Sfoglia per Autore
Interactions of polysulfanes with components of red blood cells
2011 Schneider, Thomas; Ba, Lalla A.; Khairan, Khairan; Zwergel, Clemens; Bach, Nguyen Duc; Bernhardt, Ingolf; Brandt, Wolfgang; Wessjohann, Ludger; Diederich, Marc; Jacob, Claus
Aurones: Interesting Natural and Synthetic Compounds with Emerging Biological Potential
2012 Zwergel, Clemens; F., Gaascht; Valente, Sergio; M., Diederich; D., Bagrel; G., Kirsch
Reactivity of 4-vinyl-2H-1-benzopyran-2-ones in diels-alder cycloaddition reactions: Access to coumarin-based polycycles with Cdc25 phosphatase-inhibiting activity
2013 Valente, Sergio; Zhanjie, Xu; Emilie, Bana; Zwergel, Clemens; Mai, Antonello; Jacob, Claus; Peter, Meiser; Denyse, Bagrel; Artur M. S., Silva; Kirsch, Gilbert
Novel benzofuran-chromone and -coumarin derivatives: Synthesis and biological activity in K562 human leukemia cells
2013 Zwergel, Clemens; Valente, Sergio; Salvato, Angela; Xu, Zhanjie; Talhi, Oualid; Mai, Antonello; Silva, Artur; Altucci, Lucia; Kirsch, Gilbert
Selective Non-nucleoside Inhibitors of Human DNA Methyltransferases Active in Cancer Including in Cancer Stem Cells
2014 Valente, Sergio; Yiwei, Liu; Michael, Schnekenburger; Zwergel, Clemens; Sandro, Cosconati; Christina, Gros; Maria, Tardugno; Donatella, Labella; Cristina, Florean; Steven, Minden; Hideharu, Hashimoto; Yanqi, Chang; Xing, Zhang; Gilbert, Kirsch; Ettore, Novellino; Paola B., Arimondo; Miele, Evelina; Ferretti, Elisabetta; Gulino, Alberto; Marc, Diederich; Xiaodong, Cheng; Mai, Antonello
Novel inhibitors of human histone deacetylases: Design, synthesis and bioactivity of 3-alkenoylcoumarines
2014 C., Seidel; M., Schnekenburger; Zwergel, Clemens; F., Gaascht; Mai, Antonello; M., Dicato; G., Kirsch; Valente, Sergio; M., Diederich
Novel histone deacetylase inhibitors induce growth arrest, apoptosis, and differentiation in sarcoma cancer stem cells
2015 G., Di Pompo; M., Salerno; Rotili, Dante; Valente, Sergio; Zwergel, Clemens; S., Avnet; G., Lattanzi; N., Baldini; Mai, Antonello
Emerging approaches for histone deacetylase inhibitor drug discovery
2015 Zwergel, Clemens; Valente, Sergio; Jacob, Claus; Mai, Antonello
Abstract 2946: Effects of two novel quinoline-based non-nucleoside DNA methyltransferase inhibitors against bone sarcomas
2015 Manara, Maria Cristina; Valente, Sergio; Cristalli, Camilla; Baricordi, Cristina; Zwergel, Clemens; Arimondo, Paola B; Picci, Piero; Mai, Antonello; Scotlandi, Katia
Histone deacetylase inhibitors restore IL-10 expression in lipopolysaccharide-induced cell inflammation and reduce IL-1β and IL-6 production in breast silicone implant in C57BL/6J wild-type murine model
2016 Di Liddo, Rosa; Valente, Sergio; Taurone, Samanta; Zwergel, Clemens; Marrocco, Biagina; Turchetta, Rosaria; Conconi, Maria Teresa; Scarpa, Carlotta; Bertalot, Thomas; Schrenk, Sandra; Mai, Antonello; Artico, Marco
