Ballell, Lluis; De Logu, Alessandro; Vistoli, Giulio; Biava, Mariangela
Pharmaceutical salt of BM635 with improved bioavailability
2017 Poce, Giovanna; Consalvi, Sara; Cocozza, Martina; Fernandez Menendez, Raquel; Bates, Robert H.; Ortega Muro, Fátima; Barros Aguirre, David; Ballell, Lluis; Biava, Mariangela
1,5-Diarylpyrroles as potent antitubercular and anti-inflammatory agents
2017 Venditti, Giulia; Poce, Giovanna; Consalvi, Sara; Biava, Mariangela
A series of COX-2 inhibitors endowed with NO-releasing properties: synthesis, biological evaluation, and docking analysis
2016 Consalvi, Sara; Poce, Giovanna; Ragno, Rino; Sabatino, Manuela; Lamotta, Concettina; Sartini, Stefania; Calderone, Vincenzo; Martelli, Alma; Ghelardini, Carla; Dicesaremannelli, Lorenzo; Biava, Mariangela
Synthesis and biological evaluation of fluorinated 1,5-diarylpyrrole-3-alkoxyethyl ether derivatives as selective COX-2 inhibitors endowed with anti-inflammatory activity
2016 Di Capua, Angela; Sticozzi, Claudia; Brogi, Simone; Brindisi, Margherita; Cappelli, Andrea; Sautebin, Lidia; Rossi, Antonietta; Pace, Simona; Ghelardini, Carla; Di Cesare Mannelli, Lorenzo; Valacchi, Giuseppe; Giorgi, Gianluca; Giordani, Antonio; Poce, Giovanna; Biava, Mariangela; Anzini, Maurizio
MmpL3 inhibitors: diverse chemical scaffolds inhibit the same target
2016 Poce, Giovanna; Consalvi, Sara; Biava, Mariangela
Novel inhibitors of Mycobacterium tuberculosis tryptophan biosynthetic pathway to treat tuberculosis
2016 Venditti, Giulia; Consalvi, Sara; Helena, Boshoff; Biava, Mariangela; Poce, Giovanna
(E)-3-Heteroarylidenechroman-4-ones as potent and selective monoamine oxidase-B inhibitors
2016 Desideri, Nicoletta; PROIETTI MONACO, Luca; Fioravanti, Rossella; Biava, Mariangela; Yáñez, Matilde; Alcaro, Stefano; Ortuso, Francesco
COX inhibitors: a patent review (2011 - 2014)
2015 Consalvi, Sara; Biava, Mariangela; Poce, Giovanna
Chondroprotective effect of three different classes of anti-inflammatory agents on human osteoarthritic chondrocytes exposed to IL-1β
2015 Cheleschi, Sara; Pascarelli, Nicola Antonio; Valacchi, Giuseppe; Di Capua, Angela; Biava, Mariangela; Belmonte, Giuseppe; Giordani, Antonio; Sticozzi, Claudia; Anzini, Maurizio; Fioravanti, Antonella
N-((1,3-diphenyl-1H-pyrazol-4-yl)methyl)anilines: a novel class of anti-RSV agents
2015 Fioravanti, Rossella; Desideri, Nicoletta; Biava, Mariangela; Droghini, P.; Atzori, ELENA MARIA; Ibba, C.; Collu, G.; Sanna, G.; Delogu, I.; Loddo, R.
Overcoming drug resistance for tuberculosis,
2015 Poce, Giovanna; Biava, Mariangela
Synthesis, biological evaluation and docking analysis of a new series of methylsulfonyl and sulfamoyl acetamides and ethyl acetates as potent COX-2 inhibitors
2015 Consalvi, Sara; Alfonso, Salvatore; Di Capua, Angela; Poce, Giovanna; Pirolli, Adele; Sabatino, Manuela; Ragno, Rino; Anzini, Maurizio; Sartini, Stefania; La Motta, Concettina; Di Cesare Mannelli, Lorenzo; Ghelardini, Carla; Biava, Mariangela
Activity of lipophilic and hydrophilic drugs against dormant and replicating mycobacterium tuberculosis
2015 Piccaro, G; Poce, Giovanna; Biava, Mariangela; Giannoni, F; Fattorini, L.
A novel antimycobacterial compound acts as an intracellular iron chelator
2015 Dragset Marte, S; Poce, Giovanna; Alfonso, Salvatore; Padilla Benavides, T; Ioerger, T. R.; Kaneko, T; Sacchettini, Jc; Biava, Mariangela; Parish, T; Argüello, Jm; Steigedal, M; Rubin, Ej
Enhancing the pharmacodynamic profile of a class of selective COX-2 inhibiting nitric oxide donors
2014 Biava, Mariangela; Battilocchio, Claudio; Poce, Giovanna; Alfonso, Salvatore; Consalvi, Sara; Angela Di, Capua; Vincenzo, Calderone; Alma, Martelli; Lara, Testai; Lidia, Sautebin; Antonietta, Rossi; Carla, Ghelardini; Lorenzo Di Cesare, Mannelli; Antonio, Giordani; Stefano, Persiani; Milena, Colovic; Melania, Dovizio; Paola, Patrignani; Maurizio, Anzini
SAR analysis of new anti-TB drugs currently in pre-clinical and clinical development
2014 Poce, Giovanna; Cocozza, Martina; Consalvi, Sara; Biava, Mariangela
Pharmacophore assessment through 3-D QSAR: evaluation of the predictive ability on new derivatives by the application on a series of antitubercular agents
2013 Friggeri, Laura; Ballante, Flavio; Ragno, Rino; Musmuca, Ira; DE VITA, Daniela; Manetti, F. .; Biava, Mariangela; Scipione, Luigi; DI SANTO, Roberto; Costi, Roberta; Feroci, Marta; Tortorella, Silvano
Characterization of the biotransformation pathways of clomiphene, tamoxifen and toremifene as assessed by LC-MS/(MS) following in vitro and excretion studies
2013 M., Mazzarino; Biava, Mariangela; X., de la Torre; I., Fiacco; Botre', Francesco
Inhibition of Leishmania infantum trypanothione reductase by azole-based compounds: a comparative analysis with its physiological substrate by X-ray crystallography
2013 Baiocco, P.; Poce, Giovanna; Alfonso, Salvatore; Cocozza, Martina; Porretta, Giulio Cesare; Colotti, G.; Biava, Mariangela; Moraca, F.; Botta, M.; Yardley, V.; Fiorillo, A.; Lantella, A.; Malatesta, Francesco; Ilari, Andrea
Antiproliferative effect of two novel COX-2 inhibitors on human keratinocytes
2013 Claudia, Sticozzi; Belmonte, ; G., Cervellati; F., Di Capua; A., Maioli; E., Cappelli; Antonio, Giordani; Biava, Mariangela; Anzini, ; M., Valacchi
1,5-Diphenylpenta-2,4-dien-1-ones as potent and selective monoamine oxidase-B inhibitors
2013 Desideri, Nicoletta; Fioravanti, Rossella; PROIETTI MONACO, Luca; Biava, Mariangela; Yàñez, M; Ortuso, F; Alcaro, S.
An alternative synthetic approach for the synthesis of biologically relevant 1,4-disubstituted pyrazolo[3,4-d]pyrimidines
2013 Marco, Radi; Vincenzo, Bernardo; Giulia, Vignaroli; Annalaura, Brai; Biava, Mariangela; Silvia, Schenone; Maurizio, Botta
The novel anti-inflammatory agent VA694, endowed with both NO-releasing and COX2-selective inhibiting properties, exhibits NO-mediated positive effects on blood pressure, coronary flow and endothelium in an experimental model of hypertension and endothelial dysfunction
2013 Martelli, A; Testai, L; Anzini, M; Cappelli, A; Di Capua, A; Biava, Mariangela; Poce, Giovanna; Consalvi, Sara; Giordani, A; Caselli, G; Rovati, L; Ghelardini, C; Patrignani, P; Sautebin, L; Breschi, Mc; Calderone, V.
