Sfoglia per Autore GUGLIELMI, Paolo
Novel therapeutic opportunities for Toxoplasma gondii, Trichomonas vaginalis, and Giardia intestinalis infections
2023 Arrighi, Francesca; Granese, Arianna; Chimenti, Paola; Guglielmi, Paolo
Indoleamine 2,3-dioxygenase
2023 Coluccia, Michele; Secci, Daniela; Guglielmi, Paolo
A Multitarget Approach against Neuroinflammation: Alkyl Substituted Coumarins as Inhibitors of Enzymes Involved in Neurodegeneration
2023 Berrino, E.; Carradori, S.; Carta, F.; Melfi, F.; Gallorini, M.; Poli, G.; Tuccinardi, T.; Fernandez-Bolanos, J. G.; Lopez, O.; Petzer, J. P.; Petzer, A.; Guglielmi, P.; Secci, D.; Supuran, C. T.
Kinetic Study on the Base-Catalyzed Imine-Enamine Tautomerism of a Chiral Biologically Active Isoxazoline Derivative by HPLC on Amylose Tris(3,5-dimethylphenylcarbamate) Chiral Stationary Phase
2023 Sadutto, Daniele; Guglielmi, Paolo; Carradori, Simone; Secci, Daniela; Cirilli, Roberto
Novel Insights on CAI–CORM Hybrids: Evaluation of the CO Releasing Properties and Pain-Relieving Activity of Differently Substituted Coumarins for the Treatment of Rheumatoid Arthritis
2023 Berrino, Emanuela; Micheli, Laura; Carradori, Simone; di Cesare Mannelli, Lorenzo; Guglielmi, Paolo; De Luca, Alessandro; Carta, Fabrizio; Ghelardini, Carla; Secci, Daniela; Supuran, Claudiu T.
Treatment of Toxoplasmosis: An Insight on Epigenetic Drugs
2022 Guglielmi, P.; Secci, D.
Novel Insights on Human Carbonic Anhydrase Inhibitors Based on Coumalic Acid: Design, Synthesis, Molecular Modeling Investigation, and Biological Studies
2022 Pontecorvi, Virginia; Mori, Mattia; Picarazzi, Francesca; Zara, Susi; Carradori, Simone; Cataldi, Amelia; Angeli, Andrea; Berrino, Emanuela; Chimenti, Paola; Ciogli, Alessia; Secci, Daniela; Guglielmi, Paolo; Supuran, Claudiu T.
An updated patent review on monoamine oxidase (MAO) inhibitors
2022 Guglielmi, Paolo; Carradori, Simone; D'Agostino, Ilaria; Campestre, Cristina; Petzer, Jacobus P
Metal-organic frameworks (MOFs) as biomolecules drug delivery systems for anticancer purposes
2022 Coluccia, Michele; Parisse, Valeria; Guglielmi, Paolo; Giannini, Giuseppe; Secci, Daniela
Aurone Scaffold and Structural Analogues for the Development of Monoamine Oxidase (MAO) Inhibitors
2022 Guglielmi, Paolo; Pontecorvi, Virginia; Akdemir, Atilla
New aspects of monoamine oxidase b inhibitors: The key role of halogens to open the golden door
2021 Mathew, B.; Carradori, S.; Guglielmi, P.; Uddin, M. D.; Kim, H.
Dual carbonic anhydrase ix/xii inhibitors and carbon monoxide releasing molecules modulate LPS-mediated inflammation in mouse macrophages
2021 Berrino, E.; Carradori, S.; Angeli, A.; Carta, F.; Supuran, C. T.; Guglielmi, P.; Coletti, C.; Paciotti, R.; Schweikl, H.; Maestrelli, F.; Cerbai, E.; Gallorini, M.
Synthesis and evaluation of thymol-based synthetic derivatives as dual-action inhibitors against different strains of h. pylori and AGS cell line
2021 Sisto, F.; Carradori, S.; Guglielmi, P.; Spano, M.; Secci, D.; Granese, A.; Sobolev, A. P.; Grande, R.; Campestre, C.; Di Marcantonio, M. C.; Mincione, G.
An innovative spectroscopic approach for qualitative and quantitative evaluation of Mb-CO from myoglobin carbonylation reaction through chemometrics methods
2021 Mansoldo, F. R. P.; Berrino, E.; Guglielmi, P.; Carradori, S.; Carta, F.; Secci, D.; Supuran, C. T.; Vermelho, A. B.
