Sfoglia per Autore POCE, Giovanna
Tannin microcapsules for synergy-enhanced sunscreen formulations
2023 Alfonsi, E.; Lange, H.; Zongo, L.; Poce, G.; Sgarzi, M.; Crestini, C.
Direct-Acting Antivirals and Host-Targeting Approaches against Enterovirus B Infections: Recent Advances
2023 Tammaro, Chiara; Guida, Michela; Appetecchia, Federico; Biava, Mariangela; Consalvi, Sara; Poce, Giovanna
Antiviral Mechanisms of N-Phenyl Benzamides on Coxsackie Virus A9
2023 Laajala, Mira; Kalander, Kerttu; Consalvi, Sara; Sheik Amamuddy, Olivier; Tastan Bishop, Özlem; Biava, Mariangela; Poce, Giovanna; Marjomäki, Varpu
Nano-Based Drug Delivery Systems of Potent MmpL3 Inhibitors for Tuberculosis Treatment
2022 Hanieh, P. N.; Consalvi, S.; Forte, J.; Cabiddu, G.; De Logu, A.; Poce, G.; Rinaldi, F.; Biava, M.; Carafa, M.; Marianecci, C.
Malaria transmission blocking compounds: a patent review
2022 Consalvi, Sara; Tammaro, Chiara; Appetecchia, Federico; Biava, Mariangela; Poce, Giovanna
A novel class of dual-acting DCH-CORMs counteracts oxidative stress-induced inflammation in human primary tenocytes
2021 Appetecchia, F.; Consalvi, S.; Berrino, E.; Gallorini, M.; Granese, A.; Campestre, C.; Carradori, S.; Biava, M.; Poce, G.
Therapeutic potential for coxibs-nitric oxide releasing hybrids in cystic fibrosis
2021 Consalvi, S.; Poce, G.; Ghelardini, C.; Di Cesare Mannelli, L.; Patrignani, P.; Bruno, A.; Anzini, M.; Calderone, V.; Martelli, A.; Testai, L.; Giordani, A.; Biava, M.
Dietary flavonoids: Nano delivery and nanoparticles for cancer therapy
2021 Aiello, Paola; Consalvi, Sara; Poce, Giovanna; Raguzzini, Anna; Toti, Elisabetta; Palmery, Maura; Biava, Mariangela; Bernardi, Marco; Kamale, Mohammad A.; Perry, George; Peluso, Ilaria
6-Fluorophenylbenzohydrazides inhibit Mycobacterium tuberculosis growth through alteration of tryptophan biosynthesis
2021 Consalvi, S.; Venditti, G.; Zhu, J.; Boshoff, H. I.; Arora, K.; De Logu, A.; Ioerger, T. R.; Rubin, E. J.; Biava, M.; Poce, G.
Sar analysis of small molecules interfering with energy-metabolism in mycobacterium tuberculosis
2020 Appetecchia, F.; Consalvi, S.; Scarpecci, C.; Biava, M.; Poce, G.
Overcoming drug resistance in TB: an update
2020 Consalvi, S.; Poce, G.; Scarpecci, C.; Biava, M.
Development of MmpL3 inhibitors for tuberculosis treatment
2019 Poce, Giovanna; Consalvi, Sara; Venditti, Giulia; Scarpecci, Cristina; Biava, Mariangela
Mycobacterial tryptophan biosynthesis: a promising target for tuberculosis drug development?
2019 Consalvi, Sara; Scarpecci, Cristina; Biava, Mariangela; Poce, Giovanna
Novel therapies for glaucoma: a patent review (2013-2019)
2019 Guglielmi, Paolo; Carradori, Simone; Campestre, Cristina; Poce, Giovanna
Novel pyrazole-containing compounds active against mycobacterium tuberculosis
2019 Poce, Giovanna; Consalvi, Sara; Venditti, Giulia; Alfonso, Salvatore; Desideri, Nicoletta; Fernandez-Menendez, Raquel; Bates, Robert H.; Ballell, Lluis; Barros Aguirre, David; Rullas, Joaquin; De Logu, Alessandro; Gardner, Michelle; Ioerger, Thomas R.; Rubin, Eric J.; Biava, Mariangela
Chocolate consumers and lymphocyte-to-monocyte ratio: a working hypothesis from a preliminary report of a pilot study in celiac subjects
2019 Raguzzini, A; Poce, G; Consalvi, S; Toti, E; Palmacci, F; Biava, M; Peluso, I
In vivo potent BM635 analogue with improved drug-like properties
2018 Poce, Giovanna; Cocozza, Martina; Alfonso, Salvatore; Consalvi, Sara; Venditti, Giulia; Fernandez-Menendez, Raquel; Bates, Robert H.; Barros Aguirre, David; Ballell, Lluis; De Logu, Alessandro; Vistoli, Giulio; Biava, Mariangela
Stimuli-responsive tannin–feIII hybrid microcapsules demonstrated by the active release of an anti-tuberculosis agent
2018 Bartzoka, Elisavet D.; Lange, Heiko; Poce, Giovanna; Crestini, Claudia
MmpL3 is the flippase for mycolic acids in mycobacteria
2017 Xu, Zhujun; Meshcheryakov, Vladimir A.; Poce, Giovanna; Chng, Shu-Sin
Pharmaceutical salt of BM635 with improved bioavailability
2017 Poce, Giovanna; Consalvi, Sara; Cocozza, Martina; Fernandez Menendez, Raquel; Bates, Robert H.; Ortega Muro, Fátima; Barros Aguirre, David; Ballell, Lluis; Biava, Mariangela
1,5-Diarylpyrroles as potent antitubercular and anti-inflammatory agents
2017 Venditti, Giulia; Poce, Giovanna; Consalvi, Sara; Biava, Mariangela
Novel inhibitors of Mycobacterium tuberculosis tryptophan biosynthetic pathway to treat tuberculosis
2016 Venditti, Giulia; Consalvi, Sara; Helena, Boshoff; Biava, Mariangela; Poce, Giovanna
A series of COX-2 inhibitors endowed with NO-releasing properties: synthesis, biological evaluation, and docking analysis
2016 Consalvi, Sara; Poce, Giovanna; Ragno, Rino; Sabatino, Manuela; Lamotta, Concettina; Sartini, Stefania; Calderone, Vincenzo; Martelli, Alma; Ghelardini, Carla; Dicesaremannelli, Lorenzo; Biava, Mariangela
Synthesis and biological evaluation of fluorinated 1,5-diarylpyrrole-3-alkoxyethyl ether derivatives as selective COX-2 inhibitors endowed with anti-inflammatory activity
2016 Di Capua, Angela; Sticozzi, Claudia; Brogi, Simone; Brindisi, Margherita; Cappelli, Andrea; Sautebin, Lidia; Rossi, Antonietta; Pace, Simona; Ghelardini, Carla; Di Cesare Mannelli, Lorenzo; Valacchi, Giuseppe; Giorgi, Gianluca; Giordani, Antonio; Poce, Giovanna; Biava, Mariangela; Anzini, Maurizio
MmpL3 inhibitors: diverse chemical scaffolds inhibit the same target
2016 Poce, Giovanna; Consalvi, Sara; Biava, Mariangela
COX inhibitors: a patent review (2011 - 2014)
2015 Consalvi, Sara; Biava, Mariangela; Poce, Giovanna
Synthesis, biological evaluation and docking analysis of a new series of methylsulfonyl and sulfamoyl acetamides and ethyl acetates as potent COX-2 inhibitors
2015 Consalvi, Sara; Alfonso, Salvatore; Di Capua, Angela; Poce, Giovanna; Pirolli, Adele; Sabatino, Manuela; Ragno, Rino; Anzini, Maurizio; Sartini, Stefania; La Motta, Concettina; Di Cesare Mannelli, Lorenzo; Ghelardini, Carla; Biava, Mariangela
A novel antimycobacterial compound acts as an intracellular iron chelator
2015 Dragset Marte, S; Poce, Giovanna; Alfonso, Salvatore; Padilla Benavides, T; Ioerger, T. R.; Kaneko, T; Sacchettini, Jc; Biava, Mariangela; Parish, T; Argüello, Jm; Steigedal, M; Rubin, Ej
Overcoming drug resistance for tuberculosis,
2015 Poce, Giovanna; Biava, Mariangela
Activity of lipophilic and hydrophilic drugs against dormant and replicating mycobacterium tuberculosis