Improving the solubility and the biological profile of a novel class of derivatives as selective COX-2 inhibiting nitric oxide donors
2013 Consalvi, Sara; G., Poce; Alfonso, Salvatore; Battilocchio, Claudio; G. C., Porretta; V., Calderone; A., Martelli; L., Testai; L., Sautebin; A., Rossi; C., Ghelardini; L., Di Cesare Mannelli; A., Giordani; P., Patrignani; M., Anzini; Biava, Mariangela
Novel Analgesic/Anti-inflammatory Agents: 1,5-Diarylpyrrole Nitro-oxyalkyl Ethers and Related Compounds as Cyclooxygenase-2 Inhibiting Nitric Oxide Donors
2013 Anzini, M.; Di Capua, A.; Valenti, S.; Brogi, S.; Rovin, M.; Giuliani, G.; Cappelli, A.; Vomero, S.; Chiasserini, L.; Saga, A.; Poce, Giovanna; Giorgi, G.; Calderone, V.; Martelli, A.; Testai, L.; Sautebin, L.; Rossi, A.; Papa, G.; Ghelardini, C.; Di Cesare Mannelli, L.; Benetti, V.; Giordani, A.; Anzellotti, P.; Dovizio, M.; Patrignani, P.; Biava, Mariangela
A class of pyrrole derivatives endowed with analgesic/anti-inflammatory activity
2013 Battilocchio, Claudio; Poce, Giovanna; Alfonso, Salvatore; Porretta, Giulio Cesare; Consalvi, Sara; L., Sautebin; S., Pace; A., Rossi; C., Ghelardini; L., Di Cesare Mannelli; S., Schenone; A., Giordani; L., Di Francesco; P., Patrignani; Biava, Mariangela
Identification of Hck Inhibitors As Hits for the Development of Antileukemia and Anti-HIV Agents
2013 Cristina, Tintori; Ilaria, Laurenzana; F., La Rocca; Federico, Falchi; Fabio, Carraro; Alba, Ruiz; Jose A., Este; Miroslava, Kissova; Emmanuele, Crespan; Giovanni, Maga; Biava, Mariangela; Chiara, Brullo; Silvia, Schenone; Maurizio, Botta
Flow Synthesis and Bio-Pharmacological Studies of an Adamantane Derivative that Shows Analgesic Activity and Inhibits the P2X7-Evoked Glutamate Release
2013 Battilocchio, Claudio; Guetzoyan, L; Cervetto, C; Di Cesare Mannelli, L; Frattaroli, D; Baxendale, Ir; Maura, G; Rossi, A; Sautebin, L; Biava, Mariangela; Ghelardini, C; Marcoli, M; Ley, Sv
Design, Synthesis, and in vitro hMAO-B Inhibitory Evaluation of Some 1-Methyl-3,5-diphenyl-4,5-dihydro-1H-pyrazoles
2013 Fioravanti, Rossella; Desideri, Nicoletta; Biava, Mariangela; PROIETTI MONACO, Luca; Grammatica, L; Yàñez, M.
New Improved BM212 MmpL3 Inhibitor Analogues: In Vitro and in Vivo Biological Evaluation against Mycobacterium Tuberculosis
2013 Cocozza, Martina; G., Poce; R., Férnandez; R. H., Bates; L., Ballel; Biava, Mariangela
Improved BM212 MmpL3 Inhibitor Analogue Shows Efficacy in Acute Murine Model of Tuberculosis Infection
2013 Poce, Giovanna; H. R., Bates; Alfonso, Salvatore; Cocozza, Martina; Porretta, Giulio Cesare; L., Ballel; Joaquin, Rullas; Alessandro De, Logu; Emanuela, Agus; Valentina La, Rosa; Maria Rosalia, Pasca; Edda De, Rossi; Baojie, Wae; S. J., Franzblau; Fabrizio, Manetti; Maurizio, Botta; Biava, Mariangela
MmpL3 Is the Cellular Target of the Antitubercular Pyrrole Derivative BM212
2012 V., La Rosa; Poce, Giovanna; J., Ortiz Canseco; S., Buroni; M. R., Pasca; Biava, Mariangela; R. M., Raju; Porretta, Giulio Cesare; Alfonso, Salvatore; C., Battilocchio; B., Javid; F., Sorrentino; T. R., Ioerger; J. C., Sacchettini; F., Manetti; M., Botta; A., De Logu; E. J., Rubin
Identification of a new chemical class of potent antimycobacterial compounds derived from BM 212: design, synthesis, biological evaluation and study of their mode of action.
2012 Biava, Mariangela; Poce, Giovanna; Porretta, Giulio Cesare; Alfonso, Salvatore; De Logu, A; De Rossi, E; Ballel, L; Franzblau, S; Manetti, ; Rubin, Ej; Botta, M.
Scale-up of flow-assisted synthesis of C2-symmetric chiral PyBox ligands
2012 Battilocchio, Claudio; Claudio, Baumann; Marcus, Baxendale; R., Ian; Biava, Mariangela; Matthew O., Kitching; Steven V., Ley; Rainer E., Martin; Stephan A., Ohnmacht; Nicholas D. C., Tappin
New 1,5 diarylpyrrole derivatives as antimycobacterial agents: Design, synthesis, biological evaluation and study of their mode of action
2012 Alfonso, Salvatore; Poce, Giovanna; Porretta, Giulio Cesare; Battilocchio, Claudio; Rubin, E. J.; De Rossi, E.; De Logu, A.; Franzblau, S. C.; Botta, M.; Biava, Mariangela
1,5-Diphenyl pyrroles as new antimycobacterial agents. Hit-to-lead development and target validation, New drugs for neglected diseases
2012 Poce, Giovanna; Porretta, Giulio Cesare; De Logu, A; De Rossi, A; Rubin, Ej; Ballel, L; Botta, M; Biava, Mariangela
New Pyrrole Derivatives as Anti-inflammatory and Analgesic Agents: Design, Synthesis and Biological Evaluation
2012 Biava, Mariangela; Consalvi, Sara; Poce, Giovanna; Battilocchio, Claudio; Alfonso, Salvatore; Ghelardini, C.; Sautebin, L.
New 1,5-diphenyl pyrrole derivatives as anti-inflammatory COX-2 selective compounds and their use as potential antitumoral agents.
2012 Consalvi, Sara; Battilocchio, Claudio; Poce, Giovanna; Alfonso, Salvatore; Porretta, Giulio Cesare; M., Anzini; L., Sautebin; C., Ghelardini; A., Giordani; P., Patrignani; V., Calderone; Biava, Mariangela
Analogs of BM 212: a new chemical class of antimycobacterial agents acting upon a new target
2012 Biava, Mariangela; Poce, Giovanna; Porretta, Giulio Cesare; Alfonso, Salvatore; Cocozza, Martina; De Logu, A; De Rossi, E; Ballel, L; Franzblau, S; Rubin E., J; Botta, M.
