Sfoglia per Autore BERRINO, Emanuela
A Multitarget Approach against Neuroinflammation: Alkyl Substituted Coumarins as Inhibitors of Enzymes Involved in Neurodegeneration
2023 Berrino, E.; Carradori, S.; Carta, F.; Melfi, F.; Gallorini, M.; Poli, G.; Tuccinardi, T.; Fernandez-Bolanos, J. G.; Lopez, O.; Petzer, J. P.; Petzer, A.; Guglielmi, P.; Secci, D.; Supuran, C. T.
Novel Insights on CAI–CORM Hybrids: Evaluation of the CO Releasing Properties and Pain-Relieving Activity of Differently Substituted Coumarins for the Treatment of Rheumatoid Arthritis
2023 Berrino, Emanuela; Micheli, Laura; Carradori, Simone; di Cesare Mannelli, Lorenzo; Guglielmi, Paolo; De Luca, Alessandro; Carta, Fabrizio; Ghelardini, Carla; Secci, Daniela; Supuran, Claudiu T.
Novel Insights on Human Carbonic Anhydrase Inhibitors Based on Coumalic Acid: Design, Synthesis, Molecular Modeling Investigation, and Biological Studies
2022 Pontecorvi, Virginia; Mori, Mattia; Picarazzi, Francesca; Zara, Susi; Carradori, Simone; Cataldi, Amelia; Angeli, Andrea; Berrino, Emanuela; Chimenti, Paola; Ciogli, Alessia; Secci, Daniela; Guglielmi, Paolo; Supuran, Claudiu T.
New 1 H ‐indole‐2,3‐dione 3‐thiosemicarbazones with 3‐sulfamoylphenyl moiety as selective carbonic anhydrase inhibitors
2022 Eraslan‐elma, Pınar; Akdemir, Atilla; Berrino, Emanuela; Bozdağ, Murat; Supuran, Claudiu T.; Karalı, Nilgün
A novel class of dual-acting DCH-CORMs counteracts oxidative stress-induced inflammation in human primary tenocytes
2021 Appetecchia, F.; Consalvi, S.; Berrino, E.; Gallorini, M.; Granese, A.; Campestre, C.; Carradori, S.; Biava, M.; Poce, G.
Dual carbonic anhydrase ix/xii inhibitors and carbon monoxide releasing molecules modulate LPS-mediated inflammation in mouse macrophages
2021 Berrino, E.; Carradori, S.; Angeli, A.; Carta, F.; Supuran, C. T.; Guglielmi, P.; Coletti, C.; Paciotti, R.; Schweikl, H.; Maestrelli, F.; Cerbai, E.; Gallorini, M.
Tetrahydroquinazole-based secondary sulphonamides as carbonic anhydrase inhibitors: synthesis, biological evaluation against isoforms I, II, IV, and IX, and computational studies
2021 Baglini, E; Ravichandran, R; Berrino, E; Salerno, S; Barresi, E; Marini, Am; Viviano, M; Castellano, S; Da Settimo, F; Supuran, Ct; Cosconati, S; Taliani, S.
Amine-and amino acid-based compounds as carbonic anhydrase activators
2021 Angeli, A.; Berrino, E.; Carradori, S.; Supuran, C. T.; Cirri, M.; Carta, F.; Costantino, G.
Zeta-carbonic anhydrases show CS2 hydrolase activity: A new metabolic carbon acquisition pathway in diatoms?
2021 Alterio, V; Langella, E; Buonanno, M; Esposito, D; Nocentini, A; Berrino, E; Bua, S; Polentarutti, M; Supuran, Ct; Monti, Sm; De Simone, G.
Modulating the Efficacy of Carbonic Anhydrase Inhibitors through Fluorine Substitution.
2021 Berrino, E; Michelet, B; Martin-Mingot, A; Carta, F; Supuran, Ct; Thibaudeau, S.
An innovative spectroscopic approach for qualitative and quantitative evaluation of Mb-CO from myoglobin carbonylation reaction through chemometrics methods
2021 Mansoldo, F. R. P.; Berrino, E.; Guglielmi, P.; Carradori, S.; Carta, F.; Secci, D.; Supuran, C. T.; Vermelho, A. B.