2015 Piccaro, G; Poce, Giovanna; Biava, Mariangela; Giannoni, F; Fattorini, L.
SAR analysis of new anti-TB drugs currently in pre-clinical and clinical development
2014 Poce, Giovanna; Cocozza, Martina; Consalvi, Sara; Biava, Mariangela
Enhancing the pharmacodynamic profile of a class of selective COX-2 inhibiting nitric oxide donors
2014 Biava, Mariangela; Battilocchio, Claudio; Poce, Giovanna; Alfonso, Salvatore; Consalvi, Sara; Angela Di, Capua; Vincenzo, Calderone; Alma, Martelli; Lara, Testai; Lidia, Sautebin; Antonietta, Rossi; Carla, Ghelardini; Lorenzo Di Cesare, Mannelli; Antonio, Giordani; Stefano, Persiani; Milena, Colovic; Melania, Dovizio; Paola, Patrignani; Maurizio, Anzini
A class of pyrrole derivatives endowed with analgesic/anti-inflammatory activity
2013 Battilocchio, Claudio; Poce, Giovanna; Alfonso, Salvatore; Porretta, Giulio Cesare; Consalvi, Sara; L., Sautebin; S., Pace; A., Rossi; C., Ghelardini; L., Di Cesare Mannelli; S., Schenone; A., Giordani; L., Di Francesco; P., Patrignani; Biava, Mariangela
Inhibition of Leishmania infantum trypanothione reductase by azole-based compounds: a comparative analysis with its physiological substrate by X-ray crystallography
2013 Baiocco, P.; Poce, Giovanna; Alfonso, Salvatore; Cocozza, Martina; Porretta, Giulio Cesare; Colotti, G.; Biava, Mariangela; Moraca, F.; Botta, M.; Yardley, V.; Fiorillo, A.; Lantella, A.; Malatesta, Francesco; Ilari, Andrea
Improved BM212 MmpL3 Inhibitor Analogue Shows Efficacy in Acute Murine Model of Tuberculosis Infection
2013 Poce, Giovanna; H. R., Bates; Alfonso, Salvatore; Cocozza, Martina; Porretta, Giulio Cesare; L., Ballel; Joaquin, Rullas; Alessandro De, Logu; Emanuela, Agus; Valentina La, Rosa; Maria Rosalia, Pasca; Edda De, Rossi; Baojie, Wae; S. J., Franzblau; Fabrizio, Manetti; Maurizio, Botta; Biava, Mariangela
Novel Analgesic/Anti-inflammatory Agents: 1,5-Diarylpyrrole Nitro-oxyalkyl Ethers and Related Compounds as Cyclooxygenase-2 Inhibiting Nitric Oxide Donors
2013 Anzini, M.; Di Capua, A.; Valenti, S.; Brogi, S.; Rovin, M.; Giuliani, G.; Cappelli, A.; Vomero, S.; Chiasserini, L.; Saga, A.; Poce, Giovanna; Giorgi, G.; Calderone, V.; Martelli, A.; Testai, L.; Sautebin, L.; Rossi, A.; Papa, G.; Ghelardini, C.; Di Cesare Mannelli, L.; Benetti, V.; Giordani, A.; Anzellotti, P.; Dovizio, M.; Patrignani, P.; Biava, Mariangela
The novel anti-inflammatory agent VA694, endowed with both NO-releasing and COX2-selective inhibiting properties, exhibits NO-mediated positive effects on blood pressure, coronary flow and endothelium in an experimental model of hypertension and endothelial dysfunction
2013 Martelli, A; Testai, L; Anzini, M; Cappelli, A; Di Capua, A; Biava, Mariangela; Poce, Giovanna; Consalvi, Sara; Giordani, A; Caselli, G; Rovati, L; Ghelardini, C; Patrignani, P; Sautebin, L; Breschi, Mc; Calderone, V.
New Heterocyclic Compounds Targeting Trypanothyione Metabolism in Leishmania Parasites
2012 Biava, Mariangela; Cocozza, Martina; Poce, Giovanna; Alfonso, Salvatore; Battilocchio, Claudio; Colotti, G.; Malatesta, F.; Baiocco, P.; Ilari, Andrea
New 1,5 diarylpyrrole derivatives as antimycobacterial agents: Design, synthesis, biological evaluation and study of their mode of action
2012 Alfonso, Salvatore; Poce, Giovanna; Porretta, Giulio Cesare; Battilocchio, Claudio; Rubin, E. J.; De Rossi, E.; De Logu, A.; Franzblau, S. C.; Botta, M.; Biava, Mariangela
New Pyrrole Derivatives as Anti-inflammatory and Analgesic Agents: Design, Synthesis and Biological Evaluation
2012 Biava, Mariangela; Consalvi, Sara; Poce, Giovanna; Battilocchio, Claudio; Alfonso, Salvatore; Ghelardini, C.; Sautebin, L.
MmpL3 Is the Cellular Target of the Antitubercular Pyrrole Derivative BM212
2012 V., La Rosa; Poce, Giovanna; J., Ortiz Canseco; S., Buroni; M. R., Pasca; Biava, Mariangela; R. M., Raju; Porretta, Giulio Cesare; Alfonso, Salvatore; C., Battilocchio; B., Javid; F., Sorrentino; T. R., Ioerger; J. C., Sacchettini; F., Manetti; M., Botta; A., De Logu; E. J., Rubin
Identification of a new chemical class of potent antimycobacterial compounds derived from BM 212: design, synthesis, biological evaluation and study of their mode of action.
2012 Biava, Mariangela; Poce, Giovanna; Porretta, Giulio Cesare; Alfonso, Salvatore; De Logu, A; De Rossi, E; Ballel, L; Franzblau, S; Manetti, ; Rubin, Ej; Botta, M.
1,5-Diphenyl pyrroles as new antimycobacterial agents. Hit-to-lead development and target validation, New drugs for neglected diseases
2012 Poce, Giovanna; Porretta, Giulio Cesare; De Logu, A; De Rossi, A; Rubin, Ej; Ballel, L; Botta, M; Biava, Mariangela
New 1,5-diphenyl pyrrole derivatives as anti-inflammatory COX-2 selective compounds and their use as potential antitumoral agents.
2012 Consalvi, Sara; Battilocchio, Claudio; Poce, Giovanna; Alfonso, Salvatore; Porretta, Giulio Cesare; M., Anzini; L., Sautebin; C., Ghelardini; A., Giordani; P., Patrignani; V., Calderone; Biava, Mariangela
Analogs of BM 212: a new chemical class of antimycobacterial agents acting upon a new target
2012 Biava, Mariangela; Poce, Giovanna; Porretta, Giulio Cesare; Alfonso, Salvatore; Cocozza, Martina; De Logu, A; De Rossi, E; Ballel, L; Franzblau, S; Rubin E., J; Botta, M.