Flow Based Synthesis of 2-aminoadamantane-2-carboxylic acid
2012 Battilocchio, Claudio; Baxendale, I. R.; Biava, Mariangela; Kitching, Mo; Ley, S. V.
In vitro effects of VA441, a new selective cyclooxygenase-2 inhibitor, on human osteoarthritic chondrocytes exposed to IL-1β
2012 Antonella, Fioravanti; Laura, Tinti; Nicola Antonio, Pascarelli; Angela Di, Capua; Antonello, Lamboglia; Andrea, Cappelli; Biava, Mariangela; Antonio, Giordani; Silvia, Niccolini; Mauro, Galeazzi; Maurizio, Anzini
Improving the solubility of a new class of antiinflammatory pharmacodynamic hybrids, that release nitric oxide and inhibit cycloxygenase-2 isoenzyme
2012 Biava, Mariangela; Battilocchio, Claudio; Poce, Giovanna; Alfonso, Salvatore; Porretta, Giulio Cesare; Consalvi, Sara; Vincenzo, Calderone; Alma, Martelli; Lara, Testai; Carla, Ghelardini; Lorenzo Di Cesare, Mannelli; Lidia, Sautebin; Antonietta, Rossi; Antonio, Giordani; Paola, Patrignani; Maurizio, Anzini
Preparation of 1,5-diaryl-2-alkylpyrrole-3-substituted nitro esters as selective COX-2 inhibitors and nitric oxide donors
2012 Giordani, Antonio; Biava, Mariangela; Anzini, Maurizio; Calderone, Vincenzo; Rovati Lucio, Claudio
New Heterocyclic Compounds Targeting Trypanothyione Metabolism in Leishmania Parasites
2012 Biava, Mariangela; Cocozza, Martina; Poce, Giovanna; Alfonso, Salvatore; Battilocchio, Claudio; Colotti, G.; Malatesta, F.; Baiocco, P.; Ilari, Andrea
Novel Analgesic/Anti-Inflammatory Agents: Diarylpyrrole Acetic Esters Endowed with Nitric Oxide Releasing Properties
2011 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; Alfonso, Salvatore; Michele, Rovini; Salvatore, Valenti; Gianluca, Giorgi; Vincenzo, Calderone; Alma, Martelli; Lara, Testai; Lidia, Sautebin; Antonietta, Rossi; Giuseppina, Papa; Carla, Ghelardini; Lorenzo Di Cesare, Mannelli; Antonio, Giordani; Paola, Anzellotti; Annalisa, Bruno; Paola, Patrignani; Anzini,
Developing Pyrrole-Derived Antimycobacterial Agents: a Rational Lead Optimization Approach
2011 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; Alfonso, Salvatore; A., De Logu; Fabrizio, Manetti; Maurizio, Botta
Pyrrole-based selective COX-2 inhibiting nitric oxide donors: synthesis, in vitro and in vivo evaluation
2011 Battilocchio, Claudio; Porretta, Giulio Cesare; Poce, Giovanna; Alfonso, Salvatore; Calderone, V.; Sautebin, L.; Ghelardini, C.; Giordani, A.; Anzini, M.; Biava, Mariangela
Enlarging the NSAIDs Family: Ether, Ester and Acid Derivatives of the 1,5-Diarylpyrrole Scaffold as Novel Anti-Inflammatory and Analgesic Agents
2011 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; Botta, M; Manetti, F; Rovini, M; Cappelli, A; Sautebin, L; Rossi, A; Pergola, C; Ghelardini, C; Galeotti, N; Makovec, F; Giordani, A; Anzellotti, P; Tacconelli, S; Patrignani, P; Anzini, M.
Synthesis and biological evaluation of new heterocyclic derivatives with potential antimycobacterial activity: systematic approach to lead compound optimization
2011 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Alfonso, Salvatore; Battilocchio, Claudio; De Logu, A; Manetti, F; Botta, M.
New Pyrrole-based selective COX-2 inhibiting nitric oxide donors: synthesis, in vitro and in vivo evaluation
2011 Battilocchio, Claudio; Porretta, Giulio Cesare; Poce, Giovanna; Alfonso, Salvatore; Giordani, A.; Sautebin, L.; Ghelardini, C.; Calderone, V.; Patrignani, P.; Anzini, M.; Biava, Mariangela
Fyn Kinase in Brain Diseases and Cancer: The Search for Inhibitors
2011 S., Schenone; C., Brullo; F., Musumeci; Biava, Mariangela; F., Falchi; M., Botta
Different Metabolic Routes Exhibited by the Nitrooxy-alkyl Chain of NO-Naproxene and a New NO-releasing Coxib Derivative.
2011 Calderone, V.; Martelli, A.; Testai, L.; Arcipreti, A.; Anzini, M.; Di Capua, A.; Biava, Mariangela; Battilocchio, C.; Ghelardini, C.; Giordani, A.; Rovati, L.; Breschi, M. C.
BM212 targets MmpL3, Gordon Research Conference on Tuberculosis Drug Development
2011 Poce, Giovanna; Biava, Mariangela; Porretta, Giulio Cesare; Battilocchio, Claudio; Alfonso, Salvatore; Botta, M.; Javid, B.; Sorrentino, F.; Ioerger, T. R.; Sacchettini, J. R.; Rubin, E.
Derivatives of 1-{[1,5-bis(4-chlorophenyl)-2-methyl-1H-pyrrol-3-yl]methyl}-4-methylpiperazine, synthesis process and uses thereof.
2011 Biava, Mariangela; Botta, M; Deidda, D; Manetti, F; Pompei, R; Porretta, Giulio Cesare
A fast virtual screening approach to identify structurally diverse inhibitors of trypanothione reductase
2011 Maccari, ; G., Jaeger; T., Moraca; Biava, Mariangela; Leopold, Flohe; Botta,
Identification of potent c-Src inhibitors strongly affecting the proliferation of human neuroblastoma cells
2011 Radi, M.; Brullo, C.; Crespan, E.; Tintori, C.; Musumeci, F.; Biava, Mariangela; Schenone, S.; Dreassi, E.; Zamperini, C. .; Maga, G.; Pagano, D.; Angelucci, A.; Bologna, M.; Botta, M.
Cardiovascular effects of a new NO-releasing Coxib derivative
2011 Arcipreti, A.; Martelli, A.; Testai, L.; Breschi, M. C.; Anzini, M.; Di Capua, A.; Biava, Mariangela; Alfonso, Salvatore; Ghelardini, C.; Giordani, A.; Rovati, L.; Calderone, A.
Derivatives of 1-{[1,5-bis(4-chlorophenyl)-2-methyl-1H-pyrrol-3-yl]methyl}-4-methylpiperazine, synthesis process and uses thereof
2011 Biava, Mariangela; Botta, M; Deidda, D; Manetti, F; Pompei, R; Porretta, Giulio Cesare
1,5-Diaryl-Pyrroles as New Generation of Anti-Inflammatory and Analgesic Agents: Design, Synthesis, in vitro and in vivo Evaluation
2010 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Alfonso, S; Battilocchio, Claudio; DE LOGU, A; Manetti, F; Botta, M.
Novel Ester and Acid Derivatives of the 1,5-Diarylpyrrole Scaffold as Anti-inflammatory and Analgesic Agents. Synthesis, in vitro and in vivo Biological Evaluation
2010 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; Manetti, F; Botta, M; Sautebin, L; Rossi, A; Pergola, C; Ghelardini, C; Norcini, M; Makovec, F; Anzellotti, P; Cirilli, R; Ferretti, R; Patrignani, P; Anzini, M.
Pyrrole compounds as inhibitors of mycobacteria, synthesis thereof and intermediates thereto
2010 Biava, Mariangela; Porretta, Giulio Cesare; Pompei, R; Botta, M; Manetti, F; De Logu, A.
New pyrrole derivatives of BM 212: a new class of antimycobacterial agents. Design, synthesis, biological evaluation and study of their mode of action
2010 Biava, Mariangela; Porretta, G. C.; Poce, Giovanna; Alfonso, Salvatore; Battilocchio, Claudio; De Logu, A.; De Rossi, E.; Manetti, F; Botta, M.
BM 579: a novel pyrrole derivative with improved antimycobacterial activity
2010 Biava, Mariangela; Porretta, G. C.; Poce, Giovanna; Alfonso, Salvatore; Battilocchio, Claudio; De Logu, A.; Manetti, F; Botta, M.
