Sfoglia per Autore
Novel therapeutic opportunities for Toxoplasma gondii, Trichomonas vaginalis, and Giardia intestinalis infections
2023 Arrighi, Francesca; Granese, Arianna; Chimenti, Paola; Guglielmi, Paolo
A novel class of dual-acting DCH-CORMs counteracts oxidative stress-induced inflammation in human primary tenocytes
2021 Appetecchia, F.; Consalvi, S.; Berrino, E.; Gallorini, M.; Granese, A.; Campestre, C.; Carradori, S.; Biava, M.; Poce, G.
Synthesis and evaluation of thymol-based synthetic derivatives as dual-action inhibitors against different strains of h. pylori and AGS cell line
2021 Sisto, F.; Carradori, S.; Guglielmi, P.; Spano, M.; Secci, D.; Granese, A.; Sobolev, A. P.; Grande, R.; Campestre, C.; Di Marcantonio, M. C.; Mincione, G.
Phytochemical analyses and pharmacological screening of Neem oil
2019 Cesa, S.; Sisto, F.; Zengin, G.; Scaccabarozzi, D.; Kokolakis, A. K.; Scaltrito, M. M.; Grande, R.; Locatelli, M.; Cacciagrano, F.; Angiolella, L.; Campestre, C.; Granese, A.; Chimenti, P.; Basilico, N.
Analytical procedures for secondary metabolites determination. Recent trends and future perspectives
2018 Menghini, Luigi; Bellagamba, Giuseppe; Marcelli, Fabiana; Armellani, Luca; Granese, Arianna; De Luca, Elisa; Cifelli, Roberta; Nilgun Zengin, Kucukercan; Abdurrahman, Aktumsek; Gokhan, Zengin
Antimicrobial activity, synergism and inhibition of germ tube formation by Crocus sativus-derived compounds against Candida spp
2016 Carradori, Simone; Fazzari, Marina; Granese, Arianna; Chimenti, Paola; Angiolella, Letizia
Nitric oxide donors and selective carbonic anhydrase inhibitors: A dual pharmacological approach for the treatment of glaucoma, cancer and osteoporosis
2015 Carradori, Simone; Mollica, Adriano; DE MONTE, Celeste; Granese, Arianna; Supuran, Claudiu T.
(Thiazol-2-yl)hydrazone derivatives from acetylpyridines as dual inhibitors of MAO and AChE: synthesis, biological evaluation and molecular modeling studies
2015 D’Ascenzio, M; Chimenti, Paola; Gidaro, Mc; DE MONTE, Celeste; DE VITA, Daniela; Granese, Arianna; Scipione, Luigi; DI SANTO, Roberto; Costa, G; Alcaro, S; Yáñez, M; Carradori, S.
Bioactive compounds of Crocus sativus L. and their semisynthetic derivatives as promising anti-Helicobacter pylori, anti-malarial and anti-leishmanial agents
2015 DE MONTE, Celeste; Bizzarri, Bruna; Gidaro, Maria Concetta; Carradori, Simone; Mollica, Adriano; Luisi, Grazia; Granese, Arianna; Alcaro, Stefano; Costa, Giosuè; Basilico, Nicoletta; Parapini, Silvia; Scaltrito, Maria Maddalena; Masia, Carla; Sisto, Francesca
Modern extraction techniques and their impact on the pharmacological profile of Serenoa repens extracts for the treatment of lower urinary tract symptoms.
2014 DE MONTE, Celeste; S., Carradori; Granese, Arianna; DI PIERRO, GIOVANNI BATTISTA; Leonardo, Costantino; DE NUNZIO, Cosimo
Synthesis and biological evaluation of novel 2,4-disubstituted-1,3-thiazoles as anti-Candida spp. agents
2011 Franco, Chimenti; Bizzarri, Bruna; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Granese, Arianna; Simone, Carradori; Melissa, D'Ascenzio; Lilli, Daniela; Rivanera, Daniela
Synthesis and characterization of new 3-acyl-7-hydroxy-6,8-substituted-coumarin and 3-acyl-7-benzyloxy-6,8-substituted-coumarin derivatives
2010 Chimenti, Franco; Bolasco, Adriana; Secci, Daniela; Bizzarri, Bruna; Chimenti, Paola; Granese, A; Carradori, S.
Synthesis, semipreparative HPLC separation, biological evaluation, and 3D-QSAR of hydrazothiazole derivatives as human monoamine oxidase B inhibitors
2010 Chimenti, Franco; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Arianna, Granese; Simone, Carradori; Elias, Maccioni; M., Cristina Cardia; Matilde, Yanez; Francisco, Orallo; Stefano, Alcaro; Francesco, Ortuso; Roberto, Cirilli; Rosella, Ferretti; Simona, Distinto; Johannes, Kirchmair; Thierry, Langer
Investigations on the 2-thiazolylhydrazyne scaffold: Synthesis and molecular modeling of selective human monoamine oxidase inhibitors
2010 Chimenti, Franco; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Arianna, Granese; Simone, Carradori; Matilde, Yanez; Francisco, Orallo; Francesco, Ortuso; Stefano, Alcaro
SYNTHESIS, STEREOCHEMICAL SEPARATION, AND BIOLOGICAL EVALUATION OF SELECTIVE INHIBITORS OF HUMAN MAO-B: 1-(4-ARYLTHIAZOL-2-YL)-2-(3-METHYLCYCLOHEXYLIDENE)HYDRAZINES
2010 Chimenti, Franco; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Granese, A; Carradori, S; Yanez, M; Orallo, F; Sanna, Ml; Gallinella, B; Cirilli, R.
