Sfoglia per Autore SECCI, DANIELA
Indoleamine 2,3-dioxygenase
2023 Coluccia, Michele; Secci, Daniela; Guglielmi, Paolo
A Multitarget Approach against Neuroinflammation: Alkyl Substituted Coumarins as Inhibitors of Enzymes Involved in Neurodegeneration
2023 Berrino, E.; Carradori, S.; Carta, F.; Melfi, F.; Gallorini, M.; Poli, G.; Tuccinardi, T.; Fernandez-Bolanos, J. G.; Lopez, O.; Petzer, J. P.; Petzer, A.; Guglielmi, P.; Secci, D.; Supuran, C. T.
Novel Insights on CAI–CORM Hybrids: Evaluation of the CO Releasing Properties and Pain-Relieving Activity of Differently Substituted Coumarins for the Treatment of Rheumatoid Arthritis
2023 Berrino, Emanuela; Micheli, Laura; Carradori, Simone; di Cesare Mannelli, Lorenzo; Guglielmi, Paolo; De Luca, Alessandro; Carta, Fabrizio; Ghelardini, Carla; Secci, Daniela; Supuran, Claudiu T.
Kinetic Study on the Base-Catalyzed Imine-Enamine Tautomerism of a Chiral Biologically Active Isoxazoline Derivative by HPLC on Amylose Tris(3,5-dimethylphenylcarbamate) Chiral Stationary Phase
2023 Sadutto, Daniele; Guglielmi, Paolo; Carradori, Simone; Secci, Daniela; Cirilli, Roberto
A comparative study on the suppression capacity and the environmental impact of different extinguishing agents of lithium-ion battery fires
2022 Ubaldi, Sofia; Di Bari, Cinzia; De Rosa, Armando; Quinterno, Mario; Mazzaro, Michele; Ferrigno, Gianluca; Arrighi, Francesca; Secci, Daniela; Russo, Paola
Novel Insights on Human Carbonic Anhydrase Inhibitors Based on Coumalic Acid: Design, Synthesis, Molecular Modeling Investigation, and Biological Studies
2022 Pontecorvi, Virginia; Mori, Mattia; Picarazzi, Francesca; Zara, Susi; Carradori, Simone; Cataldi, Amelia; Angeli, Andrea; Berrino, Emanuela; Chimenti, Paola; Ciogli, Alessia; Secci, Daniela; Guglielmi, Paolo; Supuran, Claudiu T.
Treatment of Toxoplasmosis: An Insight on Epigenetic Drugs
2022 Guglielmi, P.; Secci, D.
Metal-organic frameworks (MOFs) as biomolecules drug delivery systems for anticancer purposes
2022 Coluccia, Michele; Parisse, Valeria; Guglielmi, Paolo; Giannini, Giuseppe; Secci, Daniela
Synthesis and evaluation of thymol-based synthetic derivatives as dual-action inhibitors against different strains of h. pylori and AGS cell line
2021 Sisto, F.; Carradori, S.; Guglielmi, P.; Spano, M.; Secci, D.; Granese, A.; Sobolev, A. P.; Grande, R.; Campestre, C.; Di Marcantonio, M. C.; Mincione, G.
An innovative spectroscopic approach for qualitative and quantitative evaluation of Mb-CO from myoglobin carbonylation reaction through chemometrics methods
2021 Mansoldo, F. R. P.; Berrino, E.; Guglielmi, P.; Carradori, S.; Carta, F.; Secci, D.; Supuran, C. T.; Vermelho, A. B.
Chalcones: Unearthing their therapeutic possibility as monoamine oxidase B inhibitors
2020 Guglielmi, Paolo; Mathew, Bijo; Secci, Daniela; Carradori, Simone
Innovative pH-interfering agents in association with anticancer agents
2020 Secci, D.; Guglielmi, P.
Inhibition of lysine acetyltransferases impairs tumor angiogenesis acting on both endothelial and tumor cells
2020 Di Martile, Marta; Gabellini, Chiara; Desiderio, Marianna; Matraxia, Marta; Farini, Valentina; Valentini, Elisabetta; Carradori, Simone; Ercolani, Cristiana; Buglioni, Simonetta; Secci, Daniela; Andreazzoli, Massimiliano; Del Bufalo and Daniela Trisciuoglio, Donatella
Synthesis and biological evaluation of carvacrol-based derivatives as dual inhibitors of H. Pylori strains and ags cell proliferation
2020 Sisto, F.; Carradori, S.; Guglielmi, P.; Traversi, C. B.; Spano, M.; Sobolev, A. P.; Secci, D.; Di Marcantonio, M. C.; Haloci, E.; Grande, R.; Mincione, G.
Antimalarial agents from medicinal plant and fungal sources
2020 Luisi, Grazia; Carradori, Simone; Grande, Rossella; Secci, Daniela; Guglielmi, Paolo
Metabolic profiling of different wild and cultivated Allium species based on high-resolution mass spectrometry, high-performance liquid chromatography-photodiode array detector, and color analysis
2020 Maccelli, A.; Cesa, S.; Cairone, F.; Secci, D.; Menghini, L.; Chiavarino, B.; Fornarini, S.; Crestoni, M. E.; Locatelli, M.
1,3-Dipolar Cycloaddition, HPLC Enantioseparation, and Docking Studies of Saccharin/Isoxazole and Saccharin/Isoxazoline Derivatives as Selective Carbonic Anhydrase IX and XII Inhibitors
2020 D'Ascenzio, M.; Secci, D.; Carradori, S.; Zara, S.; Guglielmi, P.; Cirilli, R.; Pierini, M.; Poli, G.; Tuccinardi, T.; Angeli, A.; Supuran, C. T.
High-performance liquid chromatography enantioseparation of chiral 2-(benzylsulfinyl)benzamide derivatives on cellulose tris(3,5-dichlorophenylcarbamate) chiral stationary phase
2020 Carradori, S.; Secci, D.; Guglielmi, P.; Pierini, M.; Cirilli, R.
Synthesis and evaluation of a large library of nitroxoline derivatives as pancreatic cancer antiproliferative agents
2020 Veschi, Serena; Carradori, Simone; De Lellis, Laura; Florio, Rosalba; Brocco, Davide; Secci, Daniela; Guglielmi, Paolo; Spano, Mattia; Sobolev, Anatoly P.; Cama, Alessandro
Novel insights on saccharin- and acesulfame-based carbonic anhydrase inhibitors: design, synthesis, modelling investigations and biological activity evaluation
2020 Guglielmi, P.; Rotondi, G.; Secci, D.; Angeli, A.; Chimenti, P.; Nocentini, A.; Bonardi, A.; Gratteri, P.; Carradori, S.; Supuran, C. T.
Novel approaches to the discovery of selective human monoamine oxidase-B inhibitors: is there room for improvement?
2019 Guglielmi, P.; Carradori, S.; Ammazzalorso, A.; Secci, D.
4-(3-Nitrophenyl)thiazol-2-ylhydrazone derivatives as antioxidants and selective hMAO-B inhibitors: synthesis, biological activity and computational analysis
2019 Secci, Daniela; Carradori, Simone; Petzer, Anél; Guglielmi, Paolo; D’Ascenzio, Melissa; Chimenti, Paola; Bagetta, Donatella; Alcaro, Stefano; Zengin, Gokhan; Petzer, Jacobus P.; Ortuso, Francesco
Investigation on the stability of new biologically active thiosemicarbazone-derived compounds by a validated HPLC-PDA method
2019 Secci, Daniela; Locatelli, Marcello; Kabir, Abuzar; Salvatorelli, Erika; Macedonio, Giorgia; Mollica and Simone Carradori, Adriano
Benzo[b]tiophen-3-ol derivatives as effective inhibitors of human monoamine oxidase: design, synthesis, and biological activity
2019 Guglielmi, Paolo; Secci, Daniela; Petzer, Anél; Bagetta, Donatella; Chimenti, Paola; Rotondi, Giulia; Ferrante, Claudio; Recinella, Lucia; Leone, Sheila; Alcaro, Stefano; Zengin, Gokhan; Petzer, Jacobus P; Ortuso, Francesco; Carradori, Simone
Design, synthesis, docking studies and monoamine oxidase inhibition of a small library of 1-acetyl- and 1-thiocarbamoyl-3,5-diphenyl-4,5-dihydro-(1h)-pyrazoles
2019 Guglielmi, Paolo; Carradori, Simone; Poli, Giulio; Secci, Daniela; Cirilli, Roberto; Rotondi, Giulia; Chimenti, Paola; Petzer, Anél; Petzer, Jacobus P.
Design, synthesis and biological activity of selective hCAs inhibitors based on 2-(benzylsulfinyl)benzoic acid scaffold
2019 Rotondi, G.; Guglielmi, P.; Carradori, S.; Secci, D.; De Monte, C.; De Filippis, B.; Maccallini, C.; Amoroso, R.; Cirilli, R.; Akdemir, A.; Angeli, A.; Supuran, C. T.