Improving the solubility of a new class of antiinflammatory pharmacodynamic hybrids, that release nitric oxide and inhibit cycloxygenase-2 isoenzyme
2012 Biava, Mariangela; Battilocchio, Claudio; Poce, Giovanna; Alfonso, Salvatore; Porretta, Giulio Cesare; Consalvi, Sara; Vincenzo, Calderone; Alma, Martelli; Lara, Testai; Carla, Ghelardini; Lorenzo Di Cesare, Mannelli; Lidia, Sautebin; Antonietta, Rossi; Antonio, Giordani; Paola, Patrignani; Maurizio, Anzini
Pyrrole-based selective COX-2 inhibiting nitric oxide donors: synthesis, in vitro and in vivo evaluation
2011 Battilocchio, Claudio; Porretta, Giulio Cesare; Poce, Giovanna; Alfonso, Salvatore; Calderone, V.; Sautebin, L.; Ghelardini, C.; Giordani, A.; Anzini, M.; Biava, Mariangela
BM212 targets MmpL3, Gordon Research Conference on Tuberculosis Drug Development
2011 Poce, Giovanna; Biava, Mariangela; Porretta, Giulio Cesare; Battilocchio, Claudio; Alfonso, Salvatore; Botta, M.; Javid, B.; Sorrentino, F.; Ioerger, T. R.; Sacchettini, J. R.; Rubin, E.
Synthesis and biological evaluation of new heterocyclic derivatives with potential antimycobacterial activity: systematic approach to lead compound optimization
2011 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Alfonso, Salvatore; Battilocchio, Claudio; De Logu, A; Manetti, F; Botta, M.
New Pyrrole-based selective COX-2 inhibiting nitric oxide donors: synthesis, in vitro and in vivo evaluation
2011 Battilocchio, Claudio; Porretta, Giulio Cesare; Poce, Giovanna; Alfonso, Salvatore; Giordani, A.; Sautebin, L.; Ghelardini, C.; Calderone, V.; Patrignani, P.; Anzini, M.; Biava, Mariangela
Developing Pyrrole-Derived Antimycobacterial Agents: a Rational Lead Optimization Approach
2011 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; Alfonso, Salvatore; A., De Logu; Fabrizio, Manetti; Maurizio, Botta
Novel Analgesic/Anti-Inflammatory Agents: Diarylpyrrole Acetic Esters Endowed with Nitric Oxide Releasing Properties
2011 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; Alfonso, Salvatore; Michele, Rovini; Salvatore, Valenti; Gianluca, Giorgi; Vincenzo, Calderone; Alma, Martelli; Lara, Testai; Lidia, Sautebin; Antonietta, Rossi; Giuseppina, Papa; Carla, Ghelardini; Lorenzo Di Cesare, Mannelli; Antonio, Giordani; Paola, Anzellotti; Annalisa, Bruno; Paola, Patrignani; Anzini,
Enlarging the NSAIDs Family: Ether, Ester and Acid Derivatives of the 1,5-Diarylpyrrole Scaffold as Novel Anti-Inflammatory and Analgesic Agents
2011 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; Botta, M; Manetti, F; Rovini, M; Cappelli, A; Sautebin, L; Rossi, A; Pergola, C; Ghelardini, C; Galeotti, N; Makovec, F; Giordani, A; Anzellotti, P; Tacconelli, S; Patrignani, P; Anzini, M.
1,5-Diaryl-Pyrroles as New Generation of Anti-Inflammatory and Analgesic Agents: Design, Synthesis, in vitro and in vivo Evaluation
2010 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Alfonso, S; Battilocchio, Claudio; DE LOGU, A; Manetti, F; Botta, M.
Identification of a new Chemical Class of Potent Antimycobacterial Compounds
2010 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Alfonso, Salvatore; Battilocchio, Claudio; De Logu, A; Manetti, F; Botta, M.
Developing New Antiinflammatory and Analgesic Agents: Design, Synthesis, Biological and harmacological Evaluation
2010 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; Alfonso, Salvatore; Botta, M.; Manetti, F.; Sautebin, L; Ghelardini, C; Makovec, F; Giordani, A; Patrignani, P; Anzini, M.
Novel Ester and Acid Derivatives of the 1,5-Diarylpyrrole Scaffold as Anti-inflammatory and Analgesic Agents. Synthesis, in vitro and in vivo Biological Evaluation
2010 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; Manetti, F; Botta, M; Sautebin, L; Rossi, A; Pergola, C; Ghelardini, C; Norcini, M; Makovec, F; Anzellotti, P; Cirilli, R; Ferretti, R; Patrignani, P; Anzini, M.
New pyrrole derivatives of BM 212: a new class of antimycobacterial agents. Design, synthesis, biological evaluation and study of their mode of action
2010 Biava, Mariangela; Porretta, G. C.; Poce, Giovanna; Alfonso, Salvatore; Battilocchio, Claudio; De Logu, A.; De Rossi, E.; Manetti, F; Botta, M.
BM 579: a novel pyrrole derivative with improved antimycobacterial activity
2010 Biava, Mariangela; Porretta, G. C.; Poce, Giovanna; Alfonso, Salvatore; Battilocchio, Claudio; De Logu, A.; Manetti, F; Botta, M.
Identification of a novel pyrrole derivative endowed with antimycobacterial activity and protection index comparable to that of the current antitubercular drugs streptomycin and rifampin
2010 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; Alfonso, Salvatore; A., De Logu; Nadia, Serra; Fabrizio, Manetti; Maurizio, Botta
New heterocyclic compounds with potential activity against parasitic protozoan: Trypanosoma and Leishmania
2010 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; V., Yardley; Alfonso, Salvatore
One-pot conversions of olefins to cyclic carbonates and secondary allylic and homoallylic amines to cyclic carbamates
2010 Stephen G., Davies; Ai M., Fletcher; Wataru, Kurosawa; James A., Lee; Poce, Giovanna; Paul M., Roberts; James E., Thomson; David M., Williamson
Doubly diastereoselective conjugate addition of enantiopure lithium amides to enantiopure N-enoyl oxazolidin-2-ones: a mechanistic probe
2010 Stephen G., Davies; M. A., Fletcher; Gesine J., Hermann; Poce, Giovanna; Paul M., Roberts; Andrew D., Smith; Miles J., Sweet; James E., Thomson
Pyrrole derivatives of BM212 as novel antimycobacterial agents Design, synthesis, biological evaluation and study of their mode of action
2009 Biava, Mariangela; Porretta, Giulio Cesare; Battilocchio, Claudio; Poce, G; Pompei, R; DE LOGU, A; Manetti, F; Botta, M.
New pyrrole derivatives of BM 212: a new class of antimycobacterial agents.Design, synthesis, biological evaluation and study of their mode of action.
2009 Biava, Mariangela; Porretta, G. C.; Poce, G; DE LOGU, A; Manetti, F; Botta, M.
Potent in vitro and in vivo novel 1,5-Diarylpyrrole-3-acetic Esters COX-2 inhibitors.
2009 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Sautebin, L; Patrignani, P; Ghelardini, C; Giordani, A; Anzini, M.
Derivatives of BM 212: synthesis and biological evaluation of new derivatives with improved antimycobacterial activity.
2009 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Pompei, R; DE LOGU, A; Manetti, F; Botta, M.
C-9 Alkenylidine bridged macrolides: WO2008061189.