Synthesis and selective inhibition of human monoamine oxidases of a large scaffold of (4,5-substituted-thiazol-2-yl)hydrazones
2010 Chimenti, Franco; Secci, Daniela; Chimenti, Paola; Granese, Arianna; Carradori, Simone; D'Ascenzio, Melissa; Matilde, Yanez; Francisco, Orallo; Bolasco, Adriana
Synthesis and anti-Helicobacter pylori activity of 4-(coumarin-3-yl)thiazol-2-ylhydrazone derivatives
2010 Chimenti, F; Bizzarri, Bruna; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Granese, A; Carradori, S; D'Ascenzio, M; SCALTRITO M., M; Sisto, F.
Synthesis, selective anti-Helicobacter pylori activity, and cytotoxicity of novel N-substituted-2-oxo-2H-1-benzopyran-3-carboxamides
2010 Chimenti, Franco; Bizzarri, Bruna; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Granese, Arianna; Carradori, Simone; Rivanera, Daniela; Zicari, Alessandra; M., Maddalena Scaltrito; Francesca, Sisto
Synthesis and inhibitory activity against human monoamine oxidase of N1-thiocarbamoyl-3,5-di(hetero)aryl-4,5-dihydro-(1H)-pyrazole derivatives
2010 Chimenti, Franco; Carradori, Simone; Secci, Daniela; Bolasco, Adriana; Bizzarri, Bruna; Chimenti, Paola; Arianna, Granese; Matilde, Yanez; Francisco, Orallo
Synthesis, Molecular Modeling, and Selective Inhibitory Activity against Human Monoamine Oxidases of 3-Carboxamido-7-Substituted Coumarins.
2009 Chimenti, Franco; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Bizzarri, Bruna; Granese, Arianna; Carradori, Simone; Yanez, Matilde; Orallo, Francisco; Ortuso, Francesco; Alcaro, Stefano
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Novel therapeutic opportunities for Toxoplasma gondii, Trichomonas vaginalis, and Giardia intestinalis infections | 2023 | Arrighi, Francesca; Granese, Arianna; Chimenti, Paola; Guglielmi, Paolo | |
A novel class of dual-acting DCH-CORMs counteracts oxidative stress-induced inflammation in human primary tenocytes | 2021 | Appetecchia, F.; Consalvi, S.; Berrino, E.; Gallorini, M.; Granese, A.; Campestre, C.; Carradori, S.; Biava, M.; Poce, G. | |
Synthesis and evaluation of thymol-based synthetic derivatives as dual-action inhibitors against different strains of h. pylori and AGS cell line | 2021 | Sisto, F.; Carradori, S.; Guglielmi, P.; Spano, M.; Secci, D.; Granese, A.; Sobolev, A. P.; Grande, R.; Campestre, C.; Di Marcantonio, M. C.; Mincione, G. | |
Phytochemical analyses and pharmacological screening of Neem oil | 2019 | Cesa, S.; Sisto, F.; Zengin, G.; Scaccabarozzi, D.; Kokolakis, A. K.; Scaltrito, M. M.; Grande, R.; Locatelli, M.; Cacciagrano, F.; Angiolella, L.; Campestre, C.; Granese, A.; Chimenti, P.; Basilico, N. | |
Analytical procedures for secondary metabolites determination. Recent trends and future perspectives | 2018 | Menghini, Luigi; Bellagamba, Giuseppe; Marcelli, Fabiana; Armellani, Luca; Granese, Arianna; De Luca, Elisa; Cifelli, Roberta; Nilgun Zengin, Kucukercan; Abdurrahman, Aktumsek; Gokhan, Zengin | |
Antimicrobial activity, synergism and inhibition of germ tube formation by Crocus sativus-derived compounds against Candida spp | 2016 | Carradori, Simone; Fazzari, Marina; Granese, Arianna; Chimenti, Paola; Angiolella, Letizia | |
Nitric oxide donors and selective carbonic anhydrase inhibitors: A dual pharmacological approach for the treatment of glaucoma, cancer and osteoporosis | 2015 | Carradori, Simone; Mollica, Adriano; DE MONTE, Celeste; Granese, Arianna; Supuran, Claudiu T. | |
(Thiazol-2-yl)hydrazone derivatives from acetylpyridines as dual inhibitors of MAO and AChE: synthesis, biological evaluation and molecular modeling studies | 2015 | D’Ascenzio, M; Chimenti, Paola; Gidaro, Mc; DE MONTE, Celeste; DE VITA, Daniela; Granese, Arianna; Scipione, Luigi; DI SANTO, Roberto; Costa, G; Alcaro, S; Yáñez, M; Carradori, S. | |