Mechanisms of the Antiproliferative and Antitumor Activity of Novel Telomerase-Carbonic Anhydrase Dual-Hybrid Inhibitors
2021 Plyasova, A. A.; Berrino, E.; Khan, I. I.; Veselovsky, A. V.; Pokrovsky, V. S.; Angeli, A.; Ferraroni, M.; Supuran, C. T.; Pokrovskaya, M. V.; Alexandrova, S. S.; Gladilina, Y. A.; Sokolov, N. N.; Hilal, A.; Carta, F.; Zhdanov, D. D.
N-aryl-N′-ureido-O-sulfamates as potent and selective inhibitors of hCA VB over hCA VA: Deciphering the binding mode of new potential agents in mitochondrial dysfunctions
2020 Poli, G.; Bozdag, M.; Berrino, E.; Angeli, A.; Tuccinardi, T.; Carta, F.; Supuran, C. T.
Azidothymidine "clicked" into 1,2,3-Triazoles: First Report on Carbonic Anhydrase-Telomerase Dual-Hybrid Inhibitors
2020 Berrino, E.; Angeli, A.; Zhdanov, D. D.; Kiryukhina, A. P.; Milaneschi, A.; De Luca, A.; Bozdag, M.; Carradori, S.; Selleri, S.; Bartolucci, G.; Peat, T. S.; Ferraroni, M.; Supuran, C. T.; Carta, F.
In silico identification and biological evaluation of antioxidant food components endowed with IX and XII hCA inhibition
2020 Costa, G.; Maruca, A.; Rocca, R.; Ambrosio, F. A.; Berrino, E.; Carta, F.; Mesiti, F.; Salatino, A.; Lanzillotta, D.; Trapasso, F.; Artese, A.; Alcaro, S.; Supuran, C. T.
In Silico-Guided Identification of New Potent Inhibitors of Carbonic Anhydrases Expressed in Vibrio cholerae.
2020 Mancuso, F; De Luca, L; Angeli, A; Berrino, E; Del Prete, S; Capasso, C; Supuran, Ct; Gitto, R.
Bioorganometallic derivatives of 4-hydrazino-benzenesulfonamide as carbonic anhydrase inhibitors: Synthesis, characterization and biological evaluation
2020 Brichet, J; Arancibia, R; Berrino, E; Supuran, Ct.
A Class of Carbonic Anhydrase IX/XII - Selective Carboxylate Inhibitors
2020 Alhameed, Ra; Berrino, E; Almarhoon, Z; El-Faham, A; Supuran, Ct.
New thiopyrimidine-benzenesulfonamide conjugates as selective carbonic anhydrase II inhibitors: synthesis, in vitro biological evaluation, and molecular docking studies.
2020 Abdel-Mohsen, Ht; El Kerdawy, Am; Omar, Ma; Berrino, E; Abdelsamie, As; El Diwani, Hi; Supuran, Ct.
Toxicity evaluation of sulfamides and coumarins that efficiently inhibit human carbonic anhydrases
2020 Aspatwar, A.; Berrino, E.; Bua, S.; Carta, F.; Capasso, C.; Parkkila, S.; Supuran, C. T.
New sulfonamides containing organometallicacylhydrazones: synthesis, characterisation and biological evaluation as inhibitors of human carbonic anhydrases
2019 Huentupil, Y; Peña, L; Novoa, N; Berrino, E; Arancibia, R; Supuran, Ct.
Synthesis and carbonic anhydrase inhibitory properties of novel 4-(2-aminoethyl)benzenesulfonamide-dipeptide conjugates
2019 Küçükbay, Hasan; Buğday, Nesrin; Küçükbay, F. Zehra; Berrino, Emanuela; Bartolucci, Gian Luca; Del Prete, Sonia; Capasso, Clemente; Supuran, Claudiu T.