Synthesis and evaluation of a large library of nitroxoline derivatives as pancreatic cancer antiproliferative agents
2020 Veschi, Serena; Carradori, Simone; De Lellis, Laura; Florio, Rosalba; Brocco, Davide; Secci, Daniela; Guglielmi, Paolo; Spano, Mattia; Sobolev, Anatoly P.; Cama, Alessandro
Chalcones: Unearthing their therapeutic possibility as monoamine oxidase B inhibitors
2020 Guglielmi, Paolo; Mathew, Bijo; Secci, Daniela; Carradori, Simone
Novel insights on saccharin- and acesulfame-based carbonic anhydrase inhibitors: design, synthesis, modelling investigations and biological activity evaluation
2020 Guglielmi, P.; Rotondi, G.; Secci, D.; Angeli, A.; Chimenti, P.; Nocentini, A.; Bonardi, A.; Gratteri, P.; Carradori, S.; Supuran, C. T.
Synthesis and biological evaluation of carvacrol-based derivatives as dual inhibitors of H. Pylori strains and ags cell proliferation
2020 Sisto, F.; Carradori, S.; Guglielmi, P.; Traversi, C. B.; Spano, M.; Sobolev, A. P.; Secci, D.; Di Marcantonio, M. C.; Haloci, E.; Grande, R.; Mincione, G.
Natural compounds and extracts as novel antimicrobial agents
2020 Guglielmi, P.; Pontecorvi, V.; Rotondi, G.
Innovative pH-interfering agents in association with anticancer agents
2020 Secci, D.; Guglielmi, P.
1,3-Dipolar Cycloaddition, HPLC Enantioseparation, and Docking Studies of Saccharin/Isoxazole and Saccharin/Isoxazoline Derivatives as Selective Carbonic Anhydrase IX and XII Inhibitors
2020 D'Ascenzio, M.; Secci, D.; Carradori, S.; Zara, S.; Guglielmi, P.; Cirilli, R.; Pierini, M.; Poli, G.; Tuccinardi, T.; Angeli, A.; Supuran, C. T.
Antimalarial agents from medicinal plant and fungal sources
2020 Luisi, Grazia; Carradori, Simone; Grande, Rossella; Secci, Daniela; Guglielmi, Paolo
High-performance liquid chromatography enantioseparation of chiral 2-(benzylsulfinyl)benzamide derivatives on cellulose tris(3,5-dichlorophenylcarbamate) chiral stationary phase
2020 Carradori, S.; Secci, D.; Guglielmi, P.; Pierini, M.; Cirilli, R.
Novel approaches to the discovery of selective human monoamine oxidase-B inhibitors: is there room for improvement?
2019 Guglielmi, P.; Carradori, S.; Ammazzalorso, A.; Secci, D.
Design, synthesis and biological activity of selective hCAs inhibitors based on 2-(benzylsulfinyl)benzoic acid scaffold
2019 Rotondi, G.; Guglielmi, P.; Carradori, S.; Secci, D.; De Monte, C.; De Filippis, B.; Maccallini, C.; Amoroso, R.; Cirilli, R.; Akdemir, A.; Angeli, A.; Supuran, C. T.
Design, synthesis, docking studies and monoamine oxidase inhibition of a small library of 1-acetyl- and 1-thiocarbamoyl-3,5-diphenyl-4,5-dihydro-(1h)-pyrazoles
2019 Guglielmi, Paolo; Carradori, Simone; Poli, Giulio; Secci, Daniela; Cirilli, Roberto; Rotondi, Giulia; Chimenti, Paola; Petzer, Anél; Petzer, Jacobus P.