Atriplex mollis desf. Aerial parts: extraction procedures, secondary metabolites and color analysis
2018 Boutaoui, Nassima; Zaiter, Lahcene; Benayache, Fadila; Benayache, Samir; Cacciagrano, Francesco; Cesa, Stefania; Secci, Daniela; Carradori, Simone; Giusti, Anna Maria; Campestre, Cristina; Menghini, Luigi; Locatelli, Marcello
MAO inhibitors and their wider applications: a patent review
2018 Carradori, Simone; Secci, Daniela; Petzer, Jacques P.
A chromatographic study on the exceptional chiral recognition of 2-(benzylsulfinyl)benzamide by animmobilized-type chiral stationary phase based on cellulose tris(3,5-dichlorophenylcarbamate)
2018 Carradori, Simone; Secci, Daniela; Faggi, Cristina; Cirilli, Roberto
Bioactive isoflavones from Pueraria lobata root and starch: Different extraction techniques and carbonic anhydrase inhibition
2018 Mocan, Andrei; Carradori, Simone; Locatelli, Marcello; Secci, Daniela; Cesa, Stefania; Mollica, Adriano; Riga, Simona; Angeli, Andrea; Supuran, Claudiu T.; Celia, Christian; Di Marzio, Luisa
Magnetic metal−organic framework composite by fast and facile mechanochemical process
2018 Bellusci, M.; Guglielmi, P.; Masi, Andrea; Padella, F.; Singh, G.; Yaacoub, N.; Peddis, D.; Secci, D.
Design, synthesis and biochemical evaluation of novel multi-target inhibitors as potential anti-Parkinson agents
2018 Carradori, Simone; Ottuso, Francesco; Petzer, Anèl; Bagetta, Donatella; DE MONTE, Celeste; Secci, Daniela; DE VITA, Daniela; Guglielmi, Paolo; Zengin, Gokhan; Aktumsek, Abdurrahman; Alcaro, Stefano; Petzer, Jacobus P.
Geographical characterization by MAE-HPLC and NIR methodologies and carbonic anhydrase inhibition of Saffron components
2017 Nescatelli, Riccardo; Carradori, Simone; Marini, Federico; Caponigro, Vicky; Bucci, Remo; DE MONTE, Celeste; Mollica, Adriano; Mannina, Luisa; Ceruso, Mariangela; Supuran, CLAUDIU TRANDAFIR; Secci, Daniela
Optimization of aqueous extraction and biological activity of harpagophytum procumbens root on ex vivo rat Colon inflammatory model
2017 Locatelli, Marcello; Ferrante, Claudio; Carradori, Simone; Secci, Daniela; Leporini, Lidia; Chiavaroli, Annalisa; Leone, Sheila; Recinella, Lucia; Orlando, Giustino; Martinotti, Sara; Brunetti, Luigi; Vacca And Luigi Menghini, Michele
Open saccharin-based secondary sulfonamides as potent and selective inhibitors of cancer-related carbonic anhydrase IX and XII isoforms
2017 D'Ascenzio, M.; Guglielmi, P.; Carradori, S.; Secci, D.; Florio, R.; Mollica, A.; Ceruso, M.; Akdemir, A.; Sobolev, A. P.; Supuran, C. T.
3-(Phenyl-4-oxy)-5-phenyl-4,5-dihydro-(1H)-pyrazole: a fascinating molecular framework to study the enantioseparation ability of the amylose (3,5-dimethylphenylcarbamate) chiral stationary phase. Part II. Solvophobic effects in enantiorecognition process
2017 Pierini, Marco; Carradori, Simone; Menta, Sergio; Secci, Daniela; Cirilli, Roberto
Neem oil nanoemulsions: characterisation and antioxidant activity
2017 Rinaldi, Federica; Hanieh, PATRIZIA NADIA; Longhi, Catia; Carradori, Simone; Secci, Daniela; Zengin, Gokhan; Grazia Ammendolia, Maria; Mattia, Elena; Del Favero, Elena; Marianecci, Carlotta; Carafa, Maria
Protective effects Induced by microwave-assisted aqueous harpagophytum extract on rat cortex synaptosomes challenged with amyloid β-peptide
2017 Ferrante, Claudio; Recinella, Lucia; Locatelli, Marcello; Guglielmi, Paolo; Secci, Daniela; Leporini, Lidia; Chiavaroli, Annalisa; Leone, Sheila; Martinotti, Sara; Brunetti, Luigi; Vacca, Michele; Meneghini, Luigi; Orlando, Giustino
Synthesis, biological evaluation and quantitative structure-active relationships of 1,3-thiazolidin-4-one derivatives. A promising chemical scaffold endowed with high antifungal potency and low cytotoxicity
2017 Carradori, Simone; Bizzarri, Bruna; D'Ascenzio, Melissa; DE MONTE, Celeste; Grande, Rossella; Rivanera, Daniela; Zicari, Alessanda; Mari, Emanuela; Sabatino, Manuela; Patsilinakos, Alexandros; Ragno, Rino; Secci, Daniela
Synthesis and biological evaluation of anti-Toxoplasma gondii activity of a novel scaffold of thiazolidinone derivatives
2017 Carradori, Simone; Secci, Daniela; Bizzarri, Bruna; Chimenti, Paola; DE MONTE, Celeste; Guglielmi, Paolo; Campestre, Cristina; Rivanera, Daniela; Bordón, Claudia; Jones Brando, Lorraine
Identification of new anti-Candida compounds by ligand-based pharmacophore virtual screening
2016 Gidaro, Concetta; Alcaro, Stefano; Secci, Daniela; Rivanera, Daniela; Mollica, Adriano; Agamennone, Mariangela; Giampietro, Letizia; Simone Carradori, And
Elucidation of the mechanisms governing the thermal diastereomerization of bioactive chiral 1,3,4-thiadiazoline spiro-cyclohexyl derivatives towards their anancomeric stereoisomers
2016 Menta, Sergio; Carradori, S.; Siani, G.; Secci, Daniela; Mannina, Luisa; Sobolev, A. P.; Cirilli, R; Pierini, Marco
Novel 1,3-thiazolidin-4-one derivatives as promising anti-Candida agents endowed with anti-oxidant and chelating properties
2016 Secci, Daniela; Simone, Carradori; Bizzarri, Bruna; Chimenti, Paola; DE MONTE, Celeste; Adriano, Mollica; Rivanera, Daniela; Zicari, Alessandra; Emanuela, Mari; Gokhan, Zengin; Abdurrahman, Aktumsek
A novel library of saccharin and acesulfame derivatives as potent and selective inhibitors of carbonic anhydrase IX and XII isoforms
2016 Carradori, Simone; Secci, Daniela; DE MONTE, Celeste; Mollica, Adriano; Ceruso, Mariangela; Akdemir, Atilla; Sobolev, Anatoly P; Codispoti, Rossella; DE COSMI, Federica; Guglielmi, Paolo; Supuran, Claudiu T.
Anti-Candida activity and cytotoxicity of a large library of new N-substituted-1,3-thiazolidin-4-one derivatives
2016 DE MONTE, Celeste; Carradori, Simone; Bizzarri, Bruna; Bolasco, Adriana; Caprara, Federica; Mollica, Adriano; Rivanera, Daniela; Mari, Emanuela; Zicari, Alessandra; Akdemir, Atilla; Secci, Daniela
3-(Phenyl-4-oxy)-5-phenyl-4,5-dihydro-(1H)-pyrazole: a fascinating molecular framework to study the enantioseparation ability of the amylose (3,5-dimethylphenylcarbamate) chiral stationary phase. Part I. Structure-enantioselectivity relationships
2016 Carradori, Simone; Pierini, Marco; Menta, Sergio; Secci, Daniela; Fioravanti, Rossella; Cirilli, Roberto
Histone acetyltransferase inhibitor CPTH6 preferentially targets lung cancer stem-like cells
2016 DI MARTILE, Marta; Desideri, Marianna; DE LUCA, Teresa; Gabellini, Chiara; Buglioni, Simonetta; Eramo, Adriana; Sette, Giovanni; Milella, MICHELE STANISLAW; Rotili, Dante; Mai, Antonello; Carradori, Simone; Secci, Daniela; De Maria, Ruggero; Del Bufalo, Donatella; Trisciuoglio, Daniela