2009 Poce, Giovanna; Porretta, Giulio Cesare; Biava, Mariangela
BM212 and its derivatives: lead optimization of a new class of antimycobacterial agents.
2009 Poce, Giovanna; Porretta, Giulio Cesare; DE LOGU, A; DE ROSSI, E; Manetti, F; Botta, M; Biava, Mariangela
1,5-Diaryl-2-ethyl pyrrole derivatives as antimycobacterial agents: design, synthesis, and microbiological evaluation
2009 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; DE LOGU, A; Saddi, M; Meleddu, R; Manetti, F; DE ROSSI, E; Botta, M.
New pyrrole derivatives of BM 212: lead compound optimization strategy, Tuberculosis drug development. Targets, technologies and trials
2009 Poce, Giovanna; Porretta, Giulio Cesare; Borzi, F; DE LOGU, A; DE ROSSI, E; Manetti, F; Botta, M; Biava, Mariangela
Design and synthesis of 1,5-diaryl-2-ethyl pyrrole derivatives and their evaluation as antimycobacterial agents
2008 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; DE LOGU, A; Maleddu, R; DE ROSSI, E; Manetti, F; Botta, M.
BM212 and new derivatives as a new class of antimycobacterial agents.
2008 Poce, Giovanna; Porretta, G. C.; Borzi, F; DE LOGU, A; DE ROSSI, E; Manetti, F; Botta, M; Biava, M.
New derivatives of BM 212 with improved antimycobacterial activity.
2008 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Pompei, R; DE LOGU, A; Manetti, F; Botta, M.
Design and Synthesis of novel diarylpyrroles as p38 MAP kinase inhibitors
2008 Biava, Mariangela; Porretta, G. C.; Poce, Giovanna; Giordani, A; Menziani, C.
New oxazolidinone derivatives as antibacterial agents with improved activity
2008 Poce, Giovanna; Giovanni, Zappia; Porretta, Giulio Cesare; Botta, Bruno; Biava, Mariangela
1,5-Diphenyl Pyrrole Derivatives as Antimycobacterial Agents. Probing the Influence on Antimycobacterial Activity of Lipophilic Substituents at the Phenyl Rings
2008 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; DE LOGU, A; Saddi, M; Meleddu, R; Manetti, F; DE ROSSI, E; Botta, M.
HPLC Enantioseparation and Absolute Configuration of Novel Antiinflammatory Pyrrole Derivatives
2008 Biava, Mariangela; Cirilli, R; Fares, V; Ferretti, R; Gallinella, B; Poce, Giovanna; Porretta, Giulio Cesare; Supino, Sibilla; Villani, Claudio
Synthesis, in vitro, and in vivo biological evaluation and molecular docking simulations of chiral alcohol and ether derivatives of the 1,5-diarylpyrrole scaffold as novel anti-inflammatory and analgesic agents
2008 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Sibilla, Supino; Fabrizio, Manetti; Stefano, Forli; Maurizio, Botta; Lidia, Sautebin; Antonietta, Rossi; Carlo, Pergola; Carla, Ghelardini; Monica, Norcini; Francesco, Makovec; Paola, Anzellotti; Roberto, Cirilli; Rosella, Ferretti; Bruno, Gallinella; F., La Torre; Maurizio, Anzini; Paola, Patrignani
New 1,5-diarylpyrrole with improved antimycobacterial activity
2007 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; DE LOGU, A; Saddi, M; Botta, M.
New 1,5-diphenyl Pyrrole Derived from BM 212: a New class of Antimycobacterial Agents.
2007 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; DE LOGU, A; Manetti, F; Botta, M.
Design, synthesis and screening of new antitubercular agents derived from BM 212
2007 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Deidda, D.; Pompei, R.; Manetti, F; Botta, M.
New pyrroles with potential antimycobacterial, antifungal and COX-2 selective inhibiting activities. Synthetic methodologies
2007 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Supino, S; Sleiter, G.
Cyclooxygenase-2 Inhibitors. 1,5-Diarylpyrrol-3-acetic Esters with Enhanced Inhibitory Activity toward Cyclooxygenase-2 and Improved Cyclooxygenase-2/Cyclooxygenase-1 Selectivity
2007 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Supino, Sibilla; Cappelli, A; Vomero, S; Manetti, F; Botta, M; Sautebin, L; Rossi, A; Ghelardini, C; Vivoli, E; Makovec, F; Anzellotti, P; Patrignani, P; Anzini, M.
Synthesis of new pyrrole derivatives of BM 212, a potent antimycobacterial compound
2006 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Supino, Sibilla; Deidda, D.; Pompei, R.; Manetti, F.; Botta, M.
New 1,5-diphenyl pyrrole derived from BM 212: a new class of antimycobacterial Agents
2006 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Supino, S; Pompei, R; Manetti, F; Botta, M.
Antimycobacterial agents. Novel diarylpirrole derivatives of BM212 endowed with high activity toward Mycobacterium tuberculosis and low cytotoxicity
2006 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Supino, S; Deidda, D; Pompei, R; Molicotti, P; Manetti, F; Botta, M.
1,5-DIARYLPYRROLE DERIVATIVESAS NOVEL CLASSES OF ACTIVE AND SELECTIVE COX-2 INHIBITORS.
2005 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Tibuzzi, D; Cappelli, A; Vomero, S; Botta, M; Manetti, F; Sautebin, L; Rossi, A; Makovec, F; Anzini, A.
ENANTIOMERS OF NOVEL ANTIINFLAMMATORY PYRROLE DERIVATIVES:ANALYTICAL AND SEMIPREPARATIVE HPLC SEPARATION AND CHIROPTICAL PROPERTIES.
2005 Biava, Mariangela; Cirilli, R.; Ferretti, R.; Poce, Giovanna; Porretta, Giulio Cesare; Villani, C. .
Antimycobacterial compounds. Optimization of the BM 212 structure, the lead compound for a new pyrrole derivative class
2005 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Delia, Deidda; Raffaello, Pompei; Andrea, Tafi; Fabrizio, Manetti
Pyrrole Derivatives as New Antimycobacterial Class: Synthesis, S.A.R., Molecular Modelling Considerations and Microbiological Activity
2004 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Pompei, R; Deidda, D; Tafi, A.; Manetti, F.; Botta, M.
1,5-diarylpyrrole-3-acetic acids and esters as novel class of potent and selective COX-2 inhibitors.
2004 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Cappelli, A.; Vomero, S.; Botta, M.; Manetti, F.; Giorni, G.; Sautebin, L.; Rossi, A.; Makovec, F.; Anzini, M. .
1,5-DIARYLPYRROLE-3-ACETIC ACIDS AND ESTERS AS NOVEL CLASSES OF POTENT AND SELECTIVE COX-2 INHIBITORS.
2004 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Cappelli, A; Vomero, S; Botta, M; Manetti, F; Giorni, G; Sautebin, L; Rossi, A; Makovec, F; Anzini, M.