Benzo[b]tiophen-3-ol derivatives as effective inhibitors of human monoamine oxidase: design, synthesis, and biological activity
2019 Guglielmi, Paolo; Secci, Daniela; Petzer, Anél; Bagetta, Donatella; Chimenti, Paola; Rotondi, Giulia; Ferrante, Claudio; Recinella, Lucia; Leone, Sheila; Alcaro, Stefano; Zengin, Gokhan; Petzer, Jacobus P; Ortuso, Francesco; Carradori, Simone
4-(3-Nitrophenyl)thiazol-2-ylhydrazone derivatives as antioxidants and selective hMAO-B inhibitors: synthesis, biological activity and computational analysis
2019 Secci, Daniela; Carradori, Simone; Petzer, Anél; Guglielmi, Paolo; D’Ascenzio, Melissa; Chimenti, Paola; Bagetta, Donatella; Alcaro, Stefano; Zengin, Gokhan; Petzer, Jacobus P.; Ortuso, Francesco
Kinesin Eg5 targeting inhibitors as a new strategy for gastric adenocarcinoma treatment
2019 Marconi, G. D.; Carradori, S.; Ricci, A.; Guglielmi, P.; Cataldi, A.; Zara, S.
Novel therapies for glaucoma: a patent review (2013-2019)
2019 Guglielmi, Paolo; Carradori, Simone; Campestre, Cristina; Poce, Giovanna
The up-regulation of oxidative stress as a potential mechanism of novel MAO-B inhibitors for glioblastoma treatment
2019 Marconi, G. D.; Gallorini, M.; Carradori, S.; Guglielmi, P.; Cataldi, A.; Zara, S.
Mechanisms of action of carbonic anhydrase inhibitors: compounds that bind “out of the binding site” and compounds with an unknown mechanism of action
2019 Carradori, Simone; Guglielmi, Paolo
Synthesis and biological evaluation of new saccharin-based inhibitors of cancer-related carbonic anhydrase IX and XII isoforms & Benzo[b]tiophen-3-ol derivatives as effective inhibitors of hMAOs: design, synthesis and biological activity
2018 Guglielmi, Paolo
Design, synthesis and biochemical evaluation of novel multi-target inhibitors as potential anti-Parkinson agents
2018 Carradori, Simone; Ottuso, Francesco; Petzer, Anèl; Bagetta, Donatella; DE MONTE, Celeste; Secci, Daniela; DE VITA, Daniela; Guglielmi, Paolo; Zengin, Gokhan; Aktumsek, Abdurrahman; Alcaro, Stefano; Petzer, Jacobus P.
Crystal structure of the Eg5 - K858 complex and implications for structure-based design of thiadiazole-containing inhibitors
2018 Talapatra, Sandeep K.; Tham, Chuin Lean; Guglielmi, Paolo; Cirilli, Roberto; Chandrasekaran, Balakumar; Karpoormath, Rajshekhar; Carradori, Simone; Kozielski, Frank
Magnetic metal−organic framework composite by fast and facile mechanochemical process
2018 Bellusci, M.; Guglielmi, P.; Masi, Andrea; Padella, F.; Singh, G.; Yaacoub, N.; Peddis, D.; Secci, D.
Synthesis and biological evaluation of anti-Toxoplasma gondii activity of a novel scaffold of thiazolidinone derivatives
2017 Carradori, Simone; Secci, Daniela; Bizzarri, Bruna; Chimenti, Paola; DE MONTE, Celeste; Guglielmi, Paolo; Campestre, Cristina; Rivanera, Daniela; Bordón, Claudia; Jones Brando, Lorraine
The sodium salt of the enantiomers of ricobendazole: preparation, solubility and chiroptical properties
2017 Cirilli, Roberto; Guglielmi, Paolo; Formica, Francesca Romana; Casulli, Adriano; Carradori, Simone
Analysis of imidazoles and triazoles in biological samples after MicroExtraction by packed sorbent
2017 Campestre, Cristina; Locatelli, Marcello; Guglielmi, Paolo; De Luca, Elisa; Bellagamba, Giuseppe; Menta, Sergio; Zengin, Gokhan; Celia, Christian; Di Marzio, Luisa; Carradori, Simone
Protective effects Induced by microwave-assisted aqueous harpagophytum extract on rat cortex synaptosomes challenged with amyloid β-peptide
2017 Ferrante, Claudio; Recinella, Lucia; Locatelli, Marcello; Guglielmi, Paolo; Secci, Daniela; Leporini, Lidia; Chiavaroli, Annalisa; Leone, Sheila; Martinotti, Sara; Brunetti, Luigi; Vacca, Michele; Meneghini, Luigi; Orlando, Giustino
Enantiomers of triclabendazole sulfoxide: analytical and semipreparative HPLC separation, absolute configuration assignment, and transformation into sodium salt
2017 Ferretti, Rosella; Carradori, Simone; Guglielmi, Paolo; Pierini, Marco; Casulli, Adriano; Cirilli, Roberto
Open saccharin-based secondary sulfonamides as potent and selective inhibitors of cancer-related carbonic anhydrase IX and XII isoforms
2017 D'Ascenzio, M.; Guglielmi, P.; Carradori, S.; Secci, D.; Florio, R.; Mollica, A.; Ceruso, M.; Akdemir, A.; Sobolev, A. P.; Supuran, C. T.