Out of the active site binding pocket for carbonic anhydrase inhibitors
2015 D'Ambrosio, K.; Carradori, S.; Monti, Sm; Buonanno, M.; Secci, Daniela; Vullo, D.; Supuran, Ct; De Simone, G.
The anancomeric character of the pharmacophore 1,3,4-thiadiazoline framework in chiral spiro-cyclohexyl derivatives: effects on stereochemistry and spiro-junction lability. Thermodynamic aspects
2015 Menta, Sergio; Carradori, Simone; Secci, Daniela; Faggi, Cristina; Mannina, Luisa; Cirilli, Roberto; Pierini, Marco
Optimization of the microwave-assisted extraction of Azadirachta indica (Neem) leaves Using NMR-based metabolic fingerprinting
2015 Carradori, Simone; Mannina, Luisa; Cosmi, Federica De; Beccarini, Tamara; Secci, Daniela; Sobolevb, Anatoly P.
Metal-chelating salens and tetrahydrosalens and N- and O-substituted acesulfame and saccharin derivatives as selective inhibitors of the cancer-related carbonic anhydrases IX and XII
2015 DE MONTE, Celeste; Secci, Daniela; Simone, Carradori; Melissa, D’Ascenzio; Mariana, Farella; Claudiu T., Supuran
Synthesis and pharmacological screening of a large library of 1,3,4-thiadiazolines as innovative therapeutic tools for the treatment of prostate cancer and melanoma
2015 DE MONTE, Celeste; Carradori, Simone; Secci, Daniela; D'Ascenzio, Melissa; Guglielmi, Paolo; Mollica, Adriano; Morrone, Stefania; Scarpa, Susanna; Agliano', Anna Maria; Giantulli, Sabrina; Silvestri, Ida
Identification of the stereochemical requirements in the 4-aryl-2-cycloalkylidenhydrazinylthiazole scaffold for the design of selective human monoamine oxidase B inhibitors
2014 D'Ascenzio, M; Carradori, S; Secci, Daniela; Mannina, Luisa; Sobolev, Ap; DE MONTE, Celeste; Cirilli, R; Yanez, M; Alcaro, S; Ortuso, F.
New insights into the biological properties of Crocus sativus L.: chemical modifications, human monoamine oxidases inhibition and molecular modeling studies
2014 DE MONTE, Celeste; Carradori, Simone; Chimenti, Paola; Secci, Daniela; Mannina, Luisa; Alcaro, F; Petzer, A; N'Da, Ci; Gidaro, Mc; Costa, G; Alcaro, S; Petzer, Jp
Synthesis of a novel series of thiazole-based histone acetyltransferase inhibitors
2014 Secci, Daniela; Carradori, S.; Bizzarri, Bruna; Bolasco, Adriana; Ballario, Paola; Patramani, Z.; Fragapane, P.; Vernarecci, S.; Canzonetta, C.; Filetici, P.
Selective inhibition of human carbonic anhydrases by novel amide derivatives of probenecid: Synthesis, biological evaluation and molecular modelling studies
2014 D'Ascenzio, M; Carradori, S; Secci, Daniela; Vullo, D; Ceruso, M; Akdemir, A; Supuran, Ct
Evaluation of a large library of (thiazol-2-yl)hydrazones and analogues as histone acetyltransferase inhibitors: Enzyme and cellular studies.
2014 Carradori, S; Rotili, Dante; DE MONTE, Celeste; Lenoci, A; D'Ascenzio, M; Rodriguez, V; Filetici, Patrizia; Miceli, M; Nebbioso, A; Altucci, L; Secci, Daniela; Mai, Antonello
Design, synthesis and biological characterization of thiazolidin-4-one derivatives as promising inhibitors of Toxoplasma gondii
2014 D'Ascenzio, Melissa; Bizzarri, Bruna; DE MONTE, Celeste; Carradori, S; Bolasco, Adriana; Secci, Daniela; Rivanera, Daniela; Faulhaber, N; Bordon, C; Jones Brando, L.
Microwave and Ultrasound-Assisted Synthesis of Thiosemicarbazones and Their Corresponding (4,5-Substituted-thiazol-2-yl)hydrazines
2014 Carradori, S; Secci, Daniela; D'Ascenzio, M; Chimenti, Paola; Bolasco, Adriana
Quinoline-based p300 histone acetyltransferase inhibitors with pro-apoptotic activity in human leukemia U937 cells.
2014 Lenoci, Alessia; Tomassi, S; Conte, M; Benedetti, R; Rodriguez, V; Carradori, Simone; Secci, Daniela; Castellano, S; Sbardella, G; Filetici, P; Novellino, E; Altucci, L; Rotili, Dante; Mai, Antonello
Selective MAO-B inhibitors: a lesson from natural products
2014 Carradori, Simone; D'Ascenzio, Melissa; Chimenti, Paola; Secci, Daniela; Bolasco, Adriana
Effect of the water content on the retention and enantioselectivity of albendazole and fenbendazole sulfoxides using amylose-based chiral stationary phases in organic-acqueous conditions
2014 Materazzo, S.; Carradori, Simone; Ferretti, R.; Gallinella, B.; Secci, Daniela; Cirilli, R.
Cyclic tertiary sulfamates: Selective inhibition of the tumor-associated carbonic anhydrases IX and XII by N- and O-substituted acesulfame derivatives
2014 DE MONTE, Celeste; Carradori, Simone; Secci, Daniela; D'Ascenzio, Melissa; Vullo, D; Ceruso, M; Supuran, Ct
Design, synthesis and evaluation of N-substituted saccharin derivatives as selective inhibitors of tumor-associated carbonic anhydrase XII
2014 D'Ascenzio, M; Carradori, S; DE MONTE, Celeste; Secci, Daniela; Ceruso, M; Supuran, Ct
New thiadiazoline and thiadiazole analogues of K858: antiproliferative activity in a model of prostate carcinoma
2013 DE MONTE, Celeste; Carradori, S.; D’Ascenzio, M.; Chimenti, Paola; Secci, Daniela; Bolasco, Adriana; Nicolazzo, Chiara; Silvestri, Ida
Synthesis and Selective Human Monoamine Oxidase B Inhibition of Heterocyclic Hybrids Based on Hydrazine and Thiazole Scaffolds
2013 Simone, Carradori; Melissa, D'Ascenzio; DE MONTE, Celeste; Secci, Daniela; Matilde, Yáñez
Synthesis and cytotoxicity of novel (thiazol-2-yl)hydrazine derivatives as promising anti-Candida agents
2013 Simone, Carradori; Secci, Daniela; Bolasco, Adriana; Rivanera, Daniela; Mari, Emanuela; Zicari, Alessandra; Lotti, Lavinia Vittoria; Bizzarri, Bruna
Exploring (4-substituted-thiazol-2-yl)hydrazine derivatives of 2-, 3-, and 4-acetylpyridine as selective and reversible hMAO-B inhibitors.
2013 Chimenti, Paola; Petzer, A.; Carradori, S.; D’Ascenzio, M.; Silvestri, Romano; Alcaro, S.; Ortuso, F.; Petzer, J. J.; Secci, Daniela
Salen and tetrahydrosalen derivatives act as effective inhibitors of the tumor-associated carbonic anhydrase XII—A new scaffold for designing isoform-selective inhibitors
2013 Carradori, Simone; DE MONTE, Celeste; D'Ascenzio, Melissa; Secci, Daniela; Gulsah, Celik; Mariangela, Ceruso; Daniela, Vullo; Andrea, Scozzafava; Claudiu T., Supuran
tert-Butylcarbamate-Containing Histone Deacetylase Inhibitors: Apoptosis Induction, Cytodifferentiation, and Antiproliferative Activities in Cancer Cells.
2013 Valente, Sergio; Trisciuoglio, D; Tardugno, M; Benedetti, R; Labella, Donatella; Secci, Daniela; Mercurio, C; Boggio, R; Tomassi, S; Di Maro, S; Novellino, E; Altucci, L; Del Bufalo, D; Mai, Antonello; Cosconati, S.
The thiazole derivative CPTH6 impairs autophagy
2013 Ragazzoni, Ylenia; M., Desideri; C., Gabellini; T., De Luca; Carradori, Simone; Secci, Daniela; Nescatelli, Riccardo; A., Candiloro; M., Condello; S., Meschini; D., Del Bufalo; D., Trisciuoglio
Modulation of autophagic flux by CPTH6, a thiazole derivative with antitumoral activity
2012 Ragazzoni, Ylenia; M., Desideri; C., Gabellini; Carradori, Simone; Nescatelli, Riccardo; Secci, Daniela; A., Candiloro; D., Trisciuoglio; D., Del Bufalo
Discovery and optimization of pyrazoline derivatives as promising monoamine oxidase inhibitors
2012 Secci, Daniela; Carradori, Simone; Bolasco, Adriana; Bizzarri, Bruna; D'Ascenzio, Melissa; E., Maccioni
Synthesis and selective inhibitory activity against human COX-1 of novel 1-(4-substituted-thiazol-2-yl)-3,5-di(hetero)aryl-pyrazoline derivatives.