Nuovi derivati 1,5-difenilpirrolici derivati del BM212 attivi come agenti antitubercolari
2004 Biava, M; Porretta, G. C.; Poce, Giovanna; Deidda, D; Pompei, R; Tafi, A; Manetti, F.
Titolo | Data di pubblicazione | Autore(i) | File |
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Tannin microcapsules for synergy-enhanced sunscreen formulations | 2023 | Alfonsi, E.; Lange, H.; Zongo, L.; Poce, G.; Sgarzi, M.; Crestini, C. | |
Direct-Acting Antivirals and Host-Targeting Approaches against Enterovirus B Infections: Recent Advances | 2023 | Tammaro, Chiara; Guida, Michela; Appetecchia, Federico; Biava, Mariangela; Consalvi, Sara; Poce, Giovanna | |
Antiviral Mechanisms of N-Phenyl Benzamides on Coxsackie Virus A9 | 2023 | Laajala, Mira; Kalander, Kerttu; Consalvi, Sara; Sheik Amamuddy, Olivier; Tastan Bishop, Özlem; Biava, Mariangela; Poce, Giovanna; Marjomäki, Varpu | |
Nano-Based Drug Delivery Systems of Potent MmpL3 Inhibitors for Tuberculosis Treatment | 2022 | Hanieh, P. N.; Consalvi, S.; Forte, J.; Cabiddu, G.; De Logu, A.; Poce, G.; Rinaldi, F.; Biava, M.; Carafa, M.; Marianecci, C. | |
Malaria transmission blocking compounds: a patent review | 2022 | Consalvi, Sara; Tammaro, Chiara; Appetecchia, Federico; Biava, Mariangela; Poce, Giovanna | |
A novel class of dual-acting DCH-CORMs counteracts oxidative stress-induced inflammation in human primary tenocytes | 2021 | Appetecchia, F.; Consalvi, S.; Berrino, E.; Gallorini, M.; Granese, A.; Campestre, C.; Carradori, S.; Biava, M.; Poce, G. | |
Therapeutic potential for coxibs-nitric oxide releasing hybrids in cystic fibrosis | 2021 | Consalvi, S.; Poce, G.; Ghelardini, C.; Di Cesare Mannelli, L.; Patrignani, P.; Bruno, A.; Anzini, M.; Calderone, V.; Martelli, A.; Testai, L.; Giordani, A.; Biava, M. | |
Dietary flavonoids: Nano delivery and nanoparticles for cancer therapy | 2021 | Aiello, Paola; Consalvi, Sara; Poce, Giovanna; Raguzzini, Anna; Toti, Elisabetta; Palmery, Maura; Biava, Mariangela; Bernardi, Marco; Kamale, Mohammad A.; Perry, George; Peluso, Ilaria | |
6-Fluorophenylbenzohydrazides inhibit Mycobacterium tuberculosis growth through alteration of tryptophan biosynthesis | 2021 | Consalvi, S.; Venditti, G.; Zhu, J.; Boshoff, H. I.; Arora, K.; De Logu, A.; Ioerger, T. R.; Rubin, E. J.; Biava, M.; Poce, G. | |
Sar analysis of small molecules interfering with energy-metabolism in mycobacterium tuberculosis | 2020 | Appetecchia, F.; Consalvi, S.; Scarpecci, C.; Biava, M.; Poce, G. | |
Overcoming drug resistance in TB: an update | 2020 | Consalvi, S.; Poce, G.; Scarpecci, C.; Biava, M. | |
Development of MmpL3 inhibitors for tuberculosis treatment | 2019 | Poce, Giovanna; Consalvi, Sara; Venditti, Giulia; Scarpecci, Cristina; Biava, Mariangela | |
Mycobacterial tryptophan biosynthesis: a promising target for tuberculosis drug development? | 2019 | Consalvi, Sara; Scarpecci, Cristina; Biava, Mariangela; Poce, Giovanna | |
Novel therapies for glaucoma: a patent review (2013-2019) | 2019 | Guglielmi, Paolo; Carradori, Simone; Campestre, Cristina; Poce, Giovanna | |
Novel pyrazole-containing compounds active against mycobacterium tuberculosis | 2019 | Poce, Giovanna; Consalvi, Sara; Venditti, Giulia; Alfonso, Salvatore; Desideri, Nicoletta; Fernandez-Menendez, Raquel; Bates, Robert H.; Ballell, Lluis; Barros Aguirre, David; Rullas, Joaquin; De Logu, Alessandro; Gardner, Michelle; Ioerger, Thomas R.; Rubin, Eric J.; Biava, Mariangela | |
Chocolate consumers and lymphocyte-to-monocyte ratio: a working hypothesis from a preliminary report of a pilot study in celiac subjects | 2019 | Raguzzini, A; Poce, G; Consalvi, S; Toti, E; Palmacci, F; Biava, M; Peluso, I | |
In vivo potent BM635 analogue with improved drug-like properties | 2018 | Poce, Giovanna; Cocozza, Martina; Alfonso, Salvatore; Consalvi, Sara; Venditti, Giulia; Fernandez-Menendez, Raquel; Bates, Robert H.; Barros Aguirre, David; Ballell, Lluis; De Logu, Alessandro; Vistoli, Giulio; Biava, Mariangela | |
Stimuli-responsive tannin–feIII hybrid microcapsules demonstrated by the active release of an anti-tuberculosis agent | 2018 | Bartzoka, Elisavet D.; Lange, Heiko; Poce, Giovanna; Crestini, Claudia | |
MmpL3 is the flippase for mycolic acids in mycobacteria | 2017 | Xu, Zhujun; Meshcheryakov, Vladimir A.; Poce, Giovanna; Chng, Shu-Sin | |
Pharmaceutical salt of BM635 with improved bioavailability | 2017 | Poce, Giovanna; Consalvi, Sara; Cocozza, Martina; Fernandez Menendez, Raquel; Bates, Robert H.; Ortega Muro, Fátima; Barros Aguirre, David; Ballell, Lluis; Biava, Mariangela | |
1,5-Diarylpyrroles as potent antitubercular and anti-inflammatory agents | 2017 | Venditti, Giulia; Poce, Giovanna; Consalvi, Sara; Biava, Mariangela | |
Novel inhibitors of Mycobacterium tuberculosis tryptophan biosynthetic pathway to treat tuberculosis | 2016 | Venditti, Giulia; Consalvi, Sara; Helena, Boshoff; Biava, Mariangela; Poce, Giovanna | |
A series of COX-2 inhibitors endowed with NO-releasing properties: synthesis, biological evaluation, and docking analysis | 2016 | Consalvi, Sara; Poce, Giovanna; Ragno, Rino; Sabatino, Manuela; Lamotta, Concettina; Sartini, Stefania; Calderone, Vincenzo; Martelli, Alma; Ghelardini, Carla; Dicesaremannelli, Lorenzo; Biava, Mariangela | |
Synthesis and biological evaluation of fluorinated 1,5-diarylpyrrole-3-alkoxyethyl ether derivatives as selective COX-2 inhibitors endowed with anti-inflammatory activity | 2016 | Di Capua, Angela; Sticozzi, Claudia; Brogi, Simone; Brindisi, Margherita; Cappelli, Andrea; Sautebin, Lidia; Rossi, Antonietta; Pace, Simona; Ghelardini, Carla; Di Cesare Mannelli, Lorenzo; Valacchi, Giuseppe; Giorgi, Gianluca; Giordani, Antonio; Poce, Giovanna; Biava, Mariangela; Anzini, Maurizio | |
MmpL3 inhibitors: diverse chemical scaffolds inhibit the same target | 2016 | Poce, Giovanna; Consalvi, Sara; Biava, Mariangela | |
COX inhibitors: a patent review (2011 - 2014) | 2015 | Consalvi, Sara; Biava, Mariangela; Poce, Giovanna | |
Synthesis, biological evaluation and docking analysis of a new series of methylsulfonyl and sulfamoyl acetamides and ethyl acetates as potent COX-2 inhibitors | 2015 | Consalvi, Sara; Alfonso, Salvatore; Di Capua, Angela; Poce, Giovanna; Pirolli, Adele; Sabatino, Manuela; Ragno, Rino; Anzini, Maurizio; Sartini, Stefania; La Motta, Concettina; Di Cesare Mannelli, Lorenzo; Ghelardini, Carla; Biava, Mariangela | |
