Sfoglia per Autore
Synthesis and selective inhibition of human monoamine oxidases of a large scaffold of (4,5-substituted-thiazol-2-yl)hydrazones
2010 Chimenti, Franco; Secci, Daniela; Chimenti, Paola; Granese, Arianna; Carradori, Simone; D'Ascenzio, Melissa; Matilde, Yanez; Francisco, Orallo; Bolasco, Adriana
Discovery and optimization of pyrazoline derivatives as promising monoamine oxidase inhibitors
2012 Secci, Daniela; Carradori, Simone; Bolasco, Adriana; Bizzarri, Bruna; D'Ascenzio, Melissa; E., Maccioni
Patent-related survey on new monoamine oxidase inhibitors and their therapeutic potential
2012 Carradori, Simone; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; D'Ascenzio, Melissa
Recent advances in the development of selective human MAO-B inhibitors: (Hetero)arylidene-(4-substituted-thiazol-2- yl)hydrazines
2012 Secci, Daniela; Bolasco, Adriana; Carradori, Simone; D'Ascenzio, Melissa; Nescatelli, Riccardo; M., Yáñez
Synthesis, anti-Candida activity, and cytotoxicity of new (4-(4-iodophenyl)thiazol-2-yl)hydrazine derivatives
2012 Secci, Daniela; Bizzarri, Bruna; Bolasco, Adriana; Simone, Carradori; D'Ascenzio, Melissa; Rivanera, Daniela; Mari, Emanuela; Polletta, Lucia; Zicari, Alessandra
Salen and tetrahydrosalen derivatives act as effective inhibitors of the tumor-associated carbonic anhydrase XII—A new scaffold for designing isoform-selective inhibitors
2013 Carradori, Simone; DE MONTE, Celeste; D'Ascenzio, Melissa; Secci, Daniela; Gulsah, Celik; Mariangela, Ceruso; Daniela, Vullo; Andrea, Scozzafava; Claudiu T., Supuran
Synthesis and biological evaluation of new potential co-adjuvants for the treatment of Parkinson’s disease and a new catalytic, asymmetric approach to the synthesis of fused heterocycles of biological interest.
2013 D'Ascenzio, Melissa
Design, synthesis and biological characterization of thiazolidin-4-one derivatives as promising inhibitors of Toxoplasma gondii
2014 D'Ascenzio, Melissa; Bizzarri, Bruna; DE MONTE, Celeste; Carradori, S; Bolasco, Adriana; Secci, Daniela; Rivanera, Daniela; Faulhaber, N; Bordon, C; Jones Brando, L.
Selective MAO-B inhibitors: a lesson from natural products
2014 Carradori, Simone; D'Ascenzio, Melissa; Chimenti, Paola; Secci, Daniela; Bolasco, Adriana
Cyclic tertiary sulfamates: Selective inhibition of the tumor-associated carbonic anhydrases IX and XII by N- and O-substituted acesulfame derivatives
2014 DE MONTE, Celeste; Carradori, Simone; Secci, Daniela; D'Ascenzio, Melissa; Vullo, D; Ceruso, M; Supuran, Ct
Opening new scenarios for human MAO inhibitors
2015 DE MONTE, Celeste; D'Ascenzio, Melissa; Guglielmi, Paolo; Mancini, Veronica; Carradori, Simone
Synthesis and pharmacological screening of a large library of 1,3,4-thiadiazolines as innovative therapeutic tools for the treatment of prostate cancer and melanoma
2015 DE MONTE, Celeste; Carradori, Simone; Secci, Daniela; D'Ascenzio, Melissa; Guglielmi, Paolo; Mollica, Adriano; Morrone, Stefania; Scarpa, Susanna; Agliano', Anna Maria; Giantulli, Sabrina; Silvestri, Ida
New amide derivatives of Probenecid as selective inhibitors of carbonic anhydrase IX and XII: Biological evaluation and molecular modelling studies
2015 Carradori, Simone; Mollica, Adriano; Ceruso, Mariangela; D'Ascenzio, Melissa; DE MONTE, Celeste; Chimenti, Paola; Sabia, Rocchina; Akdemir, Atilla; Supuran, Claudiu T.