Carbonic anhydrase inhibitors of different structures dilate pre-contracted porcine retinal arteries
2019 Eysteinsson, T.; Gudmundsdottir, H.; Hardarson, A. O.; Berrino, E.; Selleri, S.; Supuran, C. T.; Carta, F.
Rho-kinase inhibitors in the management of glaucoma
2019 Berrino, E; Supuran, Ct.
Novel approaches for designing drugs that interfere with pH regulation
2019 Berrino, E; Supuran, Ct.
Synthesis and evaluation of carbonic anhydrase inhibitors with carbon monoxide releasing properties for the management of rheumatoid arthritis
2019 Berrino, E.; Milazzo, L.; Micheli, L.; Vullo, D.; Angeli, A.; Bozdag, M.; Nocentini, A.; Menicatti, M.; Bartolucci, G.; Di Cesare Mannelli, L.; Ghelardini, C.; Supuran, C. T.; Carta, F.
Carbonic anhydrase inhibitors for the treatment of epilepsy and obesity
2019 Berrino, E.; Carta, F.
SLC-0111 enaminone analogs, 3/4-(3-aryl-3-oxopropenyl) aminobenzenesulfonamides, as novel selective subnanomolar inhibitors of the tumor-associated carbonic anhydrase isoform IX
2018 Eldehna, Wm; Abo-Ashour, Mf; Berrino, E; Vullo, D; Ghabbour, Ha; Al-Rashood, St; Hassan, Gs; Alkahtani, Hm; Almehizia, Aa; Alharbi, A; Abdel-Aziz, Ha; Supuran, Ct
Inhibition of α-, β-, γ-, and δ-carbonic anhydrases from bacteria and diatoms with N'-aryl-N-hydroxy-ureas
2018 Berrino, E; Bozdag, M; Del Prete, S; Alasmary, Fas; Alqahtani, Ls; Alothman, Z; Capasso, C; Supuran, Ct.
Synthesis of novel benzenesulfamide derivatives with inhibitory activity against human cytosolic carbonic anhydrase I and II and Vibrio cholerae α- and β-class enzymes
2018 Bua, Silvia; Berrino, Emanuela; Del Prete, Sonia; Murthy, Vallabhaneni S; Vijayakumar, Vijayaparthasarathi; Tamboli, Yasinalli; Capasso, Clemente; Cerbai, Elisabetta; Mugelli, Alessandro; Carta, Fabrizio; Supuran, Claudiu T
1,2,4-Trisubstituted imidazolinones with dual carbonic anhydrase and p38 mitogen-activated protein kinase inhibitory activity.
2018 Georgey, Hh; Manhi, Fm; Mahmoud, Wr; Mohamed, Na; Berrino, E; Supuran, Ct.
4-Substituted benzenesulfonamides incorporating bi/tricyclic moieties act as potent and isoform-selective carbonic anhydrase II/IX inhibitors
2018 Salerno, S; Barresi, E; Amendola, G; Berrino, E; Milite, C; Marini, Am; Da Settimo, F; Novellino, E; Supuran, Ct; Cosconati, S; Taliani, S.
Advances in microwave-assisted synthesis and the impact of novel drug discovery
2018 Berrino, E; Supuran, Ct.
Novel sulfamide-containing compounds as selective carbonic anhydrase i inhibitors
2017 Berrino, Emanuela; Bua, Silvia; Mori, Mattia; Botta, Maurizio; Murthy, Vallabhaneni S.; Vijayakumar, Vijayaparthasarathi; Tamboli, Yasinalli; Bartolucci, GIAN LUCA; Mugelli, Alessandro; Cerbai, Elisabetta; Supuran, CLAUDIU TRANDAFIR; Carta, Fabrizio
Novel analogues of Temporin L and their potential therapeutic application
2016 Berrino, E.; Martora, F.; Merlino, F.; Loffredo, MARIA ROSA; Casciaro, Bruno; DI GRAZIA, Antonio; Yousif, A. M.; Di Carluccio, N.; Carotenuto, A.; Galdiero, M.; Novellino, E.; Iovene, M. R.; Mangoni, Maria Luisa; Grieco, P.