Developing New Antiinflammatory and Analgesic Agents: Design, Synthesis, Biological and harmacological Evaluation
2010 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; Alfonso, Salvatore; Botta, M.; Manetti, F.; Sautebin, L; Ghelardini, C; Makovec, F; Giordani, A; Patrignani, P; Anzini, M.
Identification of a novel pyrrole derivative endowed with antimycobacterial activity and protection index comparable to that of the current antitubercular drugs streptomycin and rifampin
2010 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; Alfonso, Salvatore; A., De Logu; Nadia, Serra; Fabrizio, Manetti; Maurizio, Botta
New heterocyclic compounds with potential activity against parasitic protozoan: Trypanosoma and Leishmania
2010 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; V., Yardley; Alfonso, Salvatore
Derivatives of 1-{[1,5-bis(4-chlorophenyl)-2-methyl-1H-pyrrol-3-yl]methyl}-4-methylpiperazine, synthesis process and uses thereof
2010 Biava, Mariangela; Botta, M; Deidda, D; Manetti, F; Pompei, R; Porretta, Giulio Cesare
Identification of a new Chemical Class of Potent Antimycobacterial Compounds
2010 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Alfonso, Salvatore; Battilocchio, Claudio; De Logu, A; Manetti, F; Botta, M.
1,5-Diaryl-2-ethyl pyrrole derivatives as antimycobacterial agents: design, synthesis, and microbiological evaluation
2009 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; DE LOGU, A; Saddi, M; Meleddu, R; Manetti, F; DE ROSSI, E; Botta, M.
Pyrrole derivatives of BM212 as novel antimycobacterial agents Design, synthesis, biological evaluation and study of their mode of action
2009 Biava, Mariangela; Porretta, Giulio Cesare; Battilocchio, Claudio; Poce, G; Pompei, R; DE LOGU, A; Manetti, F; Botta, M.
New pyrrole derivatives of BM 212: a new class of antimycobacterial agents.Design, synthesis, biological evaluation and study of their mode of action.
2009 Biava, Mariangela; Porretta, G. C.; Poce, G; DE LOGU, A; Manetti, F; Botta, M.
Derivatives of BM 212: synthesis and biological evaluation of new derivatives with improved antimycobacterial activity.
2009 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Pompei, R; DE LOGU, A; Manetti, F; Botta, M.
Pyrrole compounds as inhibitors of mycobacteria, synthesis thereof and intermediates thereto
2009 Biava, Mariangela; Porretta, Giulio Cesare; Pompei, R; Botta, M; Manetti, F; DE LOGU, A.
Potent in vitro and in vivo novel 1,5-Diarylpyrrole-3-acetic Esters COX-2 inhibitors.
2009 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Sautebin, L; Patrignani, P; Ghelardini, C; Giordani, A; Anzini, M.
BM212 and its derivatives: lead optimization of a new class of antimycobacterial agents.
2009 Poce, Giovanna; Porretta, Giulio Cesare; DE LOGU, A; DE ROSSI, E; Manetti, F; Botta, M; Biava, Mariangela
C-9 Alkenylidine bridged macrolides: WO2008061189.
2009 Poce, Giovanna; Porretta, Giulio Cesare; Biava, Mariangela
New pyrrole derivatives of BM 212: lead compound optimization strategy, Tuberculosis drug development. Targets, technologies and trials
2009 Poce, Giovanna; Porretta, Giulio Cesare; Borzi, F; DE LOGU, A; DE ROSSI, E; Manetti, F; Botta, M; Biava, Mariangela
Pyrrole compounds as inhibitors of mycobacteria, synthesis thereof and intermediates thereto
2009 Biava, Mariangela; Porretta, Giulio Cesare; Pompei, R; Botta, M; Manetti, F; De Logu, A.
Synthesis, Biological evaluation, and enzyme docking simulations of 1,5-diarylpyrrole-3-alkoxyethyl ethers as selective cyclooxygenase-2 inhibitors endowed with anti-inflammatory and antinociceptive activity
2008 Rovini, M; Cappelli, A; Vomero, S; Manetti, F; Botta, M; Sautebin, L; Rossi, A; Pergola, C; Ghelardini, C; Norcini, M; Goprdani, A; Makovec, F; Anzellotti, P; Patrignani, P; Biava, Mariangela; Anzini, M.
3-substituted-1,5-diaryl-2-alkyl-pyrroles highly selective and orally effective COX-2 inhibitors.
2008 Cappelli, A; Anzini, M; Biava, Mariangela; Makovec, F; Giordani, A; Caselli, G; Rovati, Lc
Design and synthesis of 1,5-diaryl-2-ethyl pyrrole derivatives and their evaluation as antimycobacterial agents
2008 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; DE LOGU, A; Maleddu, R; DE ROSSI, E; Manetti, F; Botta, M.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Direct-Acting Antivirals and Host-Targeting Approaches against Enterovirus B Infections: Recent Advances | 2023 | Tammaro, Chiara; Guida, Michela; Appetecchia, Federico; Biava, Mariangela; Consalvi, Sara; Poce, Giovanna | |
Antiviral Mechanisms of N-Phenyl Benzamides on Coxsackie Virus A9 | 2023 | Laajala, Mira; Kalander, Kerttu; Consalvi, Sara; Sheik Amamuddy, Olivier; Tastan Bishop, Özlem; Biava, Mariangela; Poce, Giovanna; Marjomäki, Varpu | |
Malaria transmission blocking compounds: a patent review | 2022 | Consalvi, Sara; Tammaro, Chiara; Appetecchia, Federico; Biava, Mariangela; Poce, Giovanna | |
Nano-Based Drug Delivery Systems of Potent MmpL3 Inhibitors for Tuberculosis Treatment | 2022 | Hanieh, P. N.; Consalvi, S.; Forte, J.; Cabiddu, G.; De Logu, A.; Poce, G.; Rinaldi, F.; Biava, M.; Carafa, M.; Marianecci, C. | |
Therapeutic potential for coxibs-nitric oxide releasing hybrids in cystic fibrosis | 2021 | Consalvi, S.; Poce, G.; Ghelardini, C.; Di Cesare Mannelli, L.; Patrignani, P.; Bruno, A.; Anzini, M.; Calderone, V.; Martelli, A.; Testai, L.; Giordani, A.; Biava, M. | |
Dietary flavonoids: Nano delivery and nanoparticles for cancer therapy | 2021 | Aiello, Paola; Consalvi, Sara; Poce, Giovanna; Raguzzini, Anna; Toti, Elisabetta; Palmery, Maura; Biava, Mariangela; Bernardi, Marco; Kamale, Mohammad A.; Perry, George; Peluso, Ilaria | |
6-Fluorophenylbenzohydrazides inhibit Mycobacterium tuberculosis growth through alteration of tryptophan biosynthesis | 2021 | Consalvi, S.; Venditti, G.; Zhu, J.; Boshoff, H. I.; Arora, K.; De Logu, A.; Ioerger, T. R.; Rubin, E. J.; Biava, M.; Poce, G. | |
Metabolomic profiling of fresh goji (Lycium barbarum l.) berries from two cultivars grown in central italy: A multi-methodological approach | 2021 | Spano, M.; Maccelli, A.; Di Matteo, G.; Ingallina, C.; Biava, M.; Crestoni, M. E.; Bardaud, J. -X.; Giusti, A. M.; Mariano, A.; Scotto D'abusco, A.; Sobolev, A. P.; Lasalvia, A.; Fornarini, S.; Mannina, L. | |
