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Novel polyamine-based Histone deacetylases-Lysine demethylase 1 dual binding inhibitors 2018 Milelli, Andrea; Marchetti, Chiara; Turrini, Eleonora; Catanzaro, Elena; Mazzone, Roberta; Tomaselli, Daniela; Fimognari, Carmela; Tumiatti, Vincenzo; Minarini, Anna
Disruptor of telomeric silencing 1-like (DOT1L): disclosing a new class of non-nucleoside inhibitors by means of ligand-based and structure-based approaches 2018 Sabatino, Manuela; Rotili, Dante; Patsilinakos, Alexandros; Forgione, Mariantonietta; Tomaselli, Daniela; Alby, Fréderic; Arimondo, Paola B.; Mai, Antonello; Ragno, Rino
Epigenetic metalloenzymes 2018 Blanquart, Christophe; Linot, Camille; Cartron, Pierre-Francois; Tomaselli, Daniela; Mai, Antonello; Bertrand, Philippe
Epigenetic polypharmacology: a new frontier for epi-drug discovery 2019 Tomaselli, Daniela; Lucidi, Alessia; Rotili, Dante; Mai, Antonello
α,γ-Diketocarboxylic acids and their esters act as carbonic anhydrase IX and XII selective inhibitors 2019 Nocentini, Alessio; Lucidi, Alessia; Perut, Francesca; Massa, Annamaria; Tomaselli, Daniela; Gratteri, Paola; Baldini, Nicola; Rotili, Dante; Mai, Antonello; Supuran, Claudiu T.
Effect of α-methoxy substitution on the anti-HIV activity of dihydropyrimidin-4(3 H)-ones 2019 Nawrozkij, Maxim B.; Forgione, Mariantonietta; Yablokov, Alexandre S.; Lucidi, Alessia; Tomaselli, Daniela; Patsilinakos, Alexandros; Panella, Cristina; Hailu, Gebremedhin S.; Kirillov, Ivan A.; Badia, Roger; Riveira-Munoz, Eva; Crespan, Emmanuele; Armijos Rivera, Jorge I.; Cirilli, Roberto; Ragno, Rino; Esté, José A.; Maga, Giovanni; Mai, Antonello; Rotili, Dante
Structure-reactivity relationships on substrates and inhibitors of the lysine deacylase sirtuin 2 from schistosoma mansoni (SmSirt2) 2019 Monaldi, Daria; Rotili, Dante; Julien Lancelot, ‡; Martin Marek, §; Nathalie Wössner, ∥; Lucidi, Alessia; Tomaselli, Daniela; Elizabeth Ramos-Morales, ‡; Christophe Romier, ∥; Pierce, ∥ Raymond J.; Mai, Antonello; and Manfred Jung, ‡
DNA Methylation: Biological Implications and Modulation of Its Aberrant Dysregulation 2019 Lucidi, Alessia; Tomaselli, Daniela; Rotili, Dante; Mai, Antonello
Recent advances in epigenetic proteolysis targeting chimeras (Epi-PROTACs) 2020 Tomaselli, D.; Mautone, N.; Mai, A.; Rotili, D.
Sirt4: a multifaceted enzyme at the crossroads of mitochondrial metabolism and cancer 2020 Tomaselli, D.; Steegborn, C.; Mai, A.; Rotili, D.
Different strategies to target the epigenome 2020 Tomaselli, Daniela
Sirtuins 2021 Zwergel, Clemens; Tomaselli, Daniela; Mai, Antonello
Specific inhibitors of mitochondrial deacylase sirtuin 4 endowed with cellular activity 2024 Pannek, M.; Alhalabi, Z.; Tomaselli, D.; Menna, M.; Fiorentino, F.; Robaa, D.; Weyand, M.; Puhlmann, M.; Tomassi, S.; Barreca, F.; Tafani, M.; Zaganjor, E.; Haigis, M. C.; Sippl, W.; Rotili, D.; Mai, A.; Steegborn, C.
Mostrati risultati da 1 a 13 di 13
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