A novel antimycobacterial compound acts as an intracellular iron chelator | 2015 | Dragset Marte, S; Poce, Giovanna; Alfonso, Salvatore; Padilla Benavides, T; Ioerger, T. R.; Kaneko, T; Sacchettini, Jc; Biava, Mariangela; Parish, T; Argüello, Jm; Steigedal, M; Rubin, Ej | |
Overcoming drug resistance for tuberculosis, | 2015 | Poce, Giovanna; Biava, Mariangela | |
Activity of lipophilic and hydrophilic drugs against dormant and replicating mycobacterium tuberculosis | 2015 | Piccaro, G; Poce, Giovanna; Biava, Mariangela; Giannoni, F; Fattorini, L. | |
SAR analysis of new anti-TB drugs currently in pre-clinical and clinical development | 2014 | Poce, Giovanna; Cocozza, Martina; Consalvi, Sara; Biava, Mariangela | |
Enhancing the pharmacodynamic profile of a class of selective COX-2 inhibiting nitric oxide donors | 2014 | Biava, Mariangela; Battilocchio, Claudio; Poce, Giovanna; Alfonso, Salvatore; Consalvi, Sara; Angela Di, Capua; Vincenzo, Calderone; Alma, Martelli; Lara, Testai; Lidia, Sautebin; Antonietta, Rossi; Carla, Ghelardini; Lorenzo Di Cesare, Mannelli; Antonio, Giordani; Stefano, Persiani; Milena, Colovic; Melania, Dovizio; Paola, Patrignani; Maurizio, Anzini | |
A class of pyrrole derivatives endowed with analgesic/anti-inflammatory activity | 2013 | Battilocchio, Claudio; Poce, Giovanna; Alfonso, Salvatore; Porretta, Giulio Cesare; Consalvi, Sara; L., Sautebin; S., Pace; A., Rossi; C., Ghelardini; L., Di Cesare Mannelli; S., Schenone; A., Giordani; L., Di Francesco; P., Patrignani; Biava, Mariangela | |
Inhibition of Leishmania infantum trypanothione reductase by azole-based compounds: a comparative analysis with its physiological substrate by X-ray crystallography | 2013 | Baiocco, P.; Poce, Giovanna; Alfonso, Salvatore; Cocozza, Martina; Porretta, Giulio Cesare; Colotti, G.; Biava, Mariangela; Moraca, F.; Botta, M.; Yardley, V.; Fiorillo, A.; Lantella, A.; Malatesta, Francesco; Ilari, Andrea | |
Improved BM212 MmpL3 Inhibitor Analogue Shows Efficacy in Acute Murine Model of Tuberculosis Infection | 2013 | Poce, Giovanna; H. R., Bates; Alfonso, Salvatore; Cocozza, Martina; Porretta, Giulio Cesare; L., Ballel; Joaquin, Rullas; Alessandro De, Logu; Emanuela, Agus; Valentina La, Rosa; Maria Rosalia, Pasca; Edda De, Rossi; Baojie, Wae; S. J., Franzblau; Fabrizio, Manetti; Maurizio, Botta; Biava, Mariangela | |
Novel Analgesic/Anti-inflammatory Agents: 1,5-Diarylpyrrole Nitro-oxyalkyl Ethers and Related Compounds as Cyclooxygenase-2 Inhibiting Nitric Oxide Donors | 2013 | Anzini, M.; Di Capua, A.; Valenti, S.; Brogi, S.; Rovin, M.; Giuliani, G.; Cappelli, A.; Vomero, S.; Chiasserini, L.; Saga, A.; Poce, Giovanna; Giorgi, G.; Calderone, V.; Martelli, A.; Testai, L.; Sautebin, L.; Rossi, A.; Papa, G.; Ghelardini, C.; Di Cesare Mannelli, L.; Benetti, V.; Giordani, A.; Anzellotti, P.; Dovizio, M.; Patrignani, P.; Biava, Mariangela | |
The novel anti-inflammatory agent VA694, endowed with both NO-releasing and COX2-selective inhibiting properties, exhibits NO-mediated positive effects on blood pressure, coronary flow and endothelium in an experimental model of hypertension and endothelial dysfunction | 2013 | Martelli, A; Testai, L; Anzini, M; Cappelli, A; Di Capua, A; Biava, Mariangela; Poce, Giovanna; Consalvi, Sara; Giordani, A; Caselli, G; Rovati, L; Ghelardini, C; Patrignani, P; Sautebin, L; Breschi, Mc; Calderone, V. | |
New Heterocyclic Compounds Targeting Trypanothyione Metabolism in Leishmania Parasites | 2012 | Biava, Mariangela; Cocozza, Martina; Poce, Giovanna; Alfonso, Salvatore; Battilocchio, Claudio; Colotti, G.; Malatesta, F.; Baiocco, P.; Ilari, Andrea | |
New 1,5 diarylpyrrole derivatives as antimycobacterial agents: Design, synthesis, biological evaluation and study of their mode of action | 2012 | Alfonso, Salvatore; Poce, Giovanna; Porretta, Giulio Cesare; Battilocchio, Claudio; Rubin, E. J.; De Rossi, E.; De Logu, A.; Franzblau, S. C.; Botta, M.; Biava, Mariangela | |
New Pyrrole Derivatives as Anti-inflammatory and Analgesic Agents: Design, Synthesis and Biological Evaluation | 2012 | Biava, Mariangela; Consalvi, Sara; Poce, Giovanna; Battilocchio, Claudio; Alfonso, Salvatore; Ghelardini, C.; Sautebin, L. | |
MmpL3 Is the Cellular Target of the Antitubercular Pyrrole Derivative BM212 | 2012 | V., La Rosa; Poce, Giovanna; J., Ortiz Canseco; S., Buroni; M. R., Pasca; Biava, Mariangela; R. M., Raju; Porretta, Giulio Cesare; Alfonso, Salvatore; C., Battilocchio; B., Javid; F., Sorrentino; T. R., Ioerger; J. C., Sacchettini; F., Manetti; M., Botta; A., De Logu; E. J., Rubin | |
Identification of a new chemical class of potent antimycobacterial compounds derived from BM 212: design, synthesis, biological evaluation and study of their mode of action. | 2012 | Biava, Mariangela; Poce, Giovanna; Porretta, Giulio Cesare; Alfonso, Salvatore; De Logu, A; De Rossi, E; Ballel, L; Franzblau, S; Manetti, ; Rubin, Ej; Botta, M. | |
1,5-Diphenyl pyrroles as new antimycobacterial agents. Hit-to-lead development and target validation, New drugs for neglected diseases | 2012 | Poce, Giovanna; Porretta, Giulio Cesare; De Logu, A; De Rossi, A; Rubin, Ej; Ballel, L; Botta, M; Biava, Mariangela | |
New 1,5-diphenyl pyrrole derivatives as anti-inflammatory COX-2 selective compounds and their use as potential antitumoral agents. | 2012 | Consalvi, Sara; Battilocchio, Claudio; Poce, Giovanna; Alfonso, Salvatore; Porretta, Giulio Cesare; M., Anzini; L., Sautebin; C., Ghelardini; A., Giordani; P., Patrignani; V., Calderone; Biava, Mariangela | |
Analogs of BM 212: a new chemical class of antimycobacterial agents acting upon a new target | 2012 | Biava, Mariangela; Poce, Giovanna; Porretta, Giulio Cesare; Alfonso, Salvatore; Cocozza, Martina; De Logu, A; De Rossi, E; Ballel, L; Franzblau, S; Rubin E., J; Botta, M. | |
Improving the solubility of a new class of antiinflammatory pharmacodynamic hybrids, that release nitric oxide and inhibit cycloxygenase-2 isoenzyme | 2012 | Biava, Mariangela; Battilocchio, Claudio; Poce, Giovanna; Alfonso, Salvatore; Porretta, Giulio Cesare; Consalvi, Sara; Vincenzo, Calderone; Alma, Martelli; Lara, Testai; Carla, Ghelardini; Lorenzo Di Cesare, Mannelli; Lidia, Sautebin; Antonietta, Rossi; Antonio, Giordani; Paola, Patrignani; Maurizio, Anzini | |