A novel class of dual-acting DCH-CORMs counteracts oxidative stress-induced inflammation in human primary tenocytes | 2021 | Appetecchia, F.; Consalvi, S.; Berrino, E.; Gallorini, M.; Granese, A.; Campestre, C.; Carradori, S.; Biava, M.; Poce, G. | |
Overcoming drug resistance in TB: an update | 2020 | Consalvi, S.; Poce, G.; Scarpecci, C.; Biava, M. | |
Sar analysis of small molecules interfering with energy-metabolism in mycobacterium tuberculosis | 2020 | Appetecchia, F.; Consalvi, S.; Scarpecci, C.; Biava, M.; Poce, G. | |
Novel pyrazole-containing compounds active against mycobacterium tuberculosis | 2019 | Poce, Giovanna; Consalvi, Sara; Venditti, Giulia; Alfonso, Salvatore; Desideri, Nicoletta; Fernandez-Menendez, Raquel; Bates, Robert H.; Ballell, Lluis; Barros Aguirre, David; Rullas, Joaquin; De Logu, Alessandro; Gardner, Michelle; Ioerger, Thomas R.; Rubin, Eric J.; Biava, Mariangela | |
Development of MmpL3 inhibitors for tuberculosis treatment | 2019 | Poce, Giovanna; Consalvi, Sara; Venditti, Giulia; Scarpecci, Cristina; Biava, Mariangela | |
Neutrophil-to-lymphocyte ratio, mediterranean diet, and bone health in coeliac disease patients: a pilot Study | 2019 | Palmacci, Francesca; Toti, Elisabetta; Raguzzini, Anna; Catasta, Giovina; Aiello, Paola; Peluso, Ilaria; Biava, Mariangela; Palmery, Maura | |
Chocolate consumers and lymphocyte-to-monocyte ratio: a working hypothesis from a preliminary report of a pilot study in celiac subjects | 2019 | Raguzzini, A; Poce, G; Consalvi, S; Toti, E; Palmacci, F; Biava, M; Peluso, I | |
Mycobacterial tryptophan biosynthesis: a promising target for tuberculosis drug development? | 2019 | Consalvi, Sara; Scarpecci, Cristina; Biava, Mariangela; Poce, Giovanna | |
Introduction to COX inhibitors | 2018 | Biava, Mariangela | |
In vitro comprehensive analysis of VA692 a new chemical entity for the treatment of osteoarthritis | 2018 | Cheleschi, Sara; Calamia, Valentina; Fernandez-Moreno, Mercedes; Biava, Mariangela; Giordani, Antonio; Fioravanti, Antonella; Anzini, Maurizio; Blanco, Francisco | |
In vivo potent BM635 analogue with improved drug-like properties | 2018 | Poce, Giovanna; Cocozza, Martina; Alfonso, Salvatore; Consalvi, Sara; Venditti, Giulia; Fernandez-Menendez, Raquel; Bates, Robert H.; Barros Aguirre, David; Ballell, Lluis; De Logu, Alessandro; Vistoli, Giulio; Biava, Mariangela | |
Pharmaceutical salt of BM635 with improved bioavailability | 2017 | Poce, Giovanna; Consalvi, Sara; Cocozza, Martina; Fernandez Menendez, Raquel; Bates, Robert H.; Ortega Muro, Fátima; Barros Aguirre, David; Ballell, Lluis; Biava, Mariangela | |
1,5-Diarylpyrroles as potent antitubercular and anti-inflammatory agents | 2017 | Venditti, Giulia; Poce, Giovanna; Consalvi, Sara; Biava, Mariangela | |
A series of COX-2 inhibitors endowed with NO-releasing properties: synthesis, biological evaluation, and docking analysis | 2016 | Consalvi, Sara; Poce, Giovanna; Ragno, Rino; Sabatino, Manuela; Lamotta, Concettina; Sartini, Stefania; Calderone, Vincenzo; Martelli, Alma; Ghelardini, Carla; Dicesaremannelli, Lorenzo; Biava, Mariangela | |
Synthesis and biological evaluation of fluorinated 1,5-diarylpyrrole-3-alkoxyethyl ether derivatives as selective COX-2 inhibitors endowed with anti-inflammatory activity | 2016 | Di Capua, Angela; Sticozzi, Claudia; Brogi, Simone; Brindisi, Margherita; Cappelli, Andrea; Sautebin, Lidia; Rossi, Antonietta; Pace, Simona; Ghelardini, Carla; Di Cesare Mannelli, Lorenzo; Valacchi, Giuseppe; Giorgi, Gianluca; Giordani, Antonio; Poce, Giovanna; Biava, Mariangela; Anzini, Maurizio | |
MmpL3 inhibitors: diverse chemical scaffolds inhibit the same target | 2016 | Poce, Giovanna; Consalvi, Sara; Biava, Mariangela | |
Novel inhibitors of Mycobacterium tuberculosis tryptophan biosynthetic pathway to treat tuberculosis | 2016 | Venditti, Giulia; Consalvi, Sara; Helena, Boshoff; Biava, Mariangela; Poce, Giovanna | |
(E)-3-Heteroarylidenechroman-4-ones as potent and selective monoamine oxidase-B inhibitors | 2016 | Desideri, Nicoletta; PROIETTI MONACO, Luca; Fioravanti, Rossella; Biava, Mariangela; Yáñez, Matilde; Alcaro, Stefano; Ortuso, Francesco | |
COX inhibitors: a patent review (2011 - 2014) | 2015 | Consalvi, Sara; Biava, Mariangela; Poce, Giovanna | |
Chondroprotective effect of three different classes of anti-inflammatory agents on human osteoarthritic chondrocytes exposed to IL-1β | 2015 | Cheleschi, Sara; Pascarelli, Nicola Antonio; Valacchi, Giuseppe; Di Capua, Angela; Biava, Mariangela; Belmonte, Giuseppe; Giordani, Antonio; Sticozzi, Claudia; Anzini, Maurizio; Fioravanti, Antonella | |
N-((1,3-diphenyl-1H-pyrazol-4-yl)methyl)anilines: a novel class of anti-RSV agents | 2015 | Fioravanti, Rossella; Desideri, Nicoletta; Biava, Mariangela; Droghini, P.; Atzori, ELENA MARIA; Ibba, C.; Collu, G.; Sanna, G.; Delogu, I.; Loddo, R. | |
Overcoming drug resistance for tuberculosis, | 2015 | Poce, Giovanna; Biava, Mariangela | |
Synthesis, biological evaluation and docking analysis of a new series of methylsulfonyl and sulfamoyl acetamides and ethyl acetates as potent COX-2 inhibitors | 2015 | Consalvi, Sara; Alfonso, Salvatore; Di Capua, Angela; Poce, Giovanna; Pirolli, Adele; Sabatino, Manuela; Ragno, Rino; Anzini, Maurizio; Sartini, Stefania; La Motta, Concettina; Di Cesare Mannelli, Lorenzo; Ghelardini, Carla; Biava, Mariangela | |
Activity of lipophilic and hydrophilic drugs against dormant and replicating mycobacterium tuberculosis | 2015 | Piccaro, G; Poce, Giovanna; Biava, Mariangela; Giannoni, F; Fattorini, L. | |
A novel antimycobacterial compound acts as an intracellular iron chelator | 2015 | Dragset Marte, S; Poce, Giovanna; Alfonso, Salvatore; Padilla Benavides, T; Ioerger, T. R.; Kaneko, T; Sacchettini, Jc; Biava, Mariangela; Parish, T; Argüello, Jm; Steigedal, M; Rubin, Ej | |
Enhancing the pharmacodynamic profile of a class of selective COX-2 inhibiting nitric oxide donors | 2014 | Biava, Mariangela; Battilocchio, Claudio; Poce, Giovanna; Alfonso, Salvatore; Consalvi, Sara; Angela Di, Capua; Vincenzo, Calderone; Alma, Martelli; Lara, Testai; Lidia, Sautebin; Antonietta, Rossi; Carla, Ghelardini; Lorenzo Di Cesare, Mannelli; Antonio, Giordani; Stefano, Persiani; Milena, Colovic; Melania, Dovizio; Paola, Patrignani; Maurizio, Anzini | |