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| A Multitarget Approach against Neuroinflammation: Alkyl Substituted Coumarins as Inhibitors of Enzymes Involved in Neurodegeneration | 2023 | Berrino, E.; Carradori, S.; Carta, F.; Melfi, F.; Gallorini, M.; Poli, G.; Tuccinardi, T.; Fernandez-Bolanos, J. G.; Lopez, O.; Petzer, J. P.; Petzer, A.; Guglielmi, P.; Secci, D.; Supuran, C. T. | |
| Novel Insights on CAI–CORM Hybrids: Evaluation of the CO Releasing Properties and Pain-Relieving Activity of Differently Substituted Coumarins for the Treatment of Rheumatoid Arthritis | 2023 | Berrino, Emanuela; Micheli, Laura; Carradori, Simone; di Cesare Mannelli, Lorenzo; Guglielmi, Paolo; De Luca, Alessandro; Carta, Fabrizio; Ghelardini, Carla; Secci, Daniela; Supuran, Claudiu T. | |
| Novel Insights on Human Carbonic Anhydrase Inhibitors Based on Coumalic Acid: Design, Synthesis, Molecular Modeling Investigation, and Biological Studies | 2022 | Pontecorvi, Virginia; Mori, Mattia; Picarazzi, Francesca; Zara, Susi; Carradori, Simone; Cataldi, Amelia; Angeli, Andrea; Berrino, Emanuela; Chimenti, Paola; Ciogli, Alessia; Secci, Daniela; Guglielmi, Paolo; Supuran, Claudiu T. | |
| New 1 H ‐indole‐2,3‐dione 3‐thiosemicarbazones with 3‐sulfamoylphenyl moiety as selective carbonic anhydrase inhibitors | 2022 | Eraslan‐elma, Pınar; Akdemir, Atilla; Berrino, Emanuela; Bozdağ, Murat; Supuran, Claudiu T.; Karalı, Nilgün | |
| A novel class of dual-acting DCH-CORMs counteracts oxidative stress-induced inflammation in human primary tenocytes | 2021 | Appetecchia, F.; Consalvi, S.; Berrino, E.; Gallorini, M.; Granese, A.; Campestre, C.; Carradori, S.; Biava, M.; Poce, G. | |
| Dual carbonic anhydrase ix/xii inhibitors and carbon monoxide releasing molecules modulate LPS-mediated inflammation in mouse macrophages | 2021 | Berrino, E.; Carradori, S.; Angeli, A.; Carta, F.; Supuran, C. T.; Guglielmi, P.; Coletti, C.; Paciotti, R.; Schweikl, H.; Maestrelli, F.; Cerbai, E.; Gallorini, M. | |
| Tetrahydroquinazole-based secondary sulphonamides as carbonic anhydrase inhibitors: synthesis, biological evaluation against isoforms I, II, IV, and IX, and computational studies | 2021 | Baglini, E; Ravichandran, R; Berrino, E; Salerno, S; Barresi, E; Marini, Am; Viviano, M; Castellano, S; Da Settimo, F; Supuran, Ct; Cosconati, S; Taliani, S. | |
| Amine-and amino acid-based compounds as carbonic anhydrase activators | 2021 | Angeli, A.; Berrino, E.; Carradori, S.; Supuran, C. T.; Cirri, M.; Carta, F.; Costantino, G. | |
| Zeta-carbonic anhydrases show CS2 hydrolase activity: A new metabolic carbon acquisition pathway in diatoms? | 2021 | Alterio, V; Langella, E; Buonanno, M; Esposito, D; Nocentini, A; Berrino, E; Bua, S; Polentarutti, M; Supuran, Ct; Monti, Sm; De Simone, G. | |
| Modulating the Efficacy of Carbonic Anhydrase Inhibitors through Fluorine Substitution. | 2021 | Berrino, E; Michelet, B; Martin-Mingot, A; Carta, F; Supuran, Ct; Thibaudeau, S. | |