1,4-Dihydropyridines Active on the SIRT1/AMPK Pathway Ameliorate Skin Repair and Mitochondrial Function and Exhibit Inhibition of Proliferation in Cancer Cells
2016 Valente, Sergio; Mellini, Paolo; Spallotta, Francesco; Carafa, Vincenzo; Nebbioso, Angela; Polletta, Lucia; Carnevale, Ilaria; Saladini, Serena; Trisciuoglio, Daniela; Gabellini, Chiara; Tardugno, Maria; Zwergel, Clemens; Cencioni, Chiara; Atlante, Sandra; Moniot, Sébastien; Steegborn, Clemens; Budriesi, Roberta; Tafani, Marco; Del Bufalo, Donatella; Altucci, Lucia; Gaetano, Carlo; Mai, Antonello
DNA methyltransferases Inhibitors from natural sources
2016 Zwergel, Clemens; Valente, Sergio; Mai, Antonello
One-pot synthesis of benzopyran-4-ones with cancer preventive and therapeutic potential
2016 Talhi, Oualid; Brodziak Jarosz, Lidia; Panning, Jana; Orlikova, Barbora; Zwergel, Clemens; Tzanova, Tzvetomira; Philippot, Stéphanie; Pinto, Diana C. G. A.; Paz, Filipe A. Almeida; Gerhaüser, Clarissa; Dick, Tobias P.; Jacob, Claus; Diederich, Marc; Bagrel, Denyse; Kirsch, Gilbert; Silva, Artur M. S.
MC1568 inhibits HDAC6/8 activity and influenza A virus replication in lung epithelial cells: Role of Hsp90 acetylation
2016 Panella, Simona; Marcocci, Maria Elena; Celestino, Ignacio; Valente, Sergio; Zwergel, Clemens; Li Puma, Domenica Donatella; Nencioni, Lucia; Mai, Antonello; Palamara, ANNA TERESA; Simonetti, Giovanna
LSD1 inhibitors: a patent review (2010-2015)
2016 Stazi, Giulia; Zwergel, Clemens; Valente, Sergio; Mai, Antonello
Novel coumarin- and quinolinone-based polycycles as cell division cycle 25-A and -C phosphatases inhibitors induce proliferation arrest and apoptosis in cancer cells
2017 Zwergel, Clemens; Czepukojc, Brigitte; Evain Bana, Emilie; Xu, Zhanjie; Stazi, Giulia; Mori, Mattia; Patsilinakos, Alexandros; Mai, Antonello; Botta, Bruno; Ragno, Rino; Bagrel, Denise; Kirsch, Gilbert; Meiser, Peter; Jacob, Claus; Montenarh, Mathias; Valente, Sergio
The histone methyltransferase EZH2 as a druggable target in SHH medulloblastoma cancer stem cells
2017 Miele, Evelina; Valente, Sergio; Alfano, Vincenzo; Silvano, Marianna; Mellini, Paolo; Borovika, Diana; Marrocco, Biagina; Po, Agnese; Besharat, Zein Mersini; Catanzaro, Giuseppina; Battaglia, Giuseppe; Abballe, Luana; Zwergel, Clemens; Stazi, Giulia; Milite, Ciro; Castellano, Sabrina; Tafani, Marco; Trapencieris, Peteris; Mai, Antonello; Ferretti, Elisabetta
Metabolite profiling of ascidian Styela plicata using LC–MS with multivariate statistical analysis and their antitumor activity
2017 Palanisamy, S. K.; Trisciuoglio, D.; Zwergel, C.; Del Bufalo, D.; Mai, A.
Epi-drugs in combination with immunotherapy: a new avenue to improve anticancer efficacy
2017 Mazzone, Roberta; Zwergel, Clemens; Mai, Antonello; Valente, Sergio
Towards the development of activity-based probes for detection of lysine-specific demethylase-1 activity.
2017 Ourailidou, Me; Lenoci, A; Zwergel, Clemens; Rotili, Dante; Mai, Antonello; Dekker, F. j. 4.
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Interactions of polysulfanes with components of red blood cells | 2011 | Schneider, Thomas; Ba, Lalla A.; Khairan, Khairan; Zwergel, Clemens; Bach, Nguyen Duc; Bernhardt, Ingolf; Brandt, Wolfgang; Wessjohann, Ludger; Diederich, Marc; Jacob, Claus | |
| Aurones: Interesting Natural and Synthetic Compounds with Emerging Biological Potential | 2012 | Zwergel, Clemens; F., Gaascht; Valente, Sergio; M., Diederich; D., Bagrel; G., Kirsch | |
| Reactivity of 4-vinyl-2H-1-benzopyran-2-ones in diels-alder cycloaddition reactions: Access to coumarin-based polycycles with Cdc25 phosphatase-inhibiting activity | 2013 | Valente, Sergio; Zhanjie, Xu; Emilie, Bana; Zwergel, Clemens; Mai, Antonello; Jacob, Claus; Peter, Meiser; Denyse, Bagrel; Artur M. S., Silva; Kirsch, Gilbert | |
| Novel benzofuran-chromone and -coumarin derivatives: Synthesis and biological activity in K562 human leukemia cells | 2013 | Zwergel, Clemens; Valente, Sergio; Salvato, Angela; Xu, Zhanjie; Talhi, Oualid; Mai, Antonello; Silva, Artur; Altucci, Lucia; Kirsch, Gilbert | |
| Selective Non-nucleoside Inhibitors of Human DNA Methyltransferases Active in Cancer Including in Cancer Stem Cells | 2014 | Valente, Sergio; Yiwei, Liu; Michael, Schnekenburger; Zwergel, Clemens; Sandro, Cosconati; Christina, Gros; Maria, Tardugno; Donatella, Labella; Cristina, Florean; Steven, Minden; Hideharu, Hashimoto; Yanqi, Chang; Xing, Zhang; Gilbert, Kirsch; Ettore, Novellino; Paola B., Arimondo; Miele, Evelina; Ferretti, Elisabetta; Gulino, Alberto; Marc, Diederich; Xiaodong, Cheng; Mai, Antonello | |
| Novel inhibitors of human histone deacetylases: Design, synthesis and bioactivity of 3-alkenoylcoumarines | 2014 | C., Seidel; M., Schnekenburger; Zwergel, Clemens; F., Gaascht; Mai, Antonello; M., Dicato; G., Kirsch; Valente, Sergio; M., Diederich | |
| Novel histone deacetylase inhibitors induce growth arrest, apoptosis, and differentiation in sarcoma cancer stem cells | 2015 | G., Di Pompo; M., Salerno; Rotili, Dante; Valente, Sergio; Zwergel, Clemens; S., Avnet; G., Lattanzi; N., Baldini; Mai, Antonello | |
| Emerging approaches for histone deacetylase inhibitor drug discovery | 2015 | Zwergel, Clemens; Valente, Sergio; Jacob, Claus; Mai, Antonello | |
| Abstract 2946: Effects of two novel quinoline-based non-nucleoside DNA methyltransferase inhibitors against bone sarcomas | 2015 | Manara, Maria Cristina; Valente, Sergio; Cristalli, Camilla; Baricordi, Cristina; Zwergel, Clemens; Arimondo, Paola B; Picci, Piero; Mai, Antonello; Scotlandi, Katia | |
| Histone deacetylase inhibitors restore IL-10 expression in lipopolysaccharide-induced cell inflammation and reduce IL-1β and IL-6 production in breast silicone implant in C57BL/6J wild-type murine model | 2016 | Di Liddo, Rosa; Valente, Sergio; Taurone, Samanta; Zwergel, Clemens; Marrocco, Biagina; Turchetta, Rosaria; Conconi, Maria Teresa; Scarpa, Carlotta; Bertalot, Thomas; Schrenk, Sandra; Mai, Antonello; Artico, Marco | |
| 1,4-Dihydropyridines Active on the SIRT1/AMPK Pathway Ameliorate Skin Repair and Mitochondrial Function and Exhibit Inhibition of Proliferation in Cancer Cells | 2016 | Valente, Sergio; Mellini, Paolo; Spallotta, Francesco; Carafa, Vincenzo; Nebbioso, Angela; Polletta, Lucia; Carnevale, Ilaria; Saladini, Serena; Trisciuoglio, Daniela; Gabellini, Chiara; Tardugno, Maria; Zwergel, Clemens; Cencioni, Chiara; Atlante, Sandra; Moniot, Sébastien; Steegborn, Clemens; Budriesi, Roberta; Tafani, Marco; Del Bufalo, Donatella; Altucci, Lucia; Gaetano, Carlo; Mai, Antonello | |
| DNA methyltransferases Inhibitors from natural sources | 2016 | Zwergel, Clemens; Valente, Sergio; Mai, Antonello | |
| One-pot synthesis of benzopyran-4-ones with cancer preventive and therapeutic potential | 2016 | Talhi, Oualid; Brodziak Jarosz, Lidia; Panning, Jana; Orlikova, Barbora; Zwergel, Clemens; Tzanova, Tzvetomira; Philippot, Stéphanie; Pinto, Diana C. G. A.; Paz, Filipe A. Almeida; Gerhaüser, Clarissa; Dick, Tobias P.; Jacob, Claus; Diederich, Marc; Bagrel, Denyse; Kirsch, Gilbert; Silva, Artur M. S. | |
| MC1568 inhibits HDAC6/8 activity and influenza A virus replication in lung epithelial cells: Role of Hsp90 acetylation | 2016 | Panella, Simona; Marcocci, Maria Elena; Celestino, Ignacio; Valente, Sergio; Zwergel, Clemens; Li Puma, Domenica Donatella; Nencioni, Lucia; Mai, Antonello; Palamara, ANNA TERESA; Simonetti, Giovanna | |
| LSD1 inhibitors: a patent review (2010-2015) | 2016 | Stazi, Giulia; Zwergel, Clemens; Valente, Sergio; Mai, Antonello | |
| Novel coumarin- and quinolinone-based polycycles as cell division cycle 25-A and -C phosphatases inhibitors induce proliferation arrest and apoptosis in cancer cells | 2017 | Zwergel, Clemens; Czepukojc, Brigitte; Evain Bana, Emilie; Xu, Zhanjie; Stazi, Giulia; Mori, Mattia; Patsilinakos, Alexandros; Mai, Antonello; Botta, Bruno; Ragno, Rino; Bagrel, Denise; Kirsch, Gilbert; Meiser, Peter; Jacob, Claus; Montenarh, Mathias; Valente, Sergio | |
| The histone methyltransferase EZH2 as a druggable target in SHH medulloblastoma cancer stem cells | 2017 | Miele, Evelina; Valente, Sergio; Alfano, Vincenzo; Silvano, Marianna; Mellini, Paolo; Borovika, Diana; Marrocco, Biagina; Po, Agnese; Besharat, Zein Mersini; Catanzaro, Giuseppina; Battaglia, Giuseppe; Abballe, Luana; Zwergel, Clemens; Stazi, Giulia; Milite, Ciro; Castellano, Sabrina; Tafani, Marco; Trapencieris, Peteris; Mai, Antonello; Ferretti, Elisabetta | |
| Metabolite profiling of ascidian Styela plicata using LC–MS with multivariate statistical analysis and their antitumor activity | 2017 | Palanisamy, S. K.; Trisciuoglio, D.; Zwergel, C.; Del Bufalo, D.; Mai, A. | |
| Epi-drugs in combination with immunotherapy: a new avenue to improve anticancer efficacy | 2017 | Mazzone, Roberta; Zwergel, Clemens; Mai, Antonello; Valente, Sergio | |
| Towards the development of activity-based probes for detection of lysine-specific demethylase-1 activity. | 2017 | Ourailidou, Me; Lenoci, A; Zwergel, Clemens; Rotili, Dante; Mai, Antonello; Dekker, F. j. 4. |
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