Sfoglia per Autore
3-(1H-pyrrol-2- and –3-yl)-2-oxazolidinones as novel potent and selective monoamine oxidase type A inhibitors.
2003 Mai, Antonello; Cervara, I.; Valente, Sergio; Artico, Marino; Sbardella, G.; Befani, Olivia; Turini, Paola; Agostinelli, Enzo
3-(1H-pyrrol-2- and –3-yl)-2-oxazolidinones as novel potent and selective monoamine oxidase type A inhibitors.
2003 Mai, Antonello; I., Cervara; Valente, Sergio; Artico, Marino; G., Sbardella; Befani, Olivia; Turini, Paola; Agostinelli, Enzo
3-(4-Aroyl-1-methyl-1H-pyrrol-2-yl)-N-hydroxy-2-propenamides as a new class of synthetic histone deacetylase inhibitors. 3. Discovery of novel lead compounds through structure-based drug design and docking studies.
2004 Ragno, Rino; Mai, Antonello; Massa, S; Cerbara, I; Valente, Sergio; Bottoni, P; Scatena, R; Jesacher, F; Loidl, P; Brosch, G.
3-(4-Aroyl-1-methyl-1H-2-pyrrolyl)-N-hydroxy-2-propenamides as a New Class of Synthetic Histone Deacetylase Inhibitors. 2. Effect of Pyrrole-C2 and/or -C4 Substitutions on Biological Activity
2004 Mai, Antonello; S., Massa; I., Cerbara; Valente, Sergio; Ragno, Rino; P., Bottoni; R., Scatena; P., Loidl; G., Brosch
Synthesis and biochemical evaluation of (R)-5-acyloxymethyl- and (S)-5-acylaminomethyl-3-(1H-pyrrol-1-yl)-2-oxazolidinones as new anti-monoamine oxidase (anti-MAO) agents.
2004 Mai, Antonello; Artico, Marino; Valente, Sergio; I., Cerbara; Befani, Olivia; Turini, Paola; L., Dalla Vedova; Agostinelli, Enzo
Antimalarial and Antileishmanial Activities of Aroyl-pyrrolyl-hydroxy-amides, a New Class of Histone Deacetylase Inhibitors
2004 Mai, Antonello; I., Cerbara; Valente, Sergio; S., Massa; L. A., Walker; B. L., Tekwani
Histone Deacetylation in Epigenetics: An Attractive Target for Anticancer Therapy
2005 Mai, Antonello; Massa, S; Rotili, Dante; Cerbara, I; Valente, Sergio; Pezzi, R; Simeoni, S; Ragno, Rino
3-(1H-Pyrrol-2-yl)-2-oxazolidinones as novel monoamine oxidase type A inhibitors.
2005 Mai, A; Artico, M.; Valente, S; Sbardella, G; Turini, P; Befani, O; DALLA VEDOVA, L; Agostinelli, E
Synthesis and biological evaluation of 2-, 3-, and 4-acylaminocinnamyl-N-hydroxyamides as novel synthetic HDAC inhibitors.
2005 Mai, Antonello; S., Massa; R., Pezzi; P., Loidl; G., Brosch; Valente, Sergio
Aroyl-pyrrolyl hydroxyamides: Influence of pyrrole C4-phenylacetyl substitution on histone deacetylase inhibition
2006 Mai, Antonello; Silvio, Massa; Valente, Sergio; Silvia, Simeoni; Ragno, Rino; Patrizia, Bottoni; Roberto, Scatena; Gerald, Brosch
3-D QSAR Studies on Histone Deacetylase Inhibitors. A GOLPE/GRID Approach on Different Series of Compounds.
2006 Ragno, Rino; Simeoni, S; Valente, Sergio; Massa, S; Mai, Antonello
New Aroyl-Pyrrolyl-Hydroxy-Amides APHAs: Class I and II Histone Deacetylase Inhibiting Activity and Binding Mode Analysis through Molecular Docking Experiments
2007 Ragno, Rino; Mai, Antonello; Simeoni, Silvia; Caroli, Antonia; Valente, Sergio; Perrone, Andrea
Novel pyrrole-containing histone deacetylase inhibitors endowed with cytodifferentiation activity
2007 Mai, Antonello; Valente, Sergio; Rotili, Dante; Silvio, Massa; Giorgia, Botta; Gerald, Brosch; Marco, Miceli; Angela, Nebbioso; Lucia, Altucci
Synthesis and biological validation of novel synthetic histone/protein methyltransferase inhibitors
2007 Mai, Antonello; Valente, Sergio; Donghang, Cheng; Andrea, Perrone; Ragno, Rino; Simeoni, Silvia; Gianluca, Sbardella; Gerald, Brosch; Mark t, Bedford
Identification of two new synthetic histone deacetylase inhibitors that modulate globin gene expression in erythroid cells from healthy donors and patients with thalassemia
2007 Mai, Antonello; K., Jelicic; Rotili, Dante; A., Di Noia; E., Alfani; Valente, Sergio; L., Altucci; A., Nebbioso; S., Massa; R., Galanello; G., Brosch; A. R., Migliaccio; G., Migliaccio
Design, synthesis and biological validation of epigenetic modulators of histone/protein deacetylation and methylation
2007 Valente, Sergio
HDAC-class II specific inhibition involves HDAC proteasome-dependent degradation mediated by RANBP2
2008 Annamaria, Scognamiglio; Angela, Nebbioso; Fabio, Manzo; Valente, Sergio; Mai, Antonello; Lucia, Altucci
Specific Activity of Class II Histone Deacetylases in Human Breast Cancer Cells
2008 V., Duong; C., Bret; L., Altucci; Mai, Antonello; C., Duraffourd; J., Loubersac; P. O., Harmand; S., Bonnet; Valente, Sergio; T., Maudelonde; V., Cavailles; N., Boulle
Novel uracil-based 2-aminoanilide and 2-aminoanilide-like derivatives: Histone deacetylase inhibition and in-cell activities
2008 Mai, Antonello; Andrea, Perrone; Angela, Nebbioso; Rotili, Dante; Valente, Sergio; Maria, Tardugno; Silvio, Massa; Floriana De, Bellis; Lucia, Altucci
Nitric oxide modulates chromatin folding in human endothelial cells via protein phosphatase 2A activation and class II histone deacetylases nuclear shuttling
2008 Illi, B.; DELLO RUSSO, Claudio; Colussi, C.; Rosati, J.; Pallaoro, M.; Spallotta, F.; Rotili, Dante; Valente, Sergio; Ragone, G.; Martelli, F.; Biglioli, P.; Steinkuhler, C.; Gallinari, P.; Mai, Antonello; Capogrossi, M. C.; Gaetano, C.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
3-(1H-pyrrol-2- and –3-yl)-2-oxazolidinones as novel potent and selective monoamine oxidase type A inhibitors. | 2003 | Mai, Antonello; Cervara, I.; Valente, Sergio; Artico, Marino; Sbardella, G.; Befani, Olivia; Turini, Paola; Agostinelli, Enzo | |
3-(1H-pyrrol-2- and –3-yl)-2-oxazolidinones as novel potent and selective monoamine oxidase type A inhibitors. | 2003 | Mai, Antonello; I., Cervara; Valente, Sergio; Artico, Marino; G., Sbardella; Befani, Olivia; Turini, Paola; Agostinelli, Enzo | |
3-(4-Aroyl-1-methyl-1H-pyrrol-2-yl)-N-hydroxy-2-propenamides as a new class of synthetic histone deacetylase inhibitors. 3. Discovery of novel lead compounds through structure-based drug design and docking studies. | 2004 | Ragno, Rino; Mai, Antonello; Massa, S; Cerbara, I; Valente, Sergio; Bottoni, P; Scatena, R; Jesacher, F; Loidl, P; Brosch, G. | |
3-(4-Aroyl-1-methyl-1H-2-pyrrolyl)-N-hydroxy-2-propenamides as a New Class of Synthetic Histone Deacetylase Inhibitors. 2. Effect of Pyrrole-C2 and/or -C4 Substitutions on Biological Activity | 2004 | Mai, Antonello; S., Massa; I., Cerbara; Valente, Sergio; Ragno, Rino; P., Bottoni; R., Scatena; P., Loidl; G., Brosch | |
Synthesis and biochemical evaluation of (R)-5-acyloxymethyl- and (S)-5-acylaminomethyl-3-(1H-pyrrol-1-yl)-2-oxazolidinones as new anti-monoamine oxidase (anti-MAO) agents. | 2004 | Mai, Antonello; Artico, Marino; Valente, Sergio; I., Cerbara; Befani, Olivia; Turini, Paola; L., Dalla Vedova; Agostinelli, Enzo | |
Antimalarial and Antileishmanial Activities of Aroyl-pyrrolyl-hydroxy-amides, a New Class of Histone Deacetylase Inhibitors | 2004 | Mai, Antonello; I., Cerbara; Valente, Sergio; S., Massa; L. A., Walker; B. L., Tekwani | |
Histone Deacetylation in Epigenetics: An Attractive Target for Anticancer Therapy | 2005 | Mai, Antonello; Massa, S; Rotili, Dante; Cerbara, I; Valente, Sergio; Pezzi, R; Simeoni, S; Ragno, Rino | |
3-(1H-Pyrrol-2-yl)-2-oxazolidinones as novel monoamine oxidase type A inhibitors. | 2005 | Mai, A; Artico, M.; Valente, S; Sbardella, G; Turini, P; Befani, O; DALLA VEDOVA, L; Agostinelli, E | |
Synthesis and biological evaluation of 2-, 3-, and 4-acylaminocinnamyl-N-hydroxyamides as novel synthetic HDAC inhibitors. | 2005 | Mai, Antonello; S., Massa; R., Pezzi; P., Loidl; G., Brosch; Valente, Sergio | |
Aroyl-pyrrolyl hydroxyamides: Influence of pyrrole C4-phenylacetyl substitution on histone deacetylase inhibition | 2006 | Mai, Antonello; Silvio, Massa; Valente, Sergio; Silvia, Simeoni; Ragno, Rino; Patrizia, Bottoni; Roberto, Scatena; Gerald, Brosch | |
3-D QSAR Studies on Histone Deacetylase Inhibitors. A GOLPE/GRID Approach on Different Series of Compounds. | 2006 | Ragno, Rino; Simeoni, S; Valente, Sergio; Massa, S; Mai, Antonello | |
New Aroyl-Pyrrolyl-Hydroxy-Amides APHAs: Class I and II Histone Deacetylase Inhibiting Activity and Binding Mode Analysis through Molecular Docking Experiments | 2007 | Ragno, Rino; Mai, Antonello; Simeoni, Silvia; Caroli, Antonia; Valente, Sergio; Perrone, Andrea | |
Novel pyrrole-containing histone deacetylase inhibitors endowed with cytodifferentiation activity | 2007 | Mai, Antonello; Valente, Sergio; Rotili, Dante; Silvio, Massa; Giorgia, Botta; Gerald, Brosch; Marco, Miceli; Angela, Nebbioso; Lucia, Altucci | |
Synthesis and biological validation of novel synthetic histone/protein methyltransferase inhibitors | 2007 | Mai, Antonello; Valente, Sergio; Donghang, Cheng; Andrea, Perrone; Ragno, Rino; Simeoni, Silvia; Gianluca, Sbardella; Gerald, Brosch; Mark t, Bedford | |
Identification of two new synthetic histone deacetylase inhibitors that modulate globin gene expression in erythroid cells from healthy donors and patients with thalassemia | 2007 | Mai, Antonello; K., Jelicic; Rotili, Dante; A., Di Noia; E., Alfani; Valente, Sergio; L., Altucci; A., Nebbioso; S., Massa; R., Galanello; G., Brosch; A. R., Migliaccio; G., Migliaccio | |
Design, synthesis and biological validation of epigenetic modulators of histone/protein deacetylation and methylation | 2007 | Valente, Sergio | |
HDAC-class II specific inhibition involves HDAC proteasome-dependent degradation mediated by RANBP2 | 2008 | Annamaria, Scognamiglio; Angela, Nebbioso; Fabio, Manzo; Valente, Sergio; Mai, Antonello; Lucia, Altucci | |
Specific Activity of Class II Histone Deacetylases in Human Breast Cancer Cells | 2008 | V., Duong; C., Bret; L., Altucci; Mai, Antonello; C., Duraffourd; J., Loubersac; P. O., Harmand; S., Bonnet; Valente, Sergio; T., Maudelonde; V., Cavailles; N., Boulle | |
Novel uracil-based 2-aminoanilide and 2-aminoanilide-like derivatives: Histone deacetylase inhibition and in-cell activities | 2008 | Mai, Antonello; Andrea, Perrone; Angela, Nebbioso; Rotili, Dante; Valente, Sergio; Maria, Tardugno; Silvio, Massa; Floriana De, Bellis; Lucia, Altucci | |
Nitric oxide modulates chromatin folding in human endothelial cells via protein phosphatase 2A activation and class II histone deacetylases nuclear shuttling | 2008 | Illi, B.; DELLO RUSSO, Claudio; Colussi, C.; Rosati, J.; Pallaoro, M.; Spallotta, F.; Rotili, Dante; Valente, Sergio; Ragone, G.; Martelli, F.; Biglioli, P.; Steinkuhler, C.; Gallinari, P.; Mai, Antonello; Capogrossi, M. C.; Gaetano, C. |
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