Inhibition of human monoamine oxidase: biological and molecular modeling studies on selected natural flavonoids
2016 Carradori, Simone; Gidaro, Maria Concetta; Petzer, Anél; Costa, Giosuè; Guglielmi, Paolo; Chimenti, Paola; Alcaro, Stefano; Petzer, Jacobus P.
A novel library of saccharin and acesulfame derivatives as potent and selective inhibitors of carbonic anhydrase IX and XII isoforms
2016 Carradori, Simone; Secci, Daniela; DE MONTE, Celeste; Mollica, Adriano; Ceruso, Mariangela; Akdemir, Atilla; Sobolev, Anatoly P; Codispoti, Rossella; DE COSMI, Federica; Guglielmi, Paolo; Supuran, Claudiu T.
Opening new scenarios for human MAO inhibitors
2015 DE MONTE, Celeste; D'Ascenzio, Melissa; Guglielmi, Paolo; Mancini, Veronica; Carradori, Simone
Synthesis and pharmacological screening of a large library of 1,3,4-thiadiazolines as innovative therapeutic tools for the treatment of prostate cancer and melanoma
2015 DE MONTE, Celeste; Carradori, Simone; Secci, Daniela; D'Ascenzio, Melissa; Guglielmi, Paolo; Mollica, Adriano; Morrone, Stefania; Scarpa, Susanna; Agliano', Anna Maria; Giantulli, Sabrina; Silvestri, Ida
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Novel therapeutic opportunities for Toxoplasma gondii, Trichomonas vaginalis, and Giardia intestinalis infections | 2023 | Arrighi, Francesca; Granese, Arianna; Chimenti, Paola; Guglielmi, Paolo | |
Indoleamine 2,3-dioxygenase | 2023 | Coluccia, Michele; Secci, Daniela; Guglielmi, Paolo | |
A Multitarget Approach against Neuroinflammation: Alkyl Substituted Coumarins as Inhibitors of Enzymes Involved in Neurodegeneration | 2023 | Berrino, E.; Carradori, S.; Carta, F.; Melfi, F.; Gallorini, M.; Poli, G.; Tuccinardi, T.; Fernandez-Bolanos, J. G.; Lopez, O.; Petzer, J. P.; Petzer, A.; Guglielmi, P.; Secci, D.; Supuran, C. T. | |
Kinetic Study on the Base-Catalyzed Imine-Enamine Tautomerism of a Chiral Biologically Active Isoxazoline Derivative by HPLC on Amylose Tris(3,5-dimethylphenylcarbamate) Chiral Stationary Phase | 2023 | Sadutto, Daniele; Guglielmi, Paolo; Carradori, Simone; Secci, Daniela; Cirilli, Roberto | |
Novel Insights on CAI–CORM Hybrids: Evaluation of the CO Releasing Properties and Pain-Relieving Activity of Differently Substituted Coumarins for the Treatment of Rheumatoid Arthritis | 2023 | Berrino, Emanuela; Micheli, Laura; Carradori, Simone; di Cesare Mannelli, Lorenzo; Guglielmi, Paolo; De Luca, Alessandro; Carta, Fabrizio; Ghelardini, Carla; Secci, Daniela; Supuran, Claudiu T. | |
Treatment of Toxoplasmosis: An Insight on Epigenetic Drugs | 2022 | Guglielmi, P.; Secci, D. | |
Novel Insights on Human Carbonic Anhydrase Inhibitors Based on Coumalic Acid: Design, Synthesis, Molecular Modeling Investigation, and Biological Studies | 2022 | Pontecorvi, Virginia; Mori, Mattia; Picarazzi, Francesca; Zara, Susi; Carradori, Simone; Cataldi, Amelia; Angeli, Andrea; Berrino, Emanuela; Chimenti, Paola; Ciogli, Alessia; Secci, Daniela; Guglielmi, Paolo; Supuran, Claudiu T. | |
An updated patent review on monoamine oxidase (MAO) inhibitors | 2022 | Guglielmi, Paolo; Carradori, Simone; D'Agostino, Ilaria; Campestre, Cristina; Petzer, Jacobus P | |
Metal-organic frameworks (MOFs) as biomolecules drug delivery systems for anticancer purposes | 2022 | Coluccia, Michele; Parisse, Valeria; Guglielmi, Paolo; Giannini, Giuseppe; Secci, Daniela | |