| An innovative spectroscopic approach for qualitative and quantitative evaluation of Mb-CO from myoglobin carbonylation reaction through chemometrics methods | 2021 | Mansoldo, F. R. P.; Berrino, E.; Guglielmi, P.; Carradori, S.; Carta, F.; Secci, D.; Supuran, C. T.; Vermelho, A. B. | |
| Mechanisms of the Antiproliferative and Antitumor Activity of Novel Telomerase-Carbonic Anhydrase Dual-Hybrid Inhibitors | 2021 | Plyasova, A. A.; Berrino, E.; Khan, I. I.; Veselovsky, A. V.; Pokrovsky, V. S.; Angeli, A.; Ferraroni, M.; Supuran, C. T.; Pokrovskaya, M. V.; Alexandrova, S. S.; Gladilina, Y. A.; Sokolov, N. N.; Hilal, A.; Carta, F.; Zhdanov, D. D. | |
| N-aryl-N′-ureido-O-sulfamates as potent and selective inhibitors of hCA VB over hCA VA: Deciphering the binding mode of new potential agents in mitochondrial dysfunctions | 2020 | Poli, G.; Bozdag, M.; Berrino, E.; Angeli, A.; Tuccinardi, T.; Carta, F.; Supuran, C. T. | |
| Azidothymidine "clicked" into 1,2,3-Triazoles: First Report on Carbonic Anhydrase-Telomerase Dual-Hybrid Inhibitors | 2020 | Berrino, E.; Angeli, A.; Zhdanov, D. D.; Kiryukhina, A. P.; Milaneschi, A.; De Luca, A.; Bozdag, M.; Carradori, S.; Selleri, S.; Bartolucci, G.; Peat, T. S.; Ferraroni, M.; Supuran, C. T.; Carta, F. | |
| In silico identification and biological evaluation of antioxidant food components endowed with IX and XII hCA inhibition | 2020 | Costa, G.; Maruca, A.; Rocca, R.; Ambrosio, F. A.; Berrino, E.; Carta, F.; Mesiti, F.; Salatino, A.; Lanzillotta, D.; Trapasso, F.; Artese, A.; Alcaro, S.; Supuran, C. T. | |
| In Silico-Guided Identification of New Potent Inhibitors of Carbonic Anhydrases Expressed in Vibrio cholerae. | 2020 | Mancuso, F; De Luca, L; Angeli, A; Berrino, E; Del Prete, S; Capasso, C; Supuran, Ct; Gitto, R. | |
| Bioorganometallic derivatives of 4-hydrazino-benzenesulfonamide as carbonic anhydrase inhibitors: Synthesis, characterization and biological evaluation | 2020 | Brichet, J; Arancibia, R; Berrino, E; Supuran, Ct. | |
| A Class of Carbonic Anhydrase IX/XII - Selective Carboxylate Inhibitors | 2020 | Alhameed, Ra; Berrino, E; Almarhoon, Z; El-Faham, A; Supuran, Ct. | |
| New thiopyrimidine-benzenesulfonamide conjugates as selective carbonic anhydrase II inhibitors: synthesis, in vitro biological evaluation, and molecular docking studies. | 2020 | Abdel-Mohsen, Ht; El Kerdawy, Am; Omar, Ma; Berrino, E; Abdelsamie, As; El Diwani, Hi; Supuran, Ct. | |
| Toxicity evaluation of sulfamides and coumarins that efficiently inhibit human carbonic anhydrases | 2020 | Aspatwar, A.; Berrino, E.; Bua, S.; Carta, F.; Capasso, C.; Parkkila, S.; Supuran, C. T. | |
| New sulfonamides containing organometallicacylhydrazones: synthesis, characterisation and biological evaluation as inhibitors of human carbonic anhydrases | 2019 | Huentupil, Y; Peña, L; Novoa, N; Berrino, E; Arancibia, R; Supuran, Ct. | |
| Synthesis and carbonic anhydrase inhibitory properties of novel 4-(2-aminoethyl)benzenesulfonamide-dipeptide conjugates | 2019 | Küçükbay, Hasan; Buğday, Nesrin; Küçükbay, F. Zehra; Berrino, Emanuela; Bartolucci, Gian Luca; Del Prete, Sonia; Capasso, Clemente; Supuran, Claudiu T. | |