2012 S., Carradori; Secci, Daniela; Bolasco, Adriana; DE MONTE, Celeste; M., Yanez
Modulation of Autophagic Flux by CPTH6, a Gcn5/pCAF Histone Acetyltransferase Inhibitor With Antitumoral Activity
2012 D., Trisciuoglio; Ragazzoni, Ylenia; M., Desideri; C., Gabellini; Nescatelli, Riccardo; Carradori, Simone; Secci, Daniela; D., Del Bufalo
Conventional and Microwave-Assisted Synthesis of Benzimidazole Derivatives and their in vitro Inhibition of human Cyclooxygenase.
2012 Secci, Daniela; Bolasco, Adriana; D’Ascenzio, M.; della Sala, F.; Yáñez, M.; Carradori, Simone
Synthesis, anti-Candida activity, and cytotoxicity of new (4-(4-iodophenyl)thiazol-2-yl)hydrazine derivatives
2012 Secci, Daniela; Bizzarri, Bruna; Bolasco, Adriana; Simone, Carradori; D'Ascenzio, Melissa; Rivanera, Daniela; Mari, Emanuela; Polletta, Lucia; Zicari, Alessandra
Current and emerging strategies in bladder cancer
2012 Carradori, Simone; Cristini, Cristiano; Secci, Daniela; Caterina, Gulia; Gentile, Vincenzo; DI PIERRO, GIOVANNI BATTISTA
METHOD FOR PRODUCTION OF AMOTPHOUS RIFAXIMIN
2012 Lavagna, Silvio Massimo; Secci, Daniela; Padella, Franco
MANGANESE IRON OXIDE SUPERPARAMAGNETIC POWDER BY MECHANOCHEMICAL PROCESSING. NANOPARTICLES FUNCTIONALIZATION AND DISPERSION IN A NANOFLUID
2012 Bellusci, Mariangela; Aliotta, C.; Fiorani, D.; LA BARBERA, A.; Padella, F.; Peddis, D.; Pilloni, M.; Secci, Daniela
Patent-related survey on new monoamine oxidase inhibitors and their therapeutic potential
2012 Carradori, Simone; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; D'Ascenzio, Melissa
3-Methylcyclohexanone thiosemicarbazone: Determination of E/Z isomerization barrier by dynamic high-performance liquid chromatography, configuration assignment and theoretical study of the mechanisms involved by the spontaneous, acid and base catalyzed processes
2012 Carradori, Simone; Cirilli, R.; Dei Cicchi, S.; Ferretti, R.; Menta, Sergio; Pierini, Marco; Secci, Daniela
Synthesis and biological assessment of novel 2-thiazolylhydrazones and computational analysis of their recognition by monoamine oxidase B
2012 Distinto, S; Yáñez, M; Alcaro, S.; Cardia M., C; Gaspari, M; Sanna M., L; Meleddu, R; Ortuso, F; Kirchmair, J; Markt, P; Bolasco, Adriana; Wolber, G; Secci, Daniela; Maccioni, E.
CPTH6, a thiazole derivative, induces histone hypoacetylation and apoptosis in human leukemia cells
2012 D., Trisciuoglio; Ragazzoni, Ylenia; A., Pelosi; M., Desideri; Carradori, Simone; C., Gabellini; G., Maresca; Nescatelli, Riccardo; Secci, Daniela; Bolasco, Adriana; Bizzarri, Bruna; Cavaliere, Chiara; I., D'Agnano; Filetici, Patrizia; L., Ricci Vitiani; M. G., Rizzo; D., Del Bufalo
Recent advances in the development of selective human MAO-B inhibitors: (Hetero)arylidene-(4-substituted-thiazol-2- yl)hydrazines
2012 Secci, Daniela; Bolasco, Adriana; Carradori, Simone; D'Ascenzio, Melissa; Nescatelli, Riccardo; M., Yáñez
CPTH6, A NOVEL Gcn5/pCAF HISTONE ACETYLTRANSFERASE INHIBITOR, INDUCES BOTH APOPTOSIS AND AUTOPHAGY IN HUMAN LEUKEMIA CELLS
2011 Ragazzoni, Y.; Trisciuoglio, D.; Gabellini, C. .; Pelosi, A.; Desideri, M.; Carradori, Simone; Secci, Daniela; Rizzo, M. G.; Del, Bufalo
The State of the Art of Pyrazole Derivatives as Monoamine Oxidase Inhibitors and Antidepressant/Anticonvulsant Agents
2011 Secci, Daniela; Bolasco, Adriana; Carradori, Simone; Chimenti, Paola
FULL AMORPHOUS RIFAXIMIN AND METHODS FOR ITS PREPARATION
2011 Lavagna, Silvio Massimo; Secci, Daniela; Padella, Franco
METHOD FOR THE PRODUCTION OF AMORPHOUS RIFAXIMIN
2011 Lavagna, Silvio Massimo; Secci, Daniela; Franco, Padella
Synthesis and selective human monoamine oxidase inhibition of 3-carbonyl, 3-acyl, and 3-carboxyhydrazido coumarin derivatives
2011 Secci, Daniela; Carradori, Simone; Bolasco, Adriana; Chimenti, Paola; Yanez, Matilde; Ortuso, Francesco; Alcaro, Stefano
Synthesis and biological evaluation of novel 2,4-disubstituted-1,3-thiazoles as anti-Candida spp. agents
2011 Franco, Chimenti; Bizzarri, Bruna; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Granese, Arianna; Simone, Carradori; Melissa, D'Ascenzio; Lilli, Daniela; Rivanera, Daniela
EPIGENETIC MODULATION OF PGC-1a ACTIVITY BY GCN5 INHIBITORS: WO2010007085
2011 Carradori, Simone; Secci, Daniela; Mai, Antonello
A new series of flavones, thioflavones, and flavanones as selective monoamine oxidase-B inhibitors
2010 Chimenti, Franco; Fioravanti, Rossella; Bolasco, Adriana; Chimenti, Paola; Secci, Daniela; Rossi, Francesca; Matilde, Yanez; Francisco, Orallo; Francesco, Ortuso; Stefano, Alcaro; Roberto, Cirilli; Rosella, Ferretti; M., Luisa Sanna
Synthesis and characterization of new 3-acyl-7-hydroxy-6,8-substituted-coumarin and 3-acyl-7-benzyloxy-6,8-substituted-coumarin derivatives
2010 Chimenti, Franco; Bolasco, Adriana; Secci, Daniela; Bizzarri, Bruna; Chimenti, Paola; Granese, A; Carradori, S.
Synthesis, semipreparative HPLC separation, biological evaluation, and 3D-QSAR of hydrazothiazole derivatives as human monoamine oxidase B inhibitors
2010 Chimenti, Franco; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Arianna, Granese; Simone, Carradori; Elias, Maccioni; M., Cristina Cardia; Matilde, Yanez; Francisco, Orallo; Stefano, Alcaro; Francesco, Ortuso; Roberto, Cirilli; Rosella, Ferretti; Simona, Distinto; Johannes, Kirchmair; Thierry, Langer
Synthesis of new 3-aryl-4,5-dihydropyrazole-1-carbothioamide derivatives. An investigation on their ability to inhibit monoamine oxidase
2010 Maccioni, E.; Alcaro, S.; Orallo, F.; Cardia, M. C.; Distinto, S.; Costa, G.; Yanez, M.; Sanna, M. L.; Vigo, S.; Meleddu, R.; Secci, D.