Pyrrole-based selective COX-2 inhibiting nitric oxide donors: synthesis, in vitro and in vivo evaluation | 2011 | Battilocchio, Claudio; Porretta, Giulio Cesare; Poce, Giovanna; Alfonso, Salvatore; Calderone, V.; Sautebin, L.; Ghelardini, C.; Giordani, A.; Anzini, M.; Biava, Mariangela | |
BM212 targets MmpL3, Gordon Research Conference on Tuberculosis Drug Development | 2011 | Poce, Giovanna; Biava, Mariangela; Porretta, Giulio Cesare; Battilocchio, Claudio; Alfonso, Salvatore; Botta, M.; Javid, B.; Sorrentino, F.; Ioerger, T. R.; Sacchettini, J. R.; Rubin, E. | |
Synthesis and biological evaluation of new heterocyclic derivatives with potential antimycobacterial activity: systematic approach to lead compound optimization | 2011 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Alfonso, Salvatore; Battilocchio, Claudio; De Logu, A; Manetti, F; Botta, M. | |
New Pyrrole-based selective COX-2 inhibiting nitric oxide donors: synthesis, in vitro and in vivo evaluation | 2011 | Battilocchio, Claudio; Porretta, Giulio Cesare; Poce, Giovanna; Alfonso, Salvatore; Giordani, A.; Sautebin, L.; Ghelardini, C.; Calderone, V.; Patrignani, P.; Anzini, M.; Biava, Mariangela | |
Developing Pyrrole-Derived Antimycobacterial Agents: a Rational Lead Optimization Approach | 2011 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; Alfonso, Salvatore; A., De Logu; Fabrizio, Manetti; Maurizio, Botta | |
Novel Analgesic/Anti-Inflammatory Agents: Diarylpyrrole Acetic Esters Endowed with Nitric Oxide Releasing Properties | 2011 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; Alfonso, Salvatore; Michele, Rovini; Salvatore, Valenti; Gianluca, Giorgi; Vincenzo, Calderone; Alma, Martelli; Lara, Testai; Lidia, Sautebin; Antonietta, Rossi; Giuseppina, Papa; Carla, Ghelardini; Lorenzo Di Cesare, Mannelli; Antonio, Giordani; Paola, Anzellotti; Annalisa, Bruno; Paola, Patrignani; Anzini, | |
Enlarging the NSAIDs Family: Ether, Ester and Acid Derivatives of the 1,5-Diarylpyrrole Scaffold as Novel Anti-Inflammatory and Analgesic Agents | 2011 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; Botta, M; Manetti, F; Rovini, M; Cappelli, A; Sautebin, L; Rossi, A; Pergola, C; Ghelardini, C; Galeotti, N; Makovec, F; Giordani, A; Anzellotti, P; Tacconelli, S; Patrignani, P; Anzini, M. | |
1,5-Diaryl-Pyrroles as New Generation of Anti-Inflammatory and Analgesic Agents: Design, Synthesis, in vitro and in vivo Evaluation | 2010 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Alfonso, S; Battilocchio, Claudio; DE LOGU, A; Manetti, F; Botta, M. | |
Identification of a new Chemical Class of Potent Antimycobacterial Compounds | 2010 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Alfonso, Salvatore; Battilocchio, Claudio; De Logu, A; Manetti, F; Botta, M. | |
Developing New Antiinflammatory and Analgesic Agents: Design, Synthesis, Biological and harmacological Evaluation | 2010 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; Alfonso, Salvatore; Botta, M.; Manetti, F.; Sautebin, L; Ghelardini, C; Makovec, F; Giordani, A; Patrignani, P; Anzini, M. | |
Novel Ester and Acid Derivatives of the 1,5-Diarylpyrrole Scaffold as Anti-inflammatory and Analgesic Agents. Synthesis, in vitro and in vivo Biological Evaluation | 2010 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; Manetti, F; Botta, M; Sautebin, L; Rossi, A; Pergola, C; Ghelardini, C; Norcini, M; Makovec, F; Anzellotti, P; Cirilli, R; Ferretti, R; Patrignani, P; Anzini, M. | |
New pyrrole derivatives of BM 212: a new class of antimycobacterial agents. Design, synthesis, biological evaluation and study of their mode of action | 2010 | Biava, Mariangela; Porretta, G. C.; Poce, Giovanna; Alfonso, Salvatore; Battilocchio, Claudio; De Logu, A.; De Rossi, E.; Manetti, F; Botta, M. | |
BM 579: a novel pyrrole derivative with improved antimycobacterial activity | 2010 | Biava, Mariangela; Porretta, G. C.; Poce, Giovanna; Alfonso, Salvatore; Battilocchio, Claudio; De Logu, A.; Manetti, F; Botta, M. | |
Identification of a novel pyrrole derivative endowed with antimycobacterial activity and protection index comparable to that of the current antitubercular drugs streptomycin and rifampin | 2010 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; Alfonso, Salvatore; A., De Logu; Nadia, Serra; Fabrizio, Manetti; Maurizio, Botta | |
New heterocyclic compounds with potential activity against parasitic protozoan: Trypanosoma and Leishmania | 2010 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; V., Yardley; Alfonso, Salvatore | |
One-pot conversions of olefins to cyclic carbonates and secondary allylic and homoallylic amines to cyclic carbamates | 2010 | Stephen G., Davies; Ai M., Fletcher; Wataru, Kurosawa; James A., Lee; Poce, Giovanna; Paul M., Roberts; James E., Thomson; David M., Williamson | |
Doubly diastereoselective conjugate addition of enantiopure lithium amides to enantiopure N-enoyl oxazolidin-2-ones: a mechanistic probe | 2010 | Stephen G., Davies; M. A., Fletcher; Gesine J., Hermann; Poce, Giovanna; Paul M., Roberts; Andrew D., Smith; Miles J., Sweet; James E., Thomson | |
Pyrrole derivatives of BM212 as novel antimycobacterial agents Design, synthesis, biological evaluation and study of their mode of action | 2009 | Biava, Mariangela; Porretta, Giulio Cesare; Battilocchio, Claudio; Poce, G; Pompei, R; DE LOGU, A; Manetti, F; Botta, M. | |
New pyrrole derivatives of BM 212: a new class of antimycobacterial agents.Design, synthesis, biological evaluation and study of their mode of action. | 2009 | Biava, Mariangela; Porretta, G. C.; Poce, G; DE LOGU, A; Manetti, F; Botta, M. | |
Potent in vitro and in vivo novel 1,5-Diarylpyrrole-3-acetic Esters COX-2 inhibitors. | 2009 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Sautebin, L; Patrignani, P; Ghelardini, C; Giordani, A; Anzini, M. | |
Derivatives of BM 212: synthesis and biological evaluation of new derivatives with improved antimycobacterial activity. | 2009 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Pompei, R; DE LOGU, A; Manetti, F; Botta, M. | |
C-9 Alkenylidine bridged macrolides: WO2008061189. | 2009 | Poce, Giovanna; Porretta, Giulio Cesare; Biava, Mariangela | |