SAR analysis of new anti-TB drugs currently in pre-clinical and clinical development | 2014 | Poce, Giovanna; Cocozza, Martina; Consalvi, Sara; Biava, Mariangela | |
Pharmacophore assessment through 3-D QSAR: evaluation of the predictive ability on new derivatives by the application on a series of antitubercular agents | 2013 | Friggeri, Laura; Ballante, Flavio; Ragno, Rino; Musmuca, Ira; DE VITA, Daniela; Manetti, F. .; Biava, Mariangela; Scipione, Luigi; DI SANTO, Roberto; Costi, Roberta; Feroci, Marta; Tortorella, Silvano | |
Characterization of the biotransformation pathways of clomiphene, tamoxifen and toremifene as assessed by LC-MS/(MS) following in vitro and excretion studies | 2013 | M., Mazzarino; Biava, Mariangela; X., de la Torre; I., Fiacco; Botre', Francesco | |
Inhibition of Leishmania infantum trypanothione reductase by azole-based compounds: a comparative analysis with its physiological substrate by X-ray crystallography | 2013 | Baiocco, P.; Poce, Giovanna; Alfonso, Salvatore; Cocozza, Martina; Porretta, Giulio Cesare; Colotti, G.; Biava, Mariangela; Moraca, F.; Botta, M.; Yardley, V.; Fiorillo, A.; Lantella, A.; Malatesta, Francesco; Ilari, Andrea | |
Antiproliferative effect of two novel COX-2 inhibitors on human keratinocytes | 2013 | Claudia, Sticozzi; Belmonte, ; G., Cervellati; F., Di Capua; A., Maioli; E., Cappelli; Antonio, Giordani; Biava, Mariangela; Anzini, ; M., Valacchi | |
1,5-Diphenylpenta-2,4-dien-1-ones as potent and selective monoamine oxidase-B inhibitors | 2013 | Desideri, Nicoletta; Fioravanti, Rossella; PROIETTI MONACO, Luca; Biava, Mariangela; Yàñez, M; Ortuso, F; Alcaro, S. | |
An alternative synthetic approach for the synthesis of biologically relevant 1,4-disubstituted pyrazolo[3,4-d]pyrimidines | 2013 | Marco, Radi; Vincenzo, Bernardo; Giulia, Vignaroli; Annalaura, Brai; Biava, Mariangela; Silvia, Schenone; Maurizio, Botta | |
The novel anti-inflammatory agent VA694, endowed with both NO-releasing and COX2-selective inhibiting properties, exhibits NO-mediated positive effects on blood pressure, coronary flow and endothelium in an experimental model of hypertension and endothelial dysfunction | 2013 | Martelli, A; Testai, L; Anzini, M; Cappelli, A; Di Capua, A; Biava, Mariangela; Poce, Giovanna; Consalvi, Sara; Giordani, A; Caselli, G; Rovati, L; Ghelardini, C; Patrignani, P; Sautebin, L; Breschi, Mc; Calderone, V. | |
Improving the solubility and the biological profile of a novel class of derivatives as selective COX-2 inhibiting nitric oxide donors | 2013 | Consalvi, Sara; G., Poce; Alfonso, Salvatore; Battilocchio, Claudio; G. C., Porretta; V., Calderone; A., Martelli; L., Testai; L., Sautebin; A., Rossi; C., Ghelardini; L., Di Cesare Mannelli; A., Giordani; P., Patrignani; M., Anzini; Biava, Mariangela | |
Novel Analgesic/Anti-inflammatory Agents: 1,5-Diarylpyrrole Nitro-oxyalkyl Ethers and Related Compounds as Cyclooxygenase-2 Inhibiting Nitric Oxide Donors | 2013 | Anzini, M.; Di Capua, A.; Valenti, S.; Brogi, S.; Rovin, M.; Giuliani, G.; Cappelli, A.; Vomero, S.; Chiasserini, L.; Saga, A.; Poce, Giovanna; Giorgi, G.; Calderone, V.; Martelli, A.; Testai, L.; Sautebin, L.; Rossi, A.; Papa, G.; Ghelardini, C.; Di Cesare Mannelli, L.; Benetti, V.; Giordani, A.; Anzellotti, P.; Dovizio, M.; Patrignani, P.; Biava, Mariangela | |
A class of pyrrole derivatives endowed with analgesic/anti-inflammatory activity | 2013 | Battilocchio, Claudio; Poce, Giovanna; Alfonso, Salvatore; Porretta, Giulio Cesare; Consalvi, Sara; L., Sautebin; S., Pace; A., Rossi; C., Ghelardini; L., Di Cesare Mannelli; S., Schenone; A., Giordani; L., Di Francesco; P., Patrignani; Biava, Mariangela | |
Identification of Hck Inhibitors As Hits for the Development of Antileukemia and Anti-HIV Agents | 2013 | Cristina, Tintori; Ilaria, Laurenzana; F., La Rocca; Federico, Falchi; Fabio, Carraro; Alba, Ruiz; Jose A., Este; Miroslava, Kissova; Emmanuele, Crespan; Giovanni, Maga; Biava, Mariangela; Chiara, Brullo; Silvia, Schenone; Maurizio, Botta | |
Flow Synthesis and Bio-Pharmacological Studies of an Adamantane Derivative that Shows Analgesic Activity and Inhibits the P2X7-Evoked Glutamate Release | 2013 | Battilocchio, Claudio; Guetzoyan, L; Cervetto, C; Di Cesare Mannelli, L; Frattaroli, D; Baxendale, Ir; Maura, G; Rossi, A; Sautebin, L; Biava, Mariangela; Ghelardini, C; Marcoli, M; Ley, Sv | |
Design, Synthesis, and in vitro hMAO-B Inhibitory Evaluation of Some 1-Methyl-3,5-diphenyl-4,5-dihydro-1H-pyrazoles | 2013 | Fioravanti, Rossella; Desideri, Nicoletta; Biava, Mariangela; PROIETTI MONACO, Luca; Grammatica, L; Yàñez, M. | |
New Improved BM212 MmpL3 Inhibitor Analogues: In Vitro and in Vivo Biological Evaluation against Mycobacterium Tuberculosis | 2013 | Cocozza, Martina; G., Poce; R., Férnandez; R. H., Bates; L., Ballel; Biava, Mariangela | |
Improved BM212 MmpL3 Inhibitor Analogue Shows Efficacy in Acute Murine Model of Tuberculosis Infection | 2013 | Poce, Giovanna; H. R., Bates; Alfonso, Salvatore; Cocozza, Martina; Porretta, Giulio Cesare; L., Ballel; Joaquin, Rullas; Alessandro De, Logu; Emanuela, Agus; Valentina La, Rosa; Maria Rosalia, Pasca; Edda De, Rossi; Baojie, Wae; S. J., Franzblau; Fabrizio, Manetti; Maurizio, Botta; Biava, Mariangela | |
MmpL3 Is the Cellular Target of the Antitubercular Pyrrole Derivative BM212 | 2012 | V., La Rosa; Poce, Giovanna; J., Ortiz Canseco; S., Buroni; M. R., Pasca; Biava, Mariangela; R. M., Raju; Porretta, Giulio Cesare; Alfonso, Salvatore; C., Battilocchio; B., Javid; F., Sorrentino; T. R., Ioerger; J. C., Sacchettini; F., Manetti; M., Botta; A., De Logu; E. J., Rubin | |
Identification of a new chemical class of potent antimycobacterial compounds derived from BM 212: design, synthesis, biological evaluation and study of their mode of action. | 2012 | Biava, Mariangela; Poce, Giovanna; Porretta, Giulio Cesare; Alfonso, Salvatore; De Logu, A; De Rossi, E; Ballel, L; Franzblau, S; Manetti, ; Rubin, Ej; Botta, M. | |
Scale-up of flow-assisted synthesis of C2-symmetric chiral PyBox ligands | 2012 | Battilocchio, Claudio; Claudio, Baumann; Marcus, Baxendale; R., Ian; Biava, Mariangela; Matthew O., Kitching; Steven V., Ley; Rainer E., Martin; Stephan A., Ohnmacht; Nicholas D. C., Tappin | |