Investigations on the 2-thiazolylhydrazyne scaffold: Synthesis and molecular modeling of selective human monoamine oxidase inhibitors
2010 Chimenti, Franco; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Arianna, Granese; Simone, Carradori; Matilde, Yanez; Francisco, Orallo; Francesco, Ortuso; Stefano, Alcaro
FULL AMORPHOUS RIFAXIMIN AND METHODS FOR ITS PREPARATION
2010 Lavagna, Silvio Massimo; Secci, Daniela; Padella, Franco
METODO PER LA PREPARAZIONE DI RIFAXIMINA IN STATO AMORFO
2010 Lavagna, Silvio Massimo; Secci, Daniela; Padella, Franco
SYNTHESIS, STEREOCHEMICAL SEPARATION, AND BIOLOGICAL EVALUATION OF SELECTIVE INHIBITORS OF HUMAN MAO-B: 1-(4-ARYLTHIAZOL-2-YL)-2-(3-METHYLCYCLOHEXYLIDENE)HYDRAZINES
2010 Chimenti, Franco; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Granese, A; Carradori, S; Yanez, M; Orallo, F; Sanna, Ml; Gallinella, B; Cirilli, R.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Indoleamine 2,3-dioxygenase | 2023 | Coluccia, Michele; Secci, Daniela; Guglielmi, Paolo | |
A Multitarget Approach against Neuroinflammation: Alkyl Substituted Coumarins as Inhibitors of Enzymes Involved in Neurodegeneration | 2023 | Berrino, E.; Carradori, S.; Carta, F.; Melfi, F.; Gallorini, M.; Poli, G.; Tuccinardi, T.; Fernandez-Bolanos, J. G.; Lopez, O.; Petzer, J. P.; Petzer, A.; Guglielmi, P.; Secci, D.; Supuran, C. T. | |
Novel Insights on CAI–CORM Hybrids: Evaluation of the CO Releasing Properties and Pain-Relieving Activity of Differently Substituted Coumarins for the Treatment of Rheumatoid Arthritis | 2023 | Berrino, Emanuela; Micheli, Laura; Carradori, Simone; di Cesare Mannelli, Lorenzo; Guglielmi, Paolo; De Luca, Alessandro; Carta, Fabrizio; Ghelardini, Carla; Secci, Daniela; Supuran, Claudiu T. | |
Kinetic Study on the Base-Catalyzed Imine-Enamine Tautomerism of a Chiral Biologically Active Isoxazoline Derivative by HPLC on Amylose Tris(3,5-dimethylphenylcarbamate) Chiral Stationary Phase | 2023 | Sadutto, Daniele; Guglielmi, Paolo; Carradori, Simone; Secci, Daniela; Cirilli, Roberto | |
A comparative study on the suppression capacity and the environmental impact of different extinguishing agents of lithium-ion battery fires | 2022 | Ubaldi, Sofia; Di Bari, Cinzia; De Rosa, Armando; Quinterno, Mario; Mazzaro, Michele; Ferrigno, Gianluca; Arrighi, Francesca; Secci, Daniela; Russo, Paola | |
Novel Insights on Human Carbonic Anhydrase Inhibitors Based on Coumalic Acid: Design, Synthesis, Molecular Modeling Investigation, and Biological Studies | 2022 | Pontecorvi, Virginia; Mori, Mattia; Picarazzi, Francesca; Zara, Susi; Carradori, Simone; Cataldi, Amelia; Angeli, Andrea; Berrino, Emanuela; Chimenti, Paola; Ciogli, Alessia; Secci, Daniela; Guglielmi, Paolo; Supuran, Claudiu T. | |
Treatment of Toxoplasmosis: An Insight on Epigenetic Drugs | 2022 | Guglielmi, P.; Secci, D. | |
Metal-organic frameworks (MOFs) as biomolecules drug delivery systems for anticancer purposes | 2022 | Coluccia, Michele; Parisse, Valeria; Guglielmi, Paolo; Giannini, Giuseppe; Secci, Daniela | |
Synthesis and evaluation of thymol-based synthetic derivatives as dual-action inhibitors against different strains of h. pylori and AGS cell line | 2021 | Sisto, F.; Carradori, S.; Guglielmi, P.; Spano, M.; Secci, D.; Granese, A.; Sobolev, A. P.; Grande, R.; Campestre, C.; Di Marcantonio, M. C.; Mincione, G. | |
An innovative spectroscopic approach for qualitative and quantitative evaluation of Mb-CO from myoglobin carbonylation reaction through chemometrics methods | 2021 | Mansoldo, F. R. P.; Berrino, E.; Guglielmi, P.; Carradori, S.; Carta, F.; Secci, D.; Supuran, C. T.; Vermelho, A. B. | |
Chalcones: Unearthing their therapeutic possibility as monoamine oxidase B inhibitors | 2020 | Guglielmi, Paolo; Mathew, Bijo; Secci, Daniela; Carradori, Simone | |
Innovative pH-interfering agents in association with anticancer agents | 2020 | Secci, D.; Guglielmi, P. | |
Inhibition of lysine acetyltransferases impairs tumor angiogenesis acting on both endothelial and tumor cells | 2020 | Di Martile, Marta; Gabellini, Chiara; Desiderio, Marianna; Matraxia, Marta; Farini, Valentina; Valentini, Elisabetta; Carradori, Simone; Ercolani, Cristiana; Buglioni, Simonetta; Secci, Daniela; Andreazzoli, Massimiliano; Del Bufalo and Daniela Trisciuoglio, Donatella | |
Synthesis and biological evaluation of carvacrol-based derivatives as dual inhibitors of H. Pylori strains and ags cell proliferation | 2020 | Sisto, F.; Carradori, S.; Guglielmi, P.; Traversi, C. B.; Spano, M.; Sobolev, A. P.; Secci, D.; Di Marcantonio, M. C.; Haloci, E.; Grande, R.; Mincione, G. | |
Antimalarial agents from medicinal plant and fungal sources | 2020 | Luisi, Grazia; Carradori, Simone; Grande, Rossella; Secci, Daniela; Guglielmi, Paolo | |
Metabolic profiling of different wild and cultivated Allium species based on high-resolution mass spectrometry, high-performance liquid chromatography-photodiode array detector, and color analysis | 2020 | Maccelli, A.; Cesa, S.; Cairone, F.; Secci, D.; Menghini, L.; Chiavarino, B.; Fornarini, S.; Crestoni, M. E.; Locatelli, M. | |
1,3-Dipolar Cycloaddition, HPLC Enantioseparation, and Docking Studies of Saccharin/Isoxazole and Saccharin/Isoxazoline Derivatives as Selective Carbonic Anhydrase IX and XII Inhibitors | 2020 | D'Ascenzio, M.; Secci, D.; Carradori, S.; Zara, S.; Guglielmi, P.; Cirilli, R.; Pierini, M.; Poli, G.; Tuccinardi, T.; Angeli, A.; Supuran, C. T. | |
High-performance liquid chromatography enantioseparation of chiral 2-(benzylsulfinyl)benzamide derivatives on cellulose tris(3,5-dichlorophenylcarbamate) chiral stationary phase | 2020 | Carradori, S.; Secci, D.; Guglielmi, P.; Pierini, M.; Cirilli, R. | |
Synthesis and evaluation of a large library of nitroxoline derivatives as pancreatic cancer antiproliferative agents | 2020 | Veschi, Serena; Carradori, Simone; De Lellis, Laura; Florio, Rosalba; Brocco, Davide; Secci, Daniela; Guglielmi, Paolo; Spano, Mattia; Sobolev, Anatoly P.; Cama, Alessandro | |
Novel insights on saccharin- and acesulfame-based carbonic anhydrase inhibitors: design, synthesis, modelling investigations and biological activity evaluation | 2020 | Guglielmi, P.; Rotondi, G.; Secci, D.; Angeli, A.; Chimenti, P.; Nocentini, A.; Bonardi, A.; Gratteri, P.; Carradori, S.; Supuran, C. T. | |
Novel approaches to the discovery of selective human monoamine oxidase-B inhibitors: is there room for improvement? | 2019 | Guglielmi, P.; Carradori, S.; Ammazzalorso, A.; Secci, D. | |
4-(3-Nitrophenyl)thiazol-2-ylhydrazone derivatives as antioxidants and selective hMAO-B inhibitors: synthesis, biological activity and computational analysis | 2019 | Secci, Daniela; Carradori, Simone; Petzer, Anél; Guglielmi, Paolo; D’Ascenzio, Melissa; Chimenti, Paola; Bagetta, Donatella; Alcaro, Stefano; Zengin, Gokhan; Petzer, Jacobus P.; Ortuso, Francesco | |
Investigation on the stability of new biologically active thiosemicarbazone-derived compounds by a validated HPLC-PDA method | 2019 | Secci, Daniela; Locatelli, Marcello; Kabir, Abuzar; Salvatorelli, Erika; Macedonio, Giorgia; Mollica and Simone Carradori, Adriano | |