BM212 and its derivatives: lead optimization of a new class of antimycobacterial agents. | 2009 | Poce, Giovanna; Porretta, Giulio Cesare; DE LOGU, A; DE ROSSI, E; Manetti, F; Botta, M; Biava, Mariangela | |
1,5-Diaryl-2-ethyl pyrrole derivatives as antimycobacterial agents: design, synthesis, and microbiological evaluation | 2009 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; DE LOGU, A; Saddi, M; Meleddu, R; Manetti, F; DE ROSSI, E; Botta, M. | |
New pyrrole derivatives of BM 212: lead compound optimization strategy, Tuberculosis drug development. Targets, technologies and trials | 2009 | Poce, Giovanna; Porretta, Giulio Cesare; Borzi, F; DE LOGU, A; DE ROSSI, E; Manetti, F; Botta, M; Biava, Mariangela | |
Design and synthesis of 1,5-diaryl-2-ethyl pyrrole derivatives and their evaluation as antimycobacterial agents | 2008 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; DE LOGU, A; Maleddu, R; DE ROSSI, E; Manetti, F; Botta, M. | |
BM212 and new derivatives as a new class of antimycobacterial agents. | 2008 | Poce, Giovanna; Porretta, G. C.; Borzi, F; DE LOGU, A; DE ROSSI, E; Manetti, F; Botta, M; Biava, M. | |
New derivatives of BM 212 with improved antimycobacterial activity. | 2008 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Pompei, R; DE LOGU, A; Manetti, F; Botta, M. | |
Design and Synthesis of novel diarylpyrroles as p38 MAP kinase inhibitors | 2008 | Biava, Mariangela; Porretta, G. C.; Poce, Giovanna; Giordani, A; Menziani, C. | |
New oxazolidinone derivatives as antibacterial agents with improved activity | 2008 | Poce, Giovanna; Giovanni, Zappia; Porretta, Giulio Cesare; Botta, Bruno; Biava, Mariangela | |
1,5-Diphenyl Pyrrole Derivatives as Antimycobacterial Agents. Probing the Influence on Antimycobacterial Activity of Lipophilic Substituents at the Phenyl Rings | 2008 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; DE LOGU, A; Saddi, M; Meleddu, R; Manetti, F; DE ROSSI, E; Botta, M. | |
HPLC Enantioseparation and Absolute Configuration of Novel Antiinflammatory Pyrrole Derivatives | 2008 | Biava, Mariangela; Cirilli, R; Fares, V; Ferretti, R; Gallinella, B; Poce, Giovanna; Porretta, Giulio Cesare; Supino, Sibilla; Villani, Claudio | |
Synthesis, in vitro, and in vivo biological evaluation and molecular docking simulations of chiral alcohol and ether derivatives of the 1,5-diarylpyrrole scaffold as novel anti-inflammatory and analgesic agents | 2008 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Sibilla, Supino; Fabrizio, Manetti; Stefano, Forli; Maurizio, Botta; Lidia, Sautebin; Antonietta, Rossi; Carlo, Pergola; Carla, Ghelardini; Monica, Norcini; Francesco, Makovec; Paola, Anzellotti; Roberto, Cirilli; Rosella, Ferretti; Bruno, Gallinella; F., La Torre; Maurizio, Anzini; Paola, Patrignani | |
New 1,5-diarylpyrrole with improved antimycobacterial activity | 2007 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; DE LOGU, A; Saddi, M; Botta, M. | |
New 1,5-diphenyl Pyrrole Derived from BM 212: a New class of Antimycobacterial Agents. | 2007 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; DE LOGU, A; Manetti, F; Botta, M. | |
Design, synthesis and screening of new antitubercular agents derived from BM 212 | 2007 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Deidda, D.; Pompei, R.; Manetti, F; Botta, M. | |
New pyrroles with potential antimycobacterial, antifungal and COX-2 selective inhibiting activities. Synthetic methodologies | 2007 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Supino, S; Sleiter, G. | |
Cyclooxygenase-2 Inhibitors. 1,5-Diarylpyrrol-3-acetic Esters with Enhanced Inhibitory Activity toward Cyclooxygenase-2 and Improved Cyclooxygenase-2/Cyclooxygenase-1 Selectivity | 2007 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Supino, Sibilla; Cappelli, A; Vomero, S; Manetti, F; Botta, M; Sautebin, L; Rossi, A; Ghelardini, C; Vivoli, E; Makovec, F; Anzellotti, P; Patrignani, P; Anzini, M. | |
Synthesis of new pyrrole derivatives of BM 212, a potent antimycobacterial compound | 2006 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Supino, Sibilla; Deidda, D.; Pompei, R.; Manetti, F.; Botta, M. | |
New 1,5-diphenyl pyrrole derived from BM 212: a new class of antimycobacterial Agents | 2006 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Supino, S; Pompei, R; Manetti, F; Botta, M. | |
Antimycobacterial agents. Novel diarylpirrole derivatives of BM212 endowed with high activity toward Mycobacterium tuberculosis and low cytotoxicity | 2006 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Supino, S; Deidda, D; Pompei, R; Molicotti, P; Manetti, F; Botta, M. | |
1,5-DIARYLPYRROLE DERIVATIVESAS NOVEL CLASSES OF ACTIVE AND SELECTIVE COX-2 INHIBITORS. | 2005 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Tibuzzi, D; Cappelli, A; Vomero, S; Botta, M; Manetti, F; Sautebin, L; Rossi, A; Makovec, F; Anzini, A. | |
ENANTIOMERS OF NOVEL ANTIINFLAMMATORY PYRROLE DERIVATIVES:ANALYTICAL AND SEMIPREPARATIVE HPLC SEPARATION AND CHIROPTICAL PROPERTIES. | 2005 | Biava, Mariangela; Cirilli, R.; Ferretti, R.; Poce, Giovanna; Porretta, Giulio Cesare; Villani, C. . | |
Antimycobacterial compounds. Optimization of the BM 212 structure, the lead compound for a new pyrrole derivative class | 2005 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Delia, Deidda; Raffaello, Pompei; Andrea, Tafi; Fabrizio, Manetti | |
Pyrrole Derivatives as New Antimycobacterial Class: Synthesis, S.A.R., Molecular Modelling Considerations and Microbiological Activity | 2004 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Pompei, R; Deidda, D; Tafi, A.; Manetti, F.; Botta, M. | |
1,5-diarylpyrrole-3-acetic acids and esters as novel class of potent and selective COX-2 inhibitors. | 2004 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Cappelli, A.; Vomero, S.; Botta, M.; Manetti, F.; Giorni, G.; Sautebin, L.; Rossi, A.; Makovec, F.; Anzini, M. . | |
1,5-DIARYLPYRROLE-3-ACETIC ACIDS AND ESTERS AS NOVEL CLASSES OF POTENT AND SELECTIVE COX-2 INHIBITORS. | 2004 | Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Cappelli, A; Vomero, S; Botta, M; Manetti, F; Giorni, G; Sautebin, L; Rossi, A; Makovec, F; Anzini, M. | |
Nuovi derivati 1,5-difenilpirrolici derivati del BM212 attivi come agenti antitubercolari | 2004 | Biava, M; Porretta, G. C.; Poce, Giovanna; Deidda, D; Pompei, R; Tafi, A; Manetti, F. |
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