New 1,5 diarylpyrrole derivatives as antimycobacterial agents: Design, synthesis, biological evaluation and study of their mode of action | 2012 | Alfonso, Salvatore; Poce, Giovanna; Porretta, Giulio Cesare; Battilocchio, Claudio; Rubin, E. J.; De Rossi, E.; De Logu, A.; Franzblau, S. C.; Botta, M.; Biava, Mariangela | |
1,5-Diphenyl pyrroles as new antimycobacterial agents. Hit-to-lead development and target validation, New drugs for neglected diseases | 2012 | Poce, Giovanna; Porretta, Giulio Cesare; De Logu, A; De Rossi, A; Rubin, Ej; Ballel, L; Botta, M; Biava, Mariangela | |
New Pyrrole Derivatives as Anti-inflammatory and Analgesic Agents: Design, Synthesis and Biological Evaluation | 2012 | Biava, Mariangela; Consalvi, Sara; Poce, Giovanna; Battilocchio, Claudio; Alfonso, Salvatore; Ghelardini, C.; Sautebin, L. | |
New 1,5-diphenyl pyrrole derivatives as anti-inflammatory COX-2 selective compounds and their use as potential antitumoral agents. | 2012 | Consalvi, Sara; Battilocchio, Claudio; Poce, Giovanna; Alfonso, Salvatore; Porretta, Giulio Cesare; M., Anzini; L., Sautebin; C., Ghelardini; A., Giordani; P., Patrignani; V., Calderone; Biava, Mariangela | |
Analogs of BM 212: a new chemical class of antimycobacterial agents acting upon a new target | 2012 | Biava, Mariangela; Poce, Giovanna; Porretta, Giulio Cesare; Alfonso, Salvatore; Cocozza, Martina; De Logu, A; De Rossi, E; Ballel, L; Franzblau, S; Rubin E., J; Botta, M. | |
Flow Based Synthesis of 2-aminoadamantane-2-carboxylic acid | 2012 | Battilocchio, Claudio; Baxendale, I. R.; Biava, Mariangela; Kitching, Mo; Ley, S. V. | |
In vitro effects of VA441, a new selective cyclooxygenase-2 inhibitor, on human osteoarthritic chondrocytes exposed to IL-1β | 2012 | Antonella, Fioravanti; Laura, Tinti; Nicola Antonio, Pascarelli; Angela Di, Capua; Antonello, Lamboglia; Andrea, Cappelli; Biava, Mariangela; Antonio, Giordani; Silvia, Niccolini; Mauro, Galeazzi; Maurizio, Anzini | |
Improving the solubility of a new class of antiinflammatory pharmacodynamic hybrids, that release nitric oxide and inhibit cycloxygenase-2 isoenzyme | 2012 | Biava, Mariangela; Battilocchio, Claudio; Poce, Giovanna; Alfonso, Salvatore; Porretta, Giulio Cesare; Consalvi, Sara; Vincenzo, Calderone; Alma, Martelli; Lara, Testai; Carla, Ghelardini; Lorenzo Di Cesare, Mannelli; Lidia, Sautebin; Antonietta, Rossi; Antonio, Giordani; Paola, Patrignani; Maurizio, Anzini | |
Preparation of 1,5-diaryl-2-alkylpyrrole-3-substituted nitro esters as selective COX-2 inhibitors and nitric oxide donors | 2012 | Giordani, Antonio; Biava, Mariangela; Anzini, Maurizio; Calderone, Vincenzo; Rovati Lucio, Claudio | |
New Heterocyclic Compounds Targeting Trypanothyione Metabolism in Leishmania Parasites | 2012 | Biava, Mariangela; Cocozza, Martina; Poce, Giovanna; Alfonso, Salvatore; Battilocchio, Claudio; Colotti, G.; Malatesta, F.; Baiocco, P.; Ilari, Andrea | |
Novel Analgesic/Anti-Inflammatory Agents: Diarylpyrrole Acetic Esters Endowed with Nitric Oxide Releasing Properties | 2011 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; Alfonso, Salvatore; Michele, Rovini; Salvatore, Valenti; Gianluca, Giorgi; Vincenzo, Calderone; Alma, Martelli; Lara, Testai; Lidia, Sautebin; Antonietta, Rossi; Giuseppina, Papa; Carla, Ghelardini; Lorenzo Di Cesare, Mannelli; Antonio, Giordani; Paola, Anzellotti; Annalisa, Bruno; Paola, Patrignani; Anzini, | |
Developing Pyrrole-Derived Antimycobacterial Agents: a Rational Lead Optimization Approach | 2011 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; Alfonso, Salvatore; A., De Logu; Fabrizio, Manetti; Maurizio, Botta | |
Pyrrole-based selective COX-2 inhibiting nitric oxide donors: synthesis, in vitro and in vivo evaluation | 2011 | Battilocchio, Claudio; Porretta, Giulio Cesare; Poce, Giovanna; Alfonso, Salvatore; Calderone, V.; Sautebin, L.; Ghelardini, C.; Giordani, A.; Anzini, M.; Biava, Mariangela | |
Enlarging the NSAIDs Family: Ether, Ester and Acid Derivatives of the 1,5-Diarylpyrrole Scaffold as Novel Anti-Inflammatory and Analgesic Agents | 2011 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; Botta, M; Manetti, F; Rovini, M; Cappelli, A; Sautebin, L; Rossi, A; Pergola, C; Ghelardini, C; Galeotti, N; Makovec, F; Giordani, A; Anzellotti, P; Tacconelli, S; Patrignani, P; Anzini, M. | |
Synthesis and biological evaluation of new heterocyclic derivatives with potential antimycobacterial activity: systematic approach to lead compound optimization | 2011 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Alfonso, Salvatore; Battilocchio, Claudio; De Logu, A; Manetti, F; Botta, M. | |
New Pyrrole-based selective COX-2 inhibiting nitric oxide donors: synthesis, in vitro and in vivo evaluation | 2011 | Battilocchio, Claudio; Porretta, Giulio Cesare; Poce, Giovanna; Alfonso, Salvatore; Giordani, A.; Sautebin, L.; Ghelardini, C.; Calderone, V.; Patrignani, P.; Anzini, M.; Biava, Mariangela | |
Fyn Kinase in Brain Diseases and Cancer: The Search for Inhibitors | 2011 | S., Schenone; C., Brullo; F., Musumeci; Biava, Mariangela; F., Falchi; M., Botta | |
Different Metabolic Routes Exhibited by the Nitrooxy-alkyl Chain of NO-Naproxene and a New NO-releasing Coxib Derivative. | 2011 | Calderone, V.; Martelli, A.; Testai, L.; Arcipreti, A.; Anzini, M.; Di Capua, A.; Biava, Mariangela; Battilocchio, C.; Ghelardini, C.; Giordani, A.; Rovati, L.; Breschi, M. C. | |
BM212 targets MmpL3, Gordon Research Conference on Tuberculosis Drug Development | 2011 | Poce, Giovanna; Biava, Mariangela; Porretta, Giulio Cesare; Battilocchio, Claudio; Alfonso, Salvatore; Botta, M.; Javid, B.; Sorrentino, F.; Ioerger, T. R.; Sacchettini, J. R.; Rubin, E. | |
Derivatives of 1-{[1,5-bis(4-chlorophenyl)-2-methyl-1H-pyrrol-3-yl]methyl}-4-methylpiperazine, synthesis process and uses thereof. | 2011 | Biava, Mariangela; Botta, M; Deidda, D; Manetti, F; Pompei, R; Porretta, Giulio Cesare | |
A fast virtual screening approach to identify structurally diverse inhibitors of trypanothione reductase | 2011 | Maccari, ; G., Jaeger; T., Moraca; Biava, Mariangela; Leopold, Flohe; Botta, | |
Identification of potent c-Src inhibitors strongly affecting the proliferation of human neuroblastoma cells | 2011 | Radi, M.; Brullo, C.; Crespan, E.; Tintori, C.; Musumeci, F.; Biava, Mariangela; Schenone, S.; Dreassi, E.; Zamperini, C. .; Maga, G.; Pagano, D.; Angelucci, A.; Bologna, M.; Botta, M. | |