Aurone Scaffold and Structural Analogues for the Development of Monoamine Oxidase (MAO) Inhibitors | 2022 | Guglielmi, Paolo; Pontecorvi, Virginia; Akdemir, Atilla | |
New aspects of monoamine oxidase b inhibitors: The key role of halogens to open the golden door | 2021 | Mathew, B.; Carradori, S.; Guglielmi, P.; Uddin, M. D.; Kim, H. | |
Dual carbonic anhydrase ix/xii inhibitors and carbon monoxide releasing molecules modulate LPS-mediated inflammation in mouse macrophages | 2021 | Berrino, E.; Carradori, S.; Angeli, A.; Carta, F.; Supuran, C. T.; Guglielmi, P.; Coletti, C.; Paciotti, R.; Schweikl, H.; Maestrelli, F.; Cerbai, E.; Gallorini, M. | |
Synthesis and evaluation of thymol-based synthetic derivatives as dual-action inhibitors against different strains of h. pylori and AGS cell line | 2021 | Sisto, F.; Carradori, S.; Guglielmi, P.; Spano, M.; Secci, D.; Granese, A.; Sobolev, A. P.; Grande, R.; Campestre, C.; Di Marcantonio, M. C.; Mincione, G. | |
An innovative spectroscopic approach for qualitative and quantitative evaluation of Mb-CO from myoglobin carbonylation reaction through chemometrics methods | 2021 | Mansoldo, F. R. P.; Berrino, E.; Guglielmi, P.; Carradori, S.; Carta, F.; Secci, D.; Supuran, C. T.; Vermelho, A. B. | |
Synthesis and evaluation of a large library of nitroxoline derivatives as pancreatic cancer antiproliferative agents | 2020 | Veschi, Serena; Carradori, Simone; De Lellis, Laura; Florio, Rosalba; Brocco, Davide; Secci, Daniela; Guglielmi, Paolo; Spano, Mattia; Sobolev, Anatoly P.; Cama, Alessandro | |
Chalcones: Unearthing their therapeutic possibility as monoamine oxidase B inhibitors | 2020 | Guglielmi, Paolo; Mathew, Bijo; Secci, Daniela; Carradori, Simone | |
Novel insights on saccharin- and acesulfame-based carbonic anhydrase inhibitors: design, synthesis, modelling investigations and biological activity evaluation | 2020 | Guglielmi, P.; Rotondi, G.; Secci, D.; Angeli, A.; Chimenti, P.; Nocentini, A.; Bonardi, A.; Gratteri, P.; Carradori, S.; Supuran, C. T. | |
Synthesis and biological evaluation of carvacrol-based derivatives as dual inhibitors of H. Pylori strains and ags cell proliferation | 2020 | Sisto, F.; Carradori, S.; Guglielmi, P.; Traversi, C. B.; Spano, M.; Sobolev, A. P.; Secci, D.; Di Marcantonio, M. C.; Haloci, E.; Grande, R.; Mincione, G. | |
Natural compounds and extracts as novel antimicrobial agents | 2020 | Guglielmi, P.; Pontecorvi, V.; Rotondi, G. | |
Innovative pH-interfering agents in association with anticancer agents | 2020 | Secci, D.; Guglielmi, P. | |
1,3-Dipolar Cycloaddition, HPLC Enantioseparation, and Docking Studies of Saccharin/Isoxazole and Saccharin/Isoxazoline Derivatives as Selective Carbonic Anhydrase IX and XII Inhibitors | 2020 | D'Ascenzio, M.; Secci, D.; Carradori, S.; Zara, S.; Guglielmi, P.; Cirilli, R.; Pierini, M.; Poli, G.; Tuccinardi, T.; Angeli, A.; Supuran, C. T. | |
Antimalarial agents from medicinal plant and fungal sources | 2020 | Luisi, Grazia; Carradori, Simone; Grande, Rossella; Secci, Daniela; Guglielmi, Paolo | |