Synthesis, biological evaluation and quantitative structure-active relationships of 1,3-thiazolidin-4-one derivatives. A promising chemical scaffold endowed with high antifungal potency and low cytotoxicity
2017 Carradori, Simone; Bizzarri, Bruna; D'Ascenzio, Melissa; DE MONTE, Celeste; Grande, Rossella; Rivanera, Daniela; Zicari, Alessanda; Mari, Emanuela; Sabatino, Manuela; Patsilinakos, Alexandros; Ragno, Rino; Secci, Daniela
4-(3-Nitrophenyl)thiazol-2-ylhydrazone derivatives as antioxidants and selective hMAO-B inhibitors: synthesis, biological activity and computational analysis
2019 Secci, Daniela; Carradori, Simone; Petzer, Anél; Guglielmi, Paolo; D’Ascenzio, Melissa; Chimenti, Paola; Bagetta, Donatella; Alcaro, Stefano; Zengin, Gokhan; Petzer, Jacobus P.; Ortuso, Francesco
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Synthesis and selective inhibition of human monoamine oxidases of a large scaffold of (4,5-substituted-thiazol-2-yl)hydrazones | 2010 | Chimenti, Franco; Secci, Daniela; Chimenti, Paola; Granese, Arianna; Carradori, Simone; D'Ascenzio, Melissa; Matilde, Yanez; Francisco, Orallo; Bolasco, Adriana | |
| Discovery and optimization of pyrazoline derivatives as promising monoamine oxidase inhibitors | 2012 | Secci, Daniela; Carradori, Simone; Bolasco, Adriana; Bizzarri, Bruna; D'Ascenzio, Melissa; E., Maccioni | |
| Patent-related survey on new monoamine oxidase inhibitors and their therapeutic potential | 2012 | Carradori, Simone; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; D'Ascenzio, Melissa | |
| Recent advances in the development of selective human MAO-B inhibitors: (Hetero)arylidene-(4-substituted-thiazol-2- yl)hydrazines | 2012 | Secci, Daniela; Bolasco, Adriana; Carradori, Simone; D'Ascenzio, Melissa; Nescatelli, Riccardo; M., Yáñez | |
| Synthesis, anti-Candida activity, and cytotoxicity of new (4-(4-iodophenyl)thiazol-2-yl)hydrazine derivatives | 2012 | Secci, Daniela; Bizzarri, Bruna; Bolasco, Adriana; Simone, Carradori; D'Ascenzio, Melissa; Rivanera, Daniela; Mari, Emanuela; Polletta, Lucia; Zicari, Alessandra | |
| Salen and tetrahydrosalen derivatives act as effective inhibitors of the tumor-associated carbonic anhydrase XII—A new scaffold for designing isoform-selective inhibitors | 2013 | Carradori, Simone; DE MONTE, Celeste; D'Ascenzio, Melissa; Secci, Daniela; Gulsah, Celik; Mariangela, Ceruso; Daniela, Vullo; Andrea, Scozzafava; Claudiu T., Supuran | |
| Synthesis and biological evaluation of new potential co-adjuvants for the treatment of Parkinson’s disease and a new catalytic, asymmetric approach to the synthesis of fused heterocycles of biological interest. | 2013 | D'Ascenzio, Melissa | |
| Design, synthesis and biological characterization of thiazolidin-4-one derivatives as promising inhibitors of Toxoplasma gondii | 2014 | D'Ascenzio, Melissa; Bizzarri, Bruna; DE MONTE, Celeste; Carradori, S; Bolasco, Adriana; Secci, Daniela; Rivanera, Daniela; Faulhaber, N; Bordon, C; Jones Brando, L. | |
| Selective MAO-B inhibitors: a lesson from natural products | 2014 | Carradori, Simone; D'Ascenzio, Melissa; Chimenti, Paola; Secci, Daniela; Bolasco, Adriana | |
| Cyclic tertiary sulfamates: Selective inhibition of the tumor-associated carbonic anhydrases IX and XII by N- and O-substituted acesulfame derivatives | 2014 | DE MONTE, Celeste; Carradori, Simone; Secci, Daniela; D'Ascenzio, Melissa; Vullo, D; Ceruso, M; Supuran, Ct | |
| Opening new scenarios for human MAO inhibitors | 2015 | DE MONTE, Celeste; D'Ascenzio, Melissa; Guglielmi, Paolo; Mancini, Veronica; Carradori, Simone | |
| Synthesis and pharmacological screening of a large library of 1,3,4-thiadiazolines as innovative therapeutic tools for the treatment of prostate cancer and melanoma | 2015 | DE MONTE, Celeste; Carradori, Simone; Secci, Daniela; D'Ascenzio, Melissa; Guglielmi, Paolo; Mollica, Adriano; Morrone, Stefania; Scarpa, Susanna; Agliano', Anna Maria; Giantulli, Sabrina; Silvestri, Ida | |
| New amide derivatives of Probenecid as selective inhibitors of carbonic anhydrase IX and XII: Biological evaluation and molecular modelling studies | 2015 | Carradori, Simone; Mollica, Adriano; Ceruso, Mariangela; D'Ascenzio, Melissa; DE MONTE, Celeste; Chimenti, Paola; Sabia, Rocchina; Akdemir, Atilla; Supuran, Claudiu T. | |
| Synthesis, biological evaluation and quantitative structure-active relationships of 1,3-thiazolidin-4-one derivatives. A promising chemical scaffold endowed with high antifungal potency and low cytotoxicity | 2017 | Carradori, Simone; Bizzarri, Bruna; D'Ascenzio, Melissa; DE MONTE, Celeste; Grande, Rossella; Rivanera, Daniela; Zicari, Alessanda; Mari, Emanuela; Sabatino, Manuela; Patsilinakos, Alexandros; Ragno, Rino; Secci, Daniela | |
| 4-(3-Nitrophenyl)thiazol-2-ylhydrazone derivatives as antioxidants and selective hMAO-B inhibitors: synthesis, biological activity and computational analysis | 2019 | Secci, Daniela; Carradori, Simone; Petzer, Anél; Guglielmi, Paolo; D’Ascenzio, Melissa; Chimenti, Paola; Bagetta, Donatella; Alcaro, Stefano; Zengin, Gokhan; Petzer, Jacobus P.; Ortuso, Francesco |
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