Cardiovascular effects of a new NO-releasing Coxib derivative | 2011 | Arcipreti, A.; Martelli, A.; Testai, L.; Breschi, M. C.; Anzini, M.; Di Capua, A.; Biava, Mariangela; Alfonso, Salvatore; Ghelardini, C.; Giordani, A.; Rovati, L.; Calderone, A. | |
Derivatives of 1-{[1,5-bis(4-chlorophenyl)-2-methyl-1H-pyrrol-3-yl]methyl}-4-methylpiperazine, synthesis process and uses thereof | 2011 | Biava, Mariangela; Botta, M; Deidda, D; Manetti, F; Pompei, R; Porretta, Giulio Cesare | |
1,5-Diaryl-Pyrroles as New Generation of Anti-Inflammatory and Analgesic Agents: Design, Synthesis, in vitro and in vivo Evaluation | 2010 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Alfonso, S; Battilocchio, Claudio; DE LOGU, A; Manetti, F; Botta, M. | |
Novel Ester and Acid Derivatives of the 1,5-Diarylpyrrole Scaffold as Anti-inflammatory and Analgesic Agents. Synthesis, in vitro and in vivo Biological Evaluation | 2010 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; Manetti, F; Botta, M; Sautebin, L; Rossi, A; Pergola, C; Ghelardini, C; Norcini, M; Makovec, F; Anzellotti, P; Cirilli, R; Ferretti, R; Patrignani, P; Anzini, M. | |
Pyrrole compounds as inhibitors of mycobacteria, synthesis thereof and intermediates thereto | 2010 | Biava, Mariangela; Porretta, Giulio Cesare; Pompei, R; Botta, M; Manetti, F; De Logu, A. | |
New pyrrole derivatives of BM 212: a new class of antimycobacterial agents. Design, synthesis, biological evaluation and study of their mode of action | 2010 | Biava, Mariangela; Porretta, G. C.; Poce, Giovanna; Alfonso, Salvatore; Battilocchio, Claudio; De Logu, A.; De Rossi, E.; Manetti, F; Botta, M. | |
BM 579: a novel pyrrole derivative with improved antimycobacterial activity | 2010 | Biava, Mariangela; Porretta, G. C.; Poce, Giovanna; Alfonso, Salvatore; Battilocchio, Claudio; De Logu, A.; Manetti, F; Botta, M. | |
Developing New Antiinflammatory and Analgesic Agents: Design, Synthesis, Biological and harmacological Evaluation | 2010 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; Alfonso, Salvatore; Botta, M.; Manetti, F.; Sautebin, L; Ghelardini, C; Makovec, F; Giordani, A; Patrignani, P; Anzini, M. | |
Identification of a novel pyrrole derivative endowed with antimycobacterial activity and protection index comparable to that of the current antitubercular drugs streptomycin and rifampin | 2010 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; Alfonso, Salvatore; A., De Logu; Nadia, Serra; Fabrizio, Manetti; Maurizio, Botta | |
New heterocyclic compounds with potential activity against parasitic protozoan: Trypanosoma and Leishmania | 2010 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; V., Yardley; Alfonso, Salvatore | |
Derivatives of 1-{[1,5-bis(4-chlorophenyl)-2-methyl-1H-pyrrol-3-yl]methyl}-4-methylpiperazine, synthesis process and uses thereof | 2010 | Biava, Mariangela; Botta, M; Deidda, D; Manetti, F; Pompei, R; Porretta, Giulio Cesare | |
Identification of a new Chemical Class of Potent Antimycobacterial Compounds | 2010 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Alfonso, Salvatore; Battilocchio, Claudio; De Logu, A; Manetti, F; Botta, M. | |
1,5-Diaryl-2-ethyl pyrrole derivatives as antimycobacterial agents: design, synthesis, and microbiological evaluation | 2009 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; DE LOGU, A; Saddi, M; Meleddu, R; Manetti, F; DE ROSSI, E; Botta, M. | |
Pyrrole derivatives of BM212 as novel antimycobacterial agents Design, synthesis, biological evaluation and study of their mode of action | 2009 | Biava, Mariangela; Porretta, Giulio Cesare; Battilocchio, Claudio; Poce, G; Pompei, R; DE LOGU, A; Manetti, F; Botta, M. | |
New pyrrole derivatives of BM 212: a new class of antimycobacterial agents.Design, synthesis, biological evaluation and study of their mode of action. | 2009 | Biava, Mariangela; Porretta, G. C.; Poce, G; DE LOGU, A; Manetti, F; Botta, M. | |
Derivatives of BM 212: synthesis and biological evaluation of new derivatives with improved antimycobacterial activity. | 2009 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Pompei, R; DE LOGU, A; Manetti, F; Botta, M. | |
Pyrrole compounds as inhibitors of mycobacteria, synthesis thereof and intermediates thereto | 2009 | Biava, Mariangela; Porretta, Giulio Cesare; Pompei, R; Botta, M; Manetti, F; DE LOGU, A. | |
Potent in vitro and in vivo novel 1,5-Diarylpyrrole-3-acetic Esters COX-2 inhibitors. | 2009 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Sautebin, L; Patrignani, P; Ghelardini, C; Giordani, A; Anzini, M. | |
BM212 and its derivatives: lead optimization of a new class of antimycobacterial agents. | 2009 | Poce, Giovanna; Porretta, Giulio Cesare; DE LOGU, A; DE ROSSI, E; Manetti, F; Botta, M; Biava, Mariangela | |
C-9 Alkenylidine bridged macrolides: WO2008061189. | 2009 | Poce, Giovanna; Porretta, Giulio Cesare; Biava, Mariangela | |
New pyrrole derivatives of BM 212: lead compound optimization strategy, Tuberculosis drug development. Targets, technologies and trials | 2009 | Poce, Giovanna; Porretta, Giulio Cesare; Borzi, F; DE LOGU, A; DE ROSSI, E; Manetti, F; Botta, M; Biava, Mariangela | |
Pyrrole compounds as inhibitors of mycobacteria, synthesis thereof and intermediates thereto | 2009 | Biava, Mariangela; Porretta, Giulio Cesare; Pompei, R; Botta, M; Manetti, F; De Logu, A. | |
Synthesis, Biological evaluation, and enzyme docking simulations of 1,5-diarylpyrrole-3-alkoxyethyl ethers as selective cyclooxygenase-2 inhibitors endowed with anti-inflammatory and antinociceptive activity | 2008 | Rovini, M; Cappelli, A; Vomero, S; Manetti, F; Botta, M; Sautebin, L; Rossi, A; Pergola, C; Ghelardini, C; Norcini, M; Goprdani, A; Makovec, F; Anzellotti, P; Patrignani, P; Biava, Mariangela; Anzini, M. | |
3-substituted-1,5-diaryl-2-alkyl-pyrroles highly selective and orally effective COX-2 inhibitors. | 2008 | Cappelli, A; Anzini, M; Biava, Mariangela; Makovec, F; Giordani, A; Caselli, G; Rovati, Lc | |
Design and synthesis of 1,5-diaryl-2-ethyl pyrrole derivatives and their evaluation as antimycobacterial agents | 2008 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; DE LOGU, A; Maleddu, R; DE ROSSI, E; Manetti, F; Botta, M. |
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