Benzo[b]tiophen-3-ol derivatives as effective inhibitors of human monoamine oxidase: design, synthesis, and biological activity | 2019 | Guglielmi, Paolo; Secci, Daniela; Petzer, Anél; Bagetta, Donatella; Chimenti, Paola; Rotondi, Giulia; Ferrante, Claudio; Recinella, Lucia; Leone, Sheila; Alcaro, Stefano; Zengin, Gokhan; Petzer, Jacobus P; Ortuso, Francesco; Carradori, Simone | |
Design, synthesis, docking studies and monoamine oxidase inhibition of a small library of 1-acetyl- and 1-thiocarbamoyl-3,5-diphenyl-4,5-dihydro-(1h)-pyrazoles | 2019 | Guglielmi, Paolo; Carradori, Simone; Poli, Giulio; Secci, Daniela; Cirilli, Roberto; Rotondi, Giulia; Chimenti, Paola; Petzer, Anél; Petzer, Jacobus P. | |
Design, synthesis and biological activity of selective hCAs inhibitors based on 2-(benzylsulfinyl)benzoic acid scaffold | 2019 | Rotondi, G.; Guglielmi, P.; Carradori, S.; Secci, D.; De Monte, C.; De Filippis, B.; Maccallini, C.; Amoroso, R.; Cirilli, R.; Akdemir, A.; Angeli, A.; Supuran, C. T. | |
Atriplex mollis desf. Aerial parts: extraction procedures, secondary metabolites and color analysis | 2018 | Boutaoui, Nassima; Zaiter, Lahcene; Benayache, Fadila; Benayache, Samir; Cacciagrano, Francesco; Cesa, Stefania; Secci, Daniela; Carradori, Simone; Giusti, Anna Maria; Campestre, Cristina; Menghini, Luigi; Locatelli, Marcello | |
MAO inhibitors and their wider applications: a patent review | 2018 | Carradori, Simone; Secci, Daniela; Petzer, Jacques P. | |
A chromatographic study on the exceptional chiral recognition of 2-(benzylsulfinyl)benzamide by animmobilized-type chiral stationary phase based on cellulose tris(3,5-dichlorophenylcarbamate) | 2018 | Carradori, Simone; Secci, Daniela; Faggi, Cristina; Cirilli, Roberto | |
Bioactive isoflavones from Pueraria lobata root and starch: Different extraction techniques and carbonic anhydrase inhibition | 2018 | Mocan, Andrei; Carradori, Simone; Locatelli, Marcello; Secci, Daniela; Cesa, Stefania; Mollica, Adriano; Riga, Simona; Angeli, Andrea; Supuran, Claudiu T.; Celia, Christian; Di Marzio, Luisa | |
Magnetic metal−organic framework composite by fast and facile mechanochemical process | 2018 | Bellusci, M.; Guglielmi, P.; Masi, Andrea; Padella, F.; Singh, G.; Yaacoub, N.; Peddis, D.; Secci, D. | |
Design, synthesis and biochemical evaluation of novel multi-target inhibitors as potential anti-Parkinson agents | 2018 | Carradori, Simone; Ottuso, Francesco; Petzer, Anèl; Bagetta, Donatella; DE MONTE, Celeste; Secci, Daniela; DE VITA, Daniela; Guglielmi, Paolo; Zengin, Gokhan; Aktumsek, Abdurrahman; Alcaro, Stefano; Petzer, Jacobus P. | |
Geographical characterization by MAE-HPLC and NIR methodologies and carbonic anhydrase inhibition of Saffron components | 2017 | Nescatelli, Riccardo; Carradori, Simone; Marini, Federico; Caponigro, Vicky; Bucci, Remo; DE MONTE, Celeste; Mollica, Adriano; Mannina, Luisa; Ceruso, Mariangela; Supuran, CLAUDIU TRANDAFIR; Secci, Daniela | |
Optimization of aqueous extraction and biological activity of harpagophytum procumbens root on ex vivo rat Colon inflammatory model | 2017 | Locatelli, Marcello; Ferrante, Claudio; Carradori, Simone; Secci, Daniela; Leporini, Lidia; Chiavaroli, Annalisa; Leone, Sheila; Recinella, Lucia; Orlando, Giustino; Martinotti, Sara; Brunetti, Luigi; Vacca And Luigi Menghini, Michele | |
Open saccharin-based secondary sulfonamides as potent and selective inhibitors of cancer-related carbonic anhydrase IX and XII isoforms | 2017 | D'Ascenzio, M.; Guglielmi, P.; Carradori, S.; Secci, D.; Florio, R.; Mollica, A.; Ceruso, M.; Akdemir, A.; Sobolev, A. P.; Supuran, C. T. | |
3-(Phenyl-4-oxy)-5-phenyl-4,5-dihydro-(1H)-pyrazole: a fascinating molecular framework to study the enantioseparation ability of the amylose (3,5-dimethylphenylcarbamate) chiral stationary phase. Part II. Solvophobic effects in enantiorecognition process | 2017 | Pierini, Marco; Carradori, Simone; Menta, Sergio; Secci, Daniela; Cirilli, Roberto | |
Neem oil nanoemulsions: characterisation and antioxidant activity | 2017 | Rinaldi, Federica; Hanieh, PATRIZIA NADIA; Longhi, Catia; Carradori, Simone; Secci, Daniela; Zengin, Gokhan; Grazia Ammendolia, Maria; Mattia, Elena; Del Favero, Elena; Marianecci, Carlotta; Carafa, Maria | |
Protective effects Induced by microwave-assisted aqueous harpagophytum extract on rat cortex synaptosomes challenged with amyloid β-peptide | 2017 | Ferrante, Claudio; Recinella, Lucia; Locatelli, Marcello; Guglielmi, Paolo; Secci, Daniela; Leporini, Lidia; Chiavaroli, Annalisa; Leone, Sheila; Martinotti, Sara; Brunetti, Luigi; Vacca, Michele; Meneghini, Luigi; Orlando, Giustino | |
Synthesis, biological evaluation and quantitative structure-active relationships of 1,3-thiazolidin-4-one derivatives. A promising chemical scaffold endowed with high antifungal potency and low cytotoxicity | 2017 | Carradori, Simone; Bizzarri, Bruna; D'Ascenzio, Melissa; DE MONTE, Celeste; Grande, Rossella; Rivanera, Daniela; Zicari, Alessanda; Mari, Emanuela; Sabatino, Manuela; Patsilinakos, Alexandros; Ragno, Rino; Secci, Daniela | |
Synthesis and biological evaluation of anti-Toxoplasma gondii activity of a novel scaffold of thiazolidinone derivatives | 2017 | Carradori, Simone; Secci, Daniela; Bizzarri, Bruna; Chimenti, Paola; DE MONTE, Celeste; Guglielmi, Paolo; Campestre, Cristina; Rivanera, Daniela; Bordón, Claudia; Jones Brando, Lorraine | |
Identification of new anti-Candida compounds by ligand-based pharmacophore virtual screening | 2016 | Gidaro, Concetta; Alcaro, Stefano; Secci, Daniela; Rivanera, Daniela; Mollica, Adriano; Agamennone, Mariangela; Giampietro, Letizia; Simone Carradori, And | |
Elucidation of the mechanisms governing the thermal diastereomerization of bioactive chiral 1,3,4-thiadiazoline spiro-cyclohexyl derivatives towards their anancomeric stereoisomers | 2016 | Menta, Sergio; Carradori, S.; Siani, G.; Secci, Daniela; Mannina, Luisa; Sobolev, A. P.; Cirilli, R; Pierini, Marco | |
Novel 1,3-thiazolidin-4-one derivatives as promising anti-Candida agents endowed with anti-oxidant and chelating properties | 2016 | Secci, Daniela; Simone, Carradori; Bizzarri, Bruna; Chimenti, Paola; DE MONTE, Celeste; Adriano, Mollica; Rivanera, Daniela; Zicari, Alessandra; Emanuela, Mari; Gokhan, Zengin; Abdurrahman, Aktumsek | |
A novel library of saccharin and acesulfame derivatives as potent and selective inhibitors of carbonic anhydrase IX and XII isoforms | 2016 | Carradori, Simone; Secci, Daniela; DE MONTE, Celeste; Mollica, Adriano; Ceruso, Mariangela; Akdemir, Atilla; Sobolev, Anatoly P; Codispoti, Rossella; DE COSMI, Federica; Guglielmi, Paolo; Supuran, Claudiu T. | |
Anti-Candida activity and cytotoxicity of a large library of new N-substituted-1,3-thiazolidin-4-one derivatives | 2016 | DE MONTE, Celeste; Carradori, Simone; Bizzarri, Bruna; Bolasco, Adriana; Caprara, Federica; Mollica, Adriano; Rivanera, Daniela; Mari, Emanuela; Zicari, Alessandra; Akdemir, Atilla; Secci, Daniela | |
3-(Phenyl-4-oxy)-5-phenyl-4,5-dihydro-(1H)-pyrazole: a fascinating molecular framework to study the enantioseparation ability of the amylose (3,5-dimethylphenylcarbamate) chiral stationary phase. Part I. Structure-enantioselectivity relationships | 2016 | Carradori, Simone; Pierini, Marco; Menta, Sergio; Secci, Daniela; Fioravanti, Rossella; Cirilli, Roberto | |