High-performance liquid chromatography enantioseparation of chiral 2-(benzylsulfinyl)benzamide derivatives on cellulose tris(3,5-dichlorophenylcarbamate) chiral stationary phase | 2020 | Carradori, S.; Secci, D.; Guglielmi, P.; Pierini, M.; Cirilli, R. | |
Novel approaches to the discovery of selective human monoamine oxidase-B inhibitors: is there room for improvement? | 2019 | Guglielmi, P.; Carradori, S.; Ammazzalorso, A.; Secci, D. | |
Design, synthesis and biological activity of selective hCAs inhibitors based on 2-(benzylsulfinyl)benzoic acid scaffold | 2019 | Rotondi, G.; Guglielmi, P.; Carradori, S.; Secci, D.; De Monte, C.; De Filippis, B.; Maccallini, C.; Amoroso, R.; Cirilli, R.; Akdemir, A.; Angeli, A.; Supuran, C. T. | |
Design, synthesis, docking studies and monoamine oxidase inhibition of a small library of 1-acetyl- and 1-thiocarbamoyl-3,5-diphenyl-4,5-dihydro-(1h)-pyrazoles | 2019 | Guglielmi, Paolo; Carradori, Simone; Poli, Giulio; Secci, Daniela; Cirilli, Roberto; Rotondi, Giulia; Chimenti, Paola; Petzer, Anél; Petzer, Jacobus P. | |
Benzo[b]tiophen-3-ol derivatives as effective inhibitors of human monoamine oxidase: design, synthesis, and biological activity | 2019 | Guglielmi, Paolo; Secci, Daniela; Petzer, Anél; Bagetta, Donatella; Chimenti, Paola; Rotondi, Giulia; Ferrante, Claudio; Recinella, Lucia; Leone, Sheila; Alcaro, Stefano; Zengin, Gokhan; Petzer, Jacobus P; Ortuso, Francesco; Carradori, Simone | |
4-(3-Nitrophenyl)thiazol-2-ylhydrazone derivatives as antioxidants and selective hMAO-B inhibitors: synthesis, biological activity and computational analysis | 2019 | Secci, Daniela; Carradori, Simone; Petzer, Anél; Guglielmi, Paolo; D’Ascenzio, Melissa; Chimenti, Paola; Bagetta, Donatella; Alcaro, Stefano; Zengin, Gokhan; Petzer, Jacobus P.; Ortuso, Francesco | |
Kinesin Eg5 targeting inhibitors as a new strategy for gastric adenocarcinoma treatment | 2019 | Marconi, G. D.; Carradori, S.; Ricci, A.; Guglielmi, P.; Cataldi, A.; Zara, S. | |
Novel therapies for glaucoma: a patent review (2013-2019) | 2019 | Guglielmi, Paolo; Carradori, Simone; Campestre, Cristina; Poce, Giovanna | |
The up-regulation of oxidative stress as a potential mechanism of novel MAO-B inhibitors for glioblastoma treatment | 2019 | Marconi, G. D.; Gallorini, M.; Carradori, S.; Guglielmi, P.; Cataldi, A.; Zara, S. | |
Mechanisms of action of carbonic anhydrase inhibitors: compounds that bind “out of the binding site” and compounds with an unknown mechanism of action | 2019 | Carradori, Simone; Guglielmi, Paolo | |
Synthesis and biological evaluation of new saccharin-based inhibitors of cancer-related carbonic anhydrase IX and XII isoforms & Benzo[b]tiophen-3-ol derivatives as effective inhibitors of hMAOs: design, synthesis and biological activity | 2018 | Guglielmi, Paolo | |
Design, synthesis and biochemical evaluation of novel multi-target inhibitors as potential anti-Parkinson agents | 2018 | Carradori, Simone; Ottuso, Francesco; Petzer, Anèl; Bagetta, Donatella; DE MONTE, Celeste; Secci, Daniela; DE VITA, Daniela; Guglielmi, Paolo; Zengin, Gokhan; Aktumsek, Abdurrahman; Alcaro, Stefano; Petzer, Jacobus P. | |
Crystal structure of the Eg5 - K858 complex and implications for structure-based design of thiadiazole-containing inhibitors | 2018 | Talapatra, Sandeep K.; Tham, Chuin Lean; Guglielmi, Paolo; Cirilli, Roberto; Chandrasekaran, Balakumar; Karpoormath, Rajshekhar; Carradori, Simone; Kozielski, Frank | |