| Carbonic anhydrase inhibitors of different structures dilate pre-contracted porcine retinal arteries | 2019 | Eysteinsson, T.; Gudmundsdottir, H.; Hardarson, A. O.; Berrino, E.; Selleri, S.; Supuran, C. T.; Carta, F. | |
| Rho-kinase inhibitors in the management of glaucoma | 2019 | Berrino, E; Supuran, Ct. | |
| Novel approaches for designing drugs that interfere with pH regulation | 2019 | Berrino, E; Supuran, Ct. | |
| Synthesis and evaluation of carbonic anhydrase inhibitors with carbon monoxide releasing properties for the management of rheumatoid arthritis | 2019 | Berrino, E.; Milazzo, L.; Micheli, L.; Vullo, D.; Angeli, A.; Bozdag, M.; Nocentini, A.; Menicatti, M.; Bartolucci, G.; Di Cesare Mannelli, L.; Ghelardini, C.; Supuran, C. T.; Carta, F. | |
| Carbonic anhydrase inhibitors for the treatment of epilepsy and obesity | 2019 | Berrino, E.; Carta, F. | |
| SLC-0111 enaminone analogs, 3/4-(3-aryl-3-oxopropenyl) aminobenzenesulfonamides, as novel selective subnanomolar inhibitors of the tumor-associated carbonic anhydrase isoform IX | 2018 | Eldehna, Wm; Abo-Ashour, Mf; Berrino, E; Vullo, D; Ghabbour, Ha; Al-Rashood, St; Hassan, Gs; Alkahtani, Hm; Almehizia, Aa; Alharbi, A; Abdel-Aziz, Ha; Supuran, Ct | |
| Inhibition of α-, β-, γ-, and δ-carbonic anhydrases from bacteria and diatoms with N'-aryl-N-hydroxy-ureas | 2018 | Berrino, E; Bozdag, M; Del Prete, S; Alasmary, Fas; Alqahtani, Ls; Alothman, Z; Capasso, C; Supuran, Ct. | |
| Synthesis of novel benzenesulfamide derivatives with inhibitory activity against human cytosolic carbonic anhydrase I and II and Vibrio cholerae α- and β-class enzymes | 2018 | Bua, Silvia; Berrino, Emanuela; Del Prete, Sonia; Murthy, Vallabhaneni S; Vijayakumar, Vijayaparthasarathi; Tamboli, Yasinalli; Capasso, Clemente; Cerbai, Elisabetta; Mugelli, Alessandro; Carta, Fabrizio; Supuran, Claudiu T | |
| 1,2,4-Trisubstituted imidazolinones with dual carbonic anhydrase and p38 mitogen-activated protein kinase inhibitory activity. | 2018 | Georgey, Hh; Manhi, Fm; Mahmoud, Wr; Mohamed, Na; Berrino, E; Supuran, Ct. | |
| 4-Substituted benzenesulfonamides incorporating bi/tricyclic moieties act as potent and isoform-selective carbonic anhydrase II/IX inhibitors | 2018 | Salerno, S; Barresi, E; Amendola, G; Berrino, E; Milite, C; Marini, Am; Da Settimo, F; Novellino, E; Supuran, Ct; Cosconati, S; Taliani, S. | |
| Advances in microwave-assisted synthesis and the impact of novel drug discovery | 2018 | Berrino, E; Supuran, Ct. | |
| Novel sulfamide-containing compounds as selective carbonic anhydrase i inhibitors | 2017 | Berrino, Emanuela; Bua, Silvia; Mori, Mattia; Botta, Maurizio; Murthy, Vallabhaneni S.; Vijayakumar, Vijayaparthasarathi; Tamboli, Yasinalli; Bartolucci, GIAN LUCA; Mugelli, Alessandro; Cerbai, Elisabetta; Supuran, CLAUDIU TRANDAFIR; Carta, Fabrizio | |
| Novel analogues of Temporin L and their potential therapeutic application | 2016 | Berrino, E.; Martora, F.; Merlino, F.; Loffredo, MARIA ROSA; Casciaro, Bruno; DI GRAZIA, Antonio; Yousif, A. M.; Di Carluccio, N.; Carotenuto, A.; Galdiero, M.; Novellino, E.; Iovene, M. R.; Mangoni, Maria Luisa; Grieco, P. |
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