Histone acetyltransferase inhibitor CPTH6 preferentially targets lung cancer stem-like cells | 2016 | DI MARTILE, Marta; Desideri, Marianna; DE LUCA, Teresa; Gabellini, Chiara; Buglioni, Simonetta; Eramo, Adriana; Sette, Giovanni; Milella, MICHELE STANISLAW; Rotili, Dante; Mai, Antonello; Carradori, Simone; Secci, Daniela; De Maria, Ruggero; Del Bufalo, Donatella; Trisciuoglio, Daniela | |
Out of the active site binding pocket for carbonic anhydrase inhibitors | 2015 | D'Ambrosio, K.; Carradori, S.; Monti, Sm; Buonanno, M.; Secci, Daniela; Vullo, D.; Supuran, Ct; De Simone, G. | |
The anancomeric character of the pharmacophore 1,3,4-thiadiazoline framework in chiral spiro-cyclohexyl derivatives: effects on stereochemistry and spiro-junction lability. Thermodynamic aspects | 2015 | Menta, Sergio; Carradori, Simone; Secci, Daniela; Faggi, Cristina; Mannina, Luisa; Cirilli, Roberto; Pierini, Marco | |
Optimization of the microwave-assisted extraction of Azadirachta indica (Neem) leaves Using NMR-based metabolic fingerprinting | 2015 | Carradori, Simone; Mannina, Luisa; Cosmi, Federica De; Beccarini, Tamara; Secci, Daniela; Sobolevb, Anatoly P. | |
Metal-chelating salens and tetrahydrosalens and N- and O-substituted acesulfame and saccharin derivatives as selective inhibitors of the cancer-related carbonic anhydrases IX and XII | 2015 | DE MONTE, Celeste; Secci, Daniela; Simone, Carradori; Melissa, D’Ascenzio; Mariana, Farella; Claudiu T., Supuran | |
Synthesis and pharmacological screening of a large library of 1,3,4-thiadiazolines as innovative therapeutic tools for the treatment of prostate cancer and melanoma | 2015 | DE MONTE, Celeste; Carradori, Simone; Secci, Daniela; D'Ascenzio, Melissa; Guglielmi, Paolo; Mollica, Adriano; Morrone, Stefania; Scarpa, Susanna; Agliano', Anna Maria; Giantulli, Sabrina; Silvestri, Ida | |
Identification of the stereochemical requirements in the 4-aryl-2-cycloalkylidenhydrazinylthiazole scaffold for the design of selective human monoamine oxidase B inhibitors | 2014 | D'Ascenzio, M; Carradori, S; Secci, Daniela; Mannina, Luisa; Sobolev, Ap; DE MONTE, Celeste; Cirilli, R; Yanez, M; Alcaro, S; Ortuso, F. | |
New insights into the biological properties of Crocus sativus L.: chemical modifications, human monoamine oxidases inhibition and molecular modeling studies | 2014 | DE MONTE, Celeste; Carradori, Simone; Chimenti, Paola; Secci, Daniela; Mannina, Luisa; Alcaro, F; Petzer, A; N'Da, Ci; Gidaro, Mc; Costa, G; Alcaro, S; Petzer, Jp | |
Synthesis of a novel series of thiazole-based histone acetyltransferase inhibitors | 2014 | Secci, Daniela; Carradori, S.; Bizzarri, Bruna; Bolasco, Adriana; Ballario, Paola; Patramani, Z.; Fragapane, P.; Vernarecci, S.; Canzonetta, C.; Filetici, P. | |
Selective inhibition of human carbonic anhydrases by novel amide derivatives of probenecid: Synthesis, biological evaluation and molecular modelling studies | 2014 | D'Ascenzio, M; Carradori, S; Secci, Daniela; Vullo, D; Ceruso, M; Akdemir, A; Supuran, Ct | |
Evaluation of a large library of (thiazol-2-yl)hydrazones and analogues as histone acetyltransferase inhibitors: Enzyme and cellular studies. | 2014 | Carradori, S; Rotili, Dante; DE MONTE, Celeste; Lenoci, A; D'Ascenzio, M; Rodriguez, V; Filetici, Patrizia; Miceli, M; Nebbioso, A; Altucci, L; Secci, Daniela; Mai, Antonello | |
Design, synthesis and biological characterization of thiazolidin-4-one derivatives as promising inhibitors of Toxoplasma gondii | 2014 | D'Ascenzio, Melissa; Bizzarri, Bruna; DE MONTE, Celeste; Carradori, S; Bolasco, Adriana; Secci, Daniela; Rivanera, Daniela; Faulhaber, N; Bordon, C; Jones Brando, L. | |
Microwave and Ultrasound-Assisted Synthesis of Thiosemicarbazones and Their Corresponding (4,5-Substituted-thiazol-2-yl)hydrazines | 2014 | Carradori, S; Secci, Daniela; D'Ascenzio, M; Chimenti, Paola; Bolasco, Adriana | |
Quinoline-based p300 histone acetyltransferase inhibitors with pro-apoptotic activity in human leukemia U937 cells. | 2014 | Lenoci, Alessia; Tomassi, S; Conte, M; Benedetti, R; Rodriguez, V; Carradori, Simone; Secci, Daniela; Castellano, S; Sbardella, G; Filetici, P; Novellino, E; Altucci, L; Rotili, Dante; Mai, Antonello | |
Selective MAO-B inhibitors: a lesson from natural products | 2014 | Carradori, Simone; D'Ascenzio, Melissa; Chimenti, Paola; Secci, Daniela; Bolasco, Adriana | |
Effect of the water content on the retention and enantioselectivity of albendazole and fenbendazole sulfoxides using amylose-based chiral stationary phases in organic-acqueous conditions | 2014 | Materazzo, S.; Carradori, Simone; Ferretti, R.; Gallinella, B.; Secci, Daniela; Cirilli, R. | |
Cyclic tertiary sulfamates: Selective inhibition of the tumor-associated carbonic anhydrases IX and XII by N- and O-substituted acesulfame derivatives | 2014 | DE MONTE, Celeste; Carradori, Simone; Secci, Daniela; D'Ascenzio, Melissa; Vullo, D; Ceruso, M; Supuran, Ct | |
Design, synthesis and evaluation of N-substituted saccharin derivatives as selective inhibitors of tumor-associated carbonic anhydrase XII | 2014 | D'Ascenzio, M; Carradori, S; DE MONTE, Celeste; Secci, Daniela; Ceruso, M; Supuran, Ct | |
New thiadiazoline and thiadiazole analogues of K858: antiproliferative activity in a model of prostate carcinoma | 2013 | DE MONTE, Celeste; Carradori, S.; D’Ascenzio, M.; Chimenti, Paola; Secci, Daniela; Bolasco, Adriana; Nicolazzo, Chiara; Silvestri, Ida | |
Synthesis and Selective Human Monoamine Oxidase B Inhibition of Heterocyclic Hybrids Based on Hydrazine and Thiazole Scaffolds | 2013 | Simone, Carradori; Melissa, D'Ascenzio; DE MONTE, Celeste; Secci, Daniela; Matilde, Yáñez | |
Synthesis and cytotoxicity of novel (thiazol-2-yl)hydrazine derivatives as promising anti-Candida agents | 2013 | Simone, Carradori; Secci, Daniela; Bolasco, Adriana; Rivanera, Daniela; Mari, Emanuela; Zicari, Alessandra; Lotti, Lavinia Vittoria; Bizzarri, Bruna | |
Exploring (4-substituted-thiazol-2-yl)hydrazine derivatives of 2-, 3-, and 4-acetylpyridine as selective and reversible hMAO-B inhibitors. | 2013 | Chimenti, Paola; Petzer, A.; Carradori, S.; D’Ascenzio, M.; Silvestri, Romano; Alcaro, S.; Ortuso, F.; Petzer, J. J.; Secci, Daniela | |
Salen and tetrahydrosalen derivatives act as effective inhibitors of the tumor-associated carbonic anhydrase XII—A new scaffold for designing isoform-selective inhibitors | 2013 | Carradori, Simone; DE MONTE, Celeste; D'Ascenzio, Melissa; Secci, Daniela; Gulsah, Celik; Mariangela, Ceruso; Daniela, Vullo; Andrea, Scozzafava; Claudiu T., Supuran | |
tert-Butylcarbamate-Containing Histone Deacetylase Inhibitors: Apoptosis Induction, Cytodifferentiation, and Antiproliferative Activities in Cancer Cells. | 2013 | Valente, Sergio; Trisciuoglio, D; Tardugno, M; Benedetti, R; Labella, Donatella; Secci, Daniela; Mercurio, C; Boggio, R; Tomassi, S; Di Maro, S; Novellino, E; Altucci, L; Del Bufalo, D; Mai, Antonello; Cosconati, S. | |
The thiazole derivative CPTH6 impairs autophagy | 2013 | Ragazzoni, Ylenia; M., Desideri; C., Gabellini; T., De Luca; Carradori, Simone; Secci, Daniela; Nescatelli, Riccardo; A., Candiloro; M., Condello; S., Meschini; D., Del Bufalo; D., Trisciuoglio | |