Magnetic metal−organic framework composite by fast and facile mechanochemical process | 2018 | Bellusci, M.; Guglielmi, P.; Masi, Andrea; Padella, F.; Singh, G.; Yaacoub, N.; Peddis, D.; Secci, D. | |
Synthesis and biological evaluation of anti-Toxoplasma gondii activity of a novel scaffold of thiazolidinone derivatives | 2017 | Carradori, Simone; Secci, Daniela; Bizzarri, Bruna; Chimenti, Paola; DE MONTE, Celeste; Guglielmi, Paolo; Campestre, Cristina; Rivanera, Daniela; Bordón, Claudia; Jones Brando, Lorraine | |
The sodium salt of the enantiomers of ricobendazole: preparation, solubility and chiroptical properties | 2017 | Cirilli, Roberto; Guglielmi, Paolo; Formica, Francesca Romana; Casulli, Adriano; Carradori, Simone | |
Analysis of imidazoles and triazoles in biological samples after MicroExtraction by packed sorbent | 2017 | Campestre, Cristina; Locatelli, Marcello; Guglielmi, Paolo; De Luca, Elisa; Bellagamba, Giuseppe; Menta, Sergio; Zengin, Gokhan; Celia, Christian; Di Marzio, Luisa; Carradori, Simone | |
Protective effects Induced by microwave-assisted aqueous harpagophytum extract on rat cortex synaptosomes challenged with amyloid β-peptide | 2017 | Ferrante, Claudio; Recinella, Lucia; Locatelli, Marcello; Guglielmi, Paolo; Secci, Daniela; Leporini, Lidia; Chiavaroli, Annalisa; Leone, Sheila; Martinotti, Sara; Brunetti, Luigi; Vacca, Michele; Meneghini, Luigi; Orlando, Giustino | |
Enantiomers of triclabendazole sulfoxide: analytical and semipreparative HPLC separation, absolute configuration assignment, and transformation into sodium salt | 2017 | Ferretti, Rosella; Carradori, Simone; Guglielmi, Paolo; Pierini, Marco; Casulli, Adriano; Cirilli, Roberto | |
Open saccharin-based secondary sulfonamides as potent and selective inhibitors of cancer-related carbonic anhydrase IX and XII isoforms | 2017 | D'Ascenzio, M.; Guglielmi, P.; Carradori, S.; Secci, D.; Florio, R.; Mollica, A.; Ceruso, M.; Akdemir, A.; Sobolev, A. P.; Supuran, C. T. | |
Inhibition of human monoamine oxidase: biological and molecular modeling studies on selected natural flavonoids | 2016 | Carradori, Simone; Gidaro, Maria Concetta; Petzer, Anél; Costa, Giosuè; Guglielmi, Paolo; Chimenti, Paola; Alcaro, Stefano; Petzer, Jacobus P. | |
A novel library of saccharin and acesulfame derivatives as potent and selective inhibitors of carbonic anhydrase IX and XII isoforms | 2016 | Carradori, Simone; Secci, Daniela; DE MONTE, Celeste; Mollica, Adriano; Ceruso, Mariangela; Akdemir, Atilla; Sobolev, Anatoly P; Codispoti, Rossella; DE COSMI, Federica; Guglielmi, Paolo; Supuran, Claudiu T. | |
Opening new scenarios for human MAO inhibitors | 2015 | DE MONTE, Celeste; D'Ascenzio, Melissa; Guglielmi, Paolo; Mancini, Veronica; Carradori, Simone | |
Synthesis and pharmacological screening of a large library of 1,3,4-thiadiazolines as innovative therapeutic tools for the treatment of prostate cancer and melanoma | 2015 | DE MONTE, Celeste; Carradori, Simone; Secci, Daniela; D'Ascenzio, Melissa; Guglielmi, Paolo; Mollica, Adriano; Morrone, Stefania; Scarpa, Susanna; Agliano', Anna Maria; Giantulli, Sabrina; Silvestri, Ida |
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