Bioactive compounds of Crocus sativus L. and their semisynthetic derivatives as promising anti-Helicobacter pylori, anti-malarial and anti-leishmanial agents | 2015 | DE MONTE, Celeste; Bizzarri, Bruna; Gidaro, Maria Concetta; Carradori, Simone; Mollica, Adriano; Luisi, Grazia; Granese, Arianna; Alcaro, Stefano; Costa, Giosuè; Basilico, Nicoletta; Parapini, Silvia; Scaltrito, Maria Maddalena; Masia, Carla; Sisto, Francesca | |
Modern extraction techniques and their impact on the pharmacological profile of Serenoa repens extracts for the treatment of lower urinary tract symptoms. | 2014 | DE MONTE, Celeste; S., Carradori; Granese, Arianna; DI PIERRO, GIOVANNI BATTISTA; Leonardo, Costantino; DE NUNZIO, Cosimo | |
Synthesis and biological evaluation of novel 2,4-disubstituted-1,3-thiazoles as anti-Candida spp. agents | 2011 | Franco, Chimenti; Bizzarri, Bruna; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Granese, Arianna; Simone, Carradori; Melissa, D'Ascenzio; Lilli, Daniela; Rivanera, Daniela | |
Synthesis and characterization of new 3-acyl-7-hydroxy-6,8-substituted-coumarin and 3-acyl-7-benzyloxy-6,8-substituted-coumarin derivatives | 2010 | Chimenti, Franco; Bolasco, Adriana; Secci, Daniela; Bizzarri, Bruna; Chimenti, Paola; Granese, A; Carradori, S. | |
Synthesis, semipreparative HPLC separation, biological evaluation, and 3D-QSAR of hydrazothiazole derivatives as human monoamine oxidase B inhibitors | 2010 | Chimenti, Franco; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Arianna, Granese; Simone, Carradori; Elias, Maccioni; M., Cristina Cardia; Matilde, Yanez; Francisco, Orallo; Stefano, Alcaro; Francesco, Ortuso; Roberto, Cirilli; Rosella, Ferretti; Simona, Distinto; Johannes, Kirchmair; Thierry, Langer | |
Investigations on the 2-thiazolylhydrazyne scaffold: Synthesis and molecular modeling of selective human monoamine oxidase inhibitors | 2010 | Chimenti, Franco; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Arianna, Granese; Simone, Carradori; Matilde, Yanez; Francisco, Orallo; Francesco, Ortuso; Stefano, Alcaro | |
SYNTHESIS, STEREOCHEMICAL SEPARATION, AND BIOLOGICAL EVALUATION OF SELECTIVE INHIBITORS OF HUMAN MAO-B: 1-(4-ARYLTHIAZOL-2-YL)-2-(3-METHYLCYCLOHEXYLIDENE)HYDRAZINES | 2010 | Chimenti, Franco; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Granese, A; Carradori, S; Yanez, M; Orallo, F; Sanna, Ml; Gallinella, B; Cirilli, R. | |
Synthesis and selective inhibition of human monoamine oxidases of a large scaffold of (4,5-substituted-thiazol-2-yl)hydrazones | 2010 | Chimenti, Franco; Secci, Daniela; Chimenti, Paola; Granese, Arianna; Carradori, Simone; D'Ascenzio, Melissa; Matilde, Yanez; Francisco, Orallo; Bolasco, Adriana | |
Synthesis and anti-Helicobacter pylori activity of 4-(coumarin-3-yl)thiazol-2-ylhydrazone derivatives | 2010 | Chimenti, F; Bizzarri, Bruna; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Granese, A; Carradori, S; D'Ascenzio, M; SCALTRITO M., M; Sisto, F. | |
Synthesis, selective anti-Helicobacter pylori activity, and cytotoxicity of novel N-substituted-2-oxo-2H-1-benzopyran-3-carboxamides | 2010 | Chimenti, Franco; Bizzarri, Bruna; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Granese, Arianna; Carradori, Simone; Rivanera, Daniela; Zicari, Alessandra; M., Maddalena Scaltrito; Francesca, Sisto | |
Synthesis and inhibitory activity against human monoamine oxidase of N1-thiocarbamoyl-3,5-di(hetero)aryl-4,5-dihydro-(1H)-pyrazole derivatives | 2010 | Chimenti, Franco; Carradori, Simone; Secci, Daniela; Bolasco, Adriana; Bizzarri, Bruna; Chimenti, Paola; Arianna, Granese; Matilde, Yanez; Francisco, Orallo | |
Synthesis, Molecular Modeling, and Selective Inhibitory Activity against Human Monoamine Oxidases of 3-Carboxamido-7-Substituted Coumarins. | 2009 | Chimenti, Franco; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Bizzarri, Bruna; Granese, Arianna; Carradori, Simone; Yanez, Matilde; Orallo, Francisco; Ortuso, Francesco; Alcaro, Stefano |
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