Modulation of autophagic flux by CPTH6, a thiazole derivative with antitumoral activity | 2012 | Ragazzoni, Ylenia; M., Desideri; C., Gabellini; Carradori, Simone; Nescatelli, Riccardo; Secci, Daniela; A., Candiloro; D., Trisciuoglio; D., Del Bufalo | |
Discovery and optimization of pyrazoline derivatives as promising monoamine oxidase inhibitors | 2012 | Secci, Daniela; Carradori, Simone; Bolasco, Adriana; Bizzarri, Bruna; D'Ascenzio, Melissa; E., Maccioni | |
Synthesis and selective inhibitory activity against human COX-1 of novel 1-(4-substituted-thiazol-2-yl)-3,5-di(hetero)aryl-pyrazoline derivatives. | 2012 | S., Carradori; Secci, Daniela; Bolasco, Adriana; DE MONTE, Celeste; M., Yanez | |
Modulation of Autophagic Flux by CPTH6, a Gcn5/pCAF Histone Acetyltransferase Inhibitor With Antitumoral Activity | 2012 | D., Trisciuoglio; Ragazzoni, Ylenia; M., Desideri; C., Gabellini; Nescatelli, Riccardo; Carradori, Simone; Secci, Daniela; D., Del Bufalo | |
Conventional and Microwave-Assisted Synthesis of Benzimidazole Derivatives and their in vitro Inhibition of human Cyclooxygenase. | 2012 | Secci, Daniela; Bolasco, Adriana; D’Ascenzio, M.; della Sala, F.; Yáñez, M.; Carradori, Simone | |
Synthesis, anti-Candida activity, and cytotoxicity of new (4-(4-iodophenyl)thiazol-2-yl)hydrazine derivatives | 2012 | Secci, Daniela; Bizzarri, Bruna; Bolasco, Adriana; Simone, Carradori; D'Ascenzio, Melissa; Rivanera, Daniela; Mari, Emanuela; Polletta, Lucia; Zicari, Alessandra | |
Current and emerging strategies in bladder cancer | 2012 | Carradori, Simone; Cristini, Cristiano; Secci, Daniela; Caterina, Gulia; Gentile, Vincenzo; DI PIERRO, GIOVANNI BATTISTA | |
METHOD FOR PRODUCTION OF AMOTPHOUS RIFAXIMIN | 2012 | Lavagna, Silvio Massimo; Secci, Daniela; Padella, Franco | |
MANGANESE IRON OXIDE SUPERPARAMAGNETIC POWDER BY MECHANOCHEMICAL PROCESSING. NANOPARTICLES FUNCTIONALIZATION AND DISPERSION IN A NANOFLUID | 2012 | Bellusci, Mariangela; Aliotta, C.; Fiorani, D.; LA BARBERA, A.; Padella, F.; Peddis, D.; Pilloni, M.; Secci, Daniela | |
Patent-related survey on new monoamine oxidase inhibitors and their therapeutic potential | 2012 | Carradori, Simone; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; D'Ascenzio, Melissa | |
3-Methylcyclohexanone thiosemicarbazone: Determination of E/Z isomerization barrier by dynamic high-performance liquid chromatography, configuration assignment and theoretical study of the mechanisms involved by the spontaneous, acid and base catalyzed processes | 2012 | Carradori, Simone; Cirilli, R.; Dei Cicchi, S.; Ferretti, R.; Menta, Sergio; Pierini, Marco; Secci, Daniela | |
Synthesis and biological assessment of novel 2-thiazolylhydrazones and computational analysis of their recognition by monoamine oxidase B | 2012 | Distinto, S; Yáñez, M; Alcaro, S.; Cardia M., C; Gaspari, M; Sanna M., L; Meleddu, R; Ortuso, F; Kirchmair, J; Markt, P; Bolasco, Adriana; Wolber, G; Secci, Daniela; Maccioni, E. | |
CPTH6, a thiazole derivative, induces histone hypoacetylation and apoptosis in human leukemia cells | 2012 | D., Trisciuoglio; Ragazzoni, Ylenia; A., Pelosi; M., Desideri; Carradori, Simone; C., Gabellini; G., Maresca; Nescatelli, Riccardo; Secci, Daniela; Bolasco, Adriana; Bizzarri, Bruna; Cavaliere, Chiara; I., D'Agnano; Filetici, Patrizia; L., Ricci Vitiani; M. G., Rizzo; D., Del Bufalo | |
Recent advances in the development of selective human MAO-B inhibitors: (Hetero)arylidene-(4-substituted-thiazol-2- yl)hydrazines | 2012 | Secci, Daniela; Bolasco, Adriana; Carradori, Simone; D'Ascenzio, Melissa; Nescatelli, Riccardo; M., Yáñez | |
CPTH6, A NOVEL Gcn5/pCAF HISTONE ACETYLTRANSFERASE INHIBITOR, INDUCES BOTH APOPTOSIS AND AUTOPHAGY IN HUMAN LEUKEMIA CELLS | 2011 | Ragazzoni, Y.; Trisciuoglio, D.; Gabellini, C. .; Pelosi, A.; Desideri, M.; Carradori, Simone; Secci, Daniela; Rizzo, M. G.; Del, Bufalo | |
The State of the Art of Pyrazole Derivatives as Monoamine Oxidase Inhibitors and Antidepressant/Anticonvulsant Agents | 2011 | Secci, Daniela; Bolasco, Adriana; Carradori, Simone; Chimenti, Paola | |
FULL AMORPHOUS RIFAXIMIN AND METHODS FOR ITS PREPARATION | 2011 | Lavagna, Silvio Massimo; Secci, Daniela; Padella, Franco | |
METHOD FOR THE PRODUCTION OF AMORPHOUS RIFAXIMIN | 2011 | Lavagna, Silvio Massimo; Secci, Daniela; Franco, Padella | |
Synthesis and selective human monoamine oxidase inhibition of 3-carbonyl, 3-acyl, and 3-carboxyhydrazido coumarin derivatives | 2011 | Secci, Daniela; Carradori, Simone; Bolasco, Adriana; Chimenti, Paola; Yanez, Matilde; Ortuso, Francesco; Alcaro, Stefano | |
Synthesis and biological evaluation of novel 2,4-disubstituted-1,3-thiazoles as anti-Candida spp. agents | 2011 | Franco, Chimenti; Bizzarri, Bruna; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Granese, Arianna; Simone, Carradori; Melissa, D'Ascenzio; Lilli, Daniela; Rivanera, Daniela | |
EPIGENETIC MODULATION OF PGC-1a ACTIVITY BY GCN5 INHIBITORS: WO2010007085 | 2011 | Carradori, Simone; Secci, Daniela; Mai, Antonello | |
A new series of flavones, thioflavones, and flavanones as selective monoamine oxidase-B inhibitors | 2010 | Chimenti, Franco; Fioravanti, Rossella; Bolasco, Adriana; Chimenti, Paola; Secci, Daniela; Rossi, Francesca; Matilde, Yanez; Francisco, Orallo; Francesco, Ortuso; Stefano, Alcaro; Roberto, Cirilli; Rosella, Ferretti; M., Luisa Sanna | |
Synthesis and characterization of new 3-acyl-7-hydroxy-6,8-substituted-coumarin and 3-acyl-7-benzyloxy-6,8-substituted-coumarin derivatives | 2010 | Chimenti, Franco; Bolasco, Adriana; Secci, Daniela; Bizzarri, Bruna; Chimenti, Paola; Granese, A; Carradori, S. | |
Synthesis, semipreparative HPLC separation, biological evaluation, and 3D-QSAR of hydrazothiazole derivatives as human monoamine oxidase B inhibitors | 2010 | Chimenti, Franco; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Arianna, Granese; Simone, Carradori; Elias, Maccioni; M., Cristina Cardia; Matilde, Yanez; Francisco, Orallo; Stefano, Alcaro; Francesco, Ortuso; Roberto, Cirilli; Rosella, Ferretti; Simona, Distinto; Johannes, Kirchmair; Thierry, Langer | |
Synthesis of new 3-aryl-4,5-dihydropyrazole-1-carbothioamide derivatives. An investigation on their ability to inhibit monoamine oxidase | 2010 | Maccioni, E.; Alcaro, S.; Orallo, F.; Cardia, M. C.; Distinto, S.; Costa, G.; Yanez, M.; Sanna, M. L.; Vigo, S.; Meleddu, R.; Secci, D. | |
Investigations on the 2-thiazolylhydrazyne scaffold: Synthesis and molecular modeling of selective human monoamine oxidase inhibitors | 2010 | Chimenti, Franco; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Arianna, Granese; Simone, Carradori; Matilde, Yanez; Francisco, Orallo; Francesco, Ortuso; Stefano, Alcaro | |
FULL AMORPHOUS RIFAXIMIN AND METHODS FOR ITS PREPARATION | 2010 | Lavagna, Silvio Massimo; Secci, Daniela; Padella, Franco | |
METODO PER LA PREPARAZIONE DI RIFAXIMINA IN STATO AMORFO | 2010 | Lavagna, Silvio Massimo; Secci, Daniela; Padella, Franco | |
SYNTHESIS, STEREOCHEMICAL SEPARATION, AND BIOLOGICAL EVALUATION OF SELECTIVE INHIBITORS OF HUMAN MAO-B: 1-(4-ARYLTHIAZOL-2-YL)-2-(3-METHYLCYCLOHEXYLIDENE)HYDRAZINES | 2010 | Chimenti, Franco; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Granese, A; Carradori, S; Yanez, M; Orallo, F; Sanna, Ml; Gallinella, B; Cirilli, R. |
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