Sfoglia per Autore
Recent development of monoamine oxidase inhibitors
2005 Bolasco, Adriana; Fioravanti, Rossella; Carradori, Simone
Synthesis, molecular modeling studies, and selective inhibitory activity against monoamine oxidase of N,N'-bis[2-oxo-2H-benzopyran]-3-carboxamides
2006 Chimenti, Franco; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Granese, Arianna; Carradori, Simone; O., Befani; Turini, Paola; S., Alcaro; F., Ortuso
Synthesis and in vitro selective anti-Helicobacter pylori activity of N-substituted-2-oxo-2H-1-benzopyran-3-carboxamides
2006 Chimenti, Franco; Bizzarri, Bruna; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Carradori, Simone; Granese, Arianna; Rivanera, Daniela; Lilli, Daniela; Maddalena Scaltrito, M.; Immacolata Brenciaglia, M.
A novel class of selective anti-Helicobacter pylori agents 2-Oxo-2H-chromene-3-carboxamide derivatives.
2007 Chimenti, Franco; Bizzarri, Bruna; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Carradori, Simone; Granese, Arianna; Rivanera, Daniela; Lilli, Daniela; Zicari, Alessandra; SCALTRITO M., M; Sisto, F.
Synthesis and in vitro activity of 2-thiazolylhydrazone derivatives compared with the activity of clotrimazole against clinical isolates of Candida spp.
2007 Chimenti, Franco; Bizzarri, Bruna; Elias, Maccioni; Secci, Daniela; Bolasco, Adriana; Fioravanti, Rossella; Chimenti, Paola; Granese, Arianna; Carradori, Simone; Rivanera, Daniela; Lilli, Daniela; Zicari, Alessandra; Simona, Distinto
High-performance liquid chromatographic separation of enantiomers and diastereomers of 2-methylcyclohexanone thiosemicarbazone, and determination of absolute configuration and configurational stability
2007 Cirilli, R.; Ferretti, R.; Torre, F. La; Secci, Daniela; Bolasco, Adriana; Carradori, Simone; Pierini, Marco
Synthesis, Stereochemical Identification, and Selective Inhibitory Activity against Human Monoamine Oxidase-B of 2-Methylcyclohexylidene-(4-arylthiazol-2-yl)hydrazones
2008 Chimenti, F.; Maccioni, E.; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Granese, Arianna; Carradori, Simone; Alcaro, S.; Ortuso, F.; Yanez, M.; Orallo, F.; Cirilli, R.; Ferretti, R.; LA TORRE, F.
Synthesis and Evaluation of 4-Acyl-2- Thiazolylhydrazone Derivatives for anti-Toxoplasma Efficacy in Vitro
2009 Chimenti, Franco; Bizzarri, Bruna; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Carradori, Simone; A., Granese; Rivanera, Daniela; N., Frishberg; C., Bordón; L., JONES BRANDO
Synthesis, Molecular Modeling, and Selective Inhibitory Activity against Human Monoamine Oxidases of 3-Carboxamido-7-Substituted Coumarins.
2009 Chimenti, Franco; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Bizzarri, Bruna; Granese, Arianna; Carradori, Simone; Yanez, Matilde; Orallo, Francisco; Ortuso, Francesco; Alcaro, Stefano
Synthesis and Biological Evaluation of Novel Conjugated Coumarin-Thiazole Systems
2009 Chimenti, Franco; Carradori, Simone; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Granese, Arianna; Bizzarri, Bruna
A Novel Histone Acetyltransferase Inhibitor Modulating Gcn5 Network: Cyclopentylidene-[4-(4′-chlorophenyl)thiazol-2-yl)hydrazone
2009 Chimenti, Franco; Bizzarri, Bruna; Elias, Maccioni; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Fioravanti, Rossella; Granese, Arianna; Carradori, Simone; Federica, Tosi; Ballario, Paola; S., Vernarecci; Patrizia, Filetici
Synthesis and selective inhibition of human monoamine oxidases of a large scaffold of (4,5-substituted-thiazol-2-yl)hydrazones
2010 Chimenti, Franco; Secci, Daniela; Chimenti, Paola; Granese, Arianna; Carradori, Simone; D'Ascenzio, Melissa; Matilde, Yanez; Francisco, Orallo; Bolasco, Adriana
Synthesis, selective anti-Helicobacter pylori activity, and cytotoxicity of novel N-substituted-2-oxo-2H-1-benzopyran-3-carboxamides
2010 Chimenti, Franco; Bizzarri, Bruna; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Granese, Arianna; Carradori, Simone; Rivanera, Daniela; Zicari, Alessandra; M., Maddalena Scaltrito; Francesca, Sisto
Synthesis and inhibitory activity against human monoamine oxidase of N1-thiocarbamoyl-3,5-di(hetero)aryl-4,5-dihydro-(1H)-pyrazole derivatives
2010 Chimenti, Franco; Carradori, Simone; Secci, Daniela; Bolasco, Adriana; Bizzarri, Bruna; Chimenti, Paola; Arianna, Granese; Matilde, Yanez; Francisco, Orallo
CPTH6, A NOVEL Gcn5/pCAF HISTONE ACETYLTRANSFERASE INHIBITOR, INDUCES BOTH APOPTOSIS AND AUTOPHAGY IN HUMAN LEUKEMIA CELLS
2011 Ragazzoni, Y.; Trisciuoglio, D.; Gabellini, C. .; Pelosi, A.; Desideri, M.; Carradori, Simone; Secci, Daniela; Rizzo, M. G.; Del, Bufalo
Synthesis and selective human monoamine oxidase inhibition of 3-carbonyl, 3-acyl, and 3-carboxyhydrazido coumarin derivatives
2011 Secci, Daniela; Carradori, Simone; Bolasco, Adriana; Chimenti, Paola; Yanez, Matilde; Ortuso, Francesco; Alcaro, Stefano
The State of the Art of Pyrazole Derivatives as Monoamine Oxidase Inhibitors and Antidepressant/Anticonvulsant Agents
2011 Secci, Daniela; Bolasco, Adriana; Carradori, Simone; Chimenti, Paola
EPIGENETIC MODULATION OF PGC-1a ACTIVITY BY GCN5 INHIBITORS: WO2010007085
2011 Carradori, Simone; Secci, Daniela; Mai, Antonello
Recent advances in the development of selective human MAO-B inhibitors: (Hetero)arylidene-(4-substituted-thiazol-2- yl)hydrazines
2012 Secci, Daniela; Bolasco, Adriana; Carradori, Simone; D'Ascenzio, Melissa; Nescatelli, Riccardo; M., Yáñez
Patent-related survey on new monoamine oxidase inhibitors and their therapeutic potential
2012 Carradori, Simone; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; D'Ascenzio, Melissa
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Recent development of monoamine oxidase inhibitors | 2005 | Bolasco, Adriana; Fioravanti, Rossella; Carradori, Simone | |
Synthesis, molecular modeling studies, and selective inhibitory activity against monoamine oxidase of N,N'-bis[2-oxo-2H-benzopyran]-3-carboxamides | 2006 | Chimenti, Franco; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Granese, Arianna; Carradori, Simone; O., Befani; Turini, Paola; S., Alcaro; F., Ortuso | |
Synthesis and in vitro selective anti-Helicobacter pylori activity of N-substituted-2-oxo-2H-1-benzopyran-3-carboxamides | 2006 | Chimenti, Franco; Bizzarri, Bruna; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Carradori, Simone; Granese, Arianna; Rivanera, Daniela; Lilli, Daniela; Maddalena Scaltrito, M.; Immacolata Brenciaglia, M. | |
A novel class of selective anti-Helicobacter pylori agents 2-Oxo-2H-chromene-3-carboxamide derivatives. | 2007 | Chimenti, Franco; Bizzarri, Bruna; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Carradori, Simone; Granese, Arianna; Rivanera, Daniela; Lilli, Daniela; Zicari, Alessandra; SCALTRITO M., M; Sisto, F. | |
Synthesis and in vitro activity of 2-thiazolylhydrazone derivatives compared with the activity of clotrimazole against clinical isolates of Candida spp. | 2007 | Chimenti, Franco; Bizzarri, Bruna; Elias, Maccioni; Secci, Daniela; Bolasco, Adriana; Fioravanti, Rossella; Chimenti, Paola; Granese, Arianna; Carradori, Simone; Rivanera, Daniela; Lilli, Daniela; Zicari, Alessandra; Simona, Distinto | |
High-performance liquid chromatographic separation of enantiomers and diastereomers of 2-methylcyclohexanone thiosemicarbazone, and determination of absolute configuration and configurational stability | 2007 | Cirilli, R.; Ferretti, R.; Torre, F. La; Secci, Daniela; Bolasco, Adriana; Carradori, Simone; Pierini, Marco | |
Synthesis, Stereochemical Identification, and Selective Inhibitory Activity against Human Monoamine Oxidase-B of 2-Methylcyclohexylidene-(4-arylthiazol-2-yl)hydrazones | 2008 | Chimenti, F.; Maccioni, E.; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Granese, Arianna; Carradori, Simone; Alcaro, S.; Ortuso, F.; Yanez, M.; Orallo, F.; Cirilli, R.; Ferretti, R.; LA TORRE, F. | |
Synthesis and Evaluation of 4-Acyl-2- Thiazolylhydrazone Derivatives for anti-Toxoplasma Efficacy in Vitro | 2009 | Chimenti, Franco; Bizzarri, Bruna; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Carradori, Simone; A., Granese; Rivanera, Daniela; N., Frishberg; C., Bordón; L., JONES BRANDO | |
Synthesis, Molecular Modeling, and Selective Inhibitory Activity against Human Monoamine Oxidases of 3-Carboxamido-7-Substituted Coumarins. | 2009 | Chimenti, Franco; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Bizzarri, Bruna; Granese, Arianna; Carradori, Simone; Yanez, Matilde; Orallo, Francisco; Ortuso, Francesco; Alcaro, Stefano | |
Synthesis and Biological Evaluation of Novel Conjugated Coumarin-Thiazole Systems | 2009 | Chimenti, Franco; Carradori, Simone; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Granese, Arianna; Bizzarri, Bruna | |
A Novel Histone Acetyltransferase Inhibitor Modulating Gcn5 Network: Cyclopentylidene-[4-(4′-chlorophenyl)thiazol-2-yl)hydrazone | 2009 | Chimenti, Franco; Bizzarri, Bruna; Elias, Maccioni; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Fioravanti, Rossella; Granese, Arianna; Carradori, Simone; Federica, Tosi; Ballario, Paola; S., Vernarecci; Patrizia, Filetici | |
Synthesis and selective inhibition of human monoamine oxidases of a large scaffold of (4,5-substituted-thiazol-2-yl)hydrazones | 2010 | Chimenti, Franco; Secci, Daniela; Chimenti, Paola; Granese, Arianna; Carradori, Simone; D'Ascenzio, Melissa; Matilde, Yanez; Francisco, Orallo; Bolasco, Adriana | |
Synthesis, selective anti-Helicobacter pylori activity, and cytotoxicity of novel N-substituted-2-oxo-2H-1-benzopyran-3-carboxamides | 2010 | Chimenti, Franco; Bizzarri, Bruna; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Granese, Arianna; Carradori, Simone; Rivanera, Daniela; Zicari, Alessandra; M., Maddalena Scaltrito; Francesca, Sisto | |
Synthesis and inhibitory activity against human monoamine oxidase of N1-thiocarbamoyl-3,5-di(hetero)aryl-4,5-dihydro-(1H)-pyrazole derivatives | 2010 | Chimenti, Franco; Carradori, Simone; Secci, Daniela; Bolasco, Adriana; Bizzarri, Bruna; Chimenti, Paola; Arianna, Granese; Matilde, Yanez; Francisco, Orallo | |
CPTH6, A NOVEL Gcn5/pCAF HISTONE ACETYLTRANSFERASE INHIBITOR, INDUCES BOTH APOPTOSIS AND AUTOPHAGY IN HUMAN LEUKEMIA CELLS | 2011 | Ragazzoni, Y.; Trisciuoglio, D.; Gabellini, C. .; Pelosi, A.; Desideri, M.; Carradori, Simone; Secci, Daniela; Rizzo, M. G.; Del, Bufalo | |
Synthesis and selective human monoamine oxidase inhibition of 3-carbonyl, 3-acyl, and 3-carboxyhydrazido coumarin derivatives | 2011 | Secci, Daniela; Carradori, Simone; Bolasco, Adriana; Chimenti, Paola; Yanez, Matilde; Ortuso, Francesco; Alcaro, Stefano | |
The State of the Art of Pyrazole Derivatives as Monoamine Oxidase Inhibitors and Antidepressant/Anticonvulsant Agents | 2011 | Secci, Daniela; Bolasco, Adriana; Carradori, Simone; Chimenti, Paola | |
EPIGENETIC MODULATION OF PGC-1a ACTIVITY BY GCN5 INHIBITORS: WO2010007085 | 2011 | Carradori, Simone; Secci, Daniela; Mai, Antonello | |
Recent advances in the development of selective human MAO-B inhibitors: (Hetero)arylidene-(4-substituted-thiazol-2- yl)hydrazines | 2012 | Secci, Daniela; Bolasco, Adriana; Carradori, Simone; D'Ascenzio, Melissa; Nescatelli, Riccardo; M., Yáñez | |
Patent-related survey on new monoamine oxidase inhibitors and their therapeutic potential | 2012 | Carradori, Simone; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; D'Ascenzio